Patents
Patents for C07D 211 - Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings (37,939)
12/2002
12/18/2002EP1265606A1 Cell adhesion inhibitors
12/18/2002EP1119564B1 Aryl- 4-fluoro-4- (2-pyridin-2-yl-ethylamino)-methyl]-piperidin-1-yl -methanone derivatives as 5-ht1 receptor antagonists
12/18/2002EP0930298B1 Fluorinated 1,4-disubstituted piperidine derivatives
12/18/2002EP0882038B1 substituted n-methyl-n-(4-(piperidin-1-yl)-2-(aryl)butyl)benzamides useful for the treatment of allergic diseases
12/18/2002EP0859607B1 Guanidino protease inhibitors
12/18/2002EP0843658B1 Didepsipeptide-based endoparasiticides, new didepsipeptides and process for preparing the same
12/18/2002CN1096460C Novel substituted N-methyl-N-(4-(piperidin-1-yl)-2-(aryl)butyl)benzamides useful for treatment of allergic diseases
12/17/2002US6495720 Preparing trisubstituted hydroxylamines, obtained from nitroxides, which can be used in particular as radical-polymerization initiators
12/17/2002US6495715 Calcium channel blockers
12/17/2002US6495694 Dissolving, precipitating
12/17/2002US6495681 Local anesthetic compounds and uses
12/17/2002US6495597 N-formyl hydroxylamine derivatives
12/17/2002US6495568 Treatment of tissue ulceration, wound repair and skin diseases
12/17/2002US6495565 For therapy of acute infection, acute phase response, age related macular degeneration, alcoholism, anorexia, asthma, autoimmune disease, autoimmune hepatitis, bechet's disease, cachexia, calcium pyrophosphate dihydrtate deposition
12/17/2002US6495549 1-heteroaryl-piperidine derivatives; moderating neuronal degeneration; promoting neuronal regeneration and outgrowth; treatog neurological disorders arising from neurodegenerative diseases or other disorders involving nerve damage
12/17/2002US6495546 Propanolamine derivatives
12/12/2002WO2002099045A2 Peptide beta-strand mimics based on 1,2-dihydro-3(6h)-pyridinone
12/12/2002WO2002098872A1 Isoindolines and process for preparation thereof
12/12/2002WO2002098850A2 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors
12/12/2002WO2002098849A2 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer’s disease and similar diseases
12/12/2002US20020188130 Alpha, alpha-dibromo-alpha-chloro-acetophenones as synthons
12/12/2002US20020188120 Such as 4-(4-methyoxy-benzenesulfonyl)-1-(3-phenyl-propyl)-piperidine-4-carboxylic acid hydroxyamide for treatment of arthritis, tumor metastasis, tissue ulceration, abnormal wound healing, periodontal disease, bone diseases, diabetes, and HIV
12/12/2002US20020188006 4-hydroxypiperidine derivatives having antiarrhythmic activity
12/12/2002CA2448834A1 Hydroxy alkyl amine derivatives as beta-secretase inhibitors and their use for the treatment of alzheimer's disease and similar diseases
12/12/2002CA2448418A1 Chemical compounds and pharmaceutical compositions as cathepsin s inhibitors
12/11/2002EP1264828A1 New inhibitor of urokinase
12/11/2002EP1264822A2 Stabiliser modification
12/11/2002EP1263760A1 Novel compounds
12/11/2002EP1263756A2 Beta-amino acid derivatives as inhibitors of matrix metalloproteases and tnf-alpha
12/11/2002EP1263730A1 Amine derivatives for the treatment of apoptosis
12/11/2002EP1263729A1 Azacyclic compounds for use in the treatment of serotonin related diseases
12/11/2002EP1263725A1 Novel compounds
12/11/2002EP1263724A1 Novel compounds
12/11/2002EP1263714A1 Novel phenylheteroalkylamine derivatives
12/11/2002EP1263712A1 3-(2,5-diaminophenyl)-acrylamide derivatives and colouring agents containing said compounds
12/11/2002EP1263711A1 Novel use of phenylheteroalkylamine derivatives
12/11/2002EP1263504A2 Compounds with 5-ht1a activity useful for treating disorders of the outer retina
12/11/2002EP1263434A1 Compounds with 5-ht 2 and 5-ht 1a agonist activity for treating glaucoma
12/11/2002EP0937064B1 Substituted oximes derivatives useful as neurokinin antagonists
12/11/2002EP0721455B1 Tetrahydropyridine-(or 4-hydroxypiperidine)alkylazoles having an affinity for sigma and/or 5ht1a receptors
12/11/2002EP0662958B1 1-(2-oxo-acetyl)-piperidine-2-carboxylic acid derivatives as multi-drug-resistent cancer cell sensitizers
12/11/2002CN1384830A Novel spiroheterocyclic compoundsus reversible inhibitors of cysteine proteases
12/11/2002CN1384743A Remedies or preventives for diseases in association with chemokines
12/11/2002CN1384100A Benzo-1,3-dioxole and benzofuran substituted pentazane derivative
12/10/2002US6492523 Subjecting a pyrrole derivative, methyl aminocrotonate and 2-chlorobenzaldehyde to a hantzsch reaction, and converting the pyrrole residue of the resulting product to an amine group by the action of hydroxylamine hydrochloride.
