Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
10/2002
10/03/2002WO2002076988A2 Tert. alkylphenoxy substituted polycyclic compounds
10/03/2002WO2002076965A1 Non peptide mimetics based on the active sequence s42fllr46 of the thrombin receptor for the treatment of thrombosis and cancer
10/03/2002WO2002076964A1 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
10/03/2002WO2002076948A1 Novel piperidine derivatives as modulators of chemokine receptors
10/03/2002WO2002076947A1 Mch antagonists and their use in the treatment of obesity
10/03/2002WO2002076940A2 Process for preparing arylpiperidine carbinol intermediates and derivatives
10/03/2002WO2002076939A2 Cysteine protease inhibitors
10/03/2002WO2002076929A1 Aryl and biaryl compounds having mch modulatory activity
10/03/2002WO2002076926A1 3,4-di-substituted cyclobutene-1, 2-diones as cxc chemokine receptor antagonists
10/03/2002WO2002076925A2 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
10/03/2002WO2002076923A1 1,3-diamino-4-(aminomethyl)-benzene derivatives and colorants containing said compounds
10/03/2002WO2002076447A1 Hallogenated aminobenzophenones and aminobenzoylpyridines as inhibitors of il-1 and tnf
10/03/2002WO2002062784A8 Piperidinee derivatives as neurokinin 1 antagonists
10/03/2002US20020143177 For inhibiting beta-secretase enzyme activity and A beta peptide production, inhibition of beta-secretase enzyme activity halts or reduces production of A beta from APP and reduces or eliminates the formation of beta-amyloid deposits
10/03/2002US20020143056 As inactivator of antigen- specific T cells is useful in the prophylaxis or therapy of autoimmune diseases, disorders involving an autoimmune component or neoplastic diseases
10/03/2002US20020143046 Used as calcium channel blockers
10/03/2002US20020143026 Induce mitotic arrest thereby making them useful as anti-cancer agents; also for therapy of diseases which can be treated by inducing mitotic arrest
10/03/2002US20020143010 Compounds for treating fibromyalgia and chronic fatigue syndrome
10/03/2002US20020143007 Donates, transfers or releases nitric oxide, elevates endogenous levels of endothelium-derived relaxing factor, stimulates endogenous synthesis of nitric oxide or is a substrate for nitric oxide synthase; for use in therapy
10/03/2002US20020143003 As serotonin, norepinephrine and dopamine reuptake inhibitors, for therapy of central nervous system and other disorders
10/03/2002US20020142969 Using didepsipeptide for the control of endoparasites in medicine and veterinary medicine
10/03/2002US20020142023 Insecticide, miticide
10/03/2002CA2443289A1 1,3-diamino-4-(aminomethyl)-benzene derivatives and colorants containing said compounds
10/03/2002CA2441080A1 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
10/03/2002CA2436351A1 3,4-di-substituted cyclobutene-1, 2-diones as cxc chemokine receptor antagonists
10/02/2002EP1245564A1 Benzamidine derivatives
10/02/2002EP1244624A1 Anthracene derivatives as anti-cancer agents
10/02/2002EP1244623A1 A process for preparing 4-substituted piperidines
10/02/2002EP1244622A1 A process for preparing trans-2,4-disubstituted piperidines
10/02/2002EP1244617A1 Substituted aminoalkylamide derivatives as antagonists of follicle stimulating hormone
10/02/2002EP1244452A1 Urotensin-ii receptor antagonists
10/02/2002EP1244451A1 Substituted piperazine and piperidine calcium channel blockers
10/02/2002EP1244448A2 Novel methods for the treatment and prevention of ileus
10/02/2002EP1098894B1 Fkbp inhibitors
10/02/2002EP0706521B1 Imides as tnf alpha inhibitors
10/02/2002DE10112040A1 Verbessertes Verfahren zur Herstellung von Sulfonylcarboxamidderivaten An improved process for the preparation of Sulfonylcarboxamidderivaten
10/02/2002CN1372548A Heterocyclic compounds and medicinal use thereof
10/02/2002CN1372541A Sulfonyl carboxamide derivatives, method for their production and their use as medicaments
10/02/2002CN1371903A Optical isomer of 3-methyl fentanyl, derivant, synthesizing and its analgesic activity
10/02/2002CN1091768C Novel benzo-1,3-dioxolyl-and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists
10/02/2002CN1091594C Use of anti-viral compound in preparing medicine for curing virus infection
10/01/2002US6458998 Naphthaleneureas as antidiabetic agents
10/01/2002US6458960 Sulfonamide derivatives
10/01/2002US6458958 Process of preparing a piperidine derivative compound of the formula: acylating an .alpha.,.alpha.-disubstituted-methylbenzene derivative having the formula:
10/01/2002US6458957 α,α-dibromo-α-chloro-acetophenones as synthons
10/01/2002US6458954 Process for preparing piperidines
10/01/2002US6458829 Substituted γ-phenyl-Δ-lactones and analogs thereof and uses related thereto
