Patents
Patents for C07K 11 - Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof (895)
10/2001
10/18/2001WO2001076616A1 Tamandarin and didemnin analogs and methods of making and using them
10/18/2001CA2405779A1 Tamandarin and didemnin analogs and methods of making and using them
10/17/2001EP1144658A2 Methods for producing polypeptides in cyclohexadepsipeptide-deficient cells
10/11/2001WO2001074884A1 Dermacentor variabilis gaba-gated chloride channels
10/11/2001WO2001074850A1 Antibiotics tripropeptins and process for producing the same
10/03/2001CN1315962A Novel process for synthesis of exochelins
09/2001
09/19/2001EP0772630B1 Streptogramine derivatives, preparation of same and pharmaceutical compositions containing same
09/12/2001EP1049481A4 Synthetic antineoplastic agents derived from dolastatin 15 and methods of making same
09/12/2001CN1312818A Chemical synthesis of exochelins
09/07/2001WO2001055306A8 Nucleic acids, proteins, and antibodies
09/05/2001CN1070481C Use of dioxomorpholines to combact endopharasites, movel dioxomopholines and process for their prodn.
08/2001
08/16/2001WO2001058934A2 Kahalalide f and related compounds
08/16/2001EP1123112A1 Ionic molecular conjugates of n-acylated derivatives of poly (2-amino-2-deoxy-d-glucose) and polypeptides
08/08/2001CN1307586A Substituted cyclooctadepsipeptides
08/02/2001WO2001055306A2 Nucleic acids, proteins, and antibodies
08/02/2001CA2395811A1 Nucleic acids, proteins, and antibodies
07/2001
07/19/2001WO2000069891A3 Previns as specific inhibitors and therapeutic agents for botulinum toxin b and tetanus neurotoxins
07/12/2001US20010007855 Antitumor drug
07/04/2001EP0773956B1 Purified form of streptogramines, preparation of same and pharmaceutical compositions containing same
07/03/2001US6255286 Depsipeptides and drugs containing the same as the active ingredient
06/2001
06/28/2001WO2001045512A1 Pest control agents / depsipeptides
06/28/2001DE19962145A1 Composition for controlling animal pests, especially lepidopteran caterpillars, comprises a cyclodepsipeptide containing a N,N-disubstituted 4-aminobenzyl group
06/21/2001WO2001044177A2 Somatostatin analogs, radiolabelled derivatives thereof and their use
06/21/2001CA2383936A1 Novel somatostatin analogs
06/14/2001WO2001042282A1 Depsipeptide and congeners thereof for use as immunosuppressants
06/13/2001EP1105416A1 Novel process for the synthesis of exochelins
06/13/2001EP1105415A1 Chemical synthesis of exochelins
05/2001
05/29/2001US6239104 Isolated and purified substance which inhibits neoplastic cell growth denominated dolastatin 16
05/09/2001CN1294134A Polypeptide structure of shark liver for preventing and curing hepatism and its purifying process
04/2001
04/11/2001EP1090031A1 Substituted cyclooctadepsipeptides
03/2001
03/22/2001WO2000063240A9 ANTIFUNGAL AGENTS ISOLATED FROM $i(PSEUDOMONAS SYRINGAE)
03/15/2001WO2001018227A1 Novel compound f-15078
03/15/2001CA2383758A1 Novel compound f-15078
03/07/2001CN1286264A Action of proinsulin associated peptide on dopamine transporter and its application in treating correlative diseases
03/07/2001CN1286261A Mimic peptide of schistosoma japonice ovum antigen and its screening and application
03/06/2001US6197536 Methodology to produce, and purify and assay polypeptides with the proteolytic activity of the HCV NS3 protease
02/2001
02/15/2001WO2001010895A1 Streptogramin derivatives, production thereof and compositions containing the same
01/2001
01/30/2001US6180392 Streptomyces strains and process to produce single streptogramin component
01/25/2001WO2001005813A1 Pseudomycin prodrugs
01/25/2001CA2379058A1 Pseudomycin prodrugs
12/2000
12/21/2000WO2000076985A1 Cyclo-imino depsipeptides and their utilization in controlling endoparasites
12/21/2000CA2374632A1 Cyclo-imino depsipeptides and their utilization in controlling endoparasites
12/14/2000WO2000042203A3 Methods for producing polypeptides in cyclohexadepsipeptide-deficient cells
12/14/2000DE19926620A1 Neue Cycloiminodepsipeptide, Verfahren zu ihrer Herstellung und ihre Verwendung zur Bekämpfung von Endoparasiten New Cycloiminodepsipeptide, processes for their preparation and their use for controlling endoparasites
11/2000
11/28/2000US6153731 Dehydrodidemnin B
11/23/2000WO2000069891A2 Previns as specific inhibitors and therapeutic agents for botulinum toxin b and tetanus neurotoxins
11/23/2000CA2372304A1 Previns as specific inhibitors and therapeutic agents for botulinum toxin b and tetanus neurotoxins
11/08/2000EP1049481A2 Synthetic antineoplastic agents derived from dolastatin 15 and methods of making same
10/2000
10/26/2000WO2000063345A1 PSEUDOMYCIN PRODUCTION BY $i(PSEUDOMONAS SYRINGAE)
10/26/2000WO2000063240A1 ANTIFUNGAL AGENTS ISOLATED FROM $i(PSEUDOMONAS SYRINGAE)
