Patents
Patents for C07D 215 - Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems (27,676)
03/2001
03/14/2001EP1082127A1 SUCCINAMIDE INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME
03/14/2001EP0681570B1 Process for preparing quinoline amines
03/14/2001CN1287553A Fused benzene heterocycle derivatives and utilization thereof
03/13/2001US6201020 Effective poly(adenosine 5'-diphospho-ribose) polymerase (parp) inhibitor for treatment of tissue damage by necrosis or apoptosis; side effect reduction
03/13/2001US6200995 Pyridyloxybenzenesulfonamide derivatives; diabetes, obesity
03/13/2001US6200976 Antithrombotic quinoxazolines
03/08/2001WO2001016108A2 Bicyclic androgen and progesterone receptor modulator compounds and methods
03/08/2001WO2001016107A1 Arylalkyloxyalkylamines and arylalkylthioalkylamines, pharmaceutical compositions containing them and their use as inhibitors of nicotinic cholinergic receptors
03/08/2001WO1999064047A8 Novel antiviral compounds
03/08/2001WO1999063930A8 Novel angiotensin receptor modulators and their uses
03/08/2001WO1999039704A8 Antibacterial agents
03/08/2001WO1999019296A8 Aminobutanoic acid derivatives
03/08/2001CA2384435A1 Bicyclic androgen and progesterone receptor modulator compounds and methods
03/08/2001CA2383307A1 Arylalkyloxyalkylamines and arylalkylthioalkylamines, pharmaceutical compositions containing them and their use as inhibitors of nicotinic cholinergic receptors
03/07/2001EP1081138A1 1,2-disubstituted 1,4-dihydro-4-oxoquinoline compounds
03/07/2001EP1080086A1 Dihydropyrimidines
03/07/2001EP1080083A1 Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
03/07/2001EP1080080A1 Novel therapeutic agents that modulate neurokinin receptors
03/07/2001EP1080074A1 New heterocyclically substituted amides, their production and their use
03/07/2001EP1079821A1 Protease inhibitors
03/07/2001EP1079764A1 The treatment of sexual dysfunction in certain patient groups
03/07/2001CN1286684A Carboxamide derivs. of pyrrolidine, piperidine and hexahydroazepine for treatment of thrombosis disorders
03/06/2001US6197968 Storage stability; colorless after solution treatment
03/06/2001US6197791 N-hdroxy-2-(alkyl, aryl, or heteroaryl, sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors
03/06/2001US6197786 Anticholesterol agents
03/06/2001US6197782 Therapy for sexual disorders
03/06/2001US6197778 Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
03/01/2001WO2001014328A2 Substituted ureas as cell adhesion inhibitors
03/01/2001DE19940394A1 New water-soluble, reactive 4,4'-cyanine dye-based fluorochromes having high quantum yield, useful as fluorescent labelling dyes for analytical use, e.g. in fluorescence immunoassays or other bioassays
02/2001
02/28/2001EP1077978A1 Novel substituted aryl hydroxamic acids as metalloproteinase inhibitors
02/28/2001EP1077957A1 Oxyiminoalkanoic acid derivatives with hypoglycemic and hypolipidemic activity
02/28/2001EP1077944A1 Carboxamide compounds, compositions, and methods for inhibiting parp activity
02/28/2001EP1077920A1 New compounds, their preparation and use
02/28/2001EP1077919A1 New compounds, their preparation and use
02/28/2001CN1285820A Metabotropic glutamate receptor antagonists for treating central nervous system disease
02/28/2001CN1062555C Substituted benzyloxy carbonyl guanidine, its prepn. method, and application of the same as medicament and medicament containing the same
02/27/2001US6194493 4-hydroxyquinoline-3-carboxylic acid derivatives as light stabilizers
02/27/2001US6194451 Prevent release tumor necrosis factor; antiinflammatory agents
02/27/2001US6194450 Polyaromatic heterocyclic compounds and pharmaceutical compositions comprised thereof
02/27/2001US6194439 Tricyclic polyhydroxylic tyrosine kinase inhibitors
02/27/2001US6194428 Use of 5-substituted pyridine and hexahydroquinoline-3 carboxylic acid derivatives for treating diseases of the central nervous system
02/27/2001US6194427 Brain disorders; psychological disorders; sleep disorders; anticonvulsants
02/27/2001CA2316662A1 Use of crf antagonists and related compositions
02/22/2001WO2001012608A1 Quinoline compounds and process for producing the same
02/22/2001WO2001012607A2 Pharmaceutical compositions comprising 4-quinolones for treating cancers
02/22/2001WO2001012606A2 Tetrahydroquinoline derivatives having retinoid-like biological activity
02/22/2001WO2001012605A1 6,7-disubstituted-5,8-quinolinedione derivatives as an antifungal agent
