Patents
Patents for C07B 51 - Introduction of protecting groups or activating groups, not provided for in groups (403)
07/1995
07/25/1995US5436331 Protection of hydroxy function with 1-N-aryl-4-alkoxy-piperidin-4-yl
06/1995
06/08/1995WO1995015308A1 Crystalline, polymorphic form of (s,s,s)-n-(1-[2-carboxy-3-(n2-mesyllysylamino)propyl]-1-cyclopentylcarbonyl)tyrosine
04/1995
04/11/1995US5405783 Removing photoremovable protective group from region of substrate, contacting with protected amino acid, repeating to form peptide
10/1994
10/27/1994WO1994024088A1 Deallylation reagent and deallylation method using said reagent
10/27/1994CA2160163A1 Deallylation reactive and deallylation process using said reactive
10/12/1994EP0619321A1 Very large scale immobilized peptide synthesis
08/1994
08/31/1994EP0476014B1 Very large scale immobilized polymer synthesis
02/1994
02/23/1994EP0583338A1 Method for synthesizing peptides, novel amino acid derivatives used therein, and methods for preparing same.
12/1993
12/14/1993CA1325216C 6-sulfonyl chromans
10/1993
10/20/1993EP0565607A1 Protection group, compoud protected by this group and device for grafting the protection group onto the compound being protected
10/16/1993CA2093989A1 Reagent and catalytic process for clearing a protected function
04/1993
04/27/1993US5206363 Process for the resolution of enantiomers of 5-heteroaryl-1,3,4-thiadiazinones
04/14/1993EP0537089A1 Reagent composition for deprotection, and its use
04/12/1993CA2080276A1 Reagent useful for breakingdown and method of use of said reagent
03/1993
03/30/1993US5198571 Monofunctionalization of phenolic hydroxy onto a polyphenol
03/10/1993EP0530657A1 Process for the separation of enantiomers of 5-hetaryl-1,3,4-thiadiazinone
03/03/1993CA2077031A1 Process for the resolution of enantiomers of 5-heteroaryl-1,3,4-thiadiazinones
12/1992
12/08/1992CA1311332C Bop reagent for solid phase peptide synthesis
11/1992
11/12/1992WO1992019643A1 Method for synthesizing peptides, novel amino acid derivatives used therein, and methods for preparing same
09/1992
09/01/1992US5143854 Large scale photolithographic solid phase synthesis of polypeptides and receptor binding screening thereof
07/1992
07/23/1992WO1992012167A1 Protection group, compoud protected by this group and device for grafting the protection group onto the compound being protected
07/23/1992CA2099120A1 Protection group, compound protected by this group and device for grafting the protection group onto the compound being protected
06/1992
06/25/1992WO1992010587A1 Sequencing of surface immobilized polymers utilizing microfluorescence detection
06/24/1992EP0491600A1 Process for the regiospecific monofunctionalisation of a phenolic hydroxy group of a polyphenol
03/1992
03/25/1992EP0476014A1 Very large scale immobilized polymer synthesis.
03/18/1992EP0475443A2 Chemical synthesis of oligonucleotides
01/1992
01/08/1992EP0464439A2 Process for the preparation of secondary or tertiary alcohols
01/07/1992US5079373 Blocking agents useful in the synthesis of polypeptides
12/1991
12/18/1991CN1015104B Deprotection of allylic esters and ethers
10/1991
10/02/1991EP0217804B1 Analogs of substances p
09/1991
09/24/1991CA1289568C Process for production of amino compounds
09/04/1991EP0444888A1 Process for the desilylation of a 4-silyloxy-tetrahydro-pyran-2-one
08/1991
08/28/1991EP0298982B1 Protecting groups for organic synthesis
02/1991
02/05/1991US4990644 Sulfonium compound and acylating agent
12/1990
12/13/1990WO1990015070A1 Very large scale immobilized peptide synthesis
12/13/1990CA2391491A1 Very large scale immobilized peptide synthesis
12/11/1990CA1277673C Substituted ethylene-silane adducts used as protective group reagents
11/1990
11/22/1990EP0398132A2 Phosphorous compounds
10/1990
10/02/1990US4960881 α-chlorinated carbonates, their method of manufacture and application in the protection of the amine functions of amino acids
09/1990
09/04/1990CA1273630A1 Deprotection of allylic esters and ethers
08/1990
08/22/1990EP0383686A1 2-Amino-7-hydroxytetraline carboxyalkyl ethers
08/21/1990US4950418 Reagent for removing protective groups in peptide synthesis
08/14/1990CA2009992A1 2-amino-7-hydroxytetralin carboxyalkyl ethers
08/07/1990US4946971 Blocking agent
05/1990
05/29/1990CA1269667A1 .alpha.-SUBSTITUTED 3,3,3-TRIFLUORO-2,2-DICHLORO-1- PROPANOLS AND THE PREPARATION THEREOF
03/1990
03/13/1990US4908469 2-Hydroxy-propanoic acid acyclic alkyl esters for benzothiazepines
01/1990
01/30/1990CA1265130A1 Process of selectively blocking amino groups
01/02/1990US4891430 Process for synthesizing active esters of carboxylic acids, new alpha-halogenated carbonates which are useful for this synthesis and the method of producing them
12/1989
12/19/1989US4888385 BOP reagent for solid phase peptide synthesis
11/1989
11/23/1989EP0342902A2 2-Hydroxy-propanoic acid acyclic alkyl esters for benzothiazepines
09/1989
09/13/1989EP0331988A1 Sulfonium compounds, as well as process for producing active esters and amides used for the production of amides
07/1989
07/05/1989EP0322973A2 Method of preparing optically active cyanohydrin derivatives and their conversion products, and optically active compounds to be obtained in this manner
05/1989
05/23/1989US4832697 Hair dye preparations containing substantive nitrodiphenylamine derivatives
01/1989
01/31/1989US4801719 Silanes, process for their preparation, and their use
01/18/1989EP0298982A1 Protecting groups for organic synthesis.
