Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
05/1992
05/26/1992US5116941 Peptide substrates for determination of enzyme activity
05/26/1992US5116861 Treatment of Hypertension and Angina Pectoris
05/26/1992US5116835 Enzyme-inhibiting urea derivatives of dipeptides, a process for the preparation thereof, agents containing these, and the use thereof
05/26/1992US5116730 Amino acid substituted 4-aminophenazones for measuring enzyme activity
05/26/1992CA1302005C Aminoacid derivatives as antihypertensives
05/22/1992WO1992009556A1 Improved matrix metalloprotease inhibitors
05/22/1992CA2096221A1 Matrix metalloprotease inhibitors
05/20/1992EP0486478A2 Renin-inhibiting peptides
05/20/1992EP0486280A2 Piperidinylcamphorsulfonyl oxytocin antagonists
05/20/1992EP0485458A1 Thioacylating reagents and intermediates, thiopeptides, and methods for preparing and using same.
05/20/1992CA2055685A1 Hiv protease inhibitors having polyether substituents
05/19/1992US5115099 Substrates for determination of enzyme activity and intermediates for synthesis of the substrates as well as process for producing the intermediates
05/19/1992US5115098 End-blocked peptides inhibiting binding capacity of gp120
05/19/1992US5114962 New amino acid esters, a process for their preparation, medicaments containing them, and the use thereof
05/19/1992US5114953 Peptides
05/19/1992US5114927 Hypotensive agents and inhibiting renin
05/19/1992US5114926 Tetrapeptide inhibiting the entry into cycle of hemopoietic stem cells processes for its preparation, and its uses
05/19/1992US5114925 Renin inhibitors containing the 2-[[(2R,3S)-3-amino-4-cyclohexyl-2-hydroxy-1-butyl]thio)alkanoyl moiety and the corresponding sulfoxide and sulfone derivatives
05/19/1992US5114921 Amphiphilic peptides and use thereof
05/19/1992CA1301181C2 Oxiranes
05/16/1992WO1992008709A1 Meta-substituted phenyl alanine derivatives
05/16/1992CA2073776A1 Meta-substituted phenyl alanine derivatives
05/14/1992WO1992007956A1 Process for amplifying nucleic acid
05/14/1992WO1992007874A1 Pharmaceutically active proteins comprising an active protein and an integrinaffinity sequence
05/14/1992WO1992007869A1 Inhibitors and substrates of thrombin
05/14/1992WO1992007576A1 Protective four amino acid epitope against plasmodium vivax malaria
05/14/1992CA2055024A1 N-phenyl piperidinylcamphorsulfonyl oxytocin antagonists
05/13/1992EP0484769A2 Improved process for crystallizing L-alpha-aspartyl-L-phenylalanine methyl ester from the solution
05/13/1992EP0484719A2 Tachykinin antagonist
05/12/1992US5112953 Radiolabeled proteins for diagnostic or therapeutic use
05/12/1992US5112947 Oligopeptides, nootropic agents
05/12/1992US5112944 Antitumor agents
05/12/1992US5112811 Sdk peptides and therapeutic compositions containing them
05/12/1992CA1300807C Heterocyclic derivatives
05/07/1992DE4034707A1 New hydroxyethyl-amine and norstatin-type pseudo:peptide(s)
05/06/1992EP0483271A1 Peptides containing diamino-glycols as transition-state mimics.
