Patents
Patents for C07K 5 - Peptides having up to four amino acids in a fully defined sequence; Derivatives thereof (30,692)
02/2004
02/26/2004WO2002038796A3 Methods for determining protease cleavage site motifs
02/26/2004US20040039160 Comprises therapeutic agent, oligopeptide having an isoleucine residue, stabilizing group, and, optionally, a linker group; prodrug is cleavable by an enzyme associated with target cell; antitumor agents
02/26/2004US20040038907 For healing wounds/tissue repair
02/26/2004US20040038905 Anticancer agents
02/26/2004US20040038897 Stimulates a sexual and/or erectile response in a mammal
02/26/2004US20040038872 Inhibitors of hepatitis C virus
02/26/2004US20040038331 Solid phase synthesis of biomolecule conjugates
02/26/2004US20040037775 Treating and preventing autoimmune diseases. The compositions and methods utilize peptides that are cell-specific. The peptides are conjugated to drugs. The peptide-drug conjugate can be internalized by the targeted cells thereby allowing for
02/25/2004EP1391518A1 Process for producing peptide
02/25/2004EP1391461A1 Bicyclic lactam inhibitors of interleukin-1-beta converting enzyme
02/25/2004EP1390405A2 Preparation of cholecystokinin agonists and antagonists and their therapeutic and diagnostic use
02/25/2004EP1390393A2 Pentapeptide compounds and uses related thereto
02/25/2004EP1390055A2 Tripeptide derivatives for the treatment of postlesional diseases of the nervous system
02/25/2004EP1390018A1 A pharmaceutical tablet having a high api content
02/25/2004EP1390011A2 Control of compactability through crystallization
02/25/2004EP1220868B1 Extracorporeal endotoxin removal method
02/25/2004CN1139599C Process for prepaing pharmacologically acceptable salts of N-(1-(S)-ethoxycarbonyl-3-phenylpropyl)-L-alanyl amino acids
02/24/2004US6696481 Immediate-release tablets; treatment of arterial hypertension and heart failure
02/24/2004US6696438 Cyclic amino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting β-amyloid peptide release and/or its synthesis by use of such compounds
02/24/2004US6696418 Somatostatin antagonists and agonists that act at the SST subtype 2 receptor
02/24/2004US6696412 Purification of daptomycin by binding to ion exchange resins in the presence of buffers and chaotropic agents, then eluting and recovering; peptide antibiotics
02/24/2004US6696303 Inhibition of amyloid protein bnding to neuronal receptor; obtain cell, incubate with modulator, monitor amyloid protein activity
02/19/2004WO2004015392A2 Improved method to identify targeting molecules
02/19/2004WO2004014944A1 Microbial-origin polyamino acids or derivatives thereof
02/19/2004WO2004014943A2 Biphalin derivates and their analgesic applications
02/19/2004WO2004014882A2 Proteasome inhibitors : peptide derivatives having c-terminal heteroaryl groups
02/19/2004WO2004014415A1 Growth hormone releasing peptides
02/19/2004WO2004014311A2 Nogo receptor antagonists
02/19/2004WO2004005326A3 Tubulysin conjugates
02/19/2004WO2003065987A3 Granzyme b inhibitors
02/19/2004WO2003045974A3 Methods and compositions for derepression of iap-inhibited caspase
02/19/2004WO2002094778A3 Peptide conjugates and fluorescence detection methods for intracellular caspase assay
02/19/2004WO2002069884A3 A sunburn treatment and sunburn prevention method
02/19/2004US20040034202 Ketone spirocyclopropaneindene compounds; antineoplastic agents to inhibit tumor cell growth in vitro or in vivo; particularly effective against solid tumors and multi-drug resistant tumors
02/19/2004US20040033958 Such as (N-((R,S)-2-(2-(N-methyl)pyrrolidinyl)ethyl)glycyl)-(N-(4 -methoxyphenethyl)glycyl)-N-(3-methylbutyl)glycinamide; for treatment of pain
02/19/2004US20040033235 Inhibitory of human and non-human retroviral, especially HIV, transmission to uninfected cells.
