Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
05/2008
05/14/2008EP1921064A1 Pharmaceutical composition
05/14/2008EP1920773A1 Compositions for inhibition of anglogenesis
05/14/2008EP1919909A2 Synthetic methods and intermediates for stereoisomeric compounds useful for the treatment of gastrointestinal and central nervous system disorders
05/14/2008EP1723114B1 Biphenyl compounds useful as muscarinic receptor antagonists
05/14/2008CN101180296A Heteroaryl-carboxylic acid (sulfamoyl alkyl) amide - derivatives as factor Xa inhibitors
05/14/2008CN101180288A Aromatic substituted pentadienoic acid amide for combination with anti-infective drugs
05/14/2008CN100387579C Graftable hindered amine light stabilizers
05/13/2008US7371867 Non-racemic trifluoroleucine, and methods of making and using
05/13/2008US7371761 Lactam-containing compounds and derivatives thereof as factor Xa inhibitors
05/13/2008US7371753 Dihydropteridinones, processes for preparing them and their use as pharmaceutical compositions
05/13/2008US7371747 Cyanoalkylamino derivatives as protease inhibitors
05/08/2008WO2008054290A1 1h-pyridine- 2 -one derivatives useful in treatment of pai-1 related disorders
05/08/2008WO2008054096A1 Crystalline s-(-)-amlodipine adipic acid salt anhydrous and preparation method thereof
05/08/2008WO2008053913A1 Sulfonylurea derivative capable of selectively inhibiting mmp-13
05/08/2008WO2008053352A2 Phenylpropionamide compounds and the use thereof
05/08/2008WO2008052899A1 Ether derivatives dual modulators of the 5-ht2a and d3 receptors
05/08/2008WO2008052769A1 Phenylamino-substituted piperidine compounds, their preparation and use as medicaments
05/08/2008WO2008024371A3 Multimediator transporter inhibitors for use in treatment of central nervous system disorders
05/08/2008WO2008010953A3 Pyridinone diketo acids: inhibitors of hiv replication in combination therapy
05/08/2008US20080108825 Compounds for treatment of inflammation, diabetes and related disorders
05/08/2008US20080108824 Has a bioactive ( being less soluble in water when the proton binding site is in the non-ionic form than when the proton binding site is in the ionic form) and having a desired rate of bioactive release
05/08/2008US20080108820 First isolated from the sponge Hemiasterella; for treatment of cancer; prevention of restenosis of blood vessels subject to traumas such as angioplasty and stenting; methods for synthetic preparation
05/08/2008US20080108691 For example, 1-(4-Cyano-2-ethyl-3-(trifluoromethyl)phenyl-1-carbamoyl)-3-hydroxy-pyrrolidine-2-carboxylic acid methyl ester; may be used in treatment of diseases or disorders associated with androgen receptor activity, such as maintenance of muscle strength and function in the elderly
05/08/2008US20080108667 [(5,6-dichloropyridin-3-yl)methyl](methyl)-oxido lambda 4-sulfanylidenecyanamide; Insecticides; potentiation; atypical mode of action; effective control in agricultural, urban and/or animal health systems by applying to a locus; control of foliar-feeding insects; aphids and other sucking insects
05/08/2008US20080108663 Cyclopropyl Piperidine Glycine Transporter Inhibitors
05/08/2008US20080108662 Biaryloxymethylarenecarboxylic acids as glycogen synthase activator
05/08/2008US20080108660 such as 4-{[4-({[(3-isopropyl-2-oxo-2,3-dihydro-1H-benzimidazol-1-yl)carbonyl]amino}methyl)piperidin-1-yl]methyl}tetrahydro-2H-pyran-4-carboxylic acid; serotonin receptor agonist; antidepressant, anxiolytic agent, analgesic, cognition activator; less toxicity, good absorption, and metabolic stability
05/08/2008US20080108618 Compounds with activity on muscarinic receptors
05/08/2008US20080108594 Antithrombotic Ethers
05/08/2008CA2667511A1 Ether derivatives dual modulators of the 5-ht2a and d3 receptors
05/08/2008CA2666750A1 Phenylpropionamide compounds and the use thereof
05/07/2008EP1918281A1 Phenylamino-substituted piperidine compounds, their preparation and use as medicaments
05/07/2008EP1918280A1 Process for the preparation of 2,5-bis-(2,2,2-trifluoroethoxy)-N-(2-piperidylmethyl)-benzamide and salts thereof
05/07/2008EP1918279A2 1-(4-piperidinyl)-1,3-dihydro-2h-benzoxazole-2-one derivatives and related compounds as nociceptin analogs and opioid receptor like receptor (ORL1) ligands for the treatment of pain
