Patents
Patents for C07B 55 - Racemisation; Complete or partial inversion (688)
07/2003
07/09/2003CN1429197A Shortened synthesis of 3,3-diarylpropylamine derivatives
07/01/2003US6586436 Serotonergic agents
07/01/2003US6586434 Method for the preparation of tetrahydrobenzothiepines
06/2003
06/11/2003EP1317426A1 Beta-thio-amino acids
06/10/2003US6576795 Racemization of optically active amines
06/04/2003EP0804417B1 Racemisation process for use in the manufacture of levobupivacaine and related piperidinecarboxanilide anaesthetic agents
05/2003
05/21/2003EP0842139B1 The preparation of chiral endo-5-norbornen-2-ol
05/08/2003US20030088105 Process for the preparation of substituted thiazolines and their intermediates
05/06/2003CA2126180C Isomerisation process
04/2003
04/23/2003EP0784603B1 Racemisation of precursors to levobupivacaine and analogues thereof
04/16/2003EP1302467A2 Process for the preparation of substituted thiazoline derivatives and their intermediate
04/15/2003US6548704 Reacting an optically active amine in the presence of hydrogen and a hydrogenation or dehydrogenation catalyst containing copper and zinc oxide catalyst on a support
04/15/2003US6548693 Nitriloxy derivatives of (R) and (S)-carnitine
04/15/2003US6548665 Asymmetric synthesis of a key intermediate for making benazepril and analogues thereof
04/11/2003WO2002032899A1 Novel anticholinergic agents that can be used as medicaments and method for the production thereof
04/02/2003CN1104416C Racemisation and asymmetric transformation process used in manufacture of levobupivacaine and analogues thereof
03/2003
03/20/2003WO2002091993A3 Estrogen receptor modulators
03/20/2003US20030055245 Kinetic resolution of a intermediate useful in the production of benazepril and analogues thereof
03/12/2003WO2002022568A1 ss-THIO-AMINO ACIDS
03/12/2003EP1289929A1 Shortened synthesis of 3,3-diarylpropylamine derivatives
03/12/2003EP1091954B1 Process for producing (8-chloro-3,10-dibromo-6,11-dihydro-5h-benzo 5,6]cyclohepta[1,2-b]pyridin-11-yl)-1-piperidine
03/05/2003EP1286984A2 Method for the preparation of tetrahydrobenzothiepines
02/2003
02/26/2003CN1399687A Method for producing optically active amines
02/19/2003EP1283898A1 Process for the preparation of enantiomerically enriched esters and alcohols
02/19/2003CN1397542A Process to enable recemation of optical rotatary vinyl substituted cyclopropane carboxylic compound
02/13/2003US20030032839 Chemical intermediate for synthetic pyrethroids
02/13/2003CA2456166A1 Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids
01/2003
01/30/2003WO2003008361A1 Process for the racemization of alcohols
01/30/2003US20030022901 Serotonergic agents
01/16/2003WO2003003972A2 Kinetic resolution of a intermediate useful in the production of benazepril and analogues thereof
01/09/2003WO2001068637A3 Method for the preparation of tetrahydrobenzothiepines
01/08/2003EP1025080B1 Process for the recycle of a waste product of diltiazem synthesis
01/03/2003WO2003000636A1 Resolution process for (r)-(-)-2-hydroxy-2-(2-chlorophenyl) acetic acid
12/2002
12/19/2002WO2002059128A3 Process for preparing clopidogrel
12/05/2002US20020183515 Asymmetric synthesis of a key intermediate for making benazepril and analogues thereof
11/2002
11/21/2002WO2002091993A2 Estrogen receptor modulators
11/21/2002CA2445922A1 Estrogen receptor modulators
10/2002
10/24/2002WO2002083694A1 Synthesis of silyl camptothecins and silyl homocamptothecins
10/22/2002US6469007 P-substituted-n-(2-(4-(2,3-dihydro-benzo(1,4)dioxin-5-yl) -piperazin-1-yl)-propyl)-n-pyridin-2-yl-benzamide,
09/2002
09/17/2002US6451854 α-amino acid phenyl ester derivatives
08/2002
08/29/2002WO2002066414A1 Method for isolating and purifying (1rs,2rs)-2-[(dimethylamino)methyl]-1-(3-methoxyphenyl)-cyclohexanol
08/29/2002WO2002022849A3 Enzymatic resolution of aryl- and thio-substituted acids
08/29/2002US20020120166 Reacting an optically active amine in the presence of hydrogen and a hydrogenation or dehydrogenation catalyst containing copper and zinc oxide catalyst on a support
08/29/2002US20020119965 Nitriloxy derivatives of (R) and (S)-carnitine
08/29/2002DE10108308A1 Verfahren zur Isolierung und Reinigung von (1RS,2RS)-2[(Dimethylamino)methyl]-1-(3-methoxyphenyl)-cyclohexanol A process for isolating and purifying (1RS, 2RS) -2 [(dimethylamino) methyl] -1- (3-methoxyphenyl) cyclohexanol
08/21/2002EP1232279A2 Method for producing optically active amines
08/20/2002US6437175 Process for racemization of n-acylamino acids by means of transition metal catalysts
08/14/2002CN1363549A Racemization of rotatory amine
08/08/2002WO2002044142A3 Piperazine derivatives, their preparation and their use for treating central nervous system (cns) disorders
08/08/2002US20020107254 P-substituted-N-(2-(4-(2,3-dihydro-benzo(1,4)dioxin-5-yl) -piperazin-1-yl)-propyl)-N-pyridin-2-yl-benzamide,
08/01/2002WO2002059128A2 Process for preparing clopidogrel
07/2002
