Patents
Patents for C07D 209 - Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom (45,780)
05/2007
05/16/2007CN1962635A Indoles compound preparation method
05/16/2007CN1315834C 6,7-dihydro-5H-pyrazolo[1,2-a]pyrazol-1-ones which control inflammatory cytokines
05/16/2007CN1315831C Direct preparation of pyrrolo [3,4-c] pyrroles compounds
05/16/2007CN1315823C New method for synthesizing Ramosetron Hydrochloride
05/16/2007CN1315821C Improvement of preparation of N-methyl-3- (1-methyl-4-piperidine)-1,4-indole-5-ethyl thiamine
05/16/2007CN1315806C Substituted 2-amino-cycloalkanecarboxamides and their use as cysteine protease inhibitors
05/16/2007CN1315805C Compositions and methods of use thereof achiral analogues of CC-1065 and duocarmycins
05/15/2007US7217840 Method for preparing 1,3,5-triaminobenzene and hydrolyzing it into high-purity phloroglucinal
05/15/2007US7217732 Cannabinoid receptor agonists
05/15/2007US7217731 Hydroisoindoline tachykinin receptor antagonists
05/15/2007US7217729 4,6-Dimethyl-3-{[3'-(N,N-dimethylaminomethyl)-4-hydroxy-4'-(3''-methoxyphenyl)-cyclohexylamino]-methyl}-1H-indole 2-carboxylic acid ethyl ester or other derivatives of substituted indoles; for treatment or prevention of neurodegenerative diseases, psychological disorders, AIDS, inflammation or allergies
05/15/2007US7217724 2-[(2-hydroxy-2-pyridinylethyl)amino]ethyl-substituted indoles, e.g., N,N-Diethyl-2-{3-[(2R)-2-((2R)-2-hydroxy-2-pyridin-3-ylethylamino)-propyl]-1H-indol-7-yloxy}acetamide; beta 3-adrenoceptor stimulants, used for treating obesity, hyperglycemia, frequent urination, and urinary incontinence
05/15/2007US7217722 Nitrogen-containing compounds having kinase inhibitory activity and drugs containing the same
05/15/2007US7217707 Amide of R-2-(aminoaryl)-propionic acid for use in the prevention of leucocyte activation
05/15/2007US7217706 Benzocycloheptenylamino derivatives; treatment of pollakiuria or urinary incontinence
05/10/2007WO2007053145A1 Haloperidol analogs
05/10/2007WO2007051619A1 N- (hetero) aryl indole derivatives as pesticides
05/10/2007WO2007030574A3 1 , 4 and 1 , 5-disubstituted indole derivatives for use as ppar active compounds
05/10/2007WO2007025709A3 Organic compounds
05/10/2007WO2007022321A3 Substituted indoles and use thereof
05/10/2007WO2007017894A3 PREPARATION OF NOVEL CRYSTALLINE η(ETA) FORM OF PERINDOPRIL ERBUMINE
05/10/2007WO2007017893A3 Preparation of novel crystalline form of perindopril erbumine monohydrate
05/10/2007WO2007007282A3 Azabicyclo derivatives as muscarinic receptor antagonists
05/10/2007WO2006127205A3 Methods of preparing 3-cyano-quinolines and intermediates made thereby
05/10/2007WO2006118607A3 Hcv inhibitors with carbazole structure
05/10/2007US20070105941 Substituted cyclohexylcarboxylic acid amide compounds
05/10/2007US20070105939 Mesylate salt of 5-(2-dimethylaminoethoxy)-1H-indole-2-carboxylic acid [3-(4-hydroxycarbamoylphenyl)prop-2-ynyl]amide
05/10/2007US20070105914 Substituted sulfonamides
05/10/2007US20070105899 Benzene compounds
05/10/2007US20070105889 Administering (S)-1-(2,3,7,8-tetrahydrofuro[2,3-g]indol-1-yl)-2-propylamine; serotonin receptor antagonists (5HT/5HT2C) for therapy of disorders of the central nervous system; damage to the central nervous system; cardiovascular disorders; gastrointestinal disorders; diabetes insipidus, and sleep apnea
05/10/2007US20070105838 Bicyclic Benzamide Compoundssa as Histamine H3 Receptor Ligand Useful in the Treatment of Neurological Diseases
05/10/2007CA2626300A1 N-(hetero) aryl indole derivatives as pesticides
05/09/2007EP1783114A1 N-(hetero)aryl indole derivatives as pesticides
