Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
01/2007
01/09/2007US7161009 Antiinflammatory agents; skin disorders; central nervous system disorders
01/09/2007US7160923 Polyamine analogues as therapeutic and diagnostic agents
01/09/2007US7160918 Substituted indole oxo-acetyl amino acetic acid derivatives as inhibitors of plasminogen activator inhibitor (PAI-1)
01/09/2007US7160917 Prepared by fermentation by microorganism Stachybotris; anticoagulants, anticarcinogenic, antitumor, antidiabetic, and antihypoxic agents; cardiovascular disorders, angina pectoris, septic shock, arteriosclerosis
01/09/2007US7160909 Cyclopenta[b]indole derivatives as sPLA2 inhibitors
01/09/2007US7160903 Sulfonylaminocarboxylic acids
01/09/2007US7160901 Antiproliferative agents; antitumor agents; kinase inhibitors
01/09/2007US7160899 Use of at least one compound with neurotrophic activity and at least one adenosine A2A receptor antagonist for the manufacture of a medicament for the treatment, prevention or alleviation of Parkinson's disease in a subject
01/09/2007US7160887 Aromatic amine derivatives, their production and use
01/09/2007US7160854 Binaphthyl peptidomimetics for treating vancomycin resistant Staphylococcus aureas infections
01/09/2007US7160684 Methods of selecting compounds for modulation of bladder function
01/09/2007US7160556 Immediate release medicinal compositions for oral use
01/09/2007US7160555 Antidiabetic agents
01/09/2007CA2407538C Novel bicyclic compounds
01/09/2007CA2169831C Cosmetic melanins
01/09/2007CA2144293C Substituted propane derivatives, a process for their preparation and the use of the compounds for treating diseases
01/09/2007CA2102780C Bis mono-and bicyclic aryl and heteroaryl compounds which inhibit egf and/or pdgf receptor tyrosine kinase
01/04/2007WO2007002314A2 Polymorphic forms of tegaserod maleate
01/04/2007WO2007002181A2 Tetrahydrocarbazole derivatives useful as androgen receptor modulators (sarm)
01/04/2007WO2007001015A1 Process for production of optically active aminopentane derivative, intermediate in the process and process for production of the intermediate
01/04/2007WO2007000339A1 Bicyclic derivatives as p38 kinase inhibitors
01/04/2007WO2007000337A1 Bicyclic derivatives as p38 kinase inhibitors
01/04/2007US20070004890 N-vinylformamide derivatives, polymers formed therefrom and synthesis thereof
01/04/2007US20070004806 Carbamic acid compounds comprising a sulfonamide linkage as HDAC inhibitors
01/04/2007US20070004791 (1 alpha ,5 alpha ,6 alpha )-N-[3-benzyl-3-azabicyclo[3.1.0]hexyl-6-(aminomethyl)-yl]-2-hydroxy-2,2-diphenyl acetamide; high affinity towards Muscarinic 3 receptors; avoiding adverse side effects; for the treatment of various diseases of the respiratory, urinary and gastrointestinal systems
01/04/2007US20070004757 Indoline derivatives substituted in the 6 position, their preparation and their use as medicaments
01/04/2007US20070004719 Inhibitors of cytosolic phospholipase A2
01/04/2007US20070004717 sarcopenia,frailty or age-related functional decline; nonsteroidal, nontoxic; side effect reduction;2-Chloro-4-(-4-hydroxy-1-oxo-hexahydrocyclopenta[c]pyrrol-2(1H)-yl)-3-methylbenzonitrile
01/04/2007US20070004703 Use of 1-(dialkoxyphenylsulfonyl)-3-(pyrrolidino)-3-(phenyl)indolin-2-one compounds to treat hypertension, cardiovascular disorders, central nervous system disorders, psychological disorders, gastrointestinal disorders; affinity for V1b and V1a receptors of arginine-vasopressin
