Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
01/1999
01/12/1999US5859184 Alpha-helix mimetics and methods relating thereto
01/12/1999US5859031 Small molecule inhibitors of rotamase enzyme activity
01/12/1999US5859002 HIV protease inhibitors
01/12/1999US5858994 Carbohydrate conjugates as inhibitors of cell adhesion
01/12/1999US5858982 Cathepsin and methods and compositions for inhibition thereof
01/12/1999US5858979 Anticoagulant peptides
01/12/1999US5858660 Parallel selex
01/07/1999WO1999032511A1 PEPTIDES, METHOD FOR ASSAYING HUMAN PEPSINOGEN II or HUMAN PEPSIN II, AND ASSAYING KIT
01/07/1999WO1999000361A1 Ace-inhibitor nitric salts
01/07/1999EP0889036A1 HIV protease inhibitors
01/07/1999EP0888459A1 Measurement of complement activation by biomaterials by means of complement convertase cleavage of peptide substrates
01/07/1999EP0888381A1 Targeted therapeutic or diagnostic agents and methods of making and using same
01/07/1999EP0888130A2 New ternary radiopharmaceutical complexes
01/07/1999CA2292794A1 Ace-inhibitor nitric salts
01/06/1999CN1204341A Oligopeptide compounds containing D-2-alkyltryptophan capable of promoting release of growth hormone
01/06/1999CN1041524C Oligopeptides derived from C-reactive protein fragments and its medical composition
01/05/1999US5856530 Antipicornaviral compounds and methods for their use and preparation
01/05/1999US5856477 Hypotensive agents; congestive heart failure
01/05/1999US5856476 Processes for preparing azepiones useful as intermediates in the preparation of inhibitors of angiotensin converting enzyme and neutral endopeptidase
01/05/1999US5856474 Cephalosporin synthesis
01/05/1999US5856439 Farnesyl transferase inhibitors, preparation thereof, and pharmaceutical compositions containing same
01/05/1999US5856353 Sulfonamide inhibitors of aspartyl protease
01/05/1999US5856310 Inhibition of farnesyltransferase
01/05/1999US5856309 Treating osteoporosis, inflammation or a disease which is due to a thromboembolic event
01/05/1999US5856307 Peptide derivatives as kininogenase inhibitors
01/05/1999US5856306 Oligopeptides modified with boron fragment
12/1998
12/30/1998WO1998058950A1 Compounds with growth hormone releasing properties
12/30/1998WO1998058949A1 Treatment of insulin resistance with growth hormone secretagogues
12/30/1998WO1998058948A1 Tartrate salt of a substituted dipeptide as growth hormone secretagogue
12/30/1998WO1998058947A1 Dipeptide derivatives as growth hormone secretagogues
12/30/1998EP0887354A2 Process of working up of 1- N2-((S)-ethoxycarbonyl)-3-phenylpropyl)-N6-trifluor-acetyl -L-lysyl-L-prolin (Lisinopril(Tfa)ethylester, LPE)
12/30/1998EP0886647A1 Serine protease inhibitors
12/30/1998EP0705105A4 Metal chelates as spacer compounds in biologically active peptides
12/30/1998CN1203602A Acylated enol derivatives of 'alpha'-ketoesters and 'alpha'-ketoamides
12/30/1998CA2294464A1 Treatment of insulin resistance
12/29/1998US5854388 Angiotensin IV peptides and receptor
12/29/1998US5854249 Opioid diarylmethylpiperazines and piperidines
12/29/1998US5854211 Compounds with growth hormone releasing properties
12/29/1998US5854029 Method for preparing antihypertensive agent
12/29/1998US5853713 Biologically compatible linear block copolymers of polyalkylene oxide and peptide units
12/29/1998US5853623 Peptidyl compounds and their therapeutic use as inhibitors of metalloproteinases
12/24/1998DE19827309A1 Tri:fluoro:acetyl lisinopril ethyl ester purification
12/23/1998EP0885904A1 Peptides as agonists and/or inhibitors of amyloid formation and/or cytotoxicity and their use against Alzheimer's disease, type II diabetes mellitus and spongiform encephalopathy
12/23/1998EP0885887A2 Sulfonamide inhibitors of HIV-Aspartyl protease
12/23/1998EP0885608A1 Remedies for brain diseases
12/23/1998EP0885243A1 Crystal structure of apopain and uses thereof
12/23/1998EP0885189A2 Method for the synthesis of poly-pyrrole and poly-imidazole carboxamides on a solid support
12/23/1998EP0885188A1 Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors
