Patents
Patents for C07H 19 - Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro derivatives thereof (20,008)
02/1995
02/15/1995EP0638586A2 Nucleoside derivatives and methods for producing them
02/15/1995EP0638123A1 Bacterial nitroreductase for the reduction of cb 1954 and analogues thereof to a cytotoxic form
02/15/1995EP0638087A1 Modified nucleotides
02/15/1995EP0638082A1 Macrocyclic immunomodulators
02/15/1995EP0638078A1 Avermectin difluoro derivatives
02/15/1995EP0637965A1 Enhanced triple-helix and double-helix formation with oligomers containing modified pyrimidines
02/14/1995CA1334392C Immunosuppressant agent
02/14/1995CA1334391C Immunosuppressant compound
02/09/1995WO1995004278A1 Process for labelling immunoglobulins
02/09/1995WO1995004162A2 Dna sequencing enzymes
02/09/1995WO1995004065A1 Processes and intermediates for phosphorous-containing covalent linkages
02/09/1995CA2168471A1 Dna sequencing enzymes
02/09/1995CA2167671A1 Processes and intermediates for phosphorous-containing covalent linkages
02/08/1995EP0637315A1 Adenosine derivatives having a 2? agonist activity
02/08/1995EP0637314A1 N-acylated 2'-deoxycytidines useful in oligonucleotide synthesis
02/08/1995EP0637244A1 A STRAIN OF $i(STREPTOMYCES AVERMITILIS) GLYCOSYLATES AVERMECTIN COMPOUNDS
02/07/1995US5387677 Forming guanidine salt, acidifying to recover free AZT
02/07/1995US5387578 Releasing drugs from bioactive agents in order to improve the therapeutic efficacy and reduce their toxic effects
02/07/1995US5387509 Antiparasitic agents
02/02/1995WO1995003317A1 Antiparasitic agents
02/01/1995EP0636372A1 Antiviral, antitumor, antimetastatic, immune system enhancing 7-thia-guanosine derivatives
02/01/1995EP0636022A1 Chemical prevention or reversal of cataract by phase separation inhibitors
02/01/1995EP0599987A4 Method for lowering blood lipid levels.
01/1995
01/31/1995US5386023 Backbone modified oligonucleotide analogs and preparation thereof through reductive coupling
01/31/1995CA1334166C Antiviral preparation containing dideoxy-nucleosides
01/26/1995WO1995002604A1 A3 adenosine receptor agonists
01/26/1995WO1995002422A1 Method for conjugating nucleotides and nucleosides to disulfide-, maleimide-, and thiol-containing compounds
01/25/1995EP0635517A1 Process for Producing 1-(2'-deoxy-beta-D-erythropentofuranosyl)-5-trifluoromethyluracil Derivatives
01/24/1995US5384396 Reaction with carbon disulfide and 3-halopropionitrile or 2-nitroethylhalide, intermediates for AZT
01/24/1995US5384316 4,16-diazatetracyclo[23.3.1.1.Hu 14,17=b . 0 Hu 4,9 triaconta-16,19-diene-2,3,10-trione derivatives
01/24/1995US5384310 2'-fluoro-2-haloarabinoadinosines and their pharmaceutical compositions
01/19/1995WO1995001986A1 Dideoxyfructonucleotides and deoxyfructonucleotides as dna polymerase substrates
01/18/1995EP0549686A4 Modified internucleoside linkages
01/12/1995WO1995001363A1 Methylphosphonic acid ester, process for preparing the same and its use
01/12/1995WO1995001362A1 Liponucleotides of desoxynucleosides, their preaparation and their use as anti-viral drugs
01/12/1995CA2165979A1 Liponucleotides of deoxynucleosides, the production thereof and their use as antiviral pharmaceutical agents
01/11/1995EP0632725A1 Alkylthio alkyl avermectins are active antiparasitic agents
01/11/1995CN1027373C Therapeutic nucleosides
01/10/1995US5380835 Chemically phosphorylating the 5'-hydroxyl terminus of an oligonucleotide
01/10/1995US5380825 AZT immunoassays, derivatives, conjugates and antibodies
01/10/1995US5380715 Ap4 A as a hypotensive agent
01/03/1995US5378825 Backbone modified oligonucleotide analogs
01/03/1995US5378696 Immunosuppressants, transplant rejection, autoimmune diseases, antitumor agents, antiinflammatory agents, fungicides
01/03/1995US5378693 Antitumor agents or viricides
01/03/1995US5378617 Process for the production of macrolide compounds
12/1994
12/28/1994EP0630905A1 Process for selectively isolating bêta-2'-deoxy-2',2'-difluorocytidine or its salts
12/28/1994EP0630898A1 Thrombocytopenia remedy
12/28/1994EP0630379A1 Cyclic ketal derivatives
12/28/1994EP0630378A1 Cyclic ketal derivatives
12/28/1994EP0378706B1 5-substituted uridine derivatives and intermediates for their preparation
12/27/1994US5376663 Immunosuppressive agents; e.g. 1,14-Dihydroxy-12-[2-(4-hydroxy-3-methoxycyclohexyl)-1-methylvinyl]-23,25-dimethoxy-13,19,21,27-tetramethyl-17-(2-oxopropyl)-11,28,-dioxa-4-azatricyclo(22.3.1.04,9)octacos-18-ene-2,3,10,16-tetraone
12/27/1994US5376644 Viricides
12/27/1994US5376642 Treatment of retroviral induced dementia by administration of 2',3'-dideoxyinosine
12/27/1994EP0638087A4 Modified nucleotides.
