Patents
Patents for C07D 521 - Heterocyclic compounds containing unspecified hetero rings (16,203)
11/2000
11/22/2000EP1054005A1 Sulfonamide derivatives, process for producing the same and utilization thereof
11/22/2000EP1054004A1 Novel pyrimidine-5-carboxamide derivatives
11/22/2000EP1052992A1 Cyclic amine modulators of chemokine receptor activity
11/21/2000US6150530 Amidation of amine with acid
11/21/2000US6150526 Piperidine derivative having renin inhibiting activity
11/21/2000US6150391 Subtype-selective 5-ht1d receptor agonists having a human 5-ht1d alpha receptor binding affiity; treatment of migraine, cluster headache, chronic paroxysmal hemicrania, vascular headache, tension headache, and pediatric migraine
11/21/2000US6150385 Viricide with activity against cytomegalo virus (cmv), herpes virus including varicella zoster virus, the epstein-barr virus, the herpes simplex virus, and the human herpes virus type 8 (hhv-8)
11/16/2000WO2000034437A3 Inhibitors of prenyl-protein transferase
11/15/2000EP1051415A1 Benzamide derivatives as vasopressin antagonists
11/15/2000EP1051407A1 2,3,4,5-tetrahydro-1h-[1,4]-benzodiazepine-3-hydroxamic acids as matrix metalloproteinase inhibitors
11/15/2000EP1051397A1 Method for preparing an n- (aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound
11/15/2000CN1273584A Imidazolyl-cyclic acetals
11/14/2000US6147083 Novel substituted 1,2-ethanediamine derivatives which antagonize the pharmacological actions of the endogenous neuropeptide tachykinins known as neurokinins, useful for the treatment of asthma, etc.
11/09/2000WO2000066580A2 Antifungal ethers
11/09/2000WO2000066120A1 Novel catechols as antimicrobial agents
11/09/2000WO2000066112A1 Cxcr-4 receptor antagonists - thrombopoietin mimetics
11/09/2000WO2000039087A3 Substituted (aminoiminomethyl or aminomethyl)benzoheteroaryl compounds as factor xa inhibitors
11/09/2000CA2372079A1 Novel catechols as antimicrobial agents
11/08/2000CN1272842A 2-acylaminopropanamines as tachykinin receptor antagonists
11/08/2000CN1272837A Process for preparation of acylated cyclic 1,3-dicarbonyl compounds
11/07/2000US6143766 Benzopyranone and quinolone inhibitors of ras farnesyl transferase
11/02/2000WO2000064873A1 Renin inhibitors
11/02/2000WO2000064445A1 Bicyclic acyl guanidine sodium/proton exchange inhibitors and method
11/02/2000EP1048641A1 Apoptosis inducer
11/02/2000EP1048640A1 Apoptosis inhibitors
11/02/2000EP1047418A1 Inhibition of raf kinase using substituted heterocyclic ureas
11/02/2000CA2370607A1 Bicyclic acyl guanidine sodium/proton exchange inhibitors and method
11/01/2000CN1058005C Triazole derivant, preparation process and medicine containing its active constituent
11/01/2000CN1058004C Heterocyclo-benzoylguanidin
11/01/2000CN1058001C 4-Mercaptobenzoylguanidine derivatives
10/2000
10/31/2000US6140504 Substituted intermediate compounds for the preparation of n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides
10/31/2000US6140349 Cyclic amine modulators of chemokine receptor activity
10/31/2000US6140347 For treatment of migraine and associated conditions, e.g. cluster headache, chronic paroxysmal hemicrania, headache associated with vascular disorders, tension headache and paediatric migraine
10/31/2000US6140340 Derivatives of 2-[3-phenyl-2-propenyl]-1,2,3,4-tetrahydro isoquinoline, their process and their use as fungicides
10/31/2000US6139596 Nitrification inhibitors and the use of polyacids to treat mineral fertilizers containing a nitrification inhibitor
10/26/2000WO2000063198A1 2,2-disubstituted cyclic ether derivatives and hair tonics containing the same
10/26/2000WO2000063183A1 Process for the preparation of substituted pyrimidines
10/26/2000WO2000063171A1 Tricyclic compounds
10/26/2000CA2370285A1 Process for the preparation of substituted pyrimidines
10/25/2000EP0842159B1 Method of prepararing sulphonyl ureas with herbicidal properties and n-pyrimidinyl or n-triazinyl carbamates as intermediates in the reaction
10/24/2000US6136826 Aminopiperidine compounds substituted with alkanoyl
10/19/2000WO2000041505A3 Anthranilic acid derivatives
10/18/2000EP1044193A1 Process for preparing triazole antimycotic compounds
10/18/2000EP1044192A1 Process for preparing triazole compounds
10/17/2000US6133485 Asymmetric synthesis of 2-(2,4-difluorophenyl)-1-heterocycl-1-yl butan-2,3-diols
10/17/2000US6133443 Optically active 1,4-dihydropyridine derivatives and process for the preparation thereof
10/17/2000US6133303 Various indene derivatives, with the exception of 5-(2-imidazole-1-yl-ethoxy)indan-1-one; treating cancer and treating or preventing restenosis or atherosclerosis
10/17/2000CA2114300C Quinoline or quinazoline derivatives, their production and use
10/12/2000WO2000059901A1 Substituted 1,4-dihydroindeno[1,2-c]pyrazoles as inhibitors of tyrosine kinase