05/09/2007EP1783110A1 Novel cyclohexane derivative, prodrug thereof and salt thereof, and therapeutic agent containing the same for diabetes
05/09/2007EP1781652A1 Pyrrolopyrimidine and pyrrolopyridine derivatives substituted with tetrahydropyridine as crf antagonists
05/09/2007EP1781630A1 Novel piperidine derivative for the treatment of depression
05/09/2007EP1781611A1 Crystalline forms of carvedilol and processes for their preparation
05/09/2007EP1781610A2 Isoindoline compounds and methods of their use
05/09/2007EP1781609A1 Small molecule inhibition of a pdz-domain interaction
05/09/2007EP1781608A1 Indole derivatives comprising an acetylene group as ppar activators
05/09/2007EP1682530B1 Pyrrole substituted indoles as inhibitors of pai-1
05/09/2007EP1501796B1 3-(pyridinyl-amino)-1h-indole-2-carboxylic acid derivatives as interleukin-4 gene expression inhibitors
05/09/2007EP1408970B1 Indolines and tetrahydro-quinolines as prodrugs for tumour treatment
05/09/2007EP1268441B1 An intermediate and process for its synthesis
05/09/2007CN1960973A 1-(1h-indol-1-yl)-3-(4-methylpiperazin-1-yl)-1-phenyl propan-2-ol derivatives and related compounds as modulators of the norepinephrine(NE) and the serotonine(5-HT) activity and the monoamine reuptake
05/09/2007CN1960727A Naphthalene derivatives useful as histamine-3-receptor ligands
05/09/2007CN1958583A Method for preparing double (N-methyl phthalimide) oxide
05/09/2007CN1958570A Method for preparing ropinirole
05/09/2007CN1958568A A kind of compound for preventing or curing infection of helicobacter pylori, preparation method, and application
05/09/2007CN1314669C 2,7-substituted indoles and their use as 5-HT6 modulators
05/09/2007CN1314656C 9,9-bis(triphenyl amino) fluorine derivatives and preparation and use thereof
05/08/2007US7214715 Substituted hydroxyl amine derivatives; inhibitors of beta-secretase, inhibit beta-secretase-mediated cleavage, inhibitors of A beta production, and/or are effective to reduce amyloid beta deposits or plaques
05/08/2007US7214704 For therapy of diabetes and related conditions
05/08/2007US7214702 Reacting the amide compound with phosphorus oxychloride in an organic solvent; treating the reaction mixture with water to form (1S,3S,5S)-2-[(2S)-2-amino-2-(3-hydroxytricyclo[3.3.1.13,7]dec-1-yl)-1-oxoethyl]-2-azabicyclo[3.1.0]hexane-3-carbonitrile-hydrochloride
05/08/2007US7214700 Administering to a human patient an 2-oxindole-3-ylidenyl) acetic acid derivatives which modulate the activity of protein kinases and effective to treat disorders related to abnormal protein kinase activity, such as cancer
05/08/2007US7214699 Indazole derivatives as CRF antagonists
05/08/2007US7214685 Antibody directed enzyme prodrug therapy
05/08/2007US7214248 Multi-component kit and method for temporarily dyeing and later decolorizing hair
05/08/2007CA2331870C Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
05/08/2007CA2276098C Tricyclic benzo[e]isoindoles and benzo[h]isoquinolines
05/08/2007CA2275479C Prevention of loss and restoration of bone mass by certain prostaglandin agonists
05/03/2007WO2007051081A1 Methods and compounds for preparing cc-1065 analogs
05/03/2007WO2007050963A1 Novel ido inhibitors and methods of use thereof
05/03/2007WO2007049736A1 Concentration crystallizer and method
05/03/2007WO2007049224A1 Novel hexahydro- or octahydro-cyclopenta[c]pyrrole derivatives
05/03/2007WO2007048841A2 Novel indole-containing beta agonists, method for producing them and their use as drugs
05/03/2007WO2007048788A1 Sulfonamide derivatives and use thereof for the modulation of metalloproteinases
05/03/2007WO2007048595A1 Compounds comprising a lactam or a lactam derivative moiety, processes for making them, and their uses
05/03/2007WO2007030939A3 Methods of modulating neurotrophin-mediated activity
05/03/2007WO2007022269A3 Compounds and compositions as tpo mimetics
05/03/2007WO2007009120A3 Heterotetracyclic compounds as tpo mimetics
05/03/2007WO2007005454A3 Improved process for preparing insecticidal (disubstitutedpropenyl) phenylalkyl substituted heterocycles
05/03/2007US20070099981 Condensed indoline derivatives and their use as 5HT, in particular 5HT2C, receptor ligands
05/03/2007US20070099980 Condensed indoline derivatives and their use as 5HT, in particular 5HT2C, receptor ligands
05/03/2007US20070099976 3-(5-tert-Butyl-2-Hydroxy-phenyl)-3-phenyl-1,3-dihydro-indol-2-one, used for treating cellular proliferative disorders, nonproliferative degenerative disorders and viral diseases or infections
05/03/2007US20070099960 Liver X receptors (LXR) modulators such as 1-[[4-(1,1-dimethylethyl)phenyl]sulfonyl]-4-methoxy-N-(2-phenyl ethyl)-2,3-dihydro-1H-)indole-2-carboxamide, used for the treatment of atherosclerosis, dyslipidemia, obesity, diabetes, hypercholesterolemia, neurodegenerative diseases and inflammatory diseases
05/03/2007US20070099916 nuclear hormone receptor inhibitors; to treat increased lipid levels, increased cholesterol levels, low HDL-cholesterol, high LDL-cholesterol, atherosclerotic diseases, diabetes, macular degeneration, Alzheimer's disease; 2-(1-benzyl-3-chloro-2-methyl-1H-indol-5-yl)-1,1,1,3,3,3-hexafluoro-propan-2-ol
05/03/2007US20070099909 N-(2-arylethyl)benzylamines as antagonists of the 5-ht6 receptor
05/03/2007US20070099826 Treatment of diseases associated with the egr-1 enhancer element
05/03/2007US20070099210 Methods of Labelling Polynucleotides with Dibenzorhodamine Dyes
05/03/2007US20070098777 Pharmaceutical or Food Composition for Treatment or Prevention of Brain Edema
05/03/2007DE102005052127A1 Neue indol-haltige Beta-Agonisten, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel New indol-containing beta-agonists, to processes for their preparation and their use as medicaments
05/03/2007DE102005051325A1 Alkoxyalkyl spirocyclische Tetram- und Tetronsäuren Alkoxyalkyl spirocyclic tetramic and tetronic acids
05/03/2007CA2627486A1 Novel indole-containing beta agonists, method for producing them and their use as drugs
05/03/2007CA2627234A1 Compounds comprising a lactam or a lactam derivative moiety, processes for making them, and their uses
05/03/2007CA2627046A1 Methods and compounds for preparing cc-1065 analogs
05/03/2007CA2623879A1 Sulfonamide derivatives and use thereof for the modulation of metalloproteinases
05/02/2007EP1780200A1 A crystalline form of fluvastatin sodium and a process for preparing it
05/02/2007EP1780196A2 Pyridine derivatives for use as vanilloid receptor ligands
05/02/2007EP1780191A1 Fluorene derivative and organic electroluminescent device using same
05/02/2007EP1778658A2 Modulators of alpha7 nicotinic acetylcholine receptors and therapeutic uses thereof
05/02/2007EP1778636A1 Oxime ester photoinitiators
05/02/2007EP1778635A2 Isoindoline compounds and methods of making and using the same
05/02/2007EP1778634A1 Isoindolone compounds and their use as metabotropic glutamate receptor potentiators
05/02/2007EP1778633A1 Indoles useful in the treatment of inflammation
05/02/2007EP1778632A1 Indoles useful in the treatment of inflammation
05/02/2007EP1778629A1 Process for the synthesis c-2, c-3 substituted n-alkylated indoles useful as cpla2 inhibitors
05/02/2007EP1549637B1 1- (indol-3-yl)carbonyl piperazine derivatives
05/02/2007EP1492766B1 Improved cc-1065 analog synthesis
05/02/2007EP1268478B1 Phenyl-substituted imidazopyridines