12/10/2002US6492522 Process and intermediates for production of donepezil and related compounds
12/10/2002US6492521 Hindered amine light stabilizers based on multi-functional carbonyl compounds and methods of making same
12/10/2002US6492423 Hepatitis c and b viricides
12/10/2002US6492400 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
12/10/2002US6492396 Substituted thioacetamides
12/10/2002US6492393 Compounds useful as anti-inflammatory agents
12/10/2002US6492375 Administering a piperidine compound
12/10/2002US6492372 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4
12/10/2002US6492367 Sulfamato hydroxamic acid metalloprotease inhibitor
12/10/2002US6492365 Microsomal triglyceride transfer protein
12/10/2002US6492362 Compounds and compositions as cathepsin S inhibitors
12/10/2002US6492355 Adamantane derivatives
12/10/2002CA2230445C Fibrinogen receptor antagonists and medicinal preparations containing the same as the active ingredient
12/10/2002CA2228752C (1s,2s)-1-(4-hydroxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)-1-propanol methanesulfonate trihydrate
12/09/2002WO2002004403A1 Biphenylcarboxylic acid amides, production thereof and use thereof as medicaments
12/09/2002CA2412116A1 Biphenylcarboxylic acid amides, the preparation thereof and the use thereof as medicaments
12/05/2002WO2002096909A1 Optical resolution of (1-benzyl-4-methylpiperidin-3-yl) -methylamine and the use thereof for the preparation of pyrrolo 2,3-pyrimidine derivatives as protein kinases inhibitors
12/05/2002WO2002096875A1 4-hydroxpiperidine derivative with analgetic activity
12/05/2002WO2002096872A1 Substituted imidates as pesticidal agents
12/05/2002WO2002096864A1 Carboxamide-substituted phenylurea derivatives and method for production thereof as medicaments
12/05/2002WO2002096420A2 Method for treating nerve injury caused by surgery
12/05/2002WO2002096351A2 Ultrashort-acting opioids for transdermal application
12/05/2002US20020183518 Use for treatment of human and animal disorders, for purification of proteins or glycoproteins, and in diagnosis
12/05/2002US20020183343 Ultrashort-acting opioids for transdermal application
12/05/2002US20020183342 For use as insecticides against a variety of insects, including larvae, such as tobacco budworm
12/05/2002US20020183334 For therapy of sleepiness, promotion of wakefulness, treatment of Parkinson's disease, cerebral ischemia, stroke, sleep apneas, eating disorders, stimulation of appetite and weight gain, treatment of attention deficit hyperactivity disorder
12/05/2002US20020183324 Monocyclic or bicyclic carbocycles and heterocycles as factor Xa inhibitors
12/05/2002US20020183321 Carbocyclic and heterocyclic substituted semicarbazones and thiosemicarbazones and the use thereof
12/05/2002US20020183316 Amidoalkyl-piperidine and amidoalkyl-piperazine derivatives useful for the treatment of nervous system disorders
12/05/2002DE10125963A1 Substituierte Imidate Substituted Imidates
12/05/2002DE10125567A1 New N-aroyl-N'-(carbamoyl-phenyl)-urea derivatives, are glycogen phosphorylase a inhibiting hypoglycemic agents, especially useful for treating type II diabetes
12/05/2002CA2449019A1 Method for treating nerve injury caused by surgery
12/05/2002CA2448509A1 4-hydroxypiperidine derivatives having analgesic activity
12/05/2002CA2448023A1 Carboxamide-substituted phenylurea derivatives and method for production thereof as medicaments
12/05/2002CA2443350A1 Ultrashort-acting opioids for transdermal application
12/04/2002EP1261731A1 Cationic amphiphilic 1,4-dihydropyridine derivatives useful for delivery of nucleotide containing compounds
12/04/2002EP1261630A2 Bacterial genes and proteins that are essential for cell viability and their uses
12/04/2002EP1261595A1 Arylpiperazines and arylpiperidines and their use as metalloproteinase inhibiting agents
12/04/2002EP1261594A1 5,10-dihydroacridines as calcium channel blockers
12/04/2002EP1261583A1 INHIBITORS OF THE ICE/Ced-3 FAMILY OF CYSTEINE PROTEASES
12/04/2002EP1261579A1 Dehydroamino acids
12/04/2002EP1261339A1 Use of n-substituted-1,5-dideoxy-1,5-imino-d-glucitol compounds for treating hepatitis virus infections
12/04/2002EP1261321A2 Carboxylic acid amides, medicaments containing these compounds and the use and production thereof
12/04/2002EP1001930B1 N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases
12/04/2002CN1382442A Method for preventing dyskinesia
12/03/2002US6489512 Method for making aryl hydrazines and substituted indoles
12/03/2002US6489482 Monomer compatibility; reacting a hindered piperidine with an acryloyl chloride
12/03/2002US6489479 Process for the preparation of mixed anhydrides
12/03/2002US6489347 Process
12/03/2002US6489334 Method for the crystallization of a tetrahydropyridin derivative and resulting crystalline forms
12/03/2002US6489327 Tryptase inhibitors
11/2002
11/28/2002WO2002094812A1 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
11/28/2002WO2002094811A1 4-(penyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
11/28/2002WO2002094810A1 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
11/28/2002WO2002094809A1 3-quinoline-2-(1h)-ylideneindolin-2-one derivatives