Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
01/2011
01/05/2011EP2268612A1 Arylsulfonamide-based matrix metalloprotease inhibitors
01/05/2011EP1948606B1 3, 5-disubstituted phenyl-piperidines as modulators of dopamine neurotransmission
01/05/2011CN101939297A Benzylpiperizine compound
01/05/2011CN101429154B Anhydrous alvimopan and medicament composition thereof
01/04/2011US7863453 salt formation of reacting isofagomine and L-(+)-tartaric acid; for treating Gaucher disease; improved Pharmacokinetics high purity, crystalline form; glucocerebrosidase inhibitors; beta glucosidase inhibitors
01/04/2011US7863452 improved process for preparation of chemical intermediate for fexofenadine; using isobutyrate or an isobutyrate equivalent
01/04/2011US7863450 e.g. 1-{3-[4-(4,4-dimethyl-4,5-dihydro-1,3-oxazol-2-yl)phenoxy]propyl}piperidine; histamine H3 receptor antagonist; anxiolytic agent, antidepressant, cognition activator; neurodegenerative diseases, eating disorder, attention deficit disorder, Alzheimer's, Parkinson's diseases, schizophrenia
01/04/2011US7863298 1 alpha ,25-dihydroxyvitamin D3 mimetics such as 3-(4-{1-ethyl-1-[4-(3-hydroxy-4,4-dimethylpentyl)-phenyl]-propyl}-2-methylphenoxy)-propane-1,2(S)-diol, used as anticarcinogenic agents or for the treatment of glandular, urogenital, bone, skin and neurodegenreative disorders; vitamin D receptor modulators
01/04/2011CA2488363C O-substituted hydroxyaryl derivatives
01/04/2011CA2479362C N-sulfonylurea apoptosis promoters
01/04/2011CA2463506C Synthesis of (4-bromophenyl) (4-piperidyl)methanone-(z)-o-ethyloxime and salts
01/04/2011CA2460822C Aralkyltetrahydropyridines, their preparation and pharmaceutical compositions containing same
01/04/2011CA2421228C Polyarylcarboxamides useful as lipid lowering agents
01/04/2011CA2412941C Piperidine compounds for use as ccr-3 inhibitors
01/04/2011CA2319672C Compounds and compositions for delivering active agents
12/2010
12/30/2010US20100331546 Method for optical resolution of alkyl piperidin-3-yl carbamate and intermediate therefor
12/30/2010US20100331375 Biphenyl compounds useful as muscarinic receptor antagonists
12/30/2010US20100331366 N-adamantyl benzamides as inhibitors of 11-beta-hydroxysteroid dehydrogenase
12/30/2010US20100331364 TREATMENT OF HFnEF
12/30/2010US20100331360 3-substituted sulfonyl piperidine derivative
12/30/2010US20100331329 Benzamide derivatives useful as histone deacetylase inhibitors
12/30/2010US20100330064 2-mercaptocyclopentanecarboxylic acid compounds, a process for their preparation and pharmaceutical compositions containing them
12/30/2010US20100327270 Novel materials for organic electroluminescent devices
12/30/2010DE10008117B4 Verfahren zur Acylierung von 4-Aminopiperidin und 4-Aminopiperidinderivaten Process for the acylation of 4-amino-piperidine and 4-aminopiperidine
12/29/2010WO2010150206A1 N-substituted-n-phenylethylsulfonamides for the identification of biological and pharmacological activity
12/29/2010WO2010150205A1 1-(sulfonyl)-n-phenylpyrrolidine-2-carboxamides for the identification of biological and pharmacological activity
12/29/2010WO2010150204A1 N-(2-oxo-1-phenylpiperidin-3-yl) sulfonamides for the identification of biological and pharmacological activity
12/29/2010WO2010149888A1 Derivatives of 2-mercaptocyclopentane carboxylic acid, method for the preparation thereof, and pharmaceutical compositions containing the same
12/29/2010WO2010149819A1 N-(1-phenyl-2-oxo-3-piperidyl sulphonamide libraries for drug discovery
12/29/2010WO2010149744A1 Method for synthesising 2-acetyl-1-pyrroline and the stable precursor thereof, optionally isotopically marked
12/29/2010WO2010149684A1 New compounds, pharmaceutical composition and methods relating thereto
12/29/2010WO2010148632A1 Dihydropyridine compounds and preparation methods, pharmaceutical compositions and uses thereof
12/29/2010WO2010132670A3 Pentacycline compounds
12/29/2010EP2265584A1 Hydroxyalkanyl amides as modulators of chemokine receptor activity
12/29/2010EP2035381B1 Process for the preparation of sterically hindered nitroxyl ethers
12/29/2010EP1292573B1 Substituted thioacetamides
12/29/2010CN101928284A Nitrogen-containing heterocyclic derivatives and drugs containing the same as the active ingredient
12/29/2010CN101928280A Pepperphentonamine derivative containing naphthalene rings
12/29/2010CN101928241A 2-mercaptopentancarboxylic acid derivatives, the method for preparing them and the pharmaceutical compositions containing them
12/29/2010CN101531629B Method for preparing levamlodipine from racemic amlodipine maleate
12/29/2010CN101503392B Aromatic aminomethane compounds, as well as preparation and medical use thereof
12/29/2010CA2766696A1 New compounds, pharmaceutical composition and methods relating thereto
12/28/2010US7858824 Aralkyltetrahydropyridines, their preparation and pharmaceutical compositions containing them
12/28/2010US7858801 Process for producing enantiomer of amlodipine in high optical purity
12/28/2010US7858799 Gelling agent, carbon nanotubes aqueous dispersing agent; simple synthesis from low cost, readily available raw materials; rapid elastic modulus recovery; environmentally friendly
12/28/2010US7858798 metabolite of ebastine
12/28/2010US7858797 Biphenyl compounds useful as muscarinic receptor antagonists
12/28/2010US7858795 or anticholinergic agents such as biphenyl-2-ylcarbamic acid 1-[2-({6-[(4-hydroxybenzylamino)methyl]pyridin-2-ylmethyl}carbamoyl)ethyl]piperidin-4-yl ester, used for the treatment of respiratory system disorders such as chronic obstructive pulmonary disease and asthma
12/28/2010US7858792 Biphenyl-2-ylcarbamic Acid 1-(2-{5-[2-(4-Hydroxyphenyl)ethylamino]pentylcarbamoyl}ethyl)piperidin-4-yl Ester, used for the treatment of respiratory system disorders such as chronic obstructive pulmonary disease and asthma
12/28/2010US7858789 Affinity for somatostatin receptors; used for the treatment of acromegalia, hypophyseal adenomas or endocrine gastroenteropancreatic tumors including carcinoid syndrome; 4-(urea or thiourea substituted)-1-alkylpiperidines
12/28/2010US7858737 Heterogeneous foldamers containing α, β, and/or γ-amino acids
12/28/2010US7858624 such as methyl 2-((R)-((R)-1-((2S,3S)-5-(butylamino)-1-cyclohexyl-3-hydroxy-5-oxopentan-2-ylcarbamoyl)piperidin-3-yl)(3-chlorophenyl)methoxy)ethylcarbamate, used as hypotensive agents or for the treatment of cardiovascular disorders, vision defects, aldosteronism and obesity
12/23/2010WO2010145037A1 Disubstituted-aminodifluorosulfinium salts, process for preparing same and method of use as deoxofluorination reagents
12/23/2010WO2010128528A3 Piperidine derivatives useful for treatment of diebetes
12/23/2010WO2010097802A3 A process for the preparation of etoricoxib
12/23/2010WO2010088450A3 Arylamide derivatives useful in the treatment of diseases associated with serca activity
12/23/2010US20100324090 Compositions of tolperisone
12/23/2010US20100324052 Novel piperidine carboxylic acid amine derivatives
12/23/2010US20100324049 Diaryl ketimine derivative having antagonism against melanin-concentrating hormone receptor
12/23/2010US20100324046 4-carboxybenzylamino derivatives as histone deacetylase inhibitors
12/23/2010US20100324025 Antibacterial Agents
12/23/2010US20100324009 Substituted Sulfonamide Compounds
12/23/2010US20100320451 Benzochrysene derivative and organic electroluminescence device using the same
