Patents
Sitemap › C07 - Organic chemistry › C07D - Heterocyclic compounds › C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
Patents for C07D 207 - Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom (40,304)
08/2010
08/19/2010WO2010047774A3 Inhibitors of mycobacterium tuberculosis malate synthase, methods of marking and uses thereof
08/19/2010US20100210838 Fluoropyrrolidines having dipeptidyl peptidase enzyme inhibitory activity
08/19/2010US20100210837 Pactamycin biosynthetic gene cluster
08/19/2010US20100210706 Pyrrolidinone anilines as progesterone receptor modulators
08/19/2010US20100210705 Pyrrole and Isoindole Carboxamide Derivatives as P2X7 Modulators
08/19/2010US20100210693 Benzylether and benzylamino beta-secretase inhibitors for the treatment of alzheimer's disease
08/19/2010US20100210633 Carboxamide compounds and their use
08/19/2010US20100210630 Diamine Derivatives as Inhibitors of Leukotriene A4 Hydrolase
08/19/2010US20100210603 Novel sulfonamide inhibitors of aspartyl protease
08/19/2010US20100210524 Novel estrogen receptor ligands
08/19/2010US20100210495 Photo-labile pro-fragrance conjugates
08/18/2010EP2218710A1 Procedure for the preparation of 2,6-diethyl-4-methylphenylacetic acid
08/18/2010EP2218330A1 Process for the preparation of 2-ethyl-4,6-dimethylphenyl acetic acid by reacting 2-ethyl-4,6-dimethylbromobenzene with tert.-butylacetate
08/18/2010EP2217568A1 Compounds for inhibiting ksp kinesin activity
08/18/2010EP2217565A1 Compounds which modulate the cb2 receptor
08/18/2010EP1351963B1 A process for the synthesis of atorvastatin form v and phenylboronates as intermediate compounds
08/18/2010EP1320526B1 Pharmaceutically active benzsulfonamide derivatives as inhibitors of protein junkinases
08/18/2010CN1795193B N-acyl nitrogen heterocyles as ligands of peroxisome proliferator-activated receptors
08/18/2010CN101808987A New disubstituted phenylpyrrolidines as modulators of cortical catecholaminergic neurotransmission
08/18/2010CN101805280A Preparation method of N,N'-m-phenylenebismaleimide
08/18/2010CN101805279A Preparation method of atorvastatin calcium
08/18/2010CN101307018B Diethylene triaminepentaacetic acid carboxyl active ester or analogues, method for synthesizing same and use
08/18/2010CN101215252B Method for preparing N-Boc or N-Cbz derivatives of chiral alpha,alpha'-disubstituted pyrrolidines containing olefinic bond and acetylene bond
08/18/2010CN101186592B Dipyrrolidine-2,5-diketone-n-alkane compound containing diene group and its synthesizing method and use
08/18/2010CN101024671B 丙型肝炎病毒抑制剂 Hepatitis C virus inhibitors
08/17/2010US7777009 for modulation of chemokines; antiinflammatory agents; cancer
08/17/2010US7776919 modulators of the interaction between the receptor for advanced glycated end products; 3-(4-Benzyloxyphenyl)propionic Acid 2,4- Di-(3-Diethylamino-1-propoxy)aniline Amide; acute and chronic inflammation; diabetic late complications; Alzheimer's disease, erectile dysfunction; metastasis
08/17/2010US7776910 Piperazinyl-substituted quinolinone compounds ;to treat nervous system diseases, neurodegenerative diseases; gastrointestinal tract disorders; cognition enhancers; 3-[4-(3-Ethylsulfanyl-benzenesulfonyl)-2-methoxy-phenyl]-pyrrolidine and 5-(3-Ethylsulfanyl-benzenesulfonyl)-2-pyrrolidin-3-yl-phenol
08/17/2010US7776909 such as (5-acetyl-1-methyl-1H-pyrrol-2-yl)acetyl methanesulphonamide, used for the of treatment of psoriasis, ulcerative colitis, melanoma, chronic obstructive pulmonary disease (COPD), skin disorders, rheumatoid arthritis, idiopathic fibrosis, glomerulonephritis and reperfusion injuries after ischemia
