Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
04/1995
04/25/1995CA1335379C Aralkylaminoalkoxyphenyl derivatives, process of preparation and compositions containing the same
04/25/1995CA1335378C Alkylaminoalkoxyphenyl derivatives, process of preparation and compositions containing the same
04/23/1995CA2132883A1 1-amino-ethylindole-derivatives
04/20/1995DE2858800C2 2-Guanidino-thiazole and imidazole derivs.
04/19/1995EP0648762A2 Bicyclic compounds as excitatory amino acid receptor antagonists
04/19/1995EP0648208A1 Indole derivatives as testosterone 5 alpha-reductase inhibitors
04/19/1995EP0550635B1 Fused ring analogs of nitrogen containing nonaromatic heterocycles
04/19/1995CA2117852A1 Bicyclic compounds as excitatory amino acid receptor antagonists
04/18/1995CA1335286C Labile ketone derivatives of 3-substituted-1-alkylamino 2-propanols and their use as .beta.-adrenergic blockers
04/13/1995WO1995009843A1 Hiv protease inhibitors
04/13/1995WO1995009835A1 Novel phenylethyl and phenylpropylamines
04/13/1995WO1995009833A1 Mercaptosulfide metalloproteinase inhibitors
04/13/1995WO1995009831A1 Nitric esters having anti-inflammatory and/or analgesic activity and process for their preparation
04/13/1995WO1995009628A1 Therapeutic application of perhydroisoindole derivatives as an anti-emetic
04/13/1995WO1995009620A1 Sulfoximine and sulfodiimine matrix metalloproteinase inhibitors
04/13/1995CA2150005A1 Novel phenylethyl and phenylpropylamines
04/12/1995EP0647874A1 Highly efficient nonlinear optical polyimides
04/12/1995EP0647644A1 Antibacterial pyrido 1,2,3-d,e 1,3,4 benzoxacin derivatives
04/12/1995EP0647625A1 Novel antibiotics with immunosuppressive activity, delaminomycins, and production thereof
04/12/1995EP0647231A1 N-substituted 3-azabicyclo 3.2.0]heptane derivates useful as neuroleptic agents, etc.
04/12/1995CN1101303A Process for preparing weakly-basic anion exchangers and reagents suitable for this purpose
04/11/1995US5405995 Difluorophthalic compounds and their preparation
04/11/1995US5405968 Useful as drugs, for producing singlet oxygen, sensitizers in electrophotographic layers and for photopolymerizations and as laser light sensitive dyes in optical recording media
04/11/1995US5405877 Water solubility; hydrolytic stability
04/11/1995US5405863 Antioxidant cardioprotective use of, and method of treatment using, hydroxycarbazole compounds
04/11/1995US5405860 Triazolyl-alkanones or triazolyl-alkanols
04/08/1995CA2132771A1 Biaryl urea and related compounds
04/06/1995WO1995009169A1 Process for the preparation of 9-amino camptothecin
04/06/1995WO1995009151A1 Acylated sulphonamides as insecticides and acaricides
04/06/1995WO1995009001A1 Inhibitors of farnesyl-protein transferase
04/06/1995CA2172125A1 Inhibitors of farnesyl-protein transferase
04/05/1995EP0646598A1 New pseudopeptides with antiviral activity containing valine
04/05/1995EP0646569A1 Novel carboxylate derivatives exhibiting phospholipase A2 inhibitory activity
04/05/1995EP0646112A1 Tertiary and secondary amines as alpha-2 antagonists and serotonin uptake inhibitors
04/05/1995EP0646110A1 N-substitued 3-azabicyclo 3.2.0]heptane derivatives useful as neuroleptic agents etc.