01/04/2007CA2613720A1 Bicyclic derivatives as p38 kinase inhibitors
01/04/2007CA2613354A1 Non-nucleoside anti-hepacivirus agents and uses thereof
01/04/2007CA2612290A1 Process for preparing optically active aminopentane derivative, intermediate and process for preparing intermediate
01/04/2007CA2612008A1 Bicyclic derivatives as p38 kinase inhibitors
01/04/2007CA2611128A1 Novel indoline compounds
01/03/2007EP1739082A1 HIV protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
01/03/2007EP1739073A1 New primary 2,3-disubstituted para-phenylendiamins and their use as oxidative colouring of keratinic fibers
01/03/2007EP1737925A1 New organic luminescent element
01/03/2007EP1737854A1 NOVEL 2-(1-AZA-BICYCLO[2.2.2]OCT-3-yl)-2,3-DIHYDROISOINDOL-l-ONE/5,6-DIHYDRO-FURO[2,3-c]PYRROL-4ONE DERIVATIVES LIGANDS FOR ALPHA 7 NICOTINIC ACETYLCHOLINE RECEPTOR
01/03/2007EP1737827A1 Process for preparing pyridazinone compounds
01/03/2007EP1737821A1 3,4-(cyclopentyl)-fused proline compounds as inhibitors of hepatitis c virus ns3 serine protease
01/03/2007EP1737820A1 Asymmetric hydrogenation process useful for the preparation of cycloalkanoindole derivatives
01/03/2007EP1737815A1 Thio-substituted biaryl-methanesulfinyl derivatives
01/03/2007EP1737813A1 Androgen modulators
01/03/2007EP1737812A1 Methods of amination
01/03/2007EP1737811A1 Cetp inhibitors
01/03/2007EP1362601B1 Method of examining effect of angionegesis inhibitor mediated by the inhibition of integrin expression
01/03/2007EP1310487B1 Processes for preparation of bicyclic compounds and intermediates therefor
01/03/2007EP1202963B1 Spla2 inhibitors
01/03/2007EP1126839B1 Substituted phenethylsulfones and method of reducing tnf-alpha and pde-iv levels
01/03/2007CN1890248A Novel compounds
01/03/2007CN1890215A Inhibitors of hepatitis c virus ns3/ns4a serine protease
01/03/2007CN1890214A Heterocyclic- or aryloxy, -thio or -amino substituted indoles-2-carboxylic acids or esters as pai-1
01/03/2007CN1890213A Process for the preparation of n-amino substituted heterocyclic compounds
01/03/2007CN1889947A Tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents
01/03/2007CN1887883A V-shaped conjugated light-absorbing organic salt compound and its use
01/03/2007CN1887865A Synthesis of 3-substituted phenyl indole compound
01/03/2007CN1293063C Substituted heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them
01/03/2007CN1293057C Ethylenediamine derivatives
01/03/2007CN1293054C Processes for preparation of bicyclic compounds and intermediates therefor
01/03/2007CN1293053C 1-sulfonyl-4-aminoalkoxy indole derivatives as 5-ht6-receptor modulators for the treatment of cns-disorders
01/03/2007CN1293042C Aromatic amino acid derivates and medicinal compositions
01/02/2007US7157585 An aromatic alkylamino compound containing a lipophilic group useful as antithrombotic agent and for use in the treatment of mast cell mediated diseases such as asthma and other allergic and inflammatory conditions
01/02/2007US7157577 5-sulfonamido-substituted indolinone compounds as protein kinase inhibitors
01/02/2007US7157489 HIV protease inhibitors
01/02/2007US7157488 N-(2-(6-Fluoro-1H-indol-3-yl)ethyl)-3-(2,2,3,3-tetrafluoropropoxy)benzylamine; treating schizophrenia, anxiety, Alzheimer's disease, and cognitive disorders
01/02/2007US7157487 Vla-4 inhibitors
01/02/2007US7157486 For therapy and prophylaxis of hepatitis C virus (HCV) infection
01/02/2007US7157485 2S, 3aS, 7aS)-1-{(2S)-2 [(tert-Butoxycarbonyl)-amino]-propionyl}-octahydro-1H-indole-2-carboxylic acid; using, as sole sources of chirality, alanine starting material and a compound readily accessible from serine
