Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
06/2008
06/25/2008EP1934186A2 Renin inhibitors nitroderivatives
06/25/2008EP1934180A2 3-cyclyl-2-(4-sulfamoyl-phenyl)-n-cyclyl-propionamide derivatives useful in the treatment of impaired glucose tolerance and diabetes
06/25/2008EP1802576B1 Process for producing enantiomer of amlodipine in high optical purity
06/25/2008CN101208352A Selective glycosidase inhibitors, methods of making inhibitors, and uses thereof
06/25/2008CN101208303A CGRP receptor antagonists
06/25/2008CN101208302A Novel 4-aminopiperidine derivatives as plasmepsin ii inhibitors
06/25/2008CN101205211A Method for preparing hydrochloric paroxetine key intermediates
06/25/2008CN100396679C Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase
06/25/2008CN100396668C Non-imidazole aryloxypiperidines
06/24/2008US7390924 Terphenyl derivatives, preparation thereof, compositions containing same
06/24/2008US7390907 Vanilloid receptor ligands and their use in treatments
06/24/2008US7390906 Forming ketone intermediates to terfenadine carboxylic acid metabolite; by use of pure regioisomer of 4-(Cyclopropyl-oxo-methyl)-alpha,alpha-dimethylphenylacetic acid
06/24/2008US7390905 Tachykinin receptor antagonists for use treating e.g. emesis, depression, urinary disorder
06/24/2008US7390904 Hydrogen peroxide catalyzed process for the preparation of sterically hindered N-hydrocarbyloxyamines
06/24/2008US7390830 MIP-1 alpha and/or MCP-1 antagonists; rheumatoid arthritis; nephritis; multiple sclerosis; nephropathy
06/24/2008US7390823 Use of saredutant and of its pharmaceutically acceptable salts for the preparation of medicinal products that are useful in the treatment or prevention of all mood disorders, adaptation disorders or mixed anxiety-depression disorders
06/24/2008US7390803 N-(3,5-bis-trifluoromethyl-benzyl)-1-(2-tert-butoxycarbonyl-amino-thiazol-4-yl)-3-(N-methyl, N-tetrahydro-4H-pyran-4-ylamino]-cyclopentanecarbamide; monocyte chemoattractant protein (MCP) receptor antagonist; antiinflammatory agent; antiallergen; autoimmune diseases; rhinitis, dermatitis, asthma
06/24/2008US7390433 Benzene derivative having long, linear conjugated structure, process for producing benzene derivative, and liquid-crystal material
06/19/2008WO2008073623A2 Soluble epoxide hydrolase inhibitors
06/19/2008WO2008072836A1 Inclusion complex comprising clopidogrel
06/19/2008WO2008072703A1 Biphenylamide derivative
06/19/2008WO2008071451A1 Dihydropyridine derivatives useful as protein kinase inhibitors
06/19/2008WO2008071421A1 Nitrate esters of carbonic anhydrase inhibitors
06/19/2008WO2008071398A1 Sulfonamides and their use as a medicament
06/19/2008WO2008051875A3 Adamantylurea compounds as soluble epoxide hydrolase inhibitors
06/19/2008WO2008051873A3 Phenylurea compounds as soluble epoxide hydrolase inhibitors
06/19/2008WO2008016643A3 Certain chemical entities, compositions, and methods
06/19/2008US20080146813 Grignard reagent (such as 4-alkylphenylmagnesium bromide) is added to a 3-cyanopyridinium salt (such as N-phenyloxycarbonyl-3-cyanopyridinium chloride) to get a 1,2-dihydropyridine which is oxidized with o-chloronil to obtain the 2-(4'-alkylphenyl)-5-cyanopyridine; display system
06/19/2008US20080146740 Process for the controlled increase in the molecular weight of polyethylenes
06/19/2008US20080146649 Substituted pyrrolidine and related compounds
06/19/2008US20080146620 Dibenzylamine Compounds and Pharmaceutical Use Thereof
06/19/2008US20080146612 Novel Biaromatic Compounds, Inhibitors of the P2X7-Receptor
06/19/2008US20080146572 N-sulfonylurea apoptosis promoters
06/19/2008US20080146569 Nicotinamide Derivatives
