Patents
Patents for C07J 71 - Steroids in which the cyclopenta[a]hydrophenanthrene skeleton is condensed with a heterocyclic ring (3,845)
05/2002
05/16/2002WO2002038584A1 Process for the production of 16,17-[(cyclohexylmethylen)bis(oxy)]-11,21-dihydroxy-pregna-1,4-dien-3,20-dion or its 21-isobutyrat by transketalisation
05/16/2002WO2002038582A2 Method for the production of 4-(17alpha substituted 3-oxoestra-4,9-dien-11-yl)benzaldehyd-(1e or 1z)-oximes
05/16/2002WO2002038581A2 Method for the production of 4-(17alpha-methyl substituted 3-oxoestra-4,9-dien-11beta-yl)benzaldehyd-(1e or 1z)-oximes
05/16/2002DE10056676A1 Preparation of estradienyl-benzaldoxime derivative preparation in high yield, for use e.g. in treating endometriosis, from epoxy-estrenone by multi-stage process including selective Grignard reaction
05/16/2002DE10056675A1 Preparation of estradienyl-benzaldoxime derivative preparation in high yield, for use e.g. in treating endometriosis, from estradienone by multi-stage process including selective Grignard reaction
05/15/2002CA2348206A1 Isomerisation of 6beta-fluorosteroids into the corresponding 6alpha-fluoro derivatives
05/10/2002WO2002036106A2 Novel medicament compositions based on anticholinergics and corticosteroids
05/10/2002WO2001029036A3 Allosteric sites on muscarinic receptors
05/07/2002US6384025 Skin disorders; reacting retinol with chloroformate compound
05/02/2002WO2001040253A3 3-methylene steroid derivative for the treatment of autoimmune diseases
05/02/2002EP0615448B1 Sex steroid activity inhibitors
04/2002
04/24/2002CN1345728A Solasodine hydrochlorate and productive method and application in medicine
04/23/2002US6376687 Steroid sulfatase inhibitors and methods for making and using the same
04/23/2002US6376657 Pharmaceutical compositions having appetite suppressant activity
04/18/2002WO2002030462A2 Hedgehog antagonists, methods and uses related thereto
04/18/2002WO2002030366A1 Melanogenesis inhibitors and whitening agents comprising ergosterol derivative and compositions containing ergosterol derivative
04/18/2002US20020045746 Form L crystalline eplerenone having a monoclinic crystal system and an X-ray powder diffraction pattern with a peak at 8. 0+-0.2 degrees 2 theta .
04/18/2002DE10049736A1 17alpha-Fluoralkylsteroide, Verfahren zu deren Herstellung und diese Verbindungen enthaltende pharmazeutische Zusammensetzungen 17alpha-Fluoroalkyl steroids, processes for their preparation and pharmaceutical compositions containing them
04/18/2002DE10048634A1 19-Nor-17alpha-pregna-1,3,5(10)-trien-17beta-ole mit einem 21, 16alpha-Laktonring 19-Nor-17alpha-pregna-1,3,5 (10) triene-17beta-ols with a 21, 16alpha-lactone
04/18/2002CA2425356A1 Hedgehog antagonists, methods and uses related thereto
04/11/2002US20020042507 Process for preparation of 9,11-epoxy steroids and intermediates useful therein
04/09/2002US6369218 Isomerisation of 6β-fluorosteroids into the corresponding 6α-fluoro derivatives
04/04/2002WO2002026763A1 19-NOR-17α-PREGNA-1,3,5 (10)-TRIEN-17β-OLS OF A 21,16α-LACTONE RING
04/04/2002WO2002026759A2 17α FLUOROALKYL STEROIDS, METHOD FOR PRODUCING THE SAME AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAID COMPOUNDS
04/04/2002CA2422056A1 17.alpha. fluoroalkyl steroids, method for producing the same and pharmaceutical compositions containing said compounds
04/03/2002CN1342657A Compound extracted from manatee for suppressing generation of new blood vessel in tumor
04/03/2002CN1342656A Cyclobornane triterpenoid saponin compound and its application in immunosuppresion and treating tumor
