Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
08/2000
08/10/2000WO2000046202A2 Process for the preparation of 1,2,3,6-tetrahydro-2,2,6,6-tetraalkylpyridines
08/10/2000WO2000046201A1 Benzamide derivatives and drugs containing the same
08/10/2000WO2000046200A1 2-n-substituted or unsubstituted-2-amino-5-methylpiperidine-3,4-diols and processes for the preparation thereof
08/10/2000WO2000046194A1 Cyclic amine derivatives and uses thereof
08/10/2000WO2000046187A2 Antizyme modulators and their use
08/10/2000WO2000046183A1 N-substituted amino acids, antioxidant pharmaceutical compositions containing same and methods using same
08/10/2000WO1999063936A9 Novel therapeutic agents that modulate endothelin receptors
08/10/2000CA2362259A1 Antizyme modulators and their use
08/10/2000CA2362230A1 Sulfamato hydroxamic acid metalloprotease inhibitor
08/10/2000CA2362077A1 Cyclic amine derivatives and uses thereof
08/10/2000CA2352507A1 Process for the preparation of 2,2,6,6-tetraalkylpiperidin-1-oxyl via 1,2,3,6-tetrahydro-2,2,6,6-tetraalkylpyridine
08/09/2000EP1026147A1 Compounds useful as intermediates in the production of piperidine derivatives
08/09/2000EP1025099A1 Bis-quaternary ammonium derivatives as neuromuscular relaxants
08/09/2000EP1025094A1 Substituted indan derivatives
08/09/2000EP1025085A1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof
08/09/2000EP1025084A1 Method for purifying 4-amino-piperidines
08/09/2000EP1024799A1 Method for treating disease-related or drug-induced dyskinesias
08/09/2000CN1262684A 2,4,4-trisubstituted-1,3-dioxolane antifungals
08/09/2000CN1262675A (+)-Norcisapride useful for 5-HT3 and 5-HT4 mediated disorbers
08/09/2000CN1262674A Gatrokinetic monocyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives
08/09/2000CN1262621A Gastrokinetic bicyclc benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives
08/09/2000CN1262618A NF-KB inhibitors containing as active ingredient phenylmethyl benzoquinone
08/09/2000CN1262272A HIV proteinase inhibitor
08/08/2000US6100420 Heterocyclylbenzonitriles
08/08/2000US6100401 Process for preparing the d-threo isomer of methylphenidate hydrochloride
08/08/2000US6100253 Tricycle substituted with azaheterocyclic carboxylic acids
08/08/2000CA2188227C Combination antiemetic therapy using nk-1 receptor antagonists
08/08/2000CA2185512C Treatment of tinnitus using neuroprotective agents
08/08/2000CA2072575C Anticholinergic agents
08/03/2000WO2000044723A1 Alkynyl containing hydroxamic acid derivatives, their preparation and their use as matrix metalloproteinase (mmp) inhibitors/tnf-alpha converting enzyme (tace) inhibitors
08/03/2000WO2000044714A1 S-nitrosothiols as agents for the treatment of circulatory dysfunctions
08/03/2000WO2000044713A1 Alkynyl containing hydroxamic acid compounds as tace inhibitors
08/03/2000WO2000044709A2 ACETYLENIC α-AMINO ACID-BASED SULFONAMIDE HYDROXAMIC ACID TACE INHIBITORS
08/03/2000WO2000044383A1 Anti-inflammatory agents and inhibitors against increase in ocular tension caused by irradiation with lasers, containing 1,4-dihydropyridine derivatives
08/03/2000WO2000044380A1 Release-regulating preparations
08/03/2000WO2000044377A1 Mono-acyloxy aralkyl neuromuscular relaxants
08/03/2000WO2000044376A1 Antidepressant heterocyclic compounds
08/03/2000WO2000008006A3 Piperidine and piperazine derivatives, process for their preparation and pharmaceutical compounds containing them
08/03/2000WO2000006146A9 Substituted anilide compounds and methods
08/03/2000WO2000005208A9 Amino-aldehyde solid support, linker therefor and methods of preparation and use thereof
08/03/2000WO2000003975A3 Aryl vinyl ether derivatives and their use as herbicides
08/03/2000DE19903126A1 New sulphur substituted sulphonylaminocarboxylic acid N-arylamide derivatives used for treating e.g. cardiovascular diseases and atherosclerosis
08/03/2000CA2360790A1 Mono-acyloxy aralkyl neuromuscular relaxants
08/03/2000CA2360689A1 Anti-inflammatory agents and inhibitors against increase in ocular tension caused by irradiation with lasers, containing 1,4-dihydropyridine derivatives
08/03/2000CA2360686A1 Release-regulating preparations
08/03/2000CA2360683A1 Antidepressant heterocyclic compounds
08/03/2000CA2356346A1 Alkynyl containing hydroxamic acid compounds as tace inhibitors
08/03/2000CA2356313A1 Alkynyl containing hydroxamic acid derivatives, their preparation and their use as matrix metalloproteinase (mmp) inhibitors/tnf-alpha converting enzyme (tace) inhibitors
08/03/2000CA2356299A1 Acetylenic .alpha.-amino acid-based sulfonamide hydroxamic acid tace inhibitors
08/02/2000EP1024134A1 Aminobutanoic acid derivatives