10/12/2000WO2000059880A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
10/12/2000WO2000059510A1 Aminopyrimidines as sorbitol dehydrogenase inhibitors
10/12/2000CA2368686A1 Substituted 1,4-dihydroindeno[1,2-c]pyrazoles as inhibitors of tyrosine kinase
10/12/2000CA2366858A1 Sorbitol dehydrogenase inhibitors
10/11/2000EP1043314A1 Novel dihydropyridine derivative
10/11/2000EP1043312A1 Heterocyclic compounds having nos inhibitory activities
10/11/2000EP1042306A1 Thiazole-, isothiazole- and thiadiazole-derivatives having microbicidal and plant immunizing activities
10/11/2000EP1042290A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
10/11/2000EP1041980A1 Acyl guanidine sodium/proton exchange inhibitors and method
10/11/2000CN1269794A 6,7-asymmetrically disubstituted quinoxalinecarboxylic acid derivatives, addition salts thereof and process for preparation of both
10/11/2000CN1269362A 1,4-dichloropyridine-3,5-carboxylic-acid derivatives and preparation method thereof
10/11/2000CN1269359A Antimer pure acetacetates, its preparation method and use
10/11/2000CN1269358A Amino-butenate compound and preparation method thereof
10/11/2000CN1269357A Benzal compound and preparation method
10/05/2000DE19903064A1 New ammonium salt derivatives of sulfonyl urea compounds, useful as herbicides or plant growth regulators providing stable formulations, especially emulsifiable concentrates
10/04/2000EP1041064A2 N-substituted alpha aminoacid amides as calcium channel modulators
10/04/2000EP1040103A1 Anilide derivative, production and use thereof
10/04/2000EP1040101A1 Substituted 2-aryl-4-amino-chinazolines, method for the production and use thereof as medicaments
10/04/2000EP1040094A1 Substituted cyclopentane and cyclopentene compounds useful as neuraminidase inhibitors
10/04/2000EP0766672B1 Arylsulfonamido-substituted hydroxamic acids as matrix metalloproteinase inhibitors
10/04/2000EP0569384B2 Fungicides
10/04/2000CN1057089C Process for preparing intermediates for synthesis of antifungal agents
10/04/2000CN1057088C Benzimidazole, prepn. method and use thereof
10/04/2000CN1057086C Phenylsulfonyl ureas, process for preparing same, and use as herbicide, herbicide composition contg. same
10/04/2000CN1056958C Pesticide composition and use thereof
10/03/2000US6127548 Preparing optionally substitued 3h-imidazole-4-carbaldehyde by protecting the 3-amino group, then formylating in presence of an organometallic compound and electrophile with formyl leaving group, deprotecting with acid or strong base
10/03/2000US6127403 An enzyme inhibitor for treating arteriosclerotic lesions of arteriosclerosis, hyperlipemia and diabetes, as well as ischemic diseases of brain, heart
10/03/2000US6127372 Sulfonamide inhibitors of aspartyl protease
09/2000
09/28/2000WO2000056726A1 Improved aqueous solubility pharmaceutical formulations
09/28/2000WO2000056718A1 Imidazole compounds
09/28/2000WO2000033839B1 Non-peptide antagonists of glp-1 receptor and methods of use
09/28/2000DE19913475A1 Use of non-volatile new and known 2-chloro-1-azolyl-ethanol compounds, as nitrification inhibitors in fertilizers
09/27/2000EP1037880A1 Retinoic acid mimetic anilides
09/27/2000EP1037878A2 Metabotropic glutamate receptor antagonists for treating central nervous system diseases
09/27/2000CN1056835C Novel selective aromatase inhibiting compounds
09/26/2000US6124416 A copolymer consisting of a monomer containing at least one isocyanate functional group and an unsaturation; useful for coating
09/26/2000US6124332 Metalloproteinase inhibitors
09/26/2000US6124330 N-[4-(Heteroarylmethyl)phenyl]-heteroarylamines
09/26/2000US6124329 Metalloproteinase inhibitors
09/26/2000US6124325 Triazole antifungal agents
09/26/2000US6124243 Method of controlling graminaceous weeds
09/21/2000WO2000055155A2 Heterocyclic compounds as adenosine deaminase inhibitors
09/21/2000WO2000055152A1 Aromatic heterocyclic compounds as anti-inflammatory agents
09/21/2000WO2000032577A3 Substituted benzo[de]isoquinoline-1,3-diones
09/21/2000DE19912690A1 New benzimidazolyl amidine or nitrile compounds, useful as thrombin inhibitors or antithrombotic agents, for treating deep leg vein thrombosis
09/20/2000EP1036058A1 Adamantane derivatives
09/20/2000EP0696288B1 Quinoxalindione derivatives, their preparation and their use in drugs
09/19/2000US6121264 Glutamate receptor antagonist, ampa receptor antagonist, nmda-glycine receptor antagonist, kainic acid neurotoxicity inhibitor, antiischemic agent, psychotropic agent
09/19/2000CA2022133C Monoclinic metazachlor and its preparation
09/14/2000WO2000053591A1 Thiazolyl urea derivatives and their utilization as antiviral agents
09/14/2000WO2000053583A1 Inhibitors of protein tyrosine phosphatase
1 ... 46 47 48 49 50 51 52 53 54 55 56 57 58 59 60 61 62 63 64 65 66 ... 163