Patents
Patents for C07D 513 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups , or (15,120)
04/2006
04/26/2006EP1648446A1 Indol-4 sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
04/26/2006EP1648445A1 Indol-5-yl sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
04/26/2006EP1648444A1 Indol-7 sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
04/26/2006CN1764641A Viral polymerase inhibitors
04/26/2006CN1253458C Process for preparing substance GM-95
04/20/2006WO2006040966A1 Aromatic-ring-fused pyrimidine derivative
04/20/2006WO2006040281A1 Thiazolyl-dihydro indazoles
04/20/2006WO2006040279A1 Pi3 kinases
04/20/2006WO2006040151A1 Subsituted hydroxyethylamine compounds for treating alzheimer’s disease
04/20/2006WO2006040149A1 Heterocyclic ketone compounds for treating alzheimer’s disease
04/20/2006WO2006040148A1 Tricyclic indole derivatives for use in the treatment of alzheimer’s disease
04/20/2006WO2005111039A3 Compounds and methods for inhibiting mitotic progression by inhibition of aurora kinase
04/20/2006US20060084680 ((1S)-5-{2-[(3-methyl-7-propyl-1,2-benzisoxazol-6-yl)oxy]ethoxy}-2,3-dihydro-1H-inden-1-yl)acetic acid; diabetes, obesity, hyperlipidemia, and atherosclerotic diseases; hyperglycemia, hyperinsulinemia, impaired glucose tolerