Patents
Patents for C07D 215 - Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems (27,676)
09/2000
09/21/2000WO2000055126A2 N-cyanomethylamides as protease inhibitors
09/21/2000WO2000055125A2 N-cyanomethyl amides as protease inhibitors
09/21/2000WO2000055116A1 Process for producing 5-amino-8- alkylquinolo necarboxylic acid derivatives and intermediates in the production thereof
09/21/2000WO2000054759A2 Lxr modulators
09/21/2000DE19911509A1 Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung Bicyclic heterocycles, pharmaceutical compositions containing them, their use and process for their preparation
09/21/2000CA2368148A1 Novel compounds and compositions as protease inhibitors
09/21/2000CA2368122A1 Novel compounds and compositions as protease inhibitors
09/21/2000CA2367595A1 Lxr modulators
09/20/2000EP1036067A2 Pdgf receptor kinase inhibitory compounds, their preparation and compositions
09/20/2000EP1035843A2 I h?-MODULATORS
09/20/2000EP1001686A4 Dehydration plant
09/20/2000CN1267284A Carbostyril derivs. for inhibiting skin erythema and/or skin pigmentation
09/20/2000CN1267281A Glucagon antagonists/inverse agonists
09/20/2000CN1056602C Esters and amides as PLAZ inhibitors
09/19/2000US6121452 Process for the preparation of quinophthalones
09/19/2000US6121450 Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors
09/19/2000US6121308 Indole and benzimidazole antithrombotic compounds, such as 1-methyl-2-(n-(4-amidinophenyl)-aminomethyl)-5-(n-(hydroxycarbonylmethyl) -quinoline-8-sulphonylamino)-indole
09/19/2000US6121287 Quinoline derivatives
09/19/2000US6121285 Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives
09/19/2000US6121284 Specified 1-(alkyl or cycloalkyl)-2-methyl-3-(alkoxycarbonyl)-4-(substituted pyridyl or aryl)-5-oxo-1,4,5,6,7,8-hexahydroquinoline compounds; treating sickle cell anemia, psychoses, depression
09/14/2000WO2000053577A1 Hydrazide inhibitors of hiv-1 integrase
09/14/2000WO2000031074A3 Indole derivatives and their use as serotonin receptor ligands
09/14/2000WO1999063999A8 H1-histamine receptor antagonists
09/13/2000EP1034173A2 Method for producing 8-methoxy-quinoline carboxylic acids
09/13/2000EP0691962B1 1-amino-3-phenoxy propane derivatives as modulators of multi-drug resistance
09/13/2000CN1266426A Microbicidal N-sulfonylglycin alkynyloxyphenemethyl amide derivatives
09/13/2000CN1056373C Process for preparation of fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles
09/12/2000US6118010 Catalytic reduction of the 1-alkoxycarbonyl-3-oxo-3-phenylpropyl derivative
09/12/2000US6118001 Anticancer agent; antiarthritic agent
09/12/2000US6117884 4-substituted quinoline derivatives having fungicidal activity
09/08/2000WO2000051991A1 4-AMINO-QUINAZOLINE AND QUINOLINE DERIVATIVES HAVING AN INHIBITORY EFFECT ON SIGNAL TRANsSDUCTION MEDIATED BY TYROSINE KINASES
09/08/2000WO2000051971A1 Oxamic acids and derivatives as thyroid receptor ligands
09/08/2000WO2000051608A1 3-thienyl and 3-furanyl pyrrolidine modulators of chemokine receptor activity
09/08/2000WO2000034260A3 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group
09/06/2000EP1032559A1 Aminoalkylphenol derivatives and related compounds
09/06/2000EP1032556A1 Pharmaceutically active compounds and methods of use
09/06/2000EP1032393A1 QUINOLINE-CONTAINING $g(a)-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS
09/06/2000EP1032377A1 Substituted 2-aminoacetamides and the use thereof
09/06/2000EP0824514B1 Dihalopropene compounds, insecticides containing them as active ingredients, and intermediates for their production
09/06/2000EP0702672B1 Substituted quinoline derivatives and their use as inhibitors of gastric acid secretion
09/06/2000EP0593766B1 Pyridonecarboxylic acid derivative
09/06/2000CN1265645A Urokinase inhibitors
09/05/2000US6114531 Reacting 7-chloro-1-(2,4-difluorophenyl)-6-fluoro-1,4-dihydro-4-oxo-1,8 -naphthyridine-3-carboxylic acid with a fused aminoaromatic salt to from trovafloxacin
09/05/2000US6114524 Process for producing halogenated heteroaryl compounds
09/05/2000US6114381 To control brain damage associated with anoxia or ischemia which typically follows stroke, cardiac arrest or perinatal asphyxia; compound is an antagonist to inhibit excitotoxic actions at excitatory amino acid receptor sites
09/05/2000US6114352 Quinolinone derivative and anti-allergic agent with said quinolinone derivative as the active ingredient
09/05/2000US6114351 N-oxides as antibacterial agents
09/05/2000US6114349 Substituted quinoline derivatives with antiviral action
08/2000
08/31/2000WO2000050428A1 Process for preparing (-)pyridobenzoxazine carboxylic acid derivatives
08/31/2000WO2000050405A1 Quinoline derivatives as tyrosine kinase inhibitors