02/19/2004CA2495121A1 Nogo receptor antagonists
02/19/2004CA2494551A1 Improved method to identify targeting molecules
02/18/2004EP1389624A1 Phosphorous-containing cysteine and serine protease inhibitors
02/18/2004EP1389200A1 Substituted n-arylsulfonyl-proline derivatives as potent cell adhesion inhibitors
02/18/2004EP1089755B1 Pharmaceutical preparations for use in combatting or preventing surface infections caused by microorganisms
02/18/2004EP1076663B1 Functionalized alkyl and alkenyl side chain derivatives of glycinamides as farnesyl transferase inhibitors
02/18/2004EP1000086B1 Alatrofloxacin parenteral compositions
02/18/2004EP0946166B1 Use of matrix metalloproteinase inhibitors for promoting wound healing
02/18/2004CN1138766C Processes for preparation of oxo-oxazoline or alloamino acid derivatives
02/18/2004CN1138472C Dipeptide apoptosis inhibitors and use thereof
02/17/2004US6693214 Intermediate for sweetener with high sweetness and process for producing the same
02/17/2004US6693199 Deprotecting carbamate group and amidating in presence of such as hydroxybenzotriazole hydrate promoter
02/17/2004US6693168 Chiral cyanoamines and methods of preparation
02/17/2004US6693167 Peptide-based gemini compounds
02/17/2004US6693165 Cyclic peptides as potent and selective melanocortin-4 receptor antagonists
02/17/2004US6693120 Spray drying of thrombin inhibitors
02/17/2004US6693099 Substituted piperazine compounds optionally containing a quinolyl moiety for treating multidrug resistance
02/17/2004US6693096 Treatment of inflammation-associated disorders using interleukin-1β-converting enzyme (ICE)/CED-3 family inhibitors
02/17/2004US6693072 Short, synthetic peptides; antiinflammatories for neutrophil associated diseases
02/17/2004CA2280279C Indole, indazole and benzimidazole derivatives as antithrombotic agents
02/12/2004WO2004013098A1 Novel gamma-lactams as beta-secretase inhibitors
02/12/2004WO2004012816A1 Antibacterial ester macrocycles
02/12/2004WO2004012756A1 New cytotoxic cyclopeptide and its use for the treatment of cancer
02/12/2004WO2004012574A2 Negative selections assays, and compositions thereof
02/12/2004WO2003062261A3 Dmt-tic di- and tri-peptidic derivatives and related compositions and methods of use
02/12/2004WO2003037916A3 Linear basic compounds having nk-2 antagonist activity and formulations thereof
02/12/2004WO2003014698A3 Biological assay detection method
02/12/2004WO2003008438A3 Cosmetic or dermatological use of peptides for promoting adhesion between skin cells
02/12/2004WO2002100344A3 Amino acid conjugates providing for sustained systemic concentrations of gaba analogues
02/12/2004US20040030105 Improved methods for synthesis of phosphinothiol reagents and novel protected reagents for use in peptide ligation
02/12/2004US20040029868 Multiple sclerosis; atherosclerosis; inflamamtory bowel diseases; asthma
02/12/2004US20040029814 Cathepins inhibitor; antiinflammatory agents; antiarthritic agents
02/12/2004US20040029813 Cardiovascular disorders; hypotensive agents; angiotensin converting enzyme inhibitor
02/12/2004US20040029812 Skin disorders; aging resistance
02/12/2004US20040029811 N-alkylglycine trimeres capable of protecting neurons against excitotoxic aggressions and compositions containing such trimeres
02/12/2004US20040029808 Binding antibody to estradiol; test device
02/12/2004US20040029778 Prostate specific antigen; immobilization; antiproliferative agents; drug delivery
02/12/2004DE10234422A1 Antibakterielle Ester-Makrozyklen Antibacterial ester macrocycles
02/12/2004CA2495479A1 Antibacterial ester macrocycles
02/11/2004EP1388537A1 Arginine derivatives
02/11/2004EP1157998B1 Heterocyclic compounds, intermediates thereof and elastase inhibitors
02/11/2004EP1086113B1 Benzothiepine-1,1-dioxide derivatives, method for producing them, medicaments containing these compounds and their use
02/11/2004CN1137891C Process for preparing growth hormone cinogenic agent
02/10/2004US6689902 Reductive alkylation
02/10/2004US6689787 Method of using an integrin antagonist and radiation therapy as combination therapy in the treatment of neoplasia
02/10/2004US6689754 Heterocyclic glycyl β-alanine derivatives
02/10/2004US6689753 Alzheimer inhibitor peptide ia beta 5 (amino acid sequence 1leu-pro-phe-phe-asp) analog
02/10/2004US6689337 Vitronectin receptor antagonist pharmaceuticals
02/10/2004CA2297134C A novel process for preparing intermediates or inhibitors of enkephalinase and angiotensin converting enzyme and intermediates thereof
02/05/2004WO2004011652A1 Process for producing tripeptide or higher peptide
02/05/2004WO2004011476A1 Glyconjugates comprising carbohydrate epitopes, methods for theirsynthesis, and their use for the treatment or prophylaxis of cancer
02/05/2004WO2003097089A3 Attenuation of metapneumovirus
02/05/2004WO2003072735A3 Use of peptide-drug conjugation to reduce inter-subject variability of drug serum levels
02/05/2004WO2003072034A3 Cyclic peptides and analogs useful to treat allergies
02/05/2004WO2003064455A3 Macrocyclic peptides active against the hepatitis c virus
02/05/2004WO2003046137A3 Hiv envelope v3-ccr5 binding site immunogen
02/05/2004WO2002100886A8 Pyrrolidin-2-one derivatives as inhibitors of factor xa
02/05/2004WO2002100883A3 Libraries of conformationally constrained peptides, chiral azacrowns, and peptidomimetics and methods of making the same
02/05/2004US20040024180 By heating suitable dipeptides in organic solvent whilst removing water by distillation; use as chiral catalysts, e.g. for the production of chiral cyanohydrines
02/05/2004US20040023888 Retinol derivatives, the method of preparations and the uses thereof
02/05/2004CA2802205A1 Drug conjugates and their use for treating cancer, an autoimmune disease or an infectious disease
02/04/2004EP1386166A2 Anti-epileptogenic agents
02/04/2004EP1385882A2 Peptides and related molecules that bind to tall-1
02/04/2004EP1385870A2 Peptides as ns3-serine protease inhibitors of hepatitis c virus