Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
06/1995
06/06/1995US5422371 Contacting a cell with a fatty acid or fatty alcohol to prevent reduction of testosterone to 5a-dihydrotestosterone
06/04/1995CA2136904A1 Excitatory amino acid receptor antagonists
06/01/1995WO1995014668A1 2-oxoindoline derivative
06/01/1995WO1995014667A1 Substituted indoles as phosphodiesterase type iv inhibitors
06/01/1995WO1995014666A1 Indolyl group containing compounds and the use thereof to promote the release of growth hormone(s)
06/01/1995WO1995014467A1 Therapeutic guanidines
06/01/1995WO1995014384A1 Inhibition of smooth muscle migration and proliferation with hydroxy carbazole compounds
06/01/1995CA2224051A1 Intermediates for producing substituted indoles as phosphodiesterase type iv inhibitors
06/01/1995CA2224049A1 Intermediates for producing substituted indoles as phosphodiesterase type iv inhibitors
06/01/1995CA2177084A1 Therapeutic guanidines
06/01/1995CA2176377A1 Inhibition of smooth muscle migration and proliferation with hydroxy carbazole compounds
06/01/1995CA2176140A1 Indolyl group containing compounds and the use thereof to promote the release of growth hormone(s)
05/1995
05/31/1995EP0655440A2 1-Aminoethylindoles
05/31/1995EP0655439A2 5,6-Bicyclic glycoprotein IIb IIIa antagonists useful in inhibition of platelet aggregation
05/31/1995EP0655243A2 Melatonin derivatives for use in treating sleep disorders
05/31/1995EP0655240A2 Immediate release tablet cores of insoluble drugs having substained-release coating
05/31/1995EP0655056A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
05/31/1995EP0655055A1 Tachykinin antagonists
05/31/1995EP0654997A1 Compositions of substituted azaspiranes and methods of treating psoriasis therewith
05/31/1995EP0654996A1 Methods of treating psoriasis employing substituted azaspiranes
05/31/1995EP0602083B1 Process for producing 5,6-dihydroxyindolines
05/31/1995CN1028592C Substituted guanidine derivatives their preparation and use
05/30/1995US5420294 Cycloalkylaminoalkoxyindoles
05/30/1995US5420289 Antiinflammatory agents, antiallergens and cytoprotective agents
05/30/1995US5420234 Polymers
05/30/1995US5420127 Morpholino-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/30/1995CA1335734C Crosslinking imidophenylamines
05/26/1995WO1995014019A1 Herbicidal pyrrolopyridine compounds
05/26/1995WO1995014017A1 Non-peptide tachykinin receptor antagonists
05/26/1995WO1995014004A1 Indole-derived azylpiperazines as ligands for 5ht1-like receptors 5ht1b and 5ht1d
05/26/1995WO1995014003A1 Propenone derivative
05/26/1995CA2176737A1 Herbicidal pyrrolopyridine compounds
05/26/1995CA2176735A1 Non-peptide tachykinin receptor antagonists
05/26/1995CA2153905A1 Propenone derivatives
05/24/1995EP0654024A1 2-thioindoles (selenoindoles) and related disulfides (selenides) which inhibit protein tyrosine kinases and which have antitumor properties
05/24/1995EP0654023A1 5-(2-oxyphenyl)-pyrrole derivatives as dopamine d3 receptor antagonists
05/23/1995US5418249 Renin inhibitors
05/23/1995US5418245 For inhibiting cell proliferation
05/23/1995US5418237 Indole derivatives
05/18/1995WO1995013266A1 Acylpyrrole-alkanoic acids and indole-2-alkanoic acids plus their derivatives for use as inhibitors of phospholipase a¿2?
