Patents
Patents for C07D 519 - Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups or (11,041)
01/1995
01/25/1995CN1097743A 9H-imidazo|1,2-a¨benzimidazole-3-acetamide derivative and preparation and pharmaceuctical application of same
01/18/1995EP0633886A1 Pharmaceutically active bicyclic-heterocyclic amines
01/18/1995CN1097423A Quinolone- and naphthyridonecarboxylic acid derivatives
01/10/1995US5380746 Bis-(1H-indol-3-YL)-maleinimide derivatives, processes for the preparation thereof and pharmaceutical compositions containing them
01/04/1995EP0632040A1 Antibacterial imidazole derivatives
01/04/1995CN1027266C Process for synthesis of dimer alkaloid compounds
01/03/1995US5378697 Cephalosporins
01/03/1995US5378276 Diketopyrrolopyrroles containing nitroxyl groups
01/03/1995CA2127318A1 Imidazole compounds and use thereof
01/03/1995CA1333809C Phenolic thiane derivatives
12/1994
12/28/1994EP0630895A1 4-Bicyclic substituted dihydropyridines, process for their preparation and their use in medicaments
12/28/1994EP0630376A1 Condensed indole derivatives as 5ht 4?-receptor antagonists
12/28/1994CN1027165C 7-(1-pyrrolidiny 1)-3-quinolone- and -naphthyridone-carboxylic acid derivatives, processes for their preparation and substituted mono- and bicyclic pyrrolidine derivatives as intermediate products....
12/27/1994US5376661 Psychological disorders
12/25/1994CA2126397A1 4-bicyclically substituted dihydropyridines, processes for their preparation and their use in medicaments
12/22/1994WO1994029321A1 Novel cephem compounds
12/14/1994EP0628562A1 Cephalospornis having in position 7 as substituted axymino radical, intermediates, processes for their preparation and their use as medicaments
12/14/1994CN1096298A New cephalosporins containing a substituted oxyimino radical in position 7, their preparation process and intermediates and their use as medicaments
12/11/1994CA2111164A1 Cephatosporins containing a 7-substituted oxyimino radic al, their preparation process and intermediates and their use as drugs
12/08/1994WO1994028002A1 36-derivatives of rifamycins and their use as antimicrobial agents
12/06/1994US5371199 Substituted porphyrins, porphyrin-containing polymers, and synthetic methods therefor
12/06/1994US5371090 Bactericides, feed additives
11/1994
11/29/1994US5369108 Potent inducers of terminal differentiation and methods of use thereof
11/23/1994EP0429464B1 Bivalent ligands effective for blocking acat enzyme
11/22/1994US5366970 Cephem compounds and pharmaceutically acceptable salts thereof
11/17/1994EP0624580A1 Styrylcoumarin compound, photosensitive resin composition, and hologram recording medium
11/16/1994CN1095068A Bicyclic amine derivatives
11/16/1994CN1026588C Novel 1-alkyl substituted benzimidazole derivatives
11/15/1994US5364855 Cardiovascular disorders or antiarrthmia agents
11/15/1994US5364854 Nervous system and gastrointestinal disorders; antiemetic, anxiolytic, and analgesic agents; cognition activators; drug abuse
11/10/1994WO1994025504A1 Tetraaroxyperylene-3,4,9,10-tetracarboxylic acid polyimides
11/10/1994WO1994025468A1 Biotin esters of rapamycin
11/10/1994WO1994025464A1 Novel quinolone carboxylic acid derivatives and process for preparing the same
11/09/1994EP0623618A2 Pyrrolo-pyridine derivatives
11/09/1994EP0623020A1 Pyropheophorbides and their use in photodynamic therapy
11/08/1994US5362722 Cephalosporin antibacterial agents
11/02/1994EP0622367A1 Novel quinolone carboxylic acid derivatives and process for preparing the same
11/02/1994EP0622365A1 2-Amino-4-heteroaryl-1,4-dihydropyridines, method for their preparation and their use in drugs
11/02/1994CN1094405A Novel quinolone carboxylic acid derivatives and process for preparing the same
11/01/1994US5360807 Substituted thiazolyl and substituted pyridinyl derivatives
10/1994
10/28/1994CA2121963A1 2-amino-4-heteroaryl-1,4- dihydropyridines, processes for their preparation and their use in medicaments
10/26/1994CN1094050A Novel heterocyclic compounds with antiasthmatic/anti-auergie, anti-inflammatory positive inotropic and blood pressure-reducing effect
10/25/1994US5359066 Certain tricyclic pyrido[3,2,1-ij]cinnoline-8-carboxylates, useful as antimicrobial agents
10/25/1994US5358953 Imidazopyridine PAF/H1 antagonists
