Patents
Patents for C07D 513 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (15,120)
09/2004
09/22/2004EP1189904B1 Substituted heterocycle fused gamma-carbolines
09/22/2004CN1531540A Heterocyclic compounds and cerebral function improvers containing same as active
09/21/2004CA2167673C Condensed benzazepine derivative and pharmaceutical composition thereof
09/16/2004WO2004078764A1 Gm-95-containing antitumor effect potentiator, combined antitumor preparation and antitumor agent
09/16/2004WO2004078758A1 Novel fused heterocycles and uses thereof
09/16/2004WO2004078682A2 Cyclic compounds and compositions as protein kinase inhibitors
09/16/2004WO2004078110A2 Fused imizadoles as transforming growth factor (tgf) inhibitors
09/16/2004WO2004058176A3 Acyclic pyrazole compounds
09/16/2004WO2004004646A3 O-derivatized nocathiacin derivatives
09/16/2004US20040181061 Controlling phytopathogenic fungi by treating plants, seeds or soil with, e.g., O-Methyl (6-chloro-3-propyl-4H-1,3-benz[e]oxazin-4(3H)-one)-2-oxime; higher activity and selectivity than previous derivatives
09/16/2004US20040180942 modulating farnesoid X receptor (FXR), liver X receptors (LXR alpha and LXR beta ) and/or orphan nuclear receptors; treatment of lipid, cardiovascular and neurodegenerative disorders
09/16/2004CA2517850A1 Gm-95-containing antitumor effect potentiator, combined antitumor preparation and antitumor agent
09/15/2004EP1455779A1 Indolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands
09/15/2004EP1455777A1 Glyt1 transporter inhibitors and uses thereof in treatment of neurological and neuropsychiatric disorders
09/15/2004EP1173440B1 Tetracyclic azepinoindole compounds as 5-ht receptor ligands
09/15/2004EP1054669B9 Use of thiadiazolo[4,3-a]pyridine derivatives
09/15/2004CN1528746A Intermediate for preparing compounds having serotonin-2 receptor antagonistic and alpha-1 blocking action and its preparing method
09/14/2004US6790850 Thiazolo(4,5-d)pyrimidine compounds
09/10/2004WO2004077367A1 Tetracyclic sulfenamide compound
09/10/2004WO2004076461A1 Porphyrin derivatives
09/10/2004WO2004076420A1 Heteroarylcarbamoylbenzene derivative
09/10/2004WO2004076411A2 Aminocyclopentyl fused heterotricylicamide modulators of chemokine receptor activity
09/10/2004CA2516705A1 Aminocyclopentyl fused heterotricylicamide modulators of chemokine receptor activity
09/10/2004CA2516407A1 Heteroarylcarbamoylbenzene derivatives
09/09/2004US20040176605 Compounds as antumor agents or immunosuppressants
09/09/2004US20040176396 anti-protoazoal; poultry feed; therapy for cytokine mediated disease i.e. osteoarthritis, cerebral malaria, chronic pulmonary inflammatory disease, silicosis, pulmonary sarcosis, bone resorption diseases, reperfusion injury, graft v. host rejection
09/09/2004US20040176390 Novel fused heteroaromatic compounds as transforming growth factor (TGF) inhibitors
09/09/2004US20040176382 treatment of inflammation, proliferative diseases, and certain cardiovascular disorders as well as Alzheimer's disease;
09/09/2004US20040176377 inhibitors of glycogen synthase kinase-3 beta; treatment of diabetes or neurodegenerative diseases such as Alzheimer's disease; 6-(2-butylamino-pyrimidin-4-yl)-3-oxo-2,3-dihydro-pyridazine-4-carboxylic acid (3-pyridin-3-yl-propyl)-amide, as example
09/09/2004US20040176362 Matrix metalloproteinase inhibitors, treatment of tumor necrosis factor mediated diseases; autoimmune and neurodegenerative disorders; anticarcinogenic and antiinflammatory agents
09/09/2004DE10308107A1 New macrocyclic peptide derivatives useful for treating bacterial infections, especially caused by Gram-positive bacteria
09/08/2004EP1453801A1 Substituted 2-amino-cycloalkanecarboxamides and their use as cysteine protease inhibitors
09/02/2004WO2004074295A1 Thiazole cycle polymers, process for producing the same, synthesis intermediates thereof and utilization of the same
09/02/2004WO2004074291A1 Triazole compounds useful in therapy
09/02/2004WO2004074283A1 N-heterocyclyl-substituted amino-thiazole derivatives as protein kinase inhibitors
09/02/2004WO2004074278A1 Novel compounds
09/02/2004WO2004074270A2 Inhibitors of hepatitis c virus rna-dependent rna polymerase, and compositions and treatments using the same
09/02/2004WO2004050036A3 Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
09/02/2004WO2004014851A3 Tyrosine kinase inhibitors
09/02/2004US20040171626 having good to very good inhibitory activity against HCV polymerase; hepatitis C virus
09/02/2004US20040171620 Nitrogen-containing bicyclic heterocycles for use as antibacterials
09/02/2004US20040171022 Methods for regulating transcription by targeting quadruplex DNA
09/02/2004US20040170866 Cyclic tertiary amine compound and organic electroluminescent device containing the compound
09/02/2004CA2516235A1 Inhibitors of hepatitis c virus rna-dependent rna polymerase, and compositions and treatments using the same
09/02/2004CA2516234A1 N-heterocyclyl-substituted amino-thiazole derivatives as protein kinase inhibitors
09/01/2004EP1452528A1 Xanthine oxidase inhibitors
09/01/2004EP1451195A1 3-biphenyl-substituted-3-substituted-4-ketolactam and ketolactone and their utilization as pesticide
08/2004