05/18/1995WO1995013262A1 Substituted phenyl compounds
05/18/1995CA2176363A1 Substituted phenyl compounds
05/18/1995CA2135811A1 Tricyclic indole-2-carboxylic acid derivatives
05/17/1995EP0652749A1 METHODS AND COMPOSITIONS FOR INHIBITING 5$g(a)-REDUCTASE ACTIVITY
05/17/1995EP0497816B1 Treatment of hiv infections and compounds useful therein
05/17/1995CN1102643A Substituted derivatives of diaminophthalimide
05/16/1995US5416221 Carbazolone derivatives
05/16/1995US5416111 Cyano-containing n-phenyl-amino-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416104 Oxazolidinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416099 Fibrinogen receptor antagonists
05/16/1995US5416095 Tetrahydro-quinolinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416092 3-azabicyclo[3.2.1]-oct-8-yl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416085 3-oxa-8-azabicyclo[3.2.1]oct-8-yl terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416083 Benzodiazepinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416068 Alpha-phenylacrylic acid derivatives, their preparation and their use for controlling pests and harmful fungi
05/16/1995CA1335595C Radiation sensitive compounds
05/16/1995CA1335590C Anhydrous, crystalline sodium salt of 5-chloro-3-(2-thenoyl)-2-oxindole-1-carboxamide
05/13/1995CA2134192A1 5, 6-bicyclic glycoprotein iib/iiia antagonists
05/11/1995WO1995012611A1 Endothelin receptor antagonists
05/11/1995WO1995012603A1 Matrix metalloprotease inhibitors________________________________
05/11/1995CA2175667A1 Matrix metalloprotease inhibitors________________________________
05/11/1995CA2173875A1 Endothelin receptor antagonists
05/10/1995EP0652212A1 Substituted fluorine-containing beta-indolebutyric acid derivatives, their preparation and their use as plant growth regulators
05/10/1995EP0652208A1 Phenylalkan(en)oic acids with leukotriene B4 antagonistic activity
05/10/1995EP0651750A1 Tetracyclic compounds process and intermediates for their preparation and their use as antitumour agents
05/10/1995EP0651743A1 Indolinyl n-hydroxyurea and n-hydroxamic acid derivatives as lipoxygenase inhibitors
05/10/1995CN1102409A Process for the preparation of indoles
05/09/1995US5414791 Thermally stable electro-optic device and method
05/09/1995US5414089 Useful for modifying enzymes or proteins
05/09/1995US5414070 Poly(amide-ether-imide)s
05/09/1995US5414017 Cardiovascular agents
05/09/1995US5414013 Trifluoromethyl mercaptan and mercaptoacyl derivatives and method of using same
05/09/1995US5414012 Indalyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/04/1995WO1995011885A1 Certain fused pyrrolecarboxanilides; a new class of gaba brain receptor ligands
05/04/1995WO1995011774A1 Abrasive articles incorporating addition polymerizable resins and reactive diluents, and methods of making said abrasive articles
05/04/1995CA2174113A1 Abrasive articles incorporating addition polymerizable resins and reactive diluents, and methods of making said abrasive articles
05/03/1995EP0650599A1 Method of colorimetric analysis of malonic dialdehyde and 4-hydroxy-2-enaldehydes as indexes of lipid peroxidation, kits for carrying out said method, substituted indoles for use in said method and their preparation
05/03/1995EP0650372A1 Compounds for cancer imaging and therapy
05/02/1995US5411962 Benzomorpholinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/02/1995US5411960 Substituted pyrroloanthracenes and -diones
05/02/1995US5411958 Benzothiomorpholinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/02/1995US5411957 3-azabicyclo[3.2.1]-nonanyl-terminated non-piptidyl alpha-succinamidoacyl aminodiols as anti-hypertensive agents
05/02/1995US5411869 Immunological analogs for captan
05/02/1995US5411743 Prevention of synovial adhesions
05/02/1995CA1335450C Indole and indazole keto sulphones as leukotriene antagonists
04/1995
04/27/1995WO1995011231A1 Amidino derivatives useful as nitric oxide synthase inhibitors
04/27/1995WO1995011224A1 Process for the preparation of a substituted 2,5-diamino-3-hydroxyhexane
04/27/1995WO1995011221A1 Calcium receptor-active arylalkyl amines
04/27/1995CA2173468A1 Amidino derivatives useful as nitric oxide synthase inhibitors
04/26/1995EP0649443A1 Oxazolone derived materials
04/26/1995EP0649406A1 Novel carbazole derivatives and their use in cosmetics, especially for make-up
04/26/1995EP0515510B1 Hydroquinone amino-acid esters, method of preparation, and pharmaceutical or cosmetic compositions containing them
04/26/1995CN1101908A Angiotensin II antagonists
04/25/1995USRE34918 Antihistamines, muscle relaxants
04/25/1995US5410067 Catalytic hydrogenation; cyclization
04/25/1995US5409949 Methylen-oxindole derivatives compositions and tyrosine kinase inhibition therewith
04/25/1995US5409941 5-heteroyl indole derivatives
04/25/1995US5409932 Antiarthritic agent for rheumatic diseases, antiinflammatory agent for gastric diseases, gastrointestinal disorders
04/25/1995US5409930 Inhibits abnoramal cell proliferation; dimethoxyquinoline/ dimethylquinoline/ quinolineoxide/ and quinoxaline derivatives
04/25/1995US5409929 Hydroisoindolines and hydroisoquinolines as psychotropic drugs