03/2002
03/28/2002WO2002000679A3 9.alpha.-chloro-6.alpha.-fluoro-17.alpha.-hydroxy-16-methyl-17-beta-methoxycarbonyl-androst-1,4-dienes esterified in position 17.alpha. by a cyclic acyl group
03/28/2002US20020038021 Eplerenone crystalline form exhibiting enhanced dissolution rate
03/21/2002WO2002022647A1 Sulphur analogues of 21-hydroxy-6,19-oxidoprogesterone (21oh-6op) for treating excess of glucocorticoids
03/21/2002WO2002022646A2 Method for the preparation of 21-hydroxy-6,19-oxidoprogesterone (21oh-6op)
03/21/2002WO2002022121A1 Fungicidal saponin, cay-1, and isolation thereof from capsicum species fruit
03/21/2002US20020035260 4-aza-steroids
03/21/2002CA2419960A1 Method for the preparation of 21-hydroxy-6,19-oxidoprogesterone (21oh-6op)
03/20/2002CN1081036C Anticarcinogen
03/14/2002US20020032179 Inhibiting the hyperproliferation of malignant or neoplastic cells by treating the cells with an antiproliferative amount of 1 alpha ,24(S)-dihydroxyvitamin D2 the cells being cancers of the lung, neck and head, pancreas, endometrium, bladder
03/13/2002CN1340056A Steroides sulfatase inhibitors and methods for making and using same
03/07/2002WO2002017895A2 Use of an aldosterone receptor antagonist to improve cognitive function
03/07/2002CA2419256A1 Use of an aldosterone receptor antagonist to improve cognitive function
03/06/2002CN1080267C Preparation of intermediat of 19, 11 beta-bridge steroid
03/05/2002US6352980 Estrenes for inducting hypothalamic effects
03/05/2002US6352697 Immunostimulating complex matrices; quil a fractions
02/2002
02/28/2002WO2001053321A3 Use of trilostane and its derivatives, optionally in combination with tamoxifen or raloxifene in the treatment of estrogen-dependent cancers e.g. breast, prostate and uterus cancers
02/28/2002US20020025951 Urogenital disorders
02/27/2002EP0970105B1 Process for preparing carboxamido-4-azasteroids
02/21/2002WO2001049703A3 Substituted sapogenins and their use
02/14/2002US20020019547 Skin disorders; reacting retinol with chloroformate compound
02/14/2002US20020019522 Steroids
02/14/2002US20020019378 Compounds
02/07/2002WO2002010188A1 16alpha-methyl or ethyl substituted estrogens
02/07/2002WO2002009760A2 Epoxy-steroidal aldosterone antagonist and beta-adrenergic antagonist combination therapy for treatment of congestive heart failure
02/07/2002WO2002009683A2 Aldosterone blocker therapy to prevent or treat inflammation-related disorders
02/07/2002US20020016481 Oxireno-, azetidino-, and methano- picene derivatives
02/07/2002US20020016455 Epoxidation of cyclopenta(a)phenanthrene derivatives
02/07/2002CA2416152A1 Aldosterone blocker therapy to prevent or treat inflammation-related disorders
02/07/2002CA2415789A1 Epoxy-steroidal aldosterone antagonist and beta-adrenergic antagonist combination therapy for treatment of congestive heart failure
02/06/2002EP1177204A2 Eplerenone crystalline form exhibiting enhanced dissolution rate
01/2002
01/30/2002EP1175434A2 Eplerenone crystalline form
01/30/2002EP1175433A1 Androgen glycosides and androgenic activity thereof
01/24/2002WO2001034132A3 Use of an aldosterone antagonist for treating restenosis
01/23/2002EP1173430A1 Enantiomers of mercapto lactones and processes for their synthesis
01/23/2002CN1078072C Use of 1 alpha, 24-dihydroxy vitamin D2
01/17/2002WO2002004410A1 Process for producing sulfamate compound
01/16/2002EP0923599B1 Process for the preparation of 17-esters of 9alpha,21-dihalo-pregnane-11beta,17alphadiol-20-ones
