Patents
Patents for A61K 31 - Medicinal preparations containing organic active ingredients (785,912)
02/2003
02/11/2003US6518435 Production method, a method of producing a compound represented by the formula (III) production method of oxyimino- alkanoic acid derivatives having an anti-diabetic activity.
02/11/2003US6518432 The invention relates to a novel process for the preparation of certain pharmaceutically active pyridyl compounds. NMDA receptor antagonist activity. The compound known as (S)-1-phenyl-2-(2- pyridyl)ethanamine is of particular
02/11/2003US6518429 Anticancer agents, treating restenosis, atherosclerosis and hepatitis virus
02/11/2003US6518428 The present invention relates to the area of platinum drugs. In particular, it relates to an improved process for preparing platinum complexes having the general formula (Ia) or (Ib): as defined of herein,
02/11/2003US6518427 Compounds are exceedingly water soluble which is useful in preparing pharmaceutical formulations of these compounds. They are also rapidly converted back to the parent amines in vivo, making them useful as prodrugs of the parent amines.
02/11/2003US6518425 A process for producing a 1,3-oxathiolane nucleoside comprising reacting a 5-halo-2-protected-oxymethyl-1,3-oxathiolane with a silylated purine or pyrimidine without the addition of a Lewis acid or an additional base to the reaction
02/11/2003US6518422 Hydrogenation of 5,5-dioxo-2,3-dihydro-1H-pyrrolo-(2,1-c)(1,2,4)benzothiadiazine with a complex of ruthenium dichloride with 2,2'-bis(diphenylphosphine)-1,1'-binaphthyl and 1,2-diphenylethylenediamine as catalyst
02/11/2003US6518421 Process for the preparation of epothilone analogs
02/11/2003US6518413 Isolated nucleic acid encoding the polypeptide which, on expression in a host cell, produces the polypeptide; use in treatment of muscular dystrophy
02/11/2003US6518410 Immunosuppressive agent, anticancer agent and DNA polymerase alpha inhibitor.
02/11/2003US6518319 Method of preparing and using compositions extracted from vegetable matter for the treatment of female symptoms
02/11/2003US6518318 Stimulating transport of glucose into animal tissue by the administration of pinitol
02/11/2003US6518317 Antiviral agents
02/11/2003US6518316 Cytokine production and tyrosine kinase inhibitors
02/11/2003US6518314 Pharmaceutical agents that impede the initiation and progression of primary and secondary DMS disruptions
02/11/2003US6518312 Activator protein (AP); treating diseases associated with immune suppressive states; benzmides such as N-((2-Diethylamino)propyl)-4-isobutyrylamino-2-methoxy-benzamide
02/11/2003US6518311 Use of branched-chain fatty acids and derivatives thereof for the treatment of pain
02/11/2003US6518310 Non-peptidic; inhibits trypsin-like protease, thrombin and embolus formation; anticoagulant
02/11/2003US6518308 Administering to the patient who will undergo surgical procedure a halogenated organic compound to prevent or retard the development of surgical adhesions
02/11/2003US6518307 Orally administering an effective amount of a peracid to an animal.
02/11/2003US6518306 PDE4 inhibitors particularly in regards to treating allergic and inflammatory diseases
02/11/2003US6518305 Five-membered carbocyclic and heterocyclic inhibitors of neuraminidases
02/11/2003US6518304 Fungicidal composition
02/11/2003US6518303 Selectively inhibit COX-2 in preference to COX-1 and are useful in the treatment of COX-2 mediated diseases, such as inflammation, pain, fever and asthma with fewer side effects
02/11/2003US6518301 Better selectivity than estrogen for the estrogen receptor-beta over receptor-alpha; treatment of Alzheimer's disease, anxiety, depression, osteoporosis, cardiovascular disease, rheumatoid arthritis, or prostate cancer
02/11/2003US6518300 Antiplipemic agent, anticholesterol agents
02/11/2003US6518298 Methods and compositions for inhibition of angiogenesis with EM-138
02/11/2003US6518297 Selective 5-HT6 receptor ligands
02/11/2003US6518295 Utilization of aryl(or heteroaryl)azolylcarbinol derivatives in the preparation of a medicament for the treatment of troubles mediated by an excess of substance P
02/11/2003US6518294 Fused pyrazolyl compounds
02/11/2003US6518293 Anti-HIV imidazolone derivatives
02/11/2003US6518292 Heterocyclic aromatic compounds usefuls as growth hormone secretagogues
02/11/2003US6518291 Inosine-5'-monophosphate dehydrogenase inhibitors
02/11/2003US6518290 Substituted oxazoles and thiazoles derivatives as HPPAr alpha activators
02/11/2003US6518289 1-substituted-1-aminomethyl-cycloalkane derivatives (=gabapentin analogues), their preparation and their use in the treatment of neurological disorders
02/11/2003US6518288 Amlodipine fumarate
02/11/2003US6518287 Substituted imidazoles as dual histamine H1 and H3 agonists or antagonists
02/11/2003US6518286 Compounds
02/11/2003US6518285 Piperidinyloxy and pyrrolidinyloxy oxazolidinone antibacterials
02/11/2003US6518283 Squaric acid derivatives
02/11/2003US6518282 4-Arylpiperidine derivatives for the treatment of pruritus
02/11/2003US6518279 Cyclopentanone dihydropyridine compounds useful as potassium channel openers
02/11/2003US6518278 Administering a synergistically effective amount of irinotecane and subsequently with a synergistically effective amount of cis-oxalato (1R,2R-diaminocyclohexane) Pt (II)