11/1988
11/30/1988EP0293073A1 Chroman-6-sulphonyl derivatives
11/29/1988US4788282 Carbapenicillins
11/08/1988CA1244452A1 .alpha.-CHLORINATED CARBONATES, THEIR METHOD OF MANUFACTURE AND APPLICATION IN THE PROTECTION OF THE AMINE FUNCTIONS OF AMINO ACIDS
11/02/1988EP0289353A2 Modified BOP reagent for solid phase peptide synthesis
11/01/1988US4782164 Reaction of acid with active carbonate
09/1988
09/21/1988EP0282749A1 Hair dyeing compositions containing direct nitrodiphenylamine derivatives
04/1988
04/20/1988EP0264063A2 Reagent for removing protective groups in peptide synthesis
01/1988
01/07/1988EP0250955A1 Process for the preparation of 2-aminoethane sulphon amide
10/1987
10/22/1987WO1987005906A3 Protecting groups for organic synthesis
10/08/1987WO1987005906A2 Protecting groups for organic synthesis
09/1987
09/22/1987US4695643 Silanes, process for their preparation, and their use
04/1987
04/15/1987EP0217804A1 Analogs of substances p.
03/1987
03/24/1987US4652665 Block amine function of amino acids; peptide synthesis
02/1987
02/04/1987CN86103521A Deprotection of allylic esters and ethers
01/1987
01/24/1987CN85101227A Process for the preparation of alpha-chlorinated carbonates and application
01/20/1987US4637902 Base precursors
01/07/1987EP0207415A1 Coupling reagent, method for its preparation and its use
10/1986
10/08/1986EP0196454A1 Process for removing an amino protecting group
07/1986
07/31/1986WO1986003495A3 Derivatives of substances p and of fragments thereof
06/1986
06/25/1986EP0185578A1 Process for the preparation of active carboxylic-acid esters, alpha-halogenated carbonates useful for this preparation and their preparation
06/19/1986WO1986003495A2 Derivatives of substances p and of fragments thereof
04/1986
04/09/1986EP0177454A2 Silanes, process for their preparation and their use
01/1986
01/14/1986US4564471 N-/benzyloxycarbonyl/aspartylphenylalanine
10/1985
10/09/1985EP0157739A1 Substituted 1-propanoles, process for their production, chloroformic-acid esters ad their use
09/1985
09/11/1985EP0154581A1 Alpha-chlorinated carbonates, process for their preparation and their application to the protection of aminic functions in amino acids
08/1985
08/27/1985US4537713 Process for the reduction of reducible groups and its use
03/1985
03/19/1985CA1184195A1 Process for preparing tert-butyl ether or ether containing polyfunctional organic compounds
12/1984
12/05/1984EP0127114A1 Process for the cleavage of phthalimides
11/1984
11/27/1984US4485253 Dissolving in sulfuric acid and ether, and reaxting with excess isobutene
10/1984
10/03/1984EP0120402A1 Base precursor
08/1983
08/23/1983CA1152496A1 Method for reductive elimination of protecting groups
04/1983
04/05/1983CA1144155A1 Process for removing an allylic group from allylic esters, carbonates and carbamates
12/1982
12/15/1982EP0066856A1 Process for the preparation of polyfunctional organic compounds with at least one tert. butyl ether group or one tert. butyl ester group
12/08/1982EP0066103A1 Process for the reduction of reducible groups, and its application
11/1982
11/17/1982EP0013663B1 Process for removing an allylic group from allylic esters, carbonates and carbamates
02/1982
02/09/1982US4314942 Deprotection of allylic esters, carbonates and carbamates catalyzed by palladium compounds
10/1981
10/07/1981EP0037373A1 Process for the elimination of alkyl and alkenyl groups
04/1981
04/22/1981EP0027319A2 Method for reductive elimination of protecting groups and preparative process using such method
02/1981
02/17/1981US4251657 Deacylation of a halogenoacetylamino compound using an n-substituted dithiocarbamic acid
07/1980
07/23/1980EP0013663A1 Process for removing an allylic group from allylic esters, carbonates and carbamates
04/1980
04/29/1980CA1076606A1 Synthesis of vicinal glycols
04/22/1980CA1076108A1 Process for the separation and/or purification of oligo- and polyhydroxy compounds
03/1980
03/25/1980CA1074300A1 Method for removal of thiol-protecting groups
10/1979
10/23/1979US4172195 Blocking
06/1979
06/27/1979EP0002586A1 Method for removing a halogenoacetyl protective group from a halogenoacetyl amino compound
1 2 3 4 5