04/05/1995EP0555283B1 Intermediates in the preparation of 4,5-difluoroanthranilic acid
04/05/1995EP0387357B1 Indolenine derivatives
04/05/1995CN1101040A Diaryl derivatives and their use as crop protection agents
04/05/1995CN1101039A 哌嗪衍生物 Piperazine derivatives
04/05/1995CN1100933A Hypoglycemic agents
04/05/1995CN1100932A Use of the substituted azaspirane in the manufacture of a medieament for the treatment of psoriasis
04/05/1995CN1028102C Process for spiro compound
04/04/1995US5403868 Capsaicin derivatives
04/04/1995US5403861 Treating or preventing nerve cell death
04/04/1995US5403851 Substituted tryptamines, phenalkylamines and related compounds
04/04/1995US5403850 Elastase inhibitors, respiratory system disorders
04/04/1995US5403702 Crystals consisting of an indolinospirobenzopyran derivative
04/04/1995CA1335102C P-hydroxy phenone derivatives and drugs containing these
04/02/1995CA2133115A1 Carboxylate derivatives exhibiting phospholipase a2 inhibitory activity
03/1995
03/29/1995EP0645391A2 Aminobenzoic acid derivatives
03/29/1995EP0645379A2 Benzoylacetylene derivatives
03/29/1995EP0645375A1 Use of benzene-sulfonyl-indole derivatives for the preparation of a medicament
03/29/1995EP0644876A1 Ultra white n,n'-ethylene-bis(tetrabromophthalimide) and its production in aqueous acetic acid
03/29/1995EP0644875A1 Ultra white n,n'-ethylene-bis(tetrabromophthalimide) and its production in acetic acid
03/29/1995CN1100720A Cyclopentadiene derivatives
03/29/1995CN1100634A Method of preventing emesis and treating sexual dyfunction using tetra hydrobenzÛCDÙ indole-6-carboxamides
03/28/1995US5401855 4-hydroxyphenylthio derivatives, their preparation and their use for the preparation of aminoalkoxyphenylsulphonyl derivatives
03/28/1995US5401854 Process for the production of indole derivatives
03/28/1995US5401766 Aminoacid derivatives, a process for their preparation, agents containing these compounds, and the use thereof
03/28/1995US5401729 7-(substituted)-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
03/28/1995US5401438 Photostabilizers
03/23/1995WO1995007950A1 Process for the production of cyanine dyes
03/23/1995WO1995007888A1 Method for the preparation of high purity substituted benz[e]indoles and the alkaline salts thereof
03/23/1995WO1995007887A1 Indole derivatives as antagonists of excitatory amino acids
03/23/1995WO1995005364A3 Inhibitors of biogenic amine transporters
03/22/1995EP0644198A1 Alpha-heteroaryloxymethyl ketones as interleukin-1beta converting enzyme inhibitors
03/22/1995EP0644187A1 Antimigraine cyclobutenedione derivatives of tryptamines
03/22/1995EP0643706A1 Compounds, compositions and methods for binding bio-affecting substances to surface membranes of bio-particles
03/22/1995EP0643695A1 Fungicidal indole derivatives.
03/22/1995EP0643694A1 A process for the preparation of eserethole
03/22/1995EP0473637B1 Peroxyacid manufacture
03/22/1995CN1100417A N-heteroaryl-n'-phenylurea derivatives, their production and use
03/21/1995US5399714 One-pot reduction; acylation
03/21/1995US5399713 Process for the production of 5,6-dihydroxyindolines
03/21/1995US5399711 Thiomarinol compounds
03/21/1995US5399707 Making salt of amino acid lysine, arginine or histidine with alpha-arylcarboxylic acid either by starting from second salt of anion and protonated cation of amino acid or by distilling water from amino acid-arylcarboxylic acid mixture
03/21/1995US5399559 Fungicidal indole derivatives
03/21/1995US5399487 6-peptidylamino-1-naphthalenesulfonamides useful as fluorogenic proteolytic enzyme substrates
03/17/1995CA2130519A1 Antimigraine cyclobutenedione derivatives of tryptamines
03/16/1995WO1995007291A1 Kininogen inhibitors
03/16/1995WO1995007276A1 Bicyclic heterocyclic sulfonamide and sulfonic ester derivatives
03/16/1995WO1995007269A1 Polar-substituted hydrocarbons
03/16/1995WO1995007261A1 Polyamidic acid derivatives with antigastrin activity, a method for their preparation, and their pharmaceutical use
03/16/1995WO1995007258A1 Cyclohexanediurea derivative and process for producing the same
03/16/1995CA2171471A1 Polar-substituted hydrocarbons
03/16/1995CA2171295A1 Cyclohexanediurea derivative and process for producing the same
03/16/1995CA2170896A1 Kininogen inhibitors
03/16/1995CA2170648A1 Polyamidic acid derivatives with antigastrin activity, a method for their preparation, and their pharmaceutical use
03/15/1995EP0643039A1 Ultraviolet ray-absorbing aromatic compound and polymeric composition containing the same
03/15/1995EP0642787A2 Cessation of tobacco use
03/15/1995EP0642496A1 Synthetic heteroaryl polyamines as excitatory amino acid neurotransmitter antagonists
03/15/1995EP0526478B1 3-indolyl thioacetate derivatives
03/15/1995CN1100095A Preparation of a sprio compound
03/15/1995CN1100094A Process for the enantioselective synthesis of alkylated oxindoles used as intermediates in the preparation of physostigmine
03/15/1995CN1027892C Improved process for preparation of substituted indolone derivatives
03/15/1995CA2131759A1 Valine-containing pseudopeptides with antiviral activity
03/14/1995US5397846 Process for preparing organic compounds carrying tert-butyloxycarbonyl groups
03/14/1995US5397819 Thermoplastic materials containing near infrared fluorophores
03/14/1995US5397801 N-sulfonylindoline derivatives, their preparation and the pharmaceutical compositions in which they are present
03/14/1995US5397800 Gastrointestinal disorders