02/11/2003US6518277 Disrupting leukocyte function
02/11/2003US6518274 Use of cyclopentabenzofuran-derivatives for combating (NF-κB)-dependent diseases
02/11/2003US6518270 Heterocyclic compounds for inhibition of gastric acid secretion, processes for their preparation and pharmaceutical compositions thereof
02/11/2003US6518269 Cancer treatment
02/11/2003US6518268 Telomerase inhibitors and methods of their use
02/11/2003US6518267 Protease inhibitors
02/11/2003US6518265 1H-imidazopyridine derivatives
02/11/2003US6518264 For treatment/prevention of psychoses, other brain disorders, and cardiovascular disorders
02/11/2003US6518263 Imidazo[4,5-b]pyridiniummethyl-containing cephem compounds having broad antibacterial spectrum
02/11/2003US6518262 22R-hydroxycholesta-8, 14-diene derivatives for the inhibition of meiosis
02/11/2003US6518261 Prostate cancer
02/11/2003US6518260 (α-aminophosphino) peptide derivatives, method for making same and therapeutic applications thereof
02/11/2003US6518259 Compositions for treating autoimmune disease
02/11/2003US6518258 6-sulphamoyl -3-quinolyphosphonic acid compounds
02/11/2003US6518253 Treatment of viral infections using the L-isomer of ribavirin
02/11/2003US6518252 Method of treating aquatic animals with an antimicrobial agent and chelating agent
02/11/2003US6518251 Macrolides
02/11/2003US6518250 Agent for preventing and curing hindrance of ischemic reperfusion
02/11/2003US6518249 Oligosaccharide derivatives and process for producing the same
02/11/2003US6518248 Method of treating gastric or colon cancer by administration of a sulfoquinovosylacylglycerol ester
02/11/2003US6518247 Method for producing an antitumoral agent and antitumoral agent thus obtained
02/11/2003US6518246 Pharmaceutical composition and method for the treatment of neoplastic cells
02/11/2003US6518245 Treatment of arrhythmias via inhibition of a multifunctional calcium/calmodulin-dependent protein kinase
02/11/2003US6518244 Cardiovascular disorders
02/11/2003US6518239 Dry powder compositions having improved dispersivity
02/11/2003US6518066 Acylated Homoserine Lactone (AHL) compounds and AHL receptors derived from bacterial quorum sensing systems; inducible or repressible promotors regulate gene expression in plants and plant cells
02/11/2003US6518063 Osf2/Cbfa1 nucleic acids and methods of use therefor
02/11/2003US6518062 Enzyme combinations for destroying proliferative cells
02/11/2003US6518043 Proteins suppressing proliferation of lympho-hematopoietic cells
02/11/2003US6518031 Hapten-carrier conjugates for treating and preventing nicotine addiction
02/11/2003US6517883 Satiety product
02/11/2003US6517871 Amorphous ammonium salt; blocking angiotensin II receptors; treating hypertension, congestive heart failure and renal failure
02/11/2003US6517870 Improved taste by reducing bitterness and saltiness
02/11/2003US6517867 Dry mix formulation for bisphosphonic acids
02/11/2003US6517866 Sertraline salts and sustained-release dosage forms of sertraline
02/11/2003US6517864 Transdermally administered tolterodine as anti-muscarinic agent for the treatment of overactive bladder
02/11/2003US6517859 Injectable, drug delivery vehicles; controlled release of bioactive agents to sites within the central nervous system; dopamine, cholecystokinin, and epidermal and basic fibroblast growth factors for Parkinson's disease
02/11/2003US6517858 Bioactive prostheses with immunosuppressive, antistenotic and antithrombotic properties
02/11/2003US6517855 Method of sterilizing
02/11/2003US6517854 Antimicrobial sanitizing lotion with skin protection properties
02/11/2003US6517849 Tissue products containing antiviral agents which are mild to the skin
02/11/2003US6517848 Method for sequestration of skin irritants with absorbent article composition
02/11/2003US6517847 Topical gel delivery system
02/11/2003US6517846 N-long chain acyl-asparagine or glutamine; effects suitable for sensitive skin, dry skin, roughening skin or skin with atopic dermatitis
02/11/2003US6517841 Solid compositions and liquid preparations for oral administration which contain cocoa polyphenols
02/11/2003US6517836 Aziridin-1-yl nitrobenzamides as prodrugs in conjunction with nitroreductase enzymes
02/11/2003US6517827 Anionic polymers as toxin binders and antibacterial agent
02/11/2003US6517826 Anionic polymers as toxin binders and antibacterial agents
02/11/2003US6517825 Polyether-based bile acid sequestrants
02/11/2003US6517822 Formulations and methods for straightening hair
02/11/2003US6517812 D1-like agonists or antagonists; SCH 23390
02/11/2003US6517811 Compounds for cancer imaging and therapy
02/11/2003US6517810 Palliation of bone pain due to cancer by the administration of a tin stannic (Sn+4) chelate complex
02/11/2003US6517809 Using a breath test; vehicle containing a sugar is powder or granules, coating vehicle with an isotope-labeled urea and encapsulating the coated vehicle in gelatin
02/11/2003US6517742 2-(butyl 4'-ylaminobenzoate)-4,6-bis((1,3,3,3-tetramethyl-1 -((trimethylsilyl)oxy)disiloxanyl)propyl-3-ylamino)-s-triazine; s-triazine derivatives substituted by at least one silicone group; from cyanuric chloride
02/11/2003CA2320129C Suspension aerosol formulations
02/11/2003CA2222361C Hydroxypropylated quaternary ammonium derivatives having an ester function, and cosmetic or dermatological compositions containing them