08/17/2010US7776903 Pharmaceutical preparations containing substituted 2,5-diaminomethyl-1H-pyrroles
08/17/2010US7776874 Cycloalkylcarbonyl-3H-spiro[2-benzofuran-1,3'-pyrrolidin]-3-ones: N-methyl-5-[4-(1-{[3-oxo-1'H,3H-spiro[2-benzofuran-1,3'-pyrrolidin]-1'-yl]carbonyl}cyclopropyl)phenyl]pyridine-2-carboxamide; 11- beta hydroxyl steroid dehydrogenase type 1 inhibitors; mineralcorticoid receptor antagonists; diabetes
08/17/2010CA2370412C Pharmaceutical compounds
08/12/2010WO2010091164A1 Inhibitors of glucosylceramide synthase
08/12/2010WO2010090344A1 Hydrazide compound and use of the same in pest control
08/12/2010WO2009082437A9 Selective androgen receptor modulators (sarms) and uses thereof
08/12/2010US20100204465 Refined routes to chlorin building blocks
08/12/2010US20100204228 Aryl Sulfonamides Useful for Modulation of the Progesterone Receptor
08/12/2010US20100204213 Arylsulfonamide derivatives for use as ccr3 antagonists in the treatment of inflammatory and immunological disorders
08/12/2010US20100204199 Cyclic 11-beta hydroxysteroid dehydrogenase type i inhibitors
08/12/2010US20100203162 Method of preparing (+)-1,4-dihydro-7-[(3S,4S)-3-methoxy-4-(methylamino)-1-pyrrolidinyl]-4-oxo-1-(2-thiazolyl)-1,8-naphthyridine-3-carboxylic acid
08/12/2010CA2750324A1 Hydrazide compound and use of the same in pest control
08/11/2010EP2215908A1 2-Alkyl-cycloalk(en)yl-carboxamides and their use as fungizides
08/11/2010EP2215084A2 Therapeutic substituted lactams
08/11/2010EP2215058A1 Substituted n-phenyl-bipyrrolidine ureas and therapeutic use thereof
08/11/2010EP2215056A2 Sulfur containing fluoroalkyl amines and isocyanates
08/11/2010EP2215055A1 New non-peptide derivatives as bradykinin b1 antagonists
08/11/2010EP1491530B1 Method of heightening optical purity of 1-benzyl-3-aminopyrrolidine and salt for use therein
08/11/2010CN201543258U Distillation apparatus of naphthol AS-BI recovered solvent
08/11/2010CN101801925A antiviral compounds
08/11/2010CN101801924A Crystalline forms of (r)-1-{2-[4'- (3-methoxy-propane-1- sulfonyl)-biphenyl-4-yl]-ethyl}-2-methyl-pyrrolidine, and compositions, and methods related thereto
08/11/2010CN101801923A Pleuromutilin derivatives and their use as antimicrobials
08/11/2010CN101798279A Method for preparing iron-catalyzed pyrrole and pyrrole cyclic compounds
08/11/2010CN101182305B Method for synthesizing 2,5-disubstituted tetrahydrofuran derivatives
08/10/2010US7772432 amidation of a heteroary substituted oxoaminobenzoic acid with an amine; for treatment of psoriasis and rheumatoid arthritis using e.g. N-(3-dimethylaminophenyl)-3-(3-methoxybenzamido)-4-methylbenzamide
08/10/2010US7772425 Vitamin D receptor modulators
08/10/2010US7772407 (1S)-1,5-anhydro-1-[3-(1-benzothien-2-ylmethyl)phenyl-D-glucitol and derivatives are Na+-glucose cotransporter inhibitors and are used to treat diabetes and related diseases such as insulin-resistance and obesity
08/10/2010US7772406 Process for production of benzyloxypyrrolidine derivative, and process for production of hydrochloride salt powder of optically active benzyloxypyrrolidine derivative
08/10/2010US7772405 3-alkyl-5- (4-alkyl-5-oxo-tetrahydrofutran-2-yl) pyrrolidin-2-one derivatives as intermediates in the synthesis of renin inhibitors
08/10/2010US7772264 Such as (S)-1-{[2-(5-Methyl-2-phenyl-oxazol-4-yl)-ethylamino]-acetyl}-pyrrolidine-2-carbonitrile mesylate; dipeptidyl peptidase IV inhibitors (DPPIV); for treatment of diabetes, non-insulin dependent diabetes mellitus, impaired glucose tolerance, bowl disease, colitis ulcerosa, morbus crohn, obesity
08/10/2010US7772237 Thio-substituted tricyclic and bicyclic aromatic methanesulfinyl derivatives