08/31/2004US6784293 Solution and solid-phase synthesis of boc-protected 3-aminohydantoins/thiohydantoins and 3-aminodihydrouracils/ dihydrothiouracils
08/31/2004US6784189 Potassium channel inhibitors and method
08/31/2004US6784174 Inhibitors of the production of cytokines such as tnf
08/26/2004WO2004072243A2 Macrocyclic hepatitis c serine protease inhibitors
08/26/2004WO2004045562A3 Mixed kappa/mu opioids and uses thereof
08/26/2004US20040167141 Anticancer agents; antidiabetic agents; Alzheimer's disease
08/26/2004US20040167123 Anti-infective agents
08/26/2004CA2515216A1 Macrocyclic hepatitis c serine protease inhibitors
08/25/2004EP1448566A2 Chemokine receptor antagonists and methods of use thereof
08/25/2004EP1448525A1 Novel piperidine derivatives as modulators of chemokine receptors
08/25/2004EP0883616B1 Dihydrobenzofuran and related compounds useful as anti-inflammatory agents
08/25/2004CN1523987A Immune response modifiers for the treatment of periodontal disease
08/19/2004WO2004069843A1 Novel tricyclic azepine derivatives, method for production therof and pharmaceutical compositions comprising the same
08/19/2004WO2004069823A1 Inhibitors of histone deacetylase
08/19/2004WO2004069245A1 Oxazolidinone derivates n-substituted by a tricyclic ring, for use as antibacterial agents
08/19/2004US20040162285 Anti-infective agents
08/19/2004CA2514241A1 Oxazolidinone derivates n-substituted by a tricyclic ring, for use as antibacterial agents
08/19/2004CA2513059A1 Novel tricyclic azepine derivatives, method for production therof and pharmaceutical compositions comprising the same
08/18/2004EP1446127A1 Triazepine derivatives as neurotrophic agents
08/18/2004EP1446110A2 Organosulfur inhibitors of tyrosine phosphatases
08/18/2004EP0876345B1 Heterocyclic compounds as h+-atpases
08/18/2004CN1521169A 2,4- dichlorophenoxy acetalimide derivatives of dithiazo pyridine with herbicidal activity and method for preparation thereof
08/17/2004US6777557 Method and composition for rejuvenating cells, tissues organs, hair and nails
08/17/2004US6777406 Substituted pyrroloquinolines and pyridoquinolines as serotinin agonists and antagonists
08/12/2004WO2004067537A1 Triazole derivatives and antifungal agents containing the same
08/12/2004WO2004048368A3 Heteroarylsulfonylmethyl hydroxamic acids and amides and their use as protease inhibitors
08/12/2004WO2004015131A3 Hepatitis c virus assays
08/12/2004US20040157893 Pyrazole compounds useful as protein kinase inhibitors
08/12/2004US20040157853 Thiazolopytimidines and their use as modulators of chemokine receptor activity
08/12/2004US20040157852 cancer, diabetes, hepatic cirrhosis, atherosclerosis, angiogenesis and renal disease
08/12/2004US20040157840 Rifalazil compositions and therapeutic regimens
08/12/2004US20040157835 selective inhibition of cyclooxygenase-2, anti-inflammatory and analgesic properties, and no side effects of causing ulcer with the treatment dosage
08/12/2004US20040157831 Therapeutic 5-HT ligand compounds
08/11/2004EP1445252A1 Sulphonamide derivatives, the preparation thereof and the application of same as medicaments
08/11/2004EP1444545A2 Controlled diffusion coefficient electrochromic materials for use in electrochromic mediums and associated electrochromic devices
08/11/2004EP1444229A1 Pyrazole derivatives as psychopharmaceuticals
08/11/2004EP1443822A1 Substituted thien-3-yl-sulfonylamino(thio)carbonyl-triazolin(thi)ones
08/11/2004CN1161120C Utilization of polycyclic 2-amino-thiazole systems in the production of medicaments for prophylasis treatment of obesity
08/10/2004US6774130 Treating chronic inflammatory disease, chronic intestinal inflammation, arthritis, psoriasis, asthma and autoimmune disorders; th1 cell-mediated disorders; for example, 1,2,3,6-tetrahydro-7h-purine-2,6-dione derivatives
08/10/2004US6774126 Pyrrolo[1,2-b][1,2,4]oxadiazine diones useful as nitric oxide synthase inhibitors
08/05/2004WO2004065395A1 Thienopyridazinones and their use in modulation of autoimmune disease
08/05/2004WO2004065394A1 Thienopyrimidinediones and their use in the modulation of autoimmune disease
08/05/2004WO2004065367A1 Viral polymerase inhibitors
08/05/2004WO2004065366A1 2.4-dihalogen-6-(c2-c3-alkyl)-phenyl substituted tetramic acid derivatives
08/05/2004WO2004064778A2 3-amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
08/05/2004WO2004064730A2 Compounds, compositions and methods
08/05/2004WO2004039776A3 A process for the preparation of benzyl 2-oxo-4- (heteroaryl) dithio-alpha-isoprenyl-1- azetidineazetate derivatives
08/05/2004WO2003059289A3 Melanin concentrating hormone receptor ligands: substituted benzoimidazole analogues
08/05/2004US20040152889 Process for the preparation of benazepril
08/05/2004US20040152739 Bone disorders; cardiovascular disorders; gastrointestinal disorders; angiogenesis inhibitors; metabolism disorders; central nervous system disorders; traumas; skin disorders; inflammatory bowel disorders; anticancer agents
08/05/2004CA2513501A1 2.4-dihalogen-6-(c2-c3-alkyl)-phenyl substituted tetramic acid derivatives
08/05/2004CA2512546A1 3-amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
08/05/2004CA2512136A1 Thienopyridazinones and their use in modulation of autoimmune disease
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