01/02/2007US7157484 Method for synthesissing (2s, 3as, 7as)-perhydroindole-2-carboxylic acid and the esters thereof and the use thereof for perindopril synthesis
01/02/2007US7157470 For use as anticoagulant agents for therapy of thromboembolic disorders
01/02/2007US7157463 Substituted piperidines/piperazines as melanocortin receptor agonists
01/02/2007US7157454 Derivatives of n-(arylsulfonyl)beta-aminoacids comprising a substituted aminomethyl group, the preparation method thereof and the pharmaceutical compositions containing same
01/02/2007US7157430 (Substituted)acyl dipeptidyl inhibitors of the ICE/CED-3 family of cysteine proteases
01/02/2007CA2211839C Use of melatonin for treating patients suffering from drug addiction
01/02/2007CA2177602C N-substituted azabicycloalkane derivatives, their preparation and use
01/02/2007CA2135709C Melatonin derivatives for use in treating sleep disorders
12/2006
12/28/2006WO2006137369A1 Reactive monomer and resin composition containing same
12/28/2006WO2006137082A1 Process for industrially viable preparation of perindopril erbumine
12/28/2006WO2006136606A2 Oxindole derivatives
12/28/2006WO2006124902A3 Synthesis of salinosporamide a and analogues thereof
12/28/2006WO2006082409A8 Tricyclic cytoprotective compounds
12/28/2006WO2006055463A3 2-amino-3-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors
12/28/2006WO2006020664A3 Ammonolysis process for the preparation of intermediates for dpp iv inhibitors
12/28/2006WO2005104711A3 Purification of progesterone receptor modulators
12/28/2006US20060293353 Matrix metalloproteinase inhibitors
12/28/2006US20060293313 Indole-3-alkyl-N-piperazine ring substituted with quinoline ring or derivatives; shows high affinity for both the dopamine D2 receptor and the serotonin reuptake site, useful for treating central nervous system disorders, such as anxiety disorders, depression, Parkinson's disease, and schizophrenia
12/28/2006US20060293306 1-Cyclopentyl-3-methyl-2-(2-pyridyl)indole-5-thio/carbonyl derivatives; hepatitis C virus infection; synergistic with another inhibitor of HCV polymerase or immunomodulatory agent such as interferons
12/28/2006DE102005030314A1 New triarylamine-derivates useful as hole transportation substance or luminescent substance in an organic electroluminescent device; and as hole transportation substance in an electrophotographic arrangement
12/28/2006CA2612451A1 Oxindole derivatives
12/27/2006EP1736468A2 Isatin derivatives with neurotrophic activity useful in the treatment of diseases mediated by the nerve growth factor (NGF) activation
12/27/2006EP1736465A1 Aniline derivatives
12/27/2006EP1735319A1 Inhibitors of histone deacetylase
12/27/2006EP1735300A1 Thio-substituted tricyclic and bicyclic aromatic methanesulfinyl derivatives
12/27/2006EP1735270A1 Diamino alcohols and their use as renin inhibitors
12/27/2006EP1734951A2 Diphenyl-indol-2-on compounds and their use in the treatment of cancer
12/27/2006EP1734942A1 Substituted urea and carbamate, phenacyl-2-hydroxy-3-diaminoalkane, and benzamide-2-hydroxy-3-diaminoalkane aspartyl-protease inhibitors
12/27/2006EP1611098B1 Compounds having activity at 5ht2c receptor and uses thereof
12/27/2006EP1436267B1 Lactam derivatives as antagonists for human 11cby receptors
12/27/2006EP1187806B1 Spermine:peptide-based surfactant compounds
12/27/2006EP1149118B1 Method of producing derivatized polymers