Patents
Patents for A61K 31 - Medicinal preparations containing organic active ingredients (785,912)
02/2003
02/05/2003CN1100537C Agonists and antagonist for nicotinic acetylcholine receptors of insects to control endoparasites
02/05/2003CN1100536C Composition for rectal administration
02/05/2003CN1100535C Pharmaceutical agents for treatment of emesis
02/05/2003CN1100533C Melatonin derivatives for usein terating desynchronization disorders
02/05/2003CN1100532C Desquamation copositions contaiig salicylic acid and zwitterionic compounds
02/05/2003CN1100531C Use of agonists of antagonist of P2 purinoceptors for prevention of glutamate evoked cytotoxicity
02/04/2003WO2002014333A1 Phosphonocephem compound
02/04/2003WO2002011734A1 Aqueous pharmaceutical compositions
02/04/2003US6515198 Transgenic animals; calibration
02/04/2003US6515173 Inhibitors of the ICE/ced-3 family of cysteine proteases
02/04/2003US6515136 To the novel intermediates prepared by these methods. The biphenyl isoxazole sulfonamides prepared by the present methods are endothelin antagonists useful, inter alia, for the treatment of hypertension.
02/04/2003US6515135 Aminoaryl oxazolidinone N-oxides
02/04/2003US6515133 Certain diaryl imidazoles act as partial agonists or antagonists for NPY receptors, in particular NPY 5 receptors. They are of use, for example in treating loss of appetite. Such compounds bear aryl groups in the 2 position.
02/04/2003US6515130 The invention relates to a process of preparing (S-(R*,S*))-beta -(((1-(1-oxo-3-(4-piperidinyl)propyl)-3-piperidinyl) carbonyl)amino)-3-pyridinepropanoic acid derivatives represented by the antagonists of the platelet fibrinogen
02/04/2003US6515129 A pharmaceutical composition which comprises, a cyclic imide derivative represented by the general formula (I): present invention relates to an aminopeptidase N inhibitor or an angiogenesis inhibitor, modulates production of tumor necrosis
02/04/2003US6515124 Dehydroamino acids
02/04/2003US6515117 C-aryl glucoside SGLT2 inhibitors and method
02/04/2003US6515116 Method of preparing form II crystals of clarithromycin
02/04/2003US6515028 Glucamine compounds for treating hepatitis virus infections
02/04/2003US6515027 Substituted benzanilides as CCR5 receptors ligands, antiinflammatory agents and antiviral agents
02/04/2003US6515025 Use of ethynyl alanine amino diol compounds to inhibit enzymatic conversion of angiotensinogen to angiotensin I
02/04/2003US6515022 Use of inhaled retinoids in the treatment of lung diseases
02/04/2003US6515021 The compounds according to the invention have pronounced activity in the fields of cell differentiation and cell proliferation
02/04/2003US6515020 Combination of carnitines and resveratrol for prevention or treatment of cerebral and ageing disorders
02/04/2003US6515019 Methods of providing symptomatic and prophylactic treatment for medical and neurological conditions
02/04/2003US6515018 Synergistic compositions for lycopene and Vitamin E for the prevention of LDL oxidation
02/04/2003US6515017 Polyamino acid conjugated paclitaxel or docetaxel have increased water solubility, efficacy and accumulation within a tumor
02/04/2003US6515016 Treating or preventing multiple sclerosis, by administering an antimicrotubule agent; treating various other inflammatory diseases
02/04/2003US6515015 Antidiabetic agents based on aryl and heteroarylacetic acids
02/04/2003US6515012 Reacting 3-benzoylthio-2-methylpropionoic acid chloride with 4-phenylthio-L-proline; hypotnsive agents
02/04/2003US6515011 Anticoagulants
02/04/2003US6515010 Carvedilol methanesulfonate
02/04/2003US6515009 Therapeutic inhibitor of vascular smooth muscle cells
02/04/2003US6515008 Formulation of H2- receptor antagonist cimetidine in liquid formulations
02/04/2003US6515007 Methods for managing scalp conditions
02/04/2003US6515006 Ophthalmic formulation which modulates dilation
02/04/2003US6515005 Substituted azole derivatives as inhibitors of corticotropin releasing factor
02/04/2003US6515004 Useful in the treatment of Alzheimer's disease, chemotherapy-induced alopecia, and cardiovascular disease
02/04/2003US6515003 Useful in the treatment of diseases related to lipid and carbohydrate metabolism
02/04/2003US6515002 Compounds and compositions for treating C1s-mediated diseases and conditions
02/04/2003US6515001 IL-8 receptor ligands-drugs for inflammatory and autoimmune diseases
02/04/2003US6514999 A substance which increases Dopamine concentration in the synaptic cleft of the neurons of the brain, in combination with an effective amount of a local anesthetic of the anilide group or derivatives thereof
02/04/2003US6514997 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
02/04/2003US6514996 Phosphodiesterase (PDE) IV inhibitors; used to treat inflammatory allergic diseases, autoimmune diseases, diseases of the central nervous system, insulin-resistant diabetes; wounds; AIDS, and the like.