08/31/2000WO2000050404A1 4-aminoquinolines as antimalarials
08/31/2000WO2000050396A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
08/31/2000WO2000040558A8 Aspartic protease inhibitors
08/31/2000DE19908567A1 New 4-amino-quinazoline or quinoline derivatives, are tyrosine kinase-mediated signal transduction inhibitors useful e.g. for treating tumors, polyps or respiratory or gastrointestinal diseases
08/31/2000CA2371876A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
08/30/2000EP1031569A1 Processes for producing 7-isoindolinequinolonecarboxylic derivatives and intermediates therefor, salts of 7-isoindolinequinolonecarboxylic acids, hydrates thereof, and composition containing the same as active ingredient
08/30/2000EP1031563A1 Sulfonyl derivatives
08/30/2000EP1031555A1 N-cyclopropyl-2-difluoromethoxy-3-halogenoanilines and intermediates for the preparation thereof
08/30/2000EP1030665A1 Therapeutic uses of quinoline derivatives
08/30/2000CN1265096A Hydrazine derivatives
08/30/2000CN1265010A Dehydration plant
08/29/2000US6110933 Amino acid derivatives and their use as phospholipase A2 inhibitor
08/29/2000US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
08/24/2000WO2000048993A1 Arylaminoalkylamides
08/24/2000WO2000031051B1 Quinoline and quinoxaline compounds as pdgf-receptor and/or lck tyrosine kinase inhibitors
08/24/2000WO1996012697A9 Calcium receptor-active compounds
08/23/2000EP1029861A1 Benzisothiazol-piperazinyl derivative and its use as neuroleptic
08/23/2000EP1028942A2 Dipeptide nitriles
08/23/2000EP0658159B1 Arylidene and heteroarylidene oxindole derivatives as tyrosine kinase inhibitors
08/23/2000CN1264378A Quinoline-4-carboxamide derivatives as NK-2 and NK-3 receptor antagonists
08/23/2000CN1264362A Method for preparing 4-(alkyl)-3-alkoxy-aniline compounds
08/22/2000US6107066 Coumarin derivative-n-linked lipid used as a fluorophore capable of undergoing energy transfer
08/17/2000WO2000047577A1 Phenyl urea and phenyl thiourea derivatives as orexin receptor antagonists
08/17/2000WO2000047576A1 Cinnamide derivatives as orexin-1 receptors antagonists
08/17/2000WO2000047574A1 Heteroaryl-substituted quinolin-2-one derivatives useful as anticancer agents
08/17/2000WO2000012076A9 Nitrosated and nitrosylated phosphodiesterase inhibitors, compositions and methods of use
08/16/2000EP1028113A1 Fused benzene heterocycle derivatives and utilization thereof
08/16/2000EP1028112A1 Phenylglycinolamides linked by a hetero-atom with antiatherosclerotic agents
08/16/2000EP1028111A1 Amide derivatives or salts thereof
08/16/2000EP1027336A1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors
08/16/2000EP0738259B1 Phenyl acetic acid derivatives, process and intermediate products for their production and agents containing them
08/16/2000CN1055468C Alkylaminoindane compounds process for preparing them and pharmaceutical compositions containing them,and use
08/15/2000US6103936 Reacting aldehyde, sulfide, sulfone, or sulfoxide with formamide in presence of acid catalyst, and optionally a dehydrating agent
08/15/2000US6103905 Quinoline-indole antimicrobial agents, uses and compositions related thereto
08/15/2000US6103904 Reacting sulfuric acid with an aniline, adding catalyst and an unsaturated aldehyde or glycerol while refluxing and increasing pressure and temperature to form quinoline with high yield
08/15/2000US6103738 Quinoline and quinazoline compounds useful in therapy
08/15/2000US6103732 Endothelin receptor inhibitors; hypotensive agents, cardiotonic agents; acute myocardial infarct, pulmonary hypertension, raynaud's syndrome, atherosclerosis; asthma; cardiovascular disorders
08/15/2000US6103721 Heteroaryl-substituted pyridazino quinoline compounds
08/15/2000US6103720 Ketobenzamides as calpain inhibitors
08/10/2000WO2000046184A1 N2-phenylamidine derivatives
08/10/2000WO1999063936A9 Novel therapeutic agents that modulate endothelin receptors
08/10/2000WO1999056666A8 The treatment of sexual dysfunction in certain patient groups
08/09/2000EP1026157A2 Method for the synthesis of huperzine A and analogs thereof and compounds useful therein
08/09/2000EP1026151A1 Aryl and heteroarylcyclopropyl oxime ethers and their use as fungicides and insecticides
08/09/2000EP1026149A1 Amidocarboxylic acid derivatives
08/09/2000EP1025846A1 Aqueous liquid preparations
08/09/2000EP1025097A1 1-(2-naphthyl) and 1-(2-azanaphthyl)-4-(1-phenylmethyl)piperazines being dopamine d 4? receptor subtype ligands
08/09/2000EP1025086A1 Benzamidine derivatives as factor xa inhibitors
08/09/2000CN1262676A 吡啶衍生物 Pyridine derivatives
08/09/2000CN1262620A Beta-Alkoxyacrylates against malaria