02/22/2001WO2001012600A1 INHIBITORS OF FACTOR Xa
02/22/2001WO2001012597A2 Method for preparing quinoline-5,8-diones
02/22/2001WO2001012591A1 Novel naphthylsulfonic acids and related compounds as glucose uptake agonists
02/22/2001WO2001012187A2 Benzoic acid derivatives and their use as ppar receptor agonists
02/22/2001WO2000071514A8 α-AMINO-β-SULFONYL HYDROXAMIC ACID COMPOUNDS
02/22/2001WO2000071500A8 Halogen compounds
02/22/2001WO2000055126A3 N-cyanomethylamides as protease inhibitors
02/22/2001WO1999063996A8 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht2 receptors
02/22/2001CA2381971A1 Amines substituted with a tetrahydroquinolinyl group, an aryl or heteroaryl group and an alkyl group, having retinoid-like biological acitity
02/22/2001CA2381968A1 Pharmaceutical compositions comprising 4-quinolones for treating cancers
02/22/2001CA2380775A1 Benzoic acid derivatives and their use as ppar receptor agonists
02/21/2001EP1076648A1 Method for the catalytic production of substituted dipyridyl derivatives
02/21/2001EP1076557A1 Ccr-3 receptor antagonists
02/21/2001CN1284878A Drugs augmenting NKT cells
02/21/2001CN1062270C Amino-acid derrivatives having benzothiophene ring, prep. thereof and use as fungus-killing agent
02/21/2001CN1062268C Alcohol to azide SN2 conversion
02/21/2001CN1062264C Amino-acid indole or quinoline derivatives, prep. thereof and use as fungus-killing agent
02/20/2001US6191157 Anticholesterol agents; cardiovascular disorders
02/20/2001US6191135 Respiratory system disorders, antiinflammatory agents; analgesics
02/15/2001WO2001010842A2 Melanocortin-4 receptor binding compounds and methods of use thereof
02/15/2001WO2001010827A1 Arylsulfonamido-substituted hydroxamic acid derivatives
02/15/2001WO2001010825A1 Carbamate derivatives and agricultural/horticultural bactericides
02/15/2001WO2000054759A3 Lxr modulators
02/15/2001DE19936472A1 Haftvermittler Adhesion promoter
02/15/2001CA2381008A1 Melanocortin-4 receptor binding compounds and methods of use thereof
02/15/2001CA2378310A1 Arylsulfonamido-substituted hydroxamic acid derivatives
02/14/2001EP0828714B1 Method for making quinolone carboxylic acids or naphthyridine carboxylic acids in free base form
02/13/2001US6187943 Catalyzing the reaction in the presence of a metal oxide catalyst containing vanadium and/or molybdenum in a fluidized bed
02/13/2001US6187926 Process for producing quinolone derivatives
02/13/2001US6187786 Antitumor and anticarcinogenic agents
02/13/2001CA2001203C Novel antimicrobial dithiocarbamoyl quinolones
02/08/2001WO2001009099A2 Bonding agent
02/08/2001WO2001009096A2 Potassium channel openers
02/08/2001WO2001009095A1 Mutilin derivatives and their use as antibacterials
02/08/2001WO2001009088A1 Urea derivatives as inhibitors of ccr-3 receptor
02/08/2001CA2378936A1 Potassium channel openers
02/07/2001EP1073662A1 Process for preparing (-)pyridobenzoxazine carboxylic acid derivatives
02/07/2001EP1073639A1 Quinoline derivatives
02/07/2001EP1073631A1 New substituted amides, their production and their use
02/07/2001EP1073624A1 Aminomethyl-benzoic ester derivatives as tryptase inhibitors
02/07/2001EP1073434A1 Ccr-3 receptor antagonists
02/07/2001EP0533882B1 2-quinolinone derivatives, methods for preparing the same and fungicides and insecticides including them
02/07/2001CN1283195A 1-(2-naphthyl) and 1(2-azanaphthyl)-4-(1-phenylmethyl)piperazines being dopamine D4 receptor subtype ligands
02/07/2001CN1283180A Inhibition of raf kinase using symmerical and unsymmerical substituted diphenyl ureas
02/07/2001CN1282737A Intermediate product used for preparing substituted quinoline-2-formamide
02/07/2001CN1282736A Method of preparing medicinal active substance derived from quinogold
02/07/2001CN1282735A Amphiphili 8-hydroxyquinoline complex, its preparing process and its application in electroluminescence
02/06/2001US6184388 Antibacterial and antimicrobial, quinoline antibiotic
02/06/2001US6184231 3-substituted-4-arylquinolin-2-one derivatives as potassium channel modulators
02/06/2001US6184230 Administering orally a quinolone antibiotic comprising 1-hydroxy-2-(2-trans-nonenyl)-3-methyl-4(1h)-quinolone or salt to treat gastrointestinal disorders, lymphomas, chronic heart disease
02/06/2001CA2126118C 5-amino-8-methyl-7-pyrrolidinylquinoline-3-carboxylic acid derivative
02/01/2001WO2001007533A1 Electron-driven chirality switches
02/01/2001WO2001007036A1 BICYCLIC ANTAGONISTS SELECTIVE FOR THE αvβ3 INTEGRIN