02/04/2003US6514994 Levobupivacaine and its use
02/04/2003US6514993 Serotonin 5-HT1A and dopamin D2 receptor ligands
02/04/2003US6514992 Caspases and apoptosis
02/04/2003US6514989 Aromatic and heteroaromatic substituted 1,2,4-triazolo pyridine derivatives
02/04/2003US6514986 Chiral fluoroquinolone arginine salt forms
02/04/2003US6514985 Induce the biosynthesis of cytokines such as interferon and tumor necrosis factor; exhibit antiviral and antitumor properties
02/04/2003US6514984 Human non-pancreatic secretory phospholipase A2 inhibitors
02/04/2003US6514983 Inhibitors of the nucleic enzyme poly(adenosine 5'-diphospho-ribose)polymerase
02/04/2003US6514982 CRF receptor antagonists and methods relating thereto
02/04/2003US6514980 Nucleoside analogs in combination therapy of herpes simplex infections
02/04/2003US6514979 For treating a viral infection, such as an HIV-1 infection
02/04/2003US6514977 For treating p38 kinase mediated disorders
02/04/2003US6514976 Arylpiperazines having activity at the serotonin 1A receptor
02/04/2003US6514975 Anti-inflammatory piperazinyl-benzyl-tetrazole derivatives and intermediates thereof
02/04/2003US6514974 Pyrido-, pyrimido-, pyridazo- and pyrazo- pyridazines having angiogenesis inhibiting activity
02/04/2003US6514973 Treatment of transmethylation disorders comprising one or more compounds selected from phosphatidyl serines, methyl transporters, and methyl and methylene donors with exipient
02/04/2003US6514971 Cinnoline derivatives and use as medicine
02/04/2003US6514970 Urotensin-II receptor antagonists
02/04/2003US6514968 Treating a disease or condition in a mammal wherein the 5-HT receptor is implicated and modulation of 5-HT function is desired comprising
02/04/2003US6514965 Substituted 1-benzazepines and derivatives thereof
02/04/2003US6514964 Treating diseases, conditions or disorders mediated by integrin receptors, such as vitronectin and fibronectin receptors
02/04/2003US6514963 Methods for the inhibition of egg production in trematodes
02/04/2003US6514962 Beta -lactam antibiotic having an esterified carboxy group directly coupled to the nucleus is mixed with a salt of phosphoric acid and oil, a dramatic improvement occurs in its stability
02/04/2003US6514961 Such as anxiety and all forms of epilepsy, particularly in humans
02/04/2003US6514960 Use of bismuth subgallate in inhibition of production of nitric oxide synthase
02/04/2003US6514959 Microbicides
02/04/2003US6514958 Dosage unit comprising tibolone and a water insoluble starch product is contained in a humid atmosphere of 50 to 70% relative humidity until administration
02/04/2003US6514957 Method of alleviating the violence and stimulating the appetite of stag in the puberty age of the fall and method of promoting the growth of stag's horn
02/04/2003US6514956 For treating diseases associated with progestogen dependence and for fertility control, abortion or contraception and for anticancer use
02/04/2003US6514953 Calcium (3S) tetrahydro-3-furanyl(1S,2R)-3-[[(4-aminophenyl)sulfonyl](isobutyl)amino]-1-benzyl-2-(phosphonooxy)propylcarbamate
