Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
09/2000
09/14/2000WO2000037068B1 Use of a 5ht2a and 5ht2a/c receptor antagonist for preparing medicines for treating snoring and high resistance syndrome of upper anatomical airways
09/14/2000WO1999063999A8 H1-histamine receptor antagonists
09/14/2000DE19911039A1 Abgewandelte Aminosäureamide, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung Modified amino acid amides, pharmaceutical compositions containing them and methods for their preparation
09/14/2000DE19910504A1 Verfahren zur Reinigung von N-substituierten Lactamen A process for purifying N-substituted lactams
09/13/2000EP1035110A1 Benzylaminodiacetamide derivatives, compositions containing the same, process for their preparation and uses
09/13/2000EP1034264A1 Splice variants for human 5-ht 4? serotonin receptor and their applications, in particular for screening
09/13/2000EP1034164A1 Substituted beta-alanine derivatives as cell adhesion inhibitors
09/13/2000EP1034162A1 9,10-dihydro-9,10-ethanoanthracene derivatives as phospholipase inhibitors
09/13/2000EP1033983A1 Cyclic amino acid derivatives as cell adhesion inhibitors
09/13/2000EP1033970A1 Novel formulation for use in pain management
09/13/2000EP0691962B1 1-amino-3-phenoxy propane derivatives as modulators of multi-drug resistance
09/13/2000CN1266428A Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same
09/13/2000CN1056373C Process for preparation of fluoroalkoxybenzylamino derivatives of nitrogen containing heterocycles
09/12/2000US6118006 Method for preparing a tetrahydropyridin derivative
09/12/2000US6118001 Anticancer agent; antiarthritic agent
09/12/2000US6117995 Oxidation of the corresponding heterocyclic amine compound
09/08/2000WO2000051985A1 Fluorides of 4-substituted piperidine derivatives
09/08/2000WO2000051971A1 Oxamic acids and derivatives as thyroid receptor ligands
09/08/2000WO2000051970A1 Amide compounds for the potentiation of cholinergic activity
09/06/2000EP1032571A1 Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance p antagonists
09/06/2000EP1032561A1 Substituted oximes as neurokinin antagonists
09/06/2000EP1032389A1 CHRONIC, BOLUS ADMINISTRATION OF D-threo METHYLPHENIDATE
09/06/2000EP1032377A1 Substituted 2-aminoacetamides and the use thereof
09/06/2000EP1032368A1 Iontophoretic devices comprising piperidin derivatives
09/06/2000CN1265647A Acrylic metalloprotease inhibitor
09/06/2000CN1265646A Aryloxyarylsulfonylamino hydroxamic acid derivatives
09/06/2000CN1056143C Piperidine derivatives and its use
09/05/2000US6114356 Method for treating gastrointestinal disorders using (+) norcisapride
09/05/2000US6114354 N-substituted azaheterocyclic compounds
09/05/2000US6113980 Applying a powder coating contining an organic polymeric binder, atleast two different compounds containing a tetramethylpiperdine residue as light stabilizer, an electron donor triboelectrically to a metal substrate
09/05/2000US6113879 Isolated d-threo-methylphenidate enantiomorph; attention deficit-hyperactivity disorder; nontoxic
09/05/2000CA2020340C Enantioselective synthesis of antifolates
08/2000
08/31/2000WO2000050397A1 Substituted piperidinedione derivatives and herbicide
08/31/2000WO2000050396A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
08/31/2000WO2000050389A1 Efficient carbamate synthesis
08/31/2000WO2000050380A1 Monoamine reuptake inhibitors for treatment of cns disorders
08/31/2000WO2000050377A1 Efficient synthesis of secondary amines by selective alkylation of primary amines
08/31/2000WO2000050376A2 Efficient synthesis of alkyl carbonates
08/31/2000WO2000040558A8 Aspartic protease inhibitors
08/31/2000WO2000012074A3 Use of piperidines and/or piperazines as inhibitors of p38-alpha kinase
08/31/2000WO2000001375A3 Calcium channel blockers
08/31/2000DE10008367A1 New 1-alkoxy-substituted hindered 2,2,6,6-tetramethylpiperidine group-containing amines useful as stabilizers for (thermoplastic) polymers, coatings, color photographic materials and printing inks
08/31/2000CA2371876A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
08/30/2000EP1031563A1 Sulfonyl derivatives
08/30/2000EP1030841A1 Process for the preparation of 1,4-dihydropyridines and compounds used in this process
08/30/2000EP1030840A1 Cyclic amine derivatives and their use as drugs
08/30/2000EP1030839A1 Use of alkylated iminosugars to treat multidrug resistance
08/30/2000EP1030836A1 Hydroxamic and carboxylic acid derivatives having mmp and tnf inhibitory activity
08/30/2000EP1030831A1 Process for the preparation of azacycloalkylalkanoyl pseudotetrapeptides