05/07/2008EP1918272A1 Pharmaceutically active compounds and methods of use
05/07/2008EP1722795B1 Piperidinyl prostaglandin e analogs
05/07/2008EP1641729B1 Use of functionalized onium salts as a soluble support for organic synthesis
05/07/2008EP1558606A4 Lactam-containing diaminoalkyl, beta-aminoacids, alpha-aminoacids and derivatives thereof as factor xa inhibitors
05/07/2008CN101175726A Process for the preparation of opioid modulators
05/07/2008CN101175725A Process for the preparation of opioid modulators
05/07/2008CN101172965A Piperidine ester compounds for producing catalyst for polymerization of olefins and catalyst thereof
05/07/2008CN101172964A 3-(4-piperidine group) substituted tetrahydronaphthalene derivative compounds and synthesis method thereof
05/07/2008CN100386313C Novel herbicides
05/06/2008US7368568 Protected 3,5-dihydroxy-2,2-dimethyl-valeroamides for the synthesis of epothilones and derivatives and process for production and the use
05/06/2008US7368462 4'-Fluoro-biphenyl-4-carboxylic acid (6-dimethylaminomethyl-naphthalen-1-ylmethyl)-amide; obesity; side effects reduction; selective binding; no stimulation of the central nervous system and no peripheral activity caused by activation of 5-HT2c receptors; improved cellular potency and pharmacokinetics
05/06/2008US7368461 Compounds and method for the treatment of overactive bladder
05/06/2008US7368443 Central nervous system disorders, drug abuse, obesity
05/02/2008WO2008051875A2 Adamantylurea compounds as soluble epoxide hydrolase inhibitors
05/02/2008WO2008051873A2 Phenylurea compounds as soluble epoxide hydrolase inhibitors
05/02/2008WO2008051056A1 Method for the separation of s-(-)-amlodipine from racemic amlodipine
05/02/2008WO2008050857A1 Amide compound or salt thereof, and biofilm formation inhibitor, biofilm remover and bactericide each using the amide compound or salt thereof
05/02/2008WO2008050351A1 NOVEL POLYMORPHIC FORMS OF l-BENZYL-4-[(5,6-DIMETHOXY-l-INDANONE)-2-YL]METHYL PIPERIDINE [DONEPEZIL] AND PROCESS FOR PREPARING THE SAME
05/02/2008WO2008050168A1 New sulfonamide derivatives as bradykinin antagonists
05/02/2008WO2008050167A1 New phenylsulfamoyl benzamide derivatives as bradykinin antagonists
05/02/2008WO2008049806A1 Piperidine or piperazine substituted tetrahydro-naphthalene-1-carboxylic acid mtp inhibiting compounds
05/02/2008CA2666482A1 Soluble epoxide hydrolase inhibitors
05/02/2008CA2664141A1 Piperidine or piperazine substituted tetrahydro-naphthalene-1-carboxylic acid mtp inhibiting compounds
05/01/2008US20080103311 Retroviral protease inhibitors
05/01/2008US20080103302 Novel acyl urea, thiourea, carbamate, thiocarbamate and related compounds are provided which are effective in inhibiting the cytokine-mediated inflammatory response in cultured cells, in ameliorating bone destruction in an animal model of arthritis and in lowering blood glucose levels in animal or cancer
05/01/2008US20080103229 Curable acrylic mixture including a hindered amine light stabilizer having a 4-Amino-2,2,6,6-tetramethylpiperidin-1 oxyl moiety linked to an acrylic moiety so as to polymerize with the primary resin
05/01/2008US20080103180 CCR9 inhibitors and methods of use thereof
05/01/2008US20080103176 N-{1-(3,5-Difluoro-benzyl)-3-[7-(2,2-dimethyl-propyl)-2-piperidin-1-yl-1,2,3,4-tetrahydro-naphthalen-1-ylamino]-2-hydroxy-propyl}-acetamide; 13-secretase inhibitor; Alzheimer's disease; inhibitors of beta-secretase, that inhibit beta-secretase-mediated cleavage of amiloid precursor protein APP
05/01/2008US20080103139 3-Carbamoyl-2-Pyridone Derivative
05/01/2008US20080103135 Histamine H3 antagonists; do not contain imidazolyl moiety; such as 1-[4-(4-piperidin-1-ylmethyl-phenyl)-but-3-ynyl]-piperidine
05/01/2008US20080103123 4-phenyl-3-substituted pyridin compounds such as tert-Butyl 4-[({5-[4-(methylsulfonyl)phenyl]pyridin-2-yl}oxy)methyl]-piperidine-1-carboxylate; agonists of the G-protein-coupled receptor GPR119; antidiabetic, antiinflammatory agent, neuropathy; use with a dipeptidyl peptidase IV (DPP IV) inhibitor
05/01/2008US20080103049 Benzoyl-Substituted Serineamides
05/01/2008US20080102031 4-[(4-N,N-diethylaminocarbonyl)phenyl]-spiro[2H,1-benzopyran-2,4'-piperidine; ligands of delta opioid receptor; analgesic, anxiolitic, antidepressant, analgesic; gastrointestinal disorders, neurodegenerative diseases; side effect reduction