02/04/2003US6514952 For the treatment and prophylaxis of diseases which are caused by an undesired extent of leucocyte adhesion and/or leucocyte migration such as rheumatoid arthritis or allergic disorders
02/04/2003US6514951 LL-F28249 alpha-lambda or a 23-oxo or 23-imino derivative of
02/04/2003US6514949 Administering A2A adenosine agonist in combination with an effective amount of a Type IV phosphodiesterase inhibitor for treatment of inflammation caused by an ischemia/reperfusion injury
02/04/2003US6514945 Azalide antibiotic compositions
02/04/2003US6514934 For treating sexual dysfunctions in males and females
02/04/2003US6514756 Human myoblast cell lines and their uses
02/04/2003US6514754 Of herpesvirus of turkeys (HVT) inserted in a non-essential region of the vector; may be manipulated to provide vaccines
02/04/2003US6514745 Oncoprotein protein kinase
02/04/2003US6514726 Aspergillus fumigatus acetyl coenzyme-A carboxylase genes and polypeptides and uses thereof
02/04/2003US6514712 Probe for the early detection of displasias in multilayer tesselated epithelium and for the diagnosis and therapy of carcinomas
02/04/2003US6514686 Alzheimer's disease
02/04/2003US6514544 Beverage for increasing the body's capacity to break down alcohol and method thereof
02/04/2003US6514537 Citric acid, magnesium hydroxide, water
02/04/2003US6514536 Drug preparations for treating sexual dysfunction
02/04/2003US6514534 Methods for forming regional tissue adherent barriers and drug delivery systems
02/04/2003US6514531 Controlled-release dosage forms comprising zolpidem or a salt thereof
02/04/2003US6514529 A compressed tablet of antibacterial oxazolidinone selected from the group consisting of linezolid, eperezolid and (S)-N-((3-(3-fluoro-4-(tetrahydro-2H-thiopyran-4-yl)phenyl-2-o xo-5-oxazolidinylmethyl)acetamide S,S-dioxide
02/04/2003US6514527 Compositions comprising a mixture of bioflavonols
02/04/2003US6514526 Coated starch capsules and a process for producing them
02/04/2003US6514525 Sustained release; mixture of non-steroid antiinflammatory drug, prostaglandin and excipient
02/04/2003US6514524 Improved absorption of hydrophilic ingredients because of particular excipients; calcium 3-acetylamino-1-propane sulfonate (calcium acamprosate); polysorbates, fatty ethers or esters of PEG, polyglycolysed glycerides
02/04/2003US6514520 Containing about 0.05 to about 5 mg/mL of an aminopolycarboxylic acid, including salts such as disodium EDTA; especially the antihistamines loratadine, descarboethoxyloratadine, and azatadine
02/04/2003US6514519 1-octadecyl-2-methyl-sn-glycero-3-phosphocholine; oral administration
02/04/2003US6514516 Local anesthetic and a biocompatible controlled release material consisting of polyanhydrides, copolymers of lactic acid and glycolic acid, poly(lactic) acid, poly(glycolic) acid, polyesters, polyorthoesters, proteins, polysaccharides
02/04/2003US6514507 Administering 10-Hydroxy-2-decenoic acid and derivatives for stimulating epidermal renewal and/or combating intrinsic aging of the skin
02/04/2003US6514499 Compositions exhibiting ADP-ribosyltransferase activity and methods for the preparation and use thereof