07/24/2002EP1224161A1 Nitroxy derivatives of (r) and (s)-carnitine
06/2002
06/20/2002DE10062729A1 Verfahren zur Racemisierung von optisch aktiven Aminen A process for the racemization of optically active amines
06/19/2002EP1215197A2 Method for the racemisation of optically active amines
06/06/2002WO2002044142A2 Piperazine derivatives, their preparation and their use for treating central nervous system (cns) disorders
06/05/2002CN1352629A Method for the recemization of optically active amines
05/2002
05/29/2002DE10028443C1 Production of optically active 3,3-diaryl-propylamine derivatives comprises six step process from 4-hydroxybenzoic acid or alkyl 4-hydroxybenzoate and cinnamic acid
05/28/2002US6395923 Antiischemic agents; cardiovascular disorders
05/23/2002US20020061565 Monitoring preferential compounds in racemic; obtain enantiomer, incubate with racemic mix, hydrolyze mix, recover preferential compound
05/22/2002EP1207165A2 Isomerisation of 6beta-fluorosteroids into the corresponding 6alpha-fluoro derivatives
05/21/2002US6392044 Using base
05/15/2002CA2348206A1 Isomerisation of 6beta-fluorosteroids into the corresponding 6alpha-fluoro derivatives
04/2002
04/18/2002DE10050994A1 New diphenylalkanoic acid azabicyclooctane ester quaternary salts useful as anticholinergic agents, especially in treatment of asthma and chronic obstructive pulmonary disease
04/16/2002US6372906 Reacting camptothecin or homocamptothecin with silyl radical precursor under conditions to generate silyl radical
04/09/2002US6369218 Isomerisation of 6β-fluorosteroids into the corresponding 6α-fluoro derivatives
03/2002
03/21/2002WO2002022849A2 Enzymatic resolution of aryl- and thio-substituted acids
03/21/2002CA2422466A1 Enzymatic resolution of aryl- and thio-substituted acids
03/20/2002EP0782569B1 Racemisation process used in the manufacture of levobupivacaine and analogues thereof
03/14/2002US20020032329 Method for the preparation of tetrahydrobenzothiepines
02/2002
02/28/2002WO2001038292A3 Method for producing optically active amines
02/27/2002CN1337934A Method for the racemization of optically active amines
02/14/2002WO2002012181A1 Novel diamines having a casr modulating activity
01/2002
01/09/2002CN1330618A Racemization of optically active amines
01/02/2002EP1167347A1 Process for racemising an enantiomer-enriched schiff base of an amino acid amide
12/2001
12/27/2001US20010056209 Using aqueous solution of a base
12/20/2001WO2001096279A1 Shortened synthesis of 3,3-diarylpropylamine derivatives
12/05/2001EP1159252A1 Method for the racemization of optically active amines
11/2001
11/29/2001WO2001090396A1 Process for the preparation of enantiomerically enriched esters and alcohols
11/29/2001CA2410529A1 Process for the preparation of enantiomerically enriched esters and alcohols
11/07/2001EP1150941A1 Method for the racemization of optically active amines
10/2001
10/18/2001US20010031890 Process for the racemization of nu-acylamino acids by means of transition metal catalysts
10/10/2001EP1140815A1 Novel thio-aminotetralin compounds useful in pain management
09/2001
09/26/2001EP1136466A2 Process for racemising N-acyl-amino acids with transition metal catalysts
09/20/2001WO2001068637A2 Method for the preparation of tetrahydrobenzothiepines
09/20/2001DE10013599A1 Verfahren zur Racemisierung von N-Acylaminosäuren mittels Übergangsmetallkatalysatoren A process for the racemisation of N-acylamino acids by means of transition metal catalysts
09/12/2001EP1131270A1 Process for converting an alcohol to the corresponding fluoride
09/11/2001US6288280 Heating compound for racemization atropisomeric bis(phosphine oxide) compounds
09/05/2001EP1129055A1 Method for racemization of optically active amines
09/05/2001CN1311770A Derivatives of alpha-amino acid phenyl ester
08/2001
08/02/2001US20010011074 Antiischemic agents; cardiovascular disorders
07/2001
07/04/2001EP1112990A1 Methods for producing and separating erythro- and threo-2-hydroxy-3-nitrobutanoic acid compounds
06/2001
06/28/2001US20010005762 Methods for producing and separating erythro- and threo-2-hydroxy-3-nitrobutanoic acid compounds
06/19/2001US6248889 Process for converting an alcohol to the corresponding fluoride
06/13/2001CN1298862A Prepn. of (+)-trans-chrysanthemic acid
05/2001
05/31/2001WO2001038292A2 Method for producing optically active amines
05/31/2001DE19956786A1 New optically active aminoalcohol and diamine derivatives useful as intermediates, e.g. for pharmaceuticals and plant protectants
05/16/2001EP1098871A1 $g(a)-AMINO ACID PHENYL ESTER DERIVATIVES
04/2001
04/18/2001EP1091954A1 Process for producing (8- chloro-3,10- dibromo-6,11- dihydro- 5h-benzo 5,6]cyclohepta 1,2-b]pyridin-11-yl)- 1-piperidine
03/2001
03/28/2001EP0741727B1 Process for isomerization of spirocyclic compounds with beta-aminocarboxyl and/or beta-aminocarbonyl systems
02/2001
02/15/2001WO2001010819A1 Nitroxy derivatives of (r) and (s)-carnitine
1 2 3 4 5 6 7