Patents
Patents for C07D 519 - Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups or (11,041)
12/1986
12/30/1986EP0206667A2 Derivatives of 4-desacetyl indole-dihydroindole alkaloids
12/30/1986EP0206666A2 Hydrazide imide derivative of indole-dihydroindole alkaloids
12/30/1986EP0206415A2 (4-Piperidinylmethyl and -hetero)purines
12/30/1986EP0206270A2 1,3,4-Tri-(het-)arylisoquinolines, process for their preparation and their use as photoconductive compounds
12/17/1986EP0205169A2 Bis-indole derivatives, process for preparing same and pharmaceutical compositions containing them
12/17/1986EP0205168A2 Furfuryl derivatives of vinblastine-type bis-indoles, a process for preparing same and pharmaceutical compositions containing them
12/04/1986WO1986007057A1 Methyl derivatives of methylated bis 7h pyridocarbazoles and farmaceutical compositions containing them
12/03/1986EP0203559A1 Penicillin derivative containing naphthyridine
12/03/1986EP0203271A2 Antibacterial compounds, their production and use
12/03/1986CN86102683A Antibacterial agents
12/02/1986US4626384 Penam derivatives
11/1986
11/26/1986EP0202763A1 5,6-Difluoronaphthyridines and 5,6,8-trifluoro-quinolines as antibacterial agents
11/26/1986EP0202703A1 Pharmaceutical compositions of the prodrug type, a process for the preparation thereof, a process for the preparation of them as prodrug functioning compounds and compounds obtained therein
11/26/1986CN86102987A Carbapenem process
11/19/1986CN85103992A Method of preparing drugs for curing tumors
11/18/1986CA1214164A1 Polycyclic hydrazones, processes for their manufacture, pharmaceutical compositions containing them, and their use
11/12/1986EP0201206A1 Penem derivatives
11/11/1986US4622402 Thienoisothiazole disulfides
11/11/1986US4622324 Cardiovascular disorders, hypotensives
11/05/1986EP0200225A2 An organ culture of catharanthus roseus capable of producing substantial amount of indole alkaloids
11/05/1986CN85109195A Process for the preparation of imidazopyridazine derivatives and their use
11/05/1986CN85108120A Process for the preparation of tricyclische pyridinderivate and their use
11/04/1986CA1213582A1 1,1-alkanediol dicarboxylate linked antibacterial agents
11/04/1986CA1213581A1 Process and intermediates for production of 1,1- dioxopenicillanoyloxymethyl 6-(2-amino-2- phenylacetamido) penicillanates
10/1986
10/29/1986EP0199490A1 Penem derivatives
10/29/1986EP0198921A1 Biologically-active xanthine derivatives
10/28/1986US4619958 Mixed 2,2,6,6-tetramethyl piperidinyl carboxylic acid ester and amide light stabilizers and stabilized synthetic polymers
10/28/1986US4619913 Treatments employing drug-containing matrices for introduction into cellular lesion areas
10/22/1986EP0198190A2 Compounds having antiplatelet aggregation activity, a process for the preparation thereof and pharmaceutical compositions containing them
10/15/1986EP0197409A1 Cephalosporin derivatives
10/14/1986US4617389 Mitomycin analogs
10/14/1986US4617300 2(N-heterocyclyl) penems
10/14/1986US4617261 Process for labeling nucleic acids and hybridization probes
10/09/1986WO1986005787A1 Antibacterial compounds
10/09/1986WO1986005786A1 Cephalosporin derivatives
10/07/1986CA1212378A1 .beta.-LACTAMASE INHIBITING 2-.beta.-SUBSTITUTED-2-.alpha.- METHYL-(5R) PENAM-3-.alpha.-CARBOXYLIC ACID 1,1- DIOXIDES AND INTERMEDIATES THEREFOR
09/1986
09/30/1986CA1212104A1 Process and intermediates for sultamicillin and analogs
09/25/1986WO1986005491A1 Synthesis of vinblastine and vincristine type compounds
09/16/1986US4612315 Biologically-active 1,3-dipropyl-8-phenylxanthine derivatives
09/12/1986WO1986005184A1 Antibacterial compound
09/12/1986WO1986005183A1 Antibacterial compounds, their production and use
09/03/1986EP0192948A1 Cholecystokinin antagonist compounds, process for their preparation and pharmaceutical compositions containing them
09/02/1986US4609731 Bromine complex of 3-bromo-6-chloro-2-methyl-imidazo(1,2-b)pyridazine
09/02/1986US4609657 Ergot peptide alkaloid derivatives, processes for their preparation and pharmaceutical compositions containing them
09/02/1986CA1210762A1 Method of producing vincristine
09/02/1986CA1210696A1 Immunoglobulin conjugates
08/1986
08/28/1986WO1986004898A1 Disulfide compounds and antineoplastic agents
08/27/1986EP0192328A1 Chromogenic compounds
08/26/1986US4608436 Piperidine compounds
08/13/1986EP0190905A2 Radio labeled dihematoporphyrin ether and its use in detecting and treating neoplastic tissue
08/13/1986EP0190709A1 Benzoxazinorifamycin derivative, process for preparing the same and anti-bacterial agent containing the same
08/13/1986EP0190587A1 Soluble quinazolino-1,4-benzodiazepin-5,13-dione derivatives, process for their preparation and pharmaceutical composition containing them
08/13/1986EP0190315A1 Dehydrated liposomes.
