Patents
Patents for C07J 41 - Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring (4,637)
01/2000
01/18/2000US6015805 Potent antiprogestational activity and are useful in the treatment of fibroids, endometriosis, cervical ripening prior to delivery, hormone replacement therapy and in the control of fertility.
01/12/2000EP0970105A1 Process for preparing carboxamido-4-azasteroids
01/12/2000EP0970104A2 Steroid sulfamates, method for the production and use thereof
01/12/2000EP0970103A1 Antigestagenic steroids with a fluorinated 17alpha-alkyl chain
01/04/2000US6011026 P-(aminoalkoxyphenyl)-steroid derivative
01/04/2000US6011025 11-(substituted phenyl)-estra-4,9-diene derivatives
01/04/2000US6011024 Steroid sulphatase inhibitors
12/1999
12/29/1999WO1999067274A1 Novel 17-halogenated 19-nor steroids, method and intermediates for preparing same, use as medicines and pharmaceutical compositions containing same
12/29/1999CA2336167A1 Novel 17-halogenated 19-nor steroids, method and intermediates for preparing same, use as medicines and pharmaceutical compositions containing same
12/23/1999WO1999033859A3 Novel anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use
12/21/1999US6005124 Method for the preparation of steroid derivative ketal
12/21/1999US6004978 Methods of treating cancer with aromatic nitro and nitroso compounds and their metabolites
12/09/1999WO1999062929A1 17β-NITRO-11β-ARYLSTEROIDS AND THEIR DERIVATIVES HAVING AGONIST OR ANTAGONIST HORMONAL PROPERTIES
12/09/1999WO1999062928A1 17β-AMINO AND HYDROXYLAMINO-11β-ARYLSTEROIDS AND THEIR DERIVATIVES HAVING AGONIST OR ANTAGONIST HORMONAL PROPERTIES
11/1999
11/30/1999US5994568 Estrenes for inducing hypothalamic effects
11/30/1999US5994336 Method of inhibiting proliferation of cells by administering an aminosterol compound
11/30/1999US5994333 Pregnane and cholane steroids as neurochemical initiators of change in human hypothalamic function and related pharmaceutical compositions and methods
11/24/1999EP0633893B1 17-substituted steroids useful in cancer treatment
11/24/1999CN1046735C Steroids for treating menopausal complaints
11/23/1999US5990328 Forming 4-nitro-3-ketosteroids which by nitration of the corresponding 3,5-dienolate, reduction of 4-nitro-3-ketosteroid forms 4-amino-3-ketosteroid
11/23/1999US5990099 Treating glc1a glaucoma by administering an angiostatic steroid of given formula
11/19/1999CA2237879A1 Nitrile derivatives of 19-nor-steroids for use in radiotherapy and/or imaging of cancer
11/18/1999WO1999058549A1 Meiosis regulating compounds
11/18/1999CA2331962A1 Meiosis regulating compounds
11/17/1999EP0957108A1 Unsaturated cholestane derivatives, pharmaceutical compositions comprising them and use of these derivatives for the preparation of meiosis regulating medicaments
11/16/1999US5986115 7α-(ξ-aminoalkyl)-estratrienes, process for their production, pharmaceutical preparations which contain these 7α-(ξ-aminoalkyl)-estratrienes as well as their use for the production of pharmaceutical agents
11/10/1999EP0954339A2 Cationic amphiphile compositions for intracellular delivery of therapeutic molecules
11/10/1999EP0954338A2 Cationic amphiphile/dna complexes
11/10/1999EP0748332B1 New cholesterol derivative for liposomal gene transfer
11/09/1999US5981516 Treating cholesterol without estrogenic activity at the uterine level in women comprising administering to women an amount of a steroid
11/02/1999US5977126 Antiangrogens, enzyme inhbitors
11/02/1999US5977096 Steroids with radical-attracting aromatic substituents, process for the production thereof and pharmaceutical compounds containing the said substances
10/1999
10/28/1999WO1999033858A9 Estrone sulfamate inhibitors of estrone sulfatase, and associated pharmaceutical compositions and methods of use
10/21/1999WO1999052932A1 Fatty acid derivatives of bile acids and bile acid derivatives
