Patents for C07D 521 - Heterocyclic compounds containing unspecified hetero rings (16,203) |
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10/26/2005 | EP1589006A1 Oxa- and thiazole derivatives useful as antidiabetics and antidiobesity agents |
10/26/2005 | EP1307431B1 Efficient ligand-mediated ullmann coupling of anilines and azoles |
10/26/2005 | EP1163234B1 Pharmaceutical formulations with improved aqueous solubility |
10/26/2005 | CN1688573A Pyrrole based inhibitors of glycogen synthase kinase 3 |
10/26/2005 | CN1224598C Naphthalene derivatives |
10/25/2005 | US6958353 Imidazole derivatives or salts thereof and drugs containing the derivatives or the salts |
10/25/2005 | US6958348 Side effect reduction |
10/25/2005 | US6958339 Pyrazole derivative |
10/25/2005 | US6958337 Crystalline antifungal polymorph |
10/25/2005 | CA2147056C Novel delta-amino-gamma-hydroxy-omega-aryl-alkanoic acid amides |
10/25/2005 | CA2059882C Sulfonylureas |
10/20/2005 | US20050234106 1-aryl-1-heteroarylaminoalkylene-substituted, e.g., 1-[fluorophenylcyclohexylmethyl]isoquinolin-1-ylamine; antiarrhythmia agents; cardiovascular disorders |
10/20/2005 | US20050234061 N-[3-(4-chlorophenyl)-2-(3-pyridyl)-1-methylpropyl]-2-(5-trifluoromethyl-2-pyridyloxy)-2-methylpropanamide; obesity; antipsychotic agents; synergistic; cannabinoid receptor antagonists |
10/20/2005 | US20050234055 Pyrazole derivative |
10/19/2005 | EP1585744A1 Process for making ondansetron and intermediates thereof |
10/19/2005 | EP1337523B1 2,4-substituted pyridine derivatives |
10/19/2005 | EP0966446B1 Bicyclic inhibitors of protein farnesyl transferase |
10/19/2005 | CN1682702A Method for preparing medicine composition capable of inhibiting post infective virus proteinase |
10/19/2005 | CN1223564C Intermediate halo phenyl derivatives and their use in process for preparing pyrrole derivatives |
10/18/2005 | US6956050 Imidazole compounds as anti-inflammatory and analgesic agents |
10/18/2005 | US6956037 Benzamide derivatives for the treatment of diseases mediated by cytokines |
10/18/2005 | CA2307581C Heterocyclic compounds having nos inhibiting action |
10/13/2005 | US20050228029 sulfonylurea derivatives, sulfonylthiourea derivatives, sulfonylguanidine derivatives, sulfonylcyanoguanidine derivatives, thioacylsulfonamide derivatives, and acylsulfonamide derivatives; effective for prevention and treatment of cardiovascular diseases, particularly those diseases related to thrombosis |
10/13/2005 | US20050228020 Beta secretase inhibitors |
10/13/2005 | US20050227979 E.g., 1-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-piperidine and 1-[4-(1-Isopropyl-piperidin-4-yloxy)-benzyl]-azepane; these compounds modulate the activity of the histamine receptor, specifically the H3 receptor, without the inherent problems associated with the presence of an imidazolyl moiety |
10/13/2005 | US20050226844 Valency platform molecules comprising carbamate linkages |
10/12/2005 | EP1583742A1 Novel cb 1 receptour inverse agonists |
10/12/2005 | CN1681788A COX-2 inhibiting pyridine derivatives |
10/12/2005 | CN1681763A Chemical compounds |
10/11/2005 | US6953807 4-substituted-picolinic acid amide derivatives useful as fungicides |
10/11/2005 | US6953806 Cyclohexane derivatives containing amine or amine oxide, useful for treating hypercholesterolemia and hyperlipemia |
10/06/2005 | WO2004072031A8 Phenylacetamides and their use as glucokinase modulators |
10/06/2005 | US20050222426 A compound selected from the group consisting of 1,2,3-benzotriazol-2-yl-L-alanine, 5-carboxy-1,2,3-benzotriazol-2-yl-L-alanine, and 5-carboxy-1,2,3-benzotriazol-1-yl-L-alanine. |