08/02/2000EP1023285A1 Azetidinylpropylpiperidine derivatives, intermediates and use as tachykinin antagonists
08/02/2000EP1023068A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
08/02/2000EP0691953B1 1-amidinophenyl-pyrrolidones/ piperidinones as platelet aggregation inhibitors
08/02/2000CN1261887A Azetidinyl propylpiperidine derivatives, intermediates and use as tachykinin antagonists
08/02/2000CN1261877A 4-bromo or 4-iodo phenylamino benzhydroxamic acid derivatives and their use as MEK inhibitors
08/02/2000CN1261876A N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases
08/02/2000CN1261795A Compounds and methods
08/01/2000US6096762 Contacting nerve cells with a neurotrophic amount of difluoroamide compound with affinity for an fk-506 binding protein for stimulating neurite grwoth in nerve cells
08/01/2000US6096761 Esters of 3-hydroxy-piperidinemethanol derivatives
08/01/2000US6096760 Solid α-phenyl-2-piperidine acetate free base, its preparation and use in medicine
08/01/2000US6096741 Oxime derivatives, hydrazone derivatives and use thereof
08/01/2000US6096729 Use of NK-1 receptor antagonists for treating amnestic disorders
08/01/2000CA2015034C Piperazine derivatives
07/2000
07/27/2000WO2000043383A1 Piperidinylquinolines as protein tyrosine kinase inhibitors
07/27/2000WO2000043372A1 Acyl derivatives which treat vla-4 related disorders
07/27/2000WO2000043369A1 Compounds which inhibit leukocyte adhesion mediated by vla-4
07/27/2000WO2000043362A1 Phenylsulphonyl derivatives as 5-ht receptor ligands
07/27/2000WO2000043352A1 A method for the synthesis of compounds of formula 1 and derivatives thereof
07/27/2000WO2000043011A1 Substituted 1-(piperidin-4-yl)-3-(aryl)-isothioureas, their preparation and therapeutic use
07/27/2000WO2000042989A2 Novel hydrogel isolated cochleate formulations, process of preparation and their use for the delivery of biologically relevant molecules
07/27/2000WO2000042852A1 Compounds and methods
07/27/2000WO2000018358A3 Method of treating hair loss using ketoamides
07/27/2000WO1999066944A9 Methods for identifying novel multimeric agents that modulate receptors
07/27/2000WO1999064033A9 Phosphodiesterase-v modulator drugs and their uses
07/27/2000WO1999063994A9 MULTIBINDING INHIBITORS OF HMG-CoA REDUCTASE
07/27/2000WO1999062881A8 Aza-heterocyclic compounds used to treat neurological disorders and hair loss
07/27/2000WO1999057098A3 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
07/27/2000CA2359983A1 Phenylsulphonyl derivatives as 5-ht receptor ligands
07/27/2000CA2359572A1 Substituted 1-(piperidin-4-yl)-3-(aryl)-isothioureas, their preparation and therapeutic use
07/27/2000CA2359113A1 Compounds which inhibit leukocyte adhesion mediated by vla-4
07/27/2000CA2359076A1 A method for the synthesis of compounds of formula 1 and derivatives thereof
07/26/2000EP1022268A1 Arylalkanoyl derivatives, processes for their preparation, their use and pharmaceutical compositions containing them
07/26/2000EP1021440A2 Antipsychotic substituted piperidine derivatives
07/26/2000EP1021425A1 N-aminoalkyl-2-anthraquinonecarboxamides; dopamine receptor subtype specific ligands
07/26/2000EP1021199A1 PEPTIDE-CONTAINING $g(a)-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS
07/26/2000EP0639976B1 Use of terfenadine derivatives as antihistaminics in a hepatically impaired patient
07/26/2000CN1261348A Dihydropyridine derivatives
07/26/2000CN1261347A Remedies/preventives for frequent urination/urinary incontinence and tropone derivatives
07/26/2000CN1261281A Peptide parathyroid hormone analogs
07/26/2000CN1054849C Process for producing quaternary glycine nitriles
07/26/2000CN1054842C 1-amidinophenyl-pyrrolidones piperidinones azetinones platelet aggregation inhibitors
07/25/2000US6093827 Process for the preparation of 10,11-dihydro-5H-dibenzo[A,D]cyclohept-5-enes and derivatives thereof
07/25/2000US6093820 Reacting an imide with a (substituted)alkoxyalkylsulfonic acid ester to form a n-alkoxyalkyl imide such as methoxymethyl ethosuximide; administering as anticonvulsant, antianxiety agent and muscle relaxant
07/25/2000US6093748 Applying to an area of skin from which reduced hair growth is desired a dermatologically acceptable composition containing a non-steroidal suppressor of angiogenesis
07/25/2000US6093733 Muscarinic receptor agonists
07/25/2000CA2197086C (azetidin-1-ylalkyl)lactams as tachykinin antagonists
07/20/2000WO2000042071A2 Compounds and methods to inhibit or augment an inflammatory response
07/20/2000WO2000042011A1 Amide compounds
07/20/2000WO2000042010A1 Contrast media for angiography
07/20/2000WO1999064048A9 Inhibitors of hiv reverse transcriptase