10/19/1999US5969168 Stimulate autonomic activity
10/13/1999CN1231670A 7 'alpha'-('xi'-aminoalkyl) estratrienes, process for preparing the same, pharmaceutical preparations containing the same, and their use for preparing medicaments
10/13/1999CN1045589C N-acylaminoglutaricamide derivative
10/12/1999US5965552 Administering androsta-4,16-dien-3-ol for treating tension, reducing anxiety; administering to the vomeronasal organ of individual
10/12/1999US5965550 Process for the preparation of 4-amino-Δ4 -3-ketosteroids via 4-nitro-Δ4 -3-ketosteroids
10/06/1999EP0946586A1 Aminosterol ester compounds
10/06/1999EP0946585A1 Steroids substituted in position 11, method of preparation, application as medicines and pharmaceutical compositions containing them
10/05/1999US5962444 Hormone inhibitor; hormone replacement therapy
10/05/1999US5962443 19-nur-pregnane steroids as neurochemical initiators of change in human hypothalamic function
10/05/1999US5962442 Administering a 3-oxo-4-azasteroid
09/1999
09/29/1999EP0944644A2 Processes for preparation of 9,11-epoxy steroids and intermediates useful therein
09/29/1999EP0944643A1 Oxyiminopregnancarbolactone
09/29/1999EP0909764B1 11 Beta-Benzaldoxim-9 Alpha, 10 Alpha-epoxy-estr-4-en-derivatives, a process for their production and pharmaceutical compositions containing them
09/28/1999US5958901 Delivery of anionic macromolecules into cells.
09/23/1999WO1999033859A9 Novel anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use
09/22/1999EP0943328A2 Combination therapy for prophylaxis and/or treatment of benign prostatic hyperplasia
09/22/1999EP0942919A2 Compound
09/22/1999EP0942918A2 Stereoselective synthesis of 24-hydroxylated compounds useful for the preparation of aminosterols, vitamin d analogs, and other compounds
09/21/1999US5955622 Method for the preparation of steroid derivative ketal
09/16/1999WO1999046280A1 Lipid compounds derived from sphingoid bases, preparation method and uses in cosmetics and dermopharmacy
09/16/1999WO1999046279A2 INHIBITORS OF TYPE 5 AND TYPE 3 17β-HYDROXYSTEROID DEHYDROGENASE AND METHODS FOR THEIR USE
09/16/1999WO1999033858A3 Estrone sulfamate inhibitors of estrone sulfatase, and associated pharmaceutical compositions and methods of use
09/16/1999CA2323089A1 Inhibitors of type 5 and type 3 17.beta.-hydroxysteroid dehydrogenase and methods for their use
09/16/1999CA2321216A1 Lipid compounds derived from sphingoid bases, preparation method and uses in cosmetics and dermopharmacy
09/15/1999EP0942001A1 Sphingoid Lipid Compounds, a Process for Their Production and Cosmetic and Dermopharmaceutical uses Thereof
09/14/1999US5952516 An intracellular delivery of a biological active material to target plasma membrane, tissue fluids, cells; gene therapy
09/14/1999US5952499 Therapeutic compound-fatty acid conjugates
09/14/1999US5952183 Synthesis of estrogen-purine base and estrogen-mercapturate adducts and development of fluorescent probes and monoclonal antibodies to assay those adducts
09/10/1999WO1999045024A1 Cholenic acid amides and pharmaceutical compositions thereof
09/10/1999WO1999045023A1 S-SUBSTITUTED 11β-BENZALDOXIME-ESTRA-4,9-DIENE-CARBONIC ACID THIOLESTERS, METHOD FOR THE PRODUCTION THEREOF AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE COMPOUNDS
09/10/1999WO1999044616A1 Steroid derived antibiotics
09/09/1999DE19809845A1 S-substituierte 11beta-Benzaldoxim-estra-4,9-dien-kohlensäurethiolester, Verfahren zu deren Herstellung und diese Verbindungen enthaltende pharmazeutische Zubereitungen For their preparation and compositions containing these compounds S-11beta-substituted benzaldoxime-estra-4,9-dien-kohlensäurethiolester, procedures pharmaceutical preparations
09/07/1999US5948925 Transport of active materials into cells