10/06/2005 | US20050222411 Method for the production of monohydro-perfluoroalkanes, bis (perfluoroalkyl) phosphinates and perfluoroalkylphosphonates |
10/06/2005 | US20050222226 N-[3-(2-Aminoethyl)-4-(4-bromophenyl)thiazol-2(3H)-ylidene]aniline; antiinflammatory agents, antiallergens; inhibit infiltration of leukocytes such as eosinophils and lymphocytes; autoimmune diseases, asthma |
10/05/2005 | EP0775110B1 Arylthio compounds as antibacterial and antiviral agents |
10/05/2005 | CN1678576A Pyrrolidine derivatives as oxytocin antagonists |
10/05/2005 | CN1221529C Substituted N-[(aminoiminomethyl or aminomethyl) phenyl] propyl amides |
10/05/2005 | CN1221524C Diphenyl ether compounds useful in therapy |
10/04/2005 | US6951886 Succinoylamino hydroxyethylamino sulfonyl urea derivatives useful as retroviral protease inhibitors |
10/04/2005 | US6951879 Heteroaromate OSC inhibitors |
10/04/2005 | US6951574 Primary intermediates for oxidative coloration of hair |
09/29/2005 | WO2005046688A3 Methods of use of thrombin receptor antagonists |
09/29/2005 | US20050215794 Group IB compounds used as condensation, amination, amidation or arylation catalysts; catalysis; efficiency; forming a carbon-carbon bond between a reactant comprising a nucleophilic carbon atom, e.g., enolate or malonate anion, and activated carbon of an aryl, heteroaryl, or vinyl halide or sulfonate |
09/28/2005 | EP1233936B1 Process for preparing ambient temperature ionic liquids |
09/28/2005 | CN1675201A N-substituted piperidine derivatives as serotonin receptor agents |
09/28/2005 | CN1674892A Hetero biaryl derivatives as matrix metalloproteinase inhibitors |
09/28/2005 | CN1220684C 2, 4, Di(hetero-)arylamino(-oxy)-5-substituted pyrimidines as antineoplastic agents |
09/28/2005 | CN1220683C Acyl derivatives for treating VLA-4 related disorders |
09/22/2005 | US20050209466 Reproducible; avoids use of 3-pyrrolidinol as a starting material |
09/22/2005 | US20050209291 Amino benzothiazole compounds with NOS inhibitory activity |
09/21/2005 | EP1575925A1 Novel carboxamides, the production and use thereof as medicaments |
09/21/2005 | CN1671717A Azole derivatives as antifungal agents |
09/21/2005 | CN1671670A Novel imidazole alcohol compound, process for producing the same, and surface-treating agent comprising the same |
09/21/2005 | CN1671667A Quinoline derivatives and their use as mycobacterial inhibitors |
09/21/2005 | CN1671386A Substituted anilinic piperidines as MCH selective antagonists |
09/20/2005 | US6946579 3-carbocycle carbonyl-3-phenylpropionaldehyde intermediates and preparation by alkylating a carbocycle benzyl ketone with an allyl halide and oxidizing the product |
09/20/2005 | US6946467 Serine protease inhibitors |
09/20/2005 | US6946460 such as cis-4-[[2-(2,4-dichlorophenyl)-2-(1H-imidazol-1-ylmethyl)-1,3-dioxolan-4-yl]methoxy]-N-methyl-N-(3-phenyl-2(E)-propenyl)-benzenemethanamine; |
09/20/2005 | US6946005 Pyrrolidinyl-substituted para-phenylenediamine derivatives substituted with a cationic radical, and use of these derivatives for dyeing keratin fibers |
09/15/2005 | US20050203093 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4 |
09/14/2005 | EP1572694A1 Pyrrolo'2,1-c!'1,4! benzodiazepines as vasopressin agonists |
09/14/2005 | EP1409440A4 A method to inhibit ethylene responses in plants |
09/14/2005 | CN1668593A Heterocyclically substituted benzoylureas, process for their preparation and their use as pharmaceuticals |
09/13/2005 | US6943183 Antiproliferative agnets; anticancer agents; skin disorders; restenosis |
09/13/2005 | US6943161 For prophylaxis and therapy of inflammation, asthma, arthritis, diabetes, atherosclerosis, ocular diseases, restenosis, autoimmune responses, multiple sclerosis, psoriasis, human cancers, fibrosis of liver, lung and kidney |
09/13/2005 | US6942966 Methods for processing chemical compounds having reactive functional groups |
09/13/2005 | CA2231105C Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives |
09/13/2005 | CA2078700C Imidazolylmethyl-pyridines |
09/07/2005 | EP1569921A1 Ionic liquids comprising n(cf sb 3 /sb ) sb 2 /sb ] sp - /sp anions |
09/07/2005 | EP1347957B1 Delta 1-pyrrolines used as pesticides |
09/07/2005 | CN1665788A Pyrimidinone compounds, compositions and methods |
09/07/2005 | CN1217933C Dihalopropene compound, insecticide/miticide containing the same and intermediate for producing the same |
09/07/2005 | CN1217928C Heterocyclic compounds having NOS inhibitory activities |
09/06/2005 | US6939974 Heating an imidazolium halide with a strong base under reduced pressure and separating the resultant products |
09/06/2005 | US6939967 Non-proteinogenic L-amino acids |
09/06/2005 | US6939875 Carbocyclic oxy sulfides such as [4-(Biphenyl-4-ylmethylsulfanyl)-5-methoxy-2-methyl-phenoxy]-acetic acid, used to control peroxisome proliferator activated receptors (PPAR), for prophylaxis of metabolic disorders |
09/01/2005 | WO2004054991A8 Ionic liquids comprising [n(cf3)2]- anions |
09/01/2005 | US20050192277 Histamine-3 receptor antagonists; 4-(2-{2-[(2R)-2-methyl-1-pyrrolidinyl]ethyl}-1-benzofuran-4-yl)benzonitrile; acute myocardial infarction, asthma, psychological disorders, gastrointestinal disorders, inflammation, jet lag, cancer, septic shock, Tourette's syndrome, neurodegenerative disorders |
08/31/2005 | EP1567498A2 Mandelic acid derivatives |
08/31/2005 | EP1278723B1 P-(sulfonyl)-aryl and -heteroaryl amines |
08/31/2005 | EP1268445B1 4-amino-5-cyano-2-anilino-pyrimidine derivatives and their use as inhibitors of cell-cycle kinases |
08/31/2005 | EP1140809B1 New biphenyl and biphenyl-analogous compounds as integrin antagonists |
08/31/2005 | CN1662525A Preparation for the production of 1, 2, 4-triazolymethyl-oxiranes |
08/31/2005 | CN1662518A Processes for producing epoxytriazole derivative and intermediate therefor |
08/31/2005 | CN1660798A Processes for preparing aminophenylsulfonylureas, and intermediates therefor |
08/30/2005 | US6936719 pyridine ring containing biaryl compound useful to treat and/or prevent clotting disorders, and as antiinflammatory and anticoagulant agents |
08/30/2005 | US6936626 Retinoic acid mimetic anilides |
08/30/2005 | US6936613 for treatment of central nervous system diseases and disorders, which are responsive to modulation of the Gamma amminobutyric acid (GABA) receptor complex, and for inducing and maintaining anesthesia, sedation and muscle relaxation |
08/30/2005 | US6936611 Serine protease inhibitors |
08/30/2005 | US6936600 Oxidoreductase enzyme inhibitors such as (R)-1-[4-(2-methyl-4-phenyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-pyrimidin-2-yl-ethanol, used as antidiabetic agents |
08/24/2005 | EP1334085B1 Sulfamides as gamma-secretase inhibitors |
08/24/2005 | EP1292190B1 N-phenyl-4-(4-pyridyl)-2-pyrimidineamine derivatives |
08/24/2005 | CN1216054C 1,4-dihydro pyridine-3,5-carboxylic-acid derivatives and preparation method thereof |
08/23/2005 | US6933311 Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor |
08/23/2005 | US6933295 Substituted isoindoles and the use thereof |
08/23/2005 | CA2370888C Renin inhibitors |
08/18/2005 | WO2005075422A1 Synthesis methods and intermediates for the manufacture of rizatriptan |
08/18/2005 | US20050182050 Therapeutic heterocyclic compounds |
08/18/2005 | CA2553652A1 Synthesis methods and intermediates for the manufacture of rizatriptan |