08/10/2010US7772190 E.g., isobutyl N-methyl-N-trimethylallophanoyl-L-alanyl-D-lactate; using parasiticides and nematocides in medicine and veterinary medicine; productive and breeding animals; foods and feeds
08/10/2010US7772159 Solution and solid phase synthesis of pyrrolinones and polypyrrolinones
08/10/2010US7771611 sufficiently soluble in common organic solvents to be used in nucleophilic displacement reactions to add the -OSF5 group; quaternary ammonium cation or metal cation complexed with crown compound or polyamine; reaction of thionyl tetrafluoride SOF4 with fluoride salt of the cation
08/10/2010CA2570482C Simple stereocontrolled synthesis of salinosporamide a
08/10/2010CA2366800C Carboxylic acid derivatives that inhibit the binding of integrins to their receptors
08/10/2010CA2237099C Sulfonylaminocarboxylic acids
08/05/2010WO2010088450A2 Methods for treating diseases associated with the modulation of serca
08/05/2010WO2010087430A1 N-acyl anthranilic acid derivative or salt thereof
08/05/2010WO2010087419A2 Ester compound and use thereof
08/05/2010WO2010086366A1 4-aryl-butane-1,3-diamides
08/05/2010WO2010086177A1 Sulfamoyl- phenyl-ureido benzamidine-derivatives as antimalarial agents
08/05/2010WO2010085968A1 Toluidine sulfonamides and their use as hif-inhibitors
08/05/2010WO2010033196A3 Simplified one-pot synthesis of [18f]sfb for radiolabeling
08/05/2010WO2010031708A3 Ortho-aminoanilides for the treatment of cancer
08/05/2010US20100197976 Catalysts
08/05/2010US20100197941 Process for the production of atorvastatin calcium in amorphous form
08/05/2010US20100197940 Method for Preparing FMOC-Based Hydrolysable Linkers
08/05/2010US20100197939 Process for the enantioselective preparation of pregabalin
08/05/2010US20100197911 Nitrogen-Containing Aromatic Derivatives
08/05/2010US20100197760 Disubstituted phenylpyrrolidines as modulators of cortical catecholaminergic neurotransmission
08/05/2010US20100197736 Cetp activity inhibitors
08/05/2010US20100197734 Pleuromutilin derivatives and their use as antimicrobials
08/05/2010US20100197680 Lactam-substituted dicarboxylic acids and use thereof
08/05/2010US20100197640 Novel sulfamoyl-phenyl-ureido compounds and their use as medicament
08/05/2010US20100196988 Bioreactive Agents
08/05/2010CA2750967A1 Sulfamoyl-phenyl-ureido benzamidine-derivatives as antimalarial agents
08/05/2010CA2750452A1 N-acyl anthranilic acid derivative or salt thereof
08/04/2010EP2212284A2 Calcium receptor modulating agents
08/04/2010EP2212283A1 Substituted n-phenyl-bipyrrolidine carboxamides and therapeutic use thereof
08/04/2010EP2212282A1 Substituted n-phenyl-bipyrrolidine carboxamides and therapeutic use thereof
08/04/2010EP2212281A1 Arylsulfonamides with analgesic activity
08/04/2010CN101795733A tyrosinase inhibitors
08/04/2010CN101792391A Polymerizable biphenyl compound
08/04/2010CN101125829B Vinylbiphenyl compounds
08/03/2010US7767831 purified polylactic acid or glycolic acid-lactic acid copolymer; insert for drugs
08/03/2010US7767830 Synthesis of antiarrhythmic vernakalant hydrochloride in stereoisomerically substantially pure form starting with microbial oxidation of a monohalobenzene to the cyclohexanediol and amination with a 3-pyrrolidinol; arrhythmia; O-benzyl protected intermediate
08/03/2010US7767695 Substituted piperidines
08/03/2010US7767679 Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
08/03/2010US7767667 Pesticidal heterocycles
08/03/2010US7767073 electrooxidation reaction using 2-(N-pyrrolidine)-N,N,N-triethylethanammonium tetrafluoroborate or 3-N-piperidine-N,N,N-triethylammoniopropanesulphonamide tetrafluoroborate; proline final product
1 ... 57 58 59 60 61 62 63 64 65 66 67 68 69 70 71 72 73 74 75 76 77 ... 404