10/26/2000CA2371363A1 Antifungal agents isolated from pseudomonas syringae
10/26/2000CA2370239A1 Pseudomycin production by pseudomonas syringae
09/2000
09/12/2000CA2029408C Antibiotic a/16686 recovery process
08/2000
08/30/2000EP0787141B1 Cyclic depsipeptide sulfonylation, sulfenylation and phosphorylation process
08/30/2000EP0687686B1 Aureobasidins
08/03/2000WO1999015130A3 Synthetic antineoplastic agents derived from dolastatin 15 and methods of making same
07/2000
07/20/2000WO2000042203A2 Methods for producing polypeptides in cyclohexadepsipeptide-deficient cells
06/2000
06/21/2000CN1053657C Didepside phthaleins based internal parasite compositions, novel didepside phthaleins and preparation process thereof
05/2000
05/31/2000CN1254596A Process for preparing composition to kill internal parasites
05/16/2000US6063919 Esterification of o-deprotected dibenzyl exochelic acid with benzyl epi-cobactin, hydrogenolytically removing the three benzyl groups to form exochelin 786sm(r)
05/03/2000EP0996458A1 Sandramycin analogs
05/02/2000CA2012480C Isolation and structural elucidation of the cytostatic linear depsipeptide dolastatin 15
04/2000
04/20/2000WO2000021567A1 Ionic molecular conjugates of n-acylated derivatives of poly(2-amino-2-deoxy-d-glucose) and polypeptides
04/20/2000CA2346066A1 Ionic molecular conjugates of n-acylated derivatives of poly(2-amino-2-deoxy-d-glucose) and polypeptides
03/2000
03/07/2000US6034058 Administering polypeptide
03/07/2000US6033879 Process for the preparation of substituted aryl lactic acid containing cyclodepsipeptides with 24 ring atoms
03/01/2000EP0981352A1 Aplidine as an l-type calcium channel enhancer
02/2000
02/24/2000WO2000009548A1 Chemical synthesis of exochelins
02/24/2000WO2000009547A1 Novel process for the synthesis of exochelins
02/24/2000CA2339184A1 Chemical synthesis of exochelins
02/24/2000CA2338781A1 Novel process for the synthesis of exochelins
01/2000
01/26/2000EP0973540A1 Isolation and structural elucidation of the cytostatic linear and cyclo-depsipeptides dolastatin 16, dolastatin 17, and dolastatin 18
01/26/2000EP0973518A1 Semi-synthetic studies toward didemnin analogues
01/11/2000US6013627 Organic compounds
01/04/2000US6011136 Inhibitor of tumor necrosis factor; antiinflammatory agents
12/1999
12/30/1999DE19828047A1 New sulfonyl-substituted cyclooctadepsipeptide derivatives useful for prevention and treatment of helminth infection
12/29/1999WO1999067281A1 Substituted cyclooctadepsipeptides
12/29/1999CA2332122A1 Substituted cyclooctadepsipeptides
12/08/1999EP0775158B1 Cyclopeptolides
12/01/1999EP0960885A1 Depsipeptides and drugs containing the same as the active ingredient
11/1999
11/17/1999EP0956033A1 Total synthesis of the amino hip analogue of didemnin a
10/1999
10/26/1999CA2029678C Isolation and structural elucidation of the cytostatic linear depsipeptide dolastatin 14
09/1999
09/21/1999CA2012867C Novel cytotoxic cyclic depsipeptides from the tunicate trididemnum solidum
09/14/1999US5952492 Reacting a mixture of diacid with dimethyl pimelate, hydrochloric acid, methanol, dibutyl ether to form intermediate, adding o-benzyl hydroxylamine hydrochloride and triethylamine, additing di-tert-butyl dicarbonate
09/14/1999US5952299 Cyclic peptide nuclei and derivatives thereof
08/1999
08/31/1999US5945316 From optically active or racemic amino acids and 2-hydroxycarboxylic acids
08/11/1999CN1225688A Novel antitumor compounds and process for producing same
06/1999
06/24/1999WO1999031127A1 Cyclopeptolides
04/1999
04/21/1999EP0909822A1 Novel antitumor compounds and process for producing the same
04/01/1999WO1999015130A2 Synthetic antineoplastic agents derived from dolastatin 15 and methods of making same
03/1999
03/16/1999CA1340447C Pipecolic acid-containing peptolides, their preparation and pharmaceutical compositions containing them
03/04/1999WO1998054211A3 Cyclodepsipeptides and pharmaceutical compositions containing them
02/1999
02/23/1999US5874530 Cyclic depsipeptide sulfonylation, sulfenylation and phosphorylation process
02/17/1999CN1208439A Process for the preparation of substituted aryl lactic acid containing cyclodepsipeptides with 24 ring atoms
01/1999
01/05/1999US5856324 Use of dioxomorpholines for combat endoparasites, dioxomorpholines and process for their production
12/1998
12/23/1998CN1202904A Cyclopeptolides
12/03/1998WO1998054211A2 Cyclodepsipeptides and pharmaceutical compositions containing them
12/01/1998US5843755 Group of antitumor compounds and method for producing the same
11/1998
11/18/1998CN1199394A Didepsipeptide-based endoparasiticides, new didepsipeptides and process for preparing same
11/10/1998US5834586 Dehydrodidemnin B
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