04/2008
04/30/2008EP1916527A1 Analysis of mass spectral data in the quiet zones
04/30/2008EP1915996A1 Agents for treating intraocular inflammation caused by irradiation with lasers, containing 1,4-dihydropyridine derivatives
04/30/2008EP1915342A1 A novel hydroxamic acid derivative as peptide deformylase inhibitor and manufacturing method thereof
04/30/2008CN101171248A 3-mono- and 3,5-disubstituted piperidine derivatives as renin inhibitors
04/30/2008CN101171230A Heterocyclic-substituted alkanamides useful as renin inhibitors
04/30/2008CN101168527A Undecane to pentadecane dicarboxylic acid di(2,2,6,6-tetramethylpiperidinyl)ester and use thereof
04/30/2008CN100384826C Preparation of sterically hindered amine ethers
04/30/2008CN100384822C 4-(2-phenylsulfanyl-phenyl)-1,2,3,6-tetrahydropyridine derivatives as serotonin reuptake inhibitors
04/30/2008CN100384821C Cetp activity inhibitors
04/30/2008CN100384421C N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines
04/29/2008US7365196 Sulphonamido-substituted bridged bicycloalkyl derivatives
04/29/2008US7365085 2-(3-{3-[[2-chloro-3-(trifluoromethyl)benzyl](2,2-dephenylethyl)amino]propoxy}phenyl)-ethanol; agonists of the nuclear receptors, LXR alpha and LXR beta used to increase ABCA1, ABCG1, and apolipoprotein E expression and inhibiting cholesterol absorption
04/29/2008US7365083 NMDA (N-methyl-D-aspartate) receptors; eg 6-(4-benzylpiperidin-1-carbonyl)-1,5-dihydro-oxazolo[4,5-f]indole-2-one
04/29/2008US7365082 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines
04/29/2008US7365076 for the prevention and treatment of conditions ameliorated by monoamine reuptake including, inter alia, vasomotor symptoms (VMS), sexual dysfunction, gastrointestinal and genitourinary disorders, chronic fatigue syndrome, fibromylagia syndrome, nervous system disorders
04/29/2008US7365070 Such as N-{2-[2-(5-Bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-butyl-guanidine; involuntary weight loss disorders
04/29/2008US7365068 Hepatitis C virus infections; -(3-cyclopropyl-4-(pentyloxy)phenyl)-3-nicotinoylthiourea;methyl 2-oxo-2-(5-((3-(4-(pentyloxy)-3-(trifluoromethyl)phenyl)thioureido)carbonyl)pyridin-2-ylamino)acetate
04/29/2008CA2394037C New derivatives of benzene sulfonamide, their preparation process and pharmaceutical compositions that contain them
04/29/2008CA2336474C C-terminal modified oxamyl dipeptides as inhibitors of the ice/ced-3 family of cysteine proteases
04/29/2008CA2254833C Pharmaceutical for treatment of neurological and neuropsychiatric disorders
04/24/2008WO2008046918A2 Addition reactions using transition metal catalysts in halogenated solvents
04/24/2008WO2008046889A1 Enantiomer-enriched alpha-,omega amino alcohol derivatives, their production and use as insect- and mite-repelling agents
04/24/2008WO2008046573A1 Substituted sulfonamide derivatives for use as bradykinin 1 receptor modulators
04/24/2008WO2008019967A3 Phenyl, pyridine and quinoline derivatives
04/24/2008US20080097117 chemical intermediates for making antiinflammatory agents treating autoimmune disease; 1-[2-(Fluoren-3-yl)ethyl]-(4-(3-trifluoromethylphenyl)-1,2,3,6-tetrahydropyridine drug
04/24/2008US20080097099 Insecticides; for human or veterinary medicine; preparing heterocyclic amide and imine derivatives
04/24/2008US20080096936 Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them
04/24/2008US20080096922 N-{[cis-1-(3-methoxyphenyl)-4-(piperidin-4-ylamino)-cyclohexyl]methyl}sulfamide diHCL; tert-butyl [({[cis-4-[(biphenyl-4-ylmethyl)amino]-1-(3-methoxyphenyl)cyclohexyl]methyl}amino)sulfonyl]carbamate; for potentiating expression of low density lipoprotein recepotr; arteriosclerosis; hyperlipidemia
04/24/2008US20080096898 Organic Compounds
04/24/2008US20080096876 Histamine receptor antagonists; 4-[3-(4-Piperidin-1-yl-but-1-ynyl)-benzyl]-thiomorpholine; antiallergens, antihistamines, antiepileptic agents; asthma, alzheimer's disease, narcolepsy, motion sickness, attention deficit disorder, schizophrenia
04/24/2008US20080096867 Imidazo[1,2-A] Pyridine Anxiolytics
04/24/2008US20080096848 Substituted N-Aryl-9-Oxo-9H-Fluorene-1-Carboxamides and Analogs as Activators of Caspases and Inducers of Apoptosis
04/24/2008US20080095708 Biphenyl compounds useful as muscarinic receptor antagonists