09/07/1999US5948767 Transport of active material into cells; drug delivery
09/01/1999EP0886645B1 New 19-nor-pregnene derivatives
08/1999
08/31/1999US5945530 17,20-epoxy steroid intermediates
08/31/1999US5945404 21-Substituted steroid compound
08/25/1999EP0937729A1 Silicon containing compounds useful as protective groups or as linkers in solid phase organic chemistry
08/24/1999US5942634 A drug delivery for gene therapy comprising a di-polyalkylamine-alkylamide or alkyl disulfide cholesterol
08/17/1999US5939570 Estrenes for inducing hypothalamic effects
08/17/1999US5939545 Method, compositions, and compounds for allosteric modulation of the gaba receptor by members of the androstane and pregnane series
08/17/1999US5939401 Cationic amphiphile compositions for intracellular delivery of therapeutic molecules
08/13/1999CA2260736A1 Linkers
08/12/1999DE19806357A1 New 11 beta-halo-7 alpha-substituted estratrienes useful for treating e.g. estrogen-dependent disease such as breast cancer
08/11/1999EP0649431B1 17-amino substituted 4-azasteroid 5-alpha-reductase inhibitors
08/03/1999US5932431 Incubating sample, solid phase coupled to antibody, labeled conjugate of steroid analogue; measuring amount of label in solution or on separated solid phase; use of slightly different steroid conjugate improves antibody performance
07/1999
07/27/1999US5929262 Method for preparing 17α-acetoxy-11β-(4-N, N-dimethylaminophyl)-19-Norpregna-4,9-diene-3, 20-dione, intermediates useful in the method, and methods for the preparation of such intermediates
07/27/1999US5929108 Detecting dna and rna sequence comprising hybridizing a probe with compementary regions of said dna and rna sequence, wherein the probe is a nucleic acid sequence labeled with digoxigenin derivative-spacer-furocoumarins complex label
07/21/1999EP0929565A2 Nitrate esters of corticoid compounds and pharmaceutical applications thereof
07/21/1999EP0565553B1 6,7-MODIFIED 11$g(b)-ARYL-4-ESTRENES
07/20/1999US5925774 Estrenes for inducing hypothalamic effects
07/20/1999US5925630 Neuroactive steroids of the androstane and pregnane series
07/20/1999US5925628 Drug delivery into cells
07/15/1999WO1999035161A1 Process for preparing carboxamido-4-azasteroids
07/15/1999CA2278487A1 Process for preparing carboxamido-4-azasteroids
07/14/1999EP0928609A2 Use of sulphamate derivatives as steroid sulphatase inhibitors
07/14/1999CN1222915A Process for alkylating and smiles rearrangement of hydroxy aromatics
07/13/1999US5922703 Useful for treating congestive heart failure
07/08/1999WO1999033859A2 Novel anti-estrogenic steroids, and associated pharmaceutical compositions and methods of use
07/08/1999WO1999033858A2 Estrone sulfamate inhibitors of estrone sulfatase, and associated pharmaceutical compositions and methods of use
07/08/1999WO1999033855A1 11β-HALOGEN-7α-SUBSTITUTED ESTRATRIENES, METHOD FOR PRODUCING PHARMACEUTICAL PREPARATIONS CONTAINING SAID 11β-HALOGEN-7α-SUBSTITUTED ESTRATRIENES AND USE OF THE SAME FOR PRODUCING MEDICAMENTS
07/08/1999CA2316444A1 11.beta.-halogen-7.alpha.-substituted estratrienes, process for the production of pharmaceutical preparations that contain these 11.beta.-halogen-7.alpha.-substituted estratrienesas well as their use for the production of pharmaceutical agents
07/07/1999CN1222160A Pregnane derivatives with no alpha-17 substitutent, their medicinal use, mfg. method and its intermediaries and related compounds
07/06/1999US5919957 For the preparation of oxoetiocholenic acid
07/01/1999WO1999032127A1 Angiostatic agents and compositions for controlling ocular hypertension
07/01/1999DE19758390A1 New 11beta-halo-7alpha-substituted-estratriene derivatives are useful for treatment e.g. various cancers, anovulatolial infertility, male hair loss, osteoporosis, and contraceptives
1 ... 15 16 17 18 19 20 21 22 23 24 25 26 27 28 29 30 31 32 33 34 35 ... 47