06/19/2008US20080145907 used for immobilization of amine-containing materials such as amino acid, peptide, protein, enzyme, immunoglobulin, DNA, RNA or fragments to substrate surfaces
06/19/2008CA2672167A1 Dihydropyridine derivatives as useful as protein kinase inhibitors
06/19/2008CA2650329A1 Terephthalamate compounds and compositions, and their use as hiv integrase inhibitors
06/18/2008EP1932830A1 Sulfonamides and their use as a medicament
06/18/2008EP1931652A2 Amido compounds and their use as pharmaceuticals
06/18/2008CN101203509A Amine-linked pyridyl and phenyl substituted piperazine-piperidines with CXCR3 antagonist activity
06/18/2008CN101203508A Substituted pyrr0lidin-2-0nes , piperidin-2-0nes and isothiazolidine-1, 1-dioxides, their use as kvl .5 potassium channel blockers and pharmaceutical preparations comprising them
06/18/2008CN101203492A Substituted butyrophenone derivatives
06/18/2008CN100395236C Piperazine and piperidine derivatives for treatment of neurological diseases
06/17/2008US7388118 Amine 1,2- and 1,3-diol compounds
06/17/2008CA2439152C Acylated piperidine derivatives as melanocortin-4 receptor agonists
06/17/2008CA2302347C 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocin-10-oles, processes for their preparation and their use for medicaments
06/17/2008CA2284732C Analogs of cocaine
06/12/2008WO2008069469A1 Crystalline s-(-)-amlodipine camsylate anhydride and preparation method thereof
06/12/2008WO2008068540A1 New benzamide derivatives as bradykinin antagonists
06/12/2008WO2008068423A2 P<0}{0pyrrol derivatives, preparation and use of the same in therapy<0}
06/12/2008WO2008042688A3 Phlorizin analogs as inhibitors of sodium glucose co-transporter 2
06/12/2008WO2007148208A3 Carbonylated (aza) cyclohexanes as dopamine d3 receptor ligands
06/12/2008WO2007123910A3 Copper-mediated functionalization of aryl c-h bonds, and compounds related thereto
06/12/2008US20080139817 Reacting 2-chloro-3-cyanopyridine with benzyl mercaptan in the presence of a sodium carbonate and an aprotic solvent; hydrolyzing resulting intermediate; no need for purification
06/12/2008US20080139811 Reacting an amino, hydroxy substituted amide with a heterocyclic substituted carboxylic acid to produce (2S,3S,5S)-2-(2,6-Dimethylphenoxyacetyl) amino-3-hydroxy-5-[2S-1-imidazolidin-2-onyl)-3-methyl-butanoyl] amino-1,6-diphenylhexane; inhibitors of HIV infection
06/12/2008US20080139630 Tissue-selective androgen receptor modulators (SARMs); male hypogonadism, prostate cancer, benign prostate hyperplasia, sarcopenia, rheumatoid arthritis and osteoarthritis; N-((5-cyclopropyl-2-fluoropyridin-3-yl)methyl)-2-phenylbutanamide for example
06/12/2008US20080139627 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides
06/12/2008US20080139625 Pyrrolidin-2-One and Piperidin-2-One Derivatives as 11-Beta Hydroxysteroid Dehydrogenase Inhibitors
06/12/2008US20080139607 Inhibitors of the serine protease PAI-1 (plasminogen activator inhibitor type 1); (3R)-8-(3,4-Difluoro-phenyl)-7-heptyl-5-oxo-2,3-dihydro-5H-thiazolo[3,2-a]pyridine-3-carboxylic acid for example; desulfurization to form corresponding 1-(1-carboxyethyl)-1,2-dihydro-2-oxopyridine compound; coadministering
06/12/2008US20080139575 Certain chemical entities, compositions, and methods
06/12/2008US20080139564 Substituted phenyl propyl amines as histamine h3 receptor and serotonin transporter modulators
06/12/2008US20080139505 Potentiators Of Glutamate Receptors
06/12/2008CA2671749A1 Bicyclic compounds and uses as antidiabetics
06/12/2008CA2671121A1 Stat3 inhibitor having anti-cancer activity and associated methods