05/06/1992CN1060848A Peptide compounds, processes for preparation thereof and pharmaceutical composition comprising same
05/05/1992USH1056 Luteinizing hormone-releasing hormone
05/05/1992US5110936 Condensation of pyroglutamic acid with ethyl ester of 4-thiazolidinecarboxylic acid
05/05/1992US5110799 Inhibition of viral ribonucleotide reductase
05/05/1992US5110798 Purine derivatives having pharmacological action
05/05/1992US5110797 Neurotropic agents
05/05/1992US5110795 Methods and compositions for the treatment of inflammatory bowel diseases and conditions
05/05/1992CA1300313C2 Amino acid derivatives
05/03/1992CA2054667A1 Cyclopeptides
04/1992
04/30/1992WO1992007265A1 Selective peptide labeling with hydrogen isotopes
04/30/1992WO1992006996A1 Peptides containing substituted 1,4-diamines as transition-state inserts
04/30/1992WO1992000284A3 Method for forming an amino acid thiohydantoin using an n-substituted ketenimine activator
04/30/1992WO1991018866A3 1,4-diamino-2,3-dihydroxybutanes
04/29/1992EP0482539A2 Peptide compounds, processes for preparation thereof and pharmaceutical composition comprising the same
04/28/1992US5109000 Thiol carboxylic acid derivatives and their use as collagenase inhibitor
04/28/1992US5108990 Glutamic acid derivatives
04/28/1992US5108890 Chromogenic compounds, processes for the preparation thereof and use thereof as enzyme substrates
04/28/1992CA1299813C METHOD OF SEPARATING .alpha.-L-ASPARTYL-L-PHENYLALANINE METHYL ESTER THROUGH CRYSTALLIZATION
04/25/1992CA2054097A1 Peptide compounds, processes for preparation thereof and pharmaceutical composition comprising the same
04/23/1992CA2053772A1 Benzolactam analogs as antagonists of cck
04/22/1992EP0481522A1 Novel mercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace
04/22/1992EP0481311A2 Aminoacid derivatives
04/22/1992EP0480969A1 Amino acid analog cck antagonists
04/22/1992EP0317573B1 Antipyretic and anti-inflammatory peptides
04/22/1992CN1060472A Tripeptide antithrombotic agents
04/22/1992CN1016341B Novel spergualin-related compounds and process for producing the same
04/21/1992US5106948 Anticarcinogenic agents
04/21/1992US5106835 Renin inhibitors
04/19/1992CA2053573A1 Amino acid derivatives
04/16/1992WO1992006108A1 Peptide compounds of laevorotatory amino acids and ring molecules, and therapeutical applications thereof
04/16/1992WO1992006090A1 Epoxysuccinamic acid derivative
04/15/1992EP0480071A1 S-(lower fatty acid)-substituted glutathione derivative
04/15/1992EP0480061A1 Hepatic disorder inhibitor
04/15/1992EP0480060A1 S-(lower fatty acid)-substituted glutathione derivative
04/15/1992EP0480044A1 Novel 4h-3,1-benzoxazin-4-one derivative
04/15/1992EP0479912A1 Inhibition of the n-end rule pathway in living cells.
04/15/1992EP0479910A1 N-SUBSTITUTED CYCLOALKYL AND POLYCYCLOALKYL ALPHA-SUBSTITUTED Trp-Phe- AND PHENETHYLAMINE DERIVATIVES
04/15/1992CN1060294A Improved oligosaccharide conjugate vaccines
04/15/1992CN1060293A Fibrinogen receptor antagonists
04/14/1992US5104852 Administering selenodiglutathione, selenodicysteine or selenodimethionone to the center of a tumor from where it diffuses outwardly
04/14/1992CA1298842C Amino acid analogs as cck-antagonists
04/13/1992WO1992007270A1 Diagnostic method
04/13/1992CA2069417A1 Diagnostic method
04/08/1992EP0479489A2 Tripeptide antithrombotic agents
04/08/1992EP0479481A2 Fibrinogen receptor antagonists
04/08/1992EP0478729A1 Process for manufacturing aspartame from a diketopiperazine and novel intermediates and derivatives therefor.
04/08/1992CN1060096A Fibrinogen receptor anlagonists
04/07/1992US5102990 Direct radiolabeling of antibodies and other proteins with technetium or rhenium
04/07/1992CA1298682C PREPARATION PROCESS OF .alpha.-L-ASPARTYL-L-PHENYL-ALANINE METHYL ESTER OR HYDROHALIDE THEREOF
04/02/1992WO1992005190A1 Deoxyhypusyl hydroxylase inhibitors
04/02/1992WO1992005179A1 Carboxylic acid esters of rapamycin
04/02/1992WO1992005160A1 4-arylsulfonyl-3,4-dihydro-2(1h)-quinoxalinone-1-alkanoic acids, esters, and salts
04/01/1992EP0477912A2 Novel N-acyldipeptides, processes for the preparation thereof and pharmaceutical compositions containing the same
04/01/1992EP0477508A1 Improved oligosaccharide conjugate vaccines
03/1992
03/31/1992US5101039 Azabicycloamino carboxylic acid intermediates
03/31/1992US5100875 Novel peptides having plateler aggregation inhibitory activity
03/31/1992US5100874 Collagenase Inhibitors
03/31/1992CA1298435C Pentapeptides with cell growth regulatory effects and a process for the preparation thereof
03/31/1992CA1298434C Process for the preparation of alpha-l-aspartyl-l- phenylalanine methyl ester
03/31/1992CA1298433C Amino acid derivatives
03/31/1992CA1298432C PROCESS FOR SEPARATION OF N-PROTECTED- .alpha. L-ASPARTYL- L-PHENYLALANINES
03/29/1992CA2051782A1 Aminoesters of rapamycin
03/28/1992CA2052057A1 Fibrinogen receptor antagonists
03/25/1992EP0476933A1 Neurotrophic peptide derivatives