01/15/2002US6339079 Steroid sulfamates, method for the production and use thereof
01/09/2002EP1170299A2 Processes for preparation of 9,11-epoxy steroids and intermediates useful therein
01/03/2002WO2002000679A2 9.alpha.-chloro-6.alpha.-fluoro-17.alpha.-hydroxy-16-methyl-17-beta-methoxycarbonyl-androst-1,4-dienes esterified in position 17.alpha. by a cyclic acyl group
01/03/2002WO2000071563A3 Taccalonolide microtubule stabilizing agents
01/02/2002EP1167381A2 Process for preparation of 7 alpha-carboxyl 9,11-epoxy steroids and Intermediates useful therein
01/02/2002EP1167380A2 11.alpha.-hydroxy-steroid-4,6-dien-3-one compounds and a process for their preparation
01/02/2002EP1167364A1 Benzopyran-containing compounds and prodrug forms thereof
01/02/2002EP1165596A1 14,15-.alpha.-methylene equilenine derivatives, methods for producing the same and medicaments containing them
01/01/2002US6335441 5β-cyano-substituted steroid compounds
12/2001
12/27/2001WO2001098322A1 Novel steroidal antiestrogens and antiandrogens and uses thereof
12/26/2001CN1076607C Process for preparing pharmaceutical composition containing novel steroid esters
12/26/2001CN1076606C Use of novel steroid esters for preparing medicaments flammatory and anti-allergic activity
12/18/2001US6331622 Processes for preparation of 9, 11-epoxy steroids and intermediates useful therein
12/18/2001US6331535 Retinyl carbonate derivatives, preparation process and uses
12/18/2001US6331534 Steroids as neurochemical stimulators of the VNO to alleviate pain
12/12/2001EP0806413B1 2-substituted vitamin d3 derivatives
12/12/2001EP0785802B1 Saponin preparations and use thereof in iscoms
12/05/2001EP1158988A2 Corticosteroid formulation
11/2001
11/29/2001WO2001042272A3 Eplerenone crystalline form exhibiting enhanced dissolution rate
11/29/2001US20010047093 Activation of a diels-alder reaction of a sterol 5,7 diene
11/22/2001WO2001041535A3 Eplerenone crystalline form
11/21/2001CN1322729A Acylated derivative of dioscin and its producing process and use
11/15/2001WO2001085174A1 Formulations containing a glucocorticoid drug for the treatment of bronchopulmonary diseases
11/15/2001CA2408647A1 Formulations containing a glucocorticoid drug for the treatment of bronchopulmonary diseases
11/14/2001EP0686613B1 Ozonide reducing agent
11/08/2001WO2001083512A1 3-nitrogen-6,7-dioxygen steroids and uses related thereto
11/08/2001CA2418748A1 3-nitrogen-6,7-dioxygen steroids and uses related thereto
11/06/2001US6313161 2,19-methyleneoxy and 2,19-methylenethio bridged steroids as aromatase, 19-hydroxylase inhibitors and methods of their use in the treatment of estrogen mediated disorders
10/2001
10/30/2001US6310225 Useful as intermediates for producing vitamin d derivates
10/30/2001US6310091 Fungicidal saponin, CAY-1, and isolation thereof from Capsium species fruit
10/24/2001EP1148061A2 Process for preparation of 9, 11- epoxy steroids and intermediates useful therein
10/24/2001EP1147124A2 Steroid sulfatase inhibitors and methods for making and using the same
10/23/2001US6306862 Treatment of liver disorders
10/11/2001WO2001074839A2 Methods of making the 4-n-butylcyclohexanoic and the undecanoic acid esters of (7 alpha, 11 beta)-dimethyl-17 beta-hydroxy-4-estren-3-one and their medical use
09/2001
09/27/2001WO2001070760A1 Process for producing diels-alder adducts of sterol 5,7-dienes using unsaturated fatty acid catalyst
09/26/2001CN1071574C Use of 1 alpha, 24-dihydroxy vitamin D2
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