06/12/2008CA2669996A1 Pyrrol derivatives, preparation and use of the same in therapy
06/11/2008EP1930330A1 Pleuromutilin derivatives as antimicrobials
06/11/2008EP1930323A1 Biphenyl compounds useful in the synthesis of muscarinic receptor antagonists
06/11/2008EP1930322A1 1-(4-piperidinyl)-1,3-dihydro-2H-benzoxazole-2-one derivatives and related compounds as nociceptin analogs and ORL1 ligands for the treatment of pain
06/11/2008EP1930308A1 Pharmaceutical agents for the treatment of cerebral amyloidosis
06/11/2008EP1930021A2 Novel amide derivatives as growth hormone secretagogues
06/11/2008EP1928875A1 2-amino-7,8-dihydro-6h-pyridoý4,3-d¨pyrimidin-5-ones
06/11/2008EP1928829A1 Piperidine derivatives as antagonists of the cc chemokine receptor ccr1 and their use as anti-inflammatory agents
06/11/2008EP1928821A1 Carboxamide derivatives as muscarinic receptor antagonists
06/11/2008EP1485348B1 Carbonylamino-derivatives as novel inhibitors of histone deacetylase
06/11/2008EP1414794B1 Allylmercaptocaptopril compounds and uses thereof
06/11/2008CN101198604A NPY antagonists, preparation and use
06/11/2008CN101198584A Benzamide derivatives and uses related thereto
06/11/2008CN101198583A Compounds which inhibit beta-secretase activity and methods of use
06/11/2008CN101195614A Production of balofloxacin and purification process thereof
06/11/2008CN101195602A 1-deoxidization nojiri toxin derivant, production method and uses thereof
06/11/2008CN100393700C Cathepsin cysteine protease inhibitors
06/10/2008US7385063 Method for preparing imidazole derivatives
06/10/2008US7385060 4-Methylpropiophenone is reacted with piperidine hydrochloride and 1,3-dioxolane in the presence of an acid serving as a catalyst, and the tolperisone obtained in the form of an acid addition salt is separated by filtering after the reaction mixture has cooled down; improved purity, simplification
06/10/2008US7385059 3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators
06/10/2008US7384967 Aryl carbonyl derivatives as therapeutic agents
06/10/2008US7384945 Indole or benzimidazole derivatives as CB1 inverse agonists
06/10/2008US7384944 Organ grafting; antiarthritic agents; inflammatory bowel disease
06/10/2008US7384929 N-aryl azaspiroalkene and azaspiroalkane compounds and methods of preparation and use thereof
06/10/2008CA2393995C Novel benzene sulfonamide derivatives, their preparation and pharmaceutical compositions containing them
06/10/2008CA2371827C Amide compounds for the potentiation of cholinergic activity
06/10/2008CA2227607C Penicillaminamide derivatives
06/10/2008CA2129046C Opioid diarylmethylpiperazines and piperidines
06/05/2008WO2008066708A2 New process for remifentanil synthesis
06/05/2008WO2008065424A1 Ramipril-amlodipine salt
06/05/2008WO2006138508B1 Benzamide derivatives and uses related thereto
06/05/2008US20080132705 Process for the preparation of 2-substituted-5-(1-alkylthio)alkylpyridines
06/05/2008US20080132683 Purification of immunoglobulins from solution (hybridoma cell culture supernatants, animal plasma or sera, or colostrum); solid phase synthesis
06/05/2008US20080132552 e.g. N-[1-(3,5-Difluoro-benzyl)-2-hydroxy-3-methylamino-propyl]-5-methyl-N',N'-dipropyl-isophthalamide; beta-secretase inhibitor; neurodegenerative diseases: Alzheimer's disease
06/05/2008US20080132543 Therapeutic and Delivery Methods of Prostaglandin Ep4, Agonists
06/05/2008US20080132539 e.g. 2-amino-5-[(naphthalen-1-ylmethyl)-aminocarbonyl]-pentanoic acid hydroxyamide; advanced glycosylation endproducts inhibitor; diabetic neurosis, diabetic retinopathy, atherosclerosis, cataract, Alzheimer's disease, rheumatic arthritis, osteoarthritis, chronic renal failure; food and cosmetics