10/01/2002US6458812 Muscarinic antagonists
10/01/2002US6458807 Methods for treating vascular dementia
10/01/2002US6458806 Aryl alkenamides derivatives as MCP-1 antagonists
10/01/2002US6458781 Blockers calcium channel antagonists for strokes, brain disorders
10/01/2002CA2245857C 1,4-dihydropyridine compounds as bradykinin antagonists
10/01/2002CA2203850C Novel n-phenyl-n-phenyliminonethylbenzamidines and their analogues as muscarinic receptor agonists
09/2002
09/26/2002WO2002074765A1 Phenyl derivatives 3
09/26/2002WO2002074744A1 Oxoammonium salts and the use thereof
09/26/2002WO2002074743A1 Aryl-substituted alicyclic compound and medical composition comprising the same
09/26/2002WO2002074735A2 Biurethane derivatives
09/26/2002WO2002074731A1 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds
09/26/2002WO2002074296A1 Remedies for solid cancer containing hydroxamic acid derivatives as the active ingredient
09/26/2002WO2002074050A2 Asymmetric synthesis of (s, s, r)-(-)-actinonin and its analogs and uses therefor
09/26/2002WO2002028810A3 Retinoids for the treatment of emphysema
09/26/2002WO2002024636A3 N-acylsulfonamide apoptosis promoters
09/26/2002WO2002018334B1 Sodium channel modulators
09/26/2002WO1997019953A8 New lh-rh antagonists with improved effectiveness
09/26/2002US20020137974 Catalysis using phosphine oxide and sulfoxide compounds
09/26/2002US20020137968 Treating with amides, ureas, amidines, carbamates, carboximidamides and other derivatives of given formula, e.g. (+)-N-((2,2-dimethylcyclopentyl)methyl)-4-hexyloxybenzamide
09/26/2002US20020137937 Process for preparing [S- (R*, S*) ] -beta- [ [ [1- [1-oxo-3- (4-piperidinyl) propyl] -3-piperidinyl] carbonyl]amino] -3-pyridinepropanoic acid and derivatives
09/26/2002US20020137932 Treating autoimmune diseases, Alzheimer's disease, atherosclerosis, osteoporosis, and asthma
09/26/2002US20020137929 1 - (3-heterocyclylphenyl) isothiourea, -isourea, -guanidine and -amidine herbicidal agents
09/26/2002US20020137770 Piperidine derivatives
09/26/2002US20020137742 Benzenesulfonamide compounds
09/26/2002US20020137686 Inhibitors of the ICE/ced-3 family of cysteine proteases
09/26/2002DE10114084A1 New 1,3-diamino-4-aminomethyl-benzene derivatives, useful as coupler substances in oxidative hair dye formulations based on a developer-coupler combination
09/26/2002DE10113710A1 Oxo-ammonium salts with a sterically-hindered oxo-ammonium group attached to an insoluble support material, used as oxidizing agents, especially for the oxidation of alcohol to ketone or aldehyde
09/26/2002DE10113402A1 New N,N'-bis-(Aminocarbonyl)-hydrazine derivatives are Factor Xa and Factor VIIa inhibitors useful e.g. for treating thrombosis, myocardial infarction, inflammation, apoplexy, restenosis or tumors
09/26/2002CA2445754A1 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds
09/26/2002CA2441822A1 Asymmetric synthesis of (s, s, r)-(-)-actinonin and its analogs and uses therefor
09/26/2002CA2441427A1 Biurethane derivatives
09/26/2002CA2440954A1 Phenyl derivatives 3
09/25/2002EP1243577A1 Novel phenylalanine derivatives
09/25/2002EP1242427A1 Novel piperidine and piperazine derivatives
09/25/2002EP1242406A1 Novel compounds
09/25/2002EP1242378A1 Novel processes
09/25/2002EP1242377A1 A process for the regioselective synthesis of 2,2-dialkyl-4-substituted piperidines
09/25/2002EP1242083A1 Phenoxypropanolamines, method for producing them and pharmaceutical compositions containing them
09/25/2002EP1242080A1 Dopamine transporter inhibitors and their use
09/25/2002EP1242075A2 Indole compounds
09/25/2002EP0912534B1 Muscarinic antagonists
09/25/2002CN1371365A Piperidine alcohols
09/25/2002CN1371364A Tetrahydropyridines as pesticides
09/25/2002CN1371356A Enatiomerically-enriched compounds having photocleavable bond(s) and methods related thereto
09/25/2002CN1371286A Use of cyclooxygenase-2 inhibitor matrix metallappoteinase inhibitor antineoplastic agent and optionally radiation as combination treatment of neoplasia
09/25/2002CN1091441C Amlo dipine mesylate and its preparation and application
09/24/2002US6455735 Reacting a tertiary or secondary amine with hydrogen peroxide in presence of a recyclable heterogeneous layered double hydroxide exchanged with one of the anions of transition metal oxides as a catalyst in a solvent
09/24/2002US6455700 Process for preparing guanidine and amidine derivatives
09/24/2002US6455671 Thrombin inhibitors, the preparation and use thereof
09/24/2002US6455581 Inhibitors of hiv protease.
09/24/2002US6455550 N-alkanoylphenylalanine derivatives
09/24/2002US6455549 Arylpiperidinol and arylpiperidine derivatives and drugs containing the same
09/24/2002US6455545 Gastrointestinal disorders