08/30/2000CN1265096A Hydrazine derivatives
08/29/2000US6110970 For treating or preventing or ameliorating cancer and other proliferative diseases as well as for inducing wound healing, treating cutaneous ulcers, treating gastrointestinal disorders, treating blood disorders such as anemias
08/29/2000US6110944 LTA4, hydrolase inhibitors
08/29/2000US6110941 Compounds analogous to thalidomide from the class comprising piperidine-2,6-diones
08/29/2000US6110937 A sodium channel blocker treating as local anesthetics and in the treatment of cardiac arrhythmias
08/29/2000US6110933 Amino acid derivatives and their use as phospholipase A2 inhibitor
08/29/2000US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
08/29/2000US6110913 N-substituted azaheterocyclic carboxylic acids and esters thereof
08/29/2000CA2012628C New fluoro-4 benzoic derivatives, process for their preparation and pharmaceutical compositions containing them
08/24/2000WO2000048993A1 Arylaminoalkylamides
08/24/2000WO2000048989A1 Mevinolin derivatives
08/24/2000WO2000048623A1 Novel amide derivatives as growth hormone secretagogues
08/24/2000WO1996012697A9 Calcium receptor-active compounds
08/24/2000CA2362290A1 Novel amide derivatives as growth hormone secretagogues
08/23/2000EP1028961A1 Pleuromutilin derivatives as antimicrobials
08/23/2000EP1028943A2 Orally-active nipecotamide glycolamide esters for the treatment of thrombosis disorders
08/23/2000EP1028942A2 Dipeptide nitriles
08/23/2000EP1028716A1 Method for treating and preventing heart failure and ventricular dilatation
08/23/2000EP0805795B1 Novel aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides
08/23/2000CN1264385A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and compositions containing same
08/23/2000CN1264300A Arylsubstituted piperazines useful in the threatement of bening prostatic hyperlasia
08/23/2000CN1055690C 4-aryloxy-and-4-arylthiopiperidine derivatives, method for preparation them, medicine compound containing them and use thereof
08/23/2000CN1055684C Method for preparing substituted pyridine
08/23/2000CN1055683C Process for producing N-allkyl-2,5-dimethyl-piperidinol-4-benzoyl ester
08/22/2000US6107345 Antidepressant; psychological disorders
08/22/2000US6107329 Hypotensive agents; cardiovascular disorders
08/17/2000WO2000047572A1 (1-phenacy-3-phenyl-3-piperidylethyl)piperidine derivatives, method for the production thereof and pharmaceutical compositions containing the same
08/17/2000WO2000047559A2 5-ht1f agonists
08/17/2000WO2000047207A1 LACTAM INHIBITORS OF FXa AND METHOD
08/17/2000WO2000047198A2 Use of substituted-1,5-dideoxy-1,5-imino-d-glucitol compounds for treating hepatitis virus infections
08/17/2000WO2000009109A3 Pipecolic acid derivatives for vision and memory disorders
08/17/2000CA2360305A1 Lactam inhibitors of fxa and method
08/17/2000CA2360164A1 5-ht1f agonists
08/16/2000EP1027713A1 Nonaqueous electrolyte for electrical storage devices
08/16/2000EP1027342A1 Cyclopentene derivatives useful as antagonists of the motilin receptor
08/16/2000EP1027339A1 Method and reagents for n-alkylating ureides
08/16/2000EP1027332A1 Novel lactam metalloprotease inhibitors
08/16/2000EP1027328A1 Substituted anilides
08/16/2000EP1027324A1 Optically active intermediates for the preparation of optically active substituted oximes, hydrazones and olefins useful as neurokinin antagonists
08/16/2000EP1026950A1 Treatment of schizophrenia with ampakines and neuroleptics
08/16/2000EP0755374B1 Process for peptide segment condensation
08/16/2000EP0738259B1 Phenyl acetic acid derivatives, process and intermediate products for their production and agents containing them
08/16/2000CN1263525A Process for preparation of amlodipine benzenesulphonate
08/16/2000CN1263093A Amlo dipine mesylate and its preparation and application
08/16/2000CN1263089A Preparation of thiol-carbamate and sulfocyanic ester compound
08/16/2000CN1055470C Paroxetine and process for preparing medical salts thereof
08/16/2000CN1055463C Process for manufacture of guanidines
08/15/2000US6103937 Producing unsaturated nitrogen containing compounds such as enamides, enamines and aryl amineslamides using as catalyst nickel and an organophosphine or carbene ligand
08/15/2000US6103720 Ketobenzamides as calpain inhibitors
08/15/2000US6103719 Neurokinin-a- or neurokinin-b tachnkinin antagonistic properties; substance p antagonism; respiratory, gastrointestinal, nervous system, skin disorders;
08/10/2000WO2000046221A1 Sulfamato hydroxamic acid metalloprotease inhibitor