12/23/1998EP0885186A1 Amino acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
12/23/1998EP0722459B1 Hemoregulatory penta- or hexapeptides
12/23/1998CN1202902A Thrombin inhibitors
12/23/1998CN1202901A Phosphonic acid derivatives with metallopeptidase inhibitory activity
12/23/1998CN1202882A New LH-RH antigonists with improved effectiveness
12/23/1998CN1041281C Polymer-bound taxol derivatives
12/22/1998US5852051 Dipeptide p-amidinobenzylamides with N-terminal sulfonyl or aminosulfonyl radicals
12/22/1998US5852045 Fibrinogen receptor antagonists
12/22/1998US5852043 HIV protease inhibitors
12/17/1998WO1998057174A1 Synthetic antibiotics
12/17/1998WO1998051325A3 Random peptides that bind to gastro-intestinal tract (git) transport receptors and related methods
12/17/1998CA2240005A1 Peptides acting as agonists and inhibitors of amyloid formation and cytotoxicity for therapeutic use with alzeheimer's disease, type ii diabetes mellitus and spongiform encephalopathies
12/16/1998EP0884326A2 Antithrombitic compound
12/16/1998EP0884325A1 Thrombin inhibitors containing a peptidyl heterocycle
12/16/1998EP0883629A1 Oligopeptides for drug delivery
12/16/1998EP0715618B1 Hydroxyethylamino sulphonamides useful as retroviral protease inhibitors
12/16/1998CN1202174A Peptide derivatives
12/16/1998CN1202161A Macrocyclic compounds as metalloprotease inhibitors
12/16/1998CN1041205C Process for crystallisation of aspartame
12/15/1998US5849954 Method of peptide synthesis
12/15/1998US5849918 Amino acid derivatives, processes for the manufacture thereof and pharmaceutical compositions containing these compounds
12/15/1998US5849908 Processes for preparing intermediates of inhibitors of enkephalinase and angiotensin converting enzyme and intermediates thereof
12/15/1998US5849893 Nucleic acid-binding oligomers possessing C-branching for therapy and diagnostics
12/15/1998US5849866 Peptidase inhibitors
12/15/1998US5849865 Peptides for altering bone resorption, angiogenesis and restenosis
12/15/1998US5849711 Cathepsin and methods and compositions for inhibition thereof
12/15/1998US5849710 Substituted indolylmethylene-oxindole analogues as tyrosine kinase inhibitors
12/15/1998US5849693 Cyclic compounds linked by a heterocyclic ring useful as inhibitors of platelet glycoprotein IIb/IIIa
12/15/1998US5849691 Peptidomimetic inhibitors of cathepsin D and plasmepsins I and II
12/15/1998US5849690 Anti-aggregatory peptides
12/15/1998US5849510 Factor Xa inhibitors
12/15/1998US5849296 Crosslinked protein crystals
12/15/1998US5849260 Technetium-99M labeled peptides for thrombus imaging
12/15/1998CA1340227C L-proline derivatives; process for preparing them and biological uses
12/15/1998CA1340186C Peptides
12/10/1998WO1998055503A1 Method for preparing salts of aspartame from n-protected aspartame
12/10/1998WO1998055449A1 Hydroxamic acid compounds having anticancer and anti-parasitic properties
12/09/1998EP0882228A1 Methods to identify modulators of cell signaling
12/09/1998EP0882128A1 Cell-based assay
12/09/1998EP0882066A1 Peptide derivatives
12/09/1998EP0751779A4 Selectively cleavable linkers based on iminodiacetic acid ester bonds
12/09/1998CN1201459A Novel pyridonecarboxylic acid derivatives or their salts and antibacterial agent comprising same as active ingredient
12/09/1998CN1201454A Meta-guanidine, urea, thiourea or azacyclic amino benzoic acid derivatives as integrin antagonists
12/08/1998US5847192 Boronic compound complexing reagents and complexes
12/08/1998US5847135 Inhibitors of interleukin-1β converting enzyme
12/08/1998US5847121 Production of nitro-benzyl-dota via direct peptide cyclization
12/08/1998US5847117 Reagent and catalytic process useful for cleaving a protected functional group
12/08/1998US5846987 Retroviral protease inhibiting compounds
12/08/1998US5846942 Cholecystokinin antagonists, their preparation and therapeutic use
12/08/1998US5846941 Isosteric antiherpes peptide derivatives II
12/08/1998US5846940 Corneal therapeutic agent
12/08/1998US5846755 Method for determining the therapeutic activity of metalloproteinase inhibitor compounds