12/22/1994WO1994029331A1 Nicotinamide ribonucleotide isosters, isosteric nad analogues. their syntheses and use in treatments of alcoholism and neoplastic diseases
12/22/1994WO1994029328A1 Antiparasitic agents
12/22/1994WO1994029312A1 O6-substituted guanine derivatives, a process for their preparation and their use in treating tumour cells
12/22/1994WO1994029279A1 Method for palladium catalyzed carbon-carbon coupling and products
12/22/1994WO1994028910A1 Immunomodulatory, anti-inflammatory, and anti-proliferative compounds: 5,6-dideoxy, 5-amino derivatives of idose and 6-deoxy, 6-amino derivatives of glucose
12/22/1994WO1994017089A3 Method for localising and measuring the proliferation of cancer and compositions for same
12/22/1994CA2164935A1 Method for palladium catalyzed carbon-carbon coupling and products
12/22/1994CA2164827A1 Immunomodulatory, anti-inflammatory, and anti-proliferative compounds: 5,6-dideoxy, 5-amino derivatives of idose and 6-deoxy, 6-amino derivatives of glucose
12/22/1994CA2163447A1 Antiparasitic agents
12/21/1994EP0629633A2 Dinucleotide analogues, intermediates therefor and oligonucleotides derived therefrom
12/21/1994EP0629208A1 Fluorosugar derivatives of macrolides
12/21/1994EP0629203A1 Desosamino derivatives of macrolides as immunosuppressants and antifungal agents
12/21/1994EP0629202A1 Antiparasitic avermectin and milbemycin derivatives.
12/21/1994EP0309560B1 Nucleosides and nucleoside analogues, pharmaceutical composition and processes for the preparation of the compounds
12/20/1994US5374655 Methods for the synthesis of monofucosylated oligosaccharides terminating in di-N-acetyllactosaminyl structures
12/20/1994US5374626 Administering nucleosides for treatment of RNA viruses
12/20/1994CA1333601C Macrolide compounds
12/20/1994CA1333600C Process for the preparation of macrolide compounds
12/20/1994CA1333599C Macrolide compounds
12/14/1994EP0628568A2 Method for the immobilisation of nucleic acids
12/14/1994EP0628567A1 Nicotine derivative
12/14/1994EP0628051A1 Applications of fluorescent n-nucleosides and fluorescent structural analogs of n-nucleosides
12/13/1994US5372816 Trehalostatin and process for the preparation thereof
12/08/1994WO1994027982A1 Use of indolocarbazole derivatives to treat a pathological condition of the prostate
12/08/1994WO1994027616A1 L-2',3'-dideoxy nucleoside analogs as anti-hepatitis b (hbv) and anti-hiv agents
12/07/1994EP0626970A1 Dihydropyrimidine nucleosides with antiviral properties
12/07/1994EP0626853A1 Use of substituted adenine derivatives for treating multiple sclerosis
12/07/1994EP0280741B1 Mitomycin derivatives
12/06/1994US5371210 Stereoselective fusion glycosylation process for preparing 2'-deoxy-2',2'-difluoronucleosides and 2'-deoxy-2'-fluoronucleosides
12/06/1994US5371203 Reacting a triester of L-fucose with trichloroacetonitrile to form corresponding trichloroacetimidate, followed by phosphating,hydrogenolysis, deprotecting, salt formation; a substrate for fucosyltransferases; tumor diagnosis
12/06/1994CA2125129A1 Dinucleotide analogues, intermediates therefor and oligonucleotides derived therefrom
12/06/1994CA1333392C Antiviral compounds
12/06/1994CA1333391C Therapeutic nucleosides
12/06/1994CA1333390C Fluorinated nucleosides and process for treating retrovirus infections therewith
12/06/1994CA1333361C Antiviral compounds
11/1994
11/30/1994EP0626387A1 Nucleosides and oligonucleotides with 2'-ether groups
11/30/1994EP0626385A1 Tetrahydropyran derivatives
11/30/1994EP0625985A1 Method and ring-opened purine compounds for labeling polynucleotides.
11/30/1994EP0427799B1 Method and compounds for aica riboside delivery and for lowering blood glucose
11/24/1994WO1994026764A1 Triester phosphorothioate oligonucleotides and method of preparation
11/24/1994WO1994026763A1 Purification of fluoronucleosides
11/24/1994WO1994026762A1 Preparation of fluoro-nucleosides and intermediates for use therein
11/24/1994WO1994026761A1 Treatment of chemotherapeutic agent and antiviral agent toxicity with acylated pyrimidine nucleosides
11/24/1994WO1994026280A1 Remedy for arthritis containing uridine as active ingredient
11/24/1994WO1994016101A3 Dna sequencing by mass spectrometry
11/24/1994CA2162684A1 Triester phosphorothioate oligonucleotides and method of preparation