08/06/1986EP0189802A1 Quinazolino-1,4-benzodiazepin-5,13-diones, processes for their preparation and pharmaceutical compositions containing them
08/05/1986US4604241 9-desoxo-9-hydroxy-pheophorbide derivatives and alkaline salts thereof
07/1986
07/30/1986CN85108556A Process for preparing novel benzoxazol-and benzothiazolamine derivatives and their use
07/29/1986US4602909 Vinca alkaloids
07/23/1986EP0188377A1 New phthalide derivatives
06/1986
06/24/1986US4596869 Pyridinyl and pyrimidinyl derivatives
06/24/1986US4596676 Bifunctional ester derivatives of 4-desacetyl indole-dihydroindole alkaloids
06/11/1986EP0184257A1 Benzoxazol- and benzothiazolamine derivatives
06/11/1986EP0184162A2 Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
06/11/1986EP0183994A1 Tricyclic pyridone derivatives
06/10/1986US4594421 Imidazopyridine compounds
06/10/1986US4594190 Quaternary salts of dibenzo[1,4]diazepinones, pyrido-[1,4]benzodiazepinones, pyrido[1,5]benzodiazepinones with antiulcer, antisecretory, spasmolytic and antimusarinic activities
06/10/1986CN85109492A Tricyclo compounds, a process for their production and a pharmaceutical composition containing the same
06/10/1986CN85107053A Process for the preparation of metal complexes of bis-indole compounds and agueous pharmaceutical compositions containing them
06/03/1986CA1205465A1 Process for manufacture of cephalosporin derivatives
05/1986
05/28/1986EP0181940A1 Cephalosporin derivatives
05/27/1986US4591459 Beta-lactamase inhibitors, penicillins, cephalosporins, bactericides
05/20/1986CA1204736A1 Process and intermediates for preparation of 1,1- dioxopenicillan-oyloxymethyl 6-beta- aminopenicillanate
05/09/1986WO1986002551A1 Biologically-active xanthine derivatives
04/1986
04/29/1986CA1203797A1 Antibacterial 6'-(2-amino-2-¬4-acyloxyphenyl|- acetamido) penicillanoyloxymethyl penicillanate 1,1- dioxide compounds
04/22/1986US4584372 Compound 3-(1,2,3,6-tetrahydro-1,3-dimethyl-2,6-dioxopurine-7-acetyl-8-(2-phenylethyl)-1-oxa-3,8-diazaspiro-(4,5)decan-2-one and a process of preparation thereof
04/16/1986EP0178089A1 2(N-heterocyclyl)penems
04/15/1986US4582829 Antibacterial 6'-(2-amino-2-[4-acyloxyphenyl]acetamido)penicillanoyloxymethyl penicillanate 1,1-dioxide compounds
04/15/1986US4582789 Containing alkylating intercalation moiety
03/1986
03/25/1986US4578378 (Oxoheterocyclic carbonamido)cephem carboxylic acid derivatives
03/19/1986EP0174858A1 Isoindolinone derivatives, production and use thereof
03/18/1986US4577016 Process for the preparation of penem derivatives
03/12/1986EP0174279A2 Improvements in relation to cyclosporin therapy
03/11/1986CA1201709A1 BIS-ESTERS OF 1,1-ALKANEDIOLS WITH 6-.beta.- HYDROXYMETHYLPENICILLANIC ACID 1,1-DIOXIDE AND .beta. LACTAM ANTIBIOTICS
03/05/1986EP0172919A1 Cephalosporin derivatives, process for their preparation, and their pharmaceutical use
02/1986
02/27/1986WO1986001103A1 Dehydrated liposomes
02/27/1986WO1986001102A1 Encapsulation of antineoplastic agents in liposomes
02/26/1986EP0172651A1 Substituted-9-fluoro-3-methyl-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de][1,4]benzoxazine-6-carboxylic acids; substituted-5-amino-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxylic acids; substituted-5-amino-6-fluoro-1,4-dihydro-4-oxo-1,8-naphthyridine-3-carboxylic acids; derivatives thereof; pharmaceutical compositions comprising the compounds; and processes for producing the compounds
02/18/1986US4571396 Antibacterial agents
02/11/1986US4569997 Polyalkylpiperidine compounds
02/11/1986CA1200545A1 Bis-esters of methanediol with penicillins and penicillanic acid 1, 1-dioxide
02/05/1986EP0170073A1 1-Methylcarbapenems having an externally alkylated mono- or bicyclic 2-quaternary heteroarylalkylthio substituent
01/1986
01/29/1986EP0169410A1 Carbapenems having a 2-quaternary pyridine altylthio or pyridine alkenylthio substituent, compositions containing the same and combinations with DHP inhibitors
01/28/1986CA1199909A1 Bis-esters of dicarboxylic acids with amoxicillin and certain hydroxymethylpenicillanate 1,1-dioxides
01/22/1986EP0168707A1 1-Methylcarbapenems having a 2-quaternary heteroarylalkylthio substituent
01/08/1986EP0167263A1 Drug-containing matrices for introduction into cellular lesion areas
01/08/1986EP0167139A1 Carbapenems having an externally alkylated 2-quaternary pyridiniumalkylthio substituent
01/08/1986EP0167100A1 Penem derivatives
01/08/1986EP0167008A2 1,4:3,6-Dianhydro-hexite derivatives, process for their preparation and their use as medicaments
01/07/1986US4563451 Quinazolino-1,4-benzodiazepin-5,13-diones
01/03/1986WO1986000070A1 Cephem compounds
12/1985
12/31/1985US4562220 Polyalkyldiazaspirodecanylacetic acid derivatives, a process for their preparation and their use as light stabilizers for organic polymers