12/23/2010CA2764241A1 Disubstituted-aminodifluorosulfinium salts, process for preparing same and method of use as deoxofluorination reagents
12/22/2010EP2264030A1 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases
12/22/2010EP1453805B1 4-piperidinyl alkylamine derivatives as muscarinic receptor antagonists
12/22/2010CN101925588A 2-cyanophenyl sulfonamide derivatives useful as pesticides
12/22/2010CN101921597A Liquid crystal alignment agent and liquid crystal display element
12/22/2010CN101921224A 1-(3-aminopropyl) piperazine-4-aminoamide compound as well as preparation method and application thereof
12/22/2010CN101080388B Piperidinesulfonylureas and -thioureas, their preparation, their use and pharmaceutical compositions comprising them
12/22/2010CN101001836B Pyrrolidin-2-one and piperidin-2-one derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors
12/21/2010CA2448896C Allylmercaptocaptopril compounds and uses thereof
12/21/2010CA2406255C Hydroxylamine esters as polymerization initiators
12/21/2010CA2397981C Azacyclic compounds for use in the treatment of serotonin related diseases
12/16/2010WO2010144446A1 (s) -2-benzyl-3- ( (3r, 4r) -4- (3 -carbamo ylphenyl) -3, 4-dimethylpiperidinyl) propanoic acid and salt therof as antagonists of the opioid receptors
12/16/2010WO2010144380A1 Process for the preparation of 6-(aryl)-4-aminopicolinates
12/16/2010WO2010144379A1 3-halo-(arly)-4-iminotetrahydropicolinates and their use as herbicides
12/16/2010WO2010144371A1 Alkanoylamino benzamide aniline hdac inihibitor compounds
12/16/2010WO2010142985A1 Substituted n-[1-cyano-2-(phenyl)ethyl]piperidin-2-ylcarboxmide compounds 761
12/16/2010WO2010142650A1 Novel cyclopentane derivatives
12/16/2010WO2010142572A1 Sterically hindered amine stabilizers
12/16/2010WO2010142241A1 High penetration compositions or prodrugs of antimicrobials and antimicrobial-related compounds
12/16/2010WO2010122580A3 Piperidine derivatives as inhibitors of renin
12/16/2010WO2010104306A3 Pharmaceutical compositions for treating or preventing diseases caused by the translocation of gsk3 from the cell nucleus to the cytoplasm, containing compounds for inhibiting the translocation of gsk3 from the cell nucleus to the cytoplasm
12/16/2010US20100317697 Renin Inhibitors
12/16/2010US20100317690 Treatment of protein folding disorders
12/16/2010US20100317678 Hydroxamates as inhibitors of histone deacetylase
12/16/2010US20100317647 Novel cyclopentane derivatives
12/16/2010US20100317644 Substituted Sulfonamide Compounds
12/16/2010US20100317630 Novel heterocyclic compounds as mglu5 antagonists
12/16/2010CA2802334A1 Compositions and methods for imaging tissues, organs and tumors
12/16/2010CA2764981A1 (s) -2-benzyl-3- ( (3r, 4r) -4- (3 -carbamoylphenyl) -3, 4-dimethylpiperidinyl) propanoic acid and salt therof as antagonists of the opioid receptors
12/16/2010CA2764376A1 High penetration compositions or prodrugs of antimicrobials and antimicrobial-related compounds
12/16/2010CA2763786A1 Alkanoylamino benzamide aniline hdac inihibitor compounds
12/16/2010CA2763167A1 Cycloalkylcarbamate benzamide aniline hdac inhibitor compounds
12/16/2010CA2762930A1 Sterically hindered amine stabilizers
12/16/2010CA2762619A1 Novel cyclopentane derivatives
12/16/2010CA2761229A1 3-halo-6-(aryl)-4-iminotetrahydropicolinates and their use as herbicides
12/15/2010EP2261210A1 3-substituted sulfonyl piperazine derivative
12/15/2010EP2261209A1 Novel crystalline forms of 4-[4-[4- hydroxydiphenylmethyl)-1-piperidinyl]-1-hydroxybutyl]-alpha, alpha-dimethylbenene acetic acid and its hydrochloride
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