10/19/1994EP0619821A1 HEXAHYDROFURO(2,3-b)FURANS AS PAF ANTAGONISTS
10/18/1994US5356888 1,1-dioxo-cephem-4-carbothiolic acid derivatives
10/13/1994WO1994022863A1 Second messenger cell signaling inhibitors
10/12/1994EP0425566B1 New photosensitizing agents
10/11/1994US5354766 2-Ethoxy-1-((2'(2,5-dihydro-5-oxo-1,2,4-oxadiazol-3-yl) biphenyl-4-yl)methyl)benzimidazole-7-carboxylic acid; hypotensive agents; CNS activity
10/05/1994CN1026115C Novel S-adenosyl methionine inhibitors
10/04/1994US5352685 Gastrointestinal disorders
09/1994
09/28/1994EP0340243B1 Cc-1065 analogs
09/28/1994CN1092776A 2-(9-fluorenonyl)-carbapenem intermediates
09/28/1994CN1092775A Pharmaceuticals
09/21/1994EP0615977A1 Spiro piperidines and homologs which promote release of growth hormone
09/20/1994US5348952 Antibiotics for antiinflammatory agents, degenerative diseases caused by proteolytic enzymes and respiratory system disorders
09/15/1994WO1994020497A1 Pyrrolo-pyridine derivatives
09/14/1994EP0614664A1 Quinolonecarboxylic acid derivatives, their preparation and their use as cell adhesion inhibitors
09/14/1994CN1092071A Spiro piperidines and homologs which promote release of growth hormone
09/14/1994CN1092069A Novel quinolone derivatives and processes for preparing the same
09/10/1994CA2117224A1 Quinolonecarboxylic acid derivatives, their production and use
09/07/1994CN1025855C Process and intermediates for the preparation of oxophthalazinyl acetic acids and analogs thereof
09/02/1994CA2116213A1 Pyrrolo-pyridine derivatives
09/01/1994WO1994019367A1 Spiro piperidines and homologs promote release of growth hormone
08/1994
08/31/1994EP0612752A1 Organic charge transfer complex
08/31/1994EP0612751A2 Compounds for the preparation of cephem derivatives
08/31/1994EP0612747A2 Nitroxyl groups-containing diketopyrrolopyrroles
08/31/1994EP0505413B1 Beta-lactam derivatives
08/24/1994CA2116064A1 Diketopyrrolopyrroles containing nitroxyl groups
08/23/1994US5340814 Hypotensive agents
08/10/1994EP0609278A1 Imidazopyridines and indolizines as 5-ht 4 antagonists
08/09/1994US5336768 Bactericides
08/09/1994US5336674 2-phenanthridinyl carbaphenem antibacterial agent
08/09/1994CA1331381C Antibacterial agents - ii
08/04/1994WO1994017066A1 2-phenanthridinyl carbapenem antibacterial agents
08/04/1994CA2154276A1 2-phenanthridinyl carbapenem antibacterial agents
08/03/1994EP0572425B1 Imidazopyridine paf/h 1 antagonists
08/03/1994CN1090285A Quinolonecarboxylic acids
08/02/1994US5334385 New alkaloid derivatives, their use and pharmaceutical formulations containing them
07/1994
07/27/1994EP0607825A1 6-H-4-OXO-3-quinoline-carboxylic acids and their analogues as antibacterial agents
07/27/1994EP0607233A1 3,9-diazabicyclo(3.3.1)nonane derivatives with 5-ht3 receptor antagonist activity
07/26/1994US5332837 CC-1065 analogs
07/21/1994WO1994015938A1 Novel quinolone derivatives and processes for preparing the same
07/20/1994EP0607076A1 9H-Imidazo 1,2-a benzimidazole derivatives with GABA activity
07/20/1994EP0606421A1 Derivatives of imidazo 5,1-c] 1, 4]benzoxazin-1-one as 5 ht3 antagonists
07/20/1994CN1089611A Optical active isoindolinone derivatives, their production and use
07/20/1994CA2113513A1 Quinolone- und naphthyridonecarboxylic acid derivatives
07/19/1994CA1330798C Benzo- and thieno-3,4-dihydro-pyridine derivatives
07/16/1994CA2113490A1 9h-imidazo[1,2-a]benzimidazole-3-acetamide derivatives, their preparation and their therapeutic application
07/13/1994EP0605836A1 Cephalosporin derivatives
07/13/1994CN1089267A Chemical compounds
07/12/1994US5329002 Antibacterial cephalosporin compounds
07/12/1994US5328908 Antimicrobial quinolone thioureas
07/07/1994WO1994014813A1 Novel quinolone derivatives and processes for preparing the same
07/05/1994US5326874 Process for preparing trans-piperidine-2,5-dicarboxylates
07/05/1994US5326768 5-hydroxytryptamine antagonists
06/1994
06/29/1994EP0603887A2 Bicyclic amine derivatives
06/23/1994WO1994013696A1 Spiro piperidines and homologs which promote release of growth hormone
06/23/1994WO1994013681A1 Antiallergic triazolo(pyrrolo, thieno or furano)azepine derivatives
06/23/1994WO1994013680A1 ANTIALLERGIC IMIDAZO[1,2-a](PYRROLO, THIENO OR FURANO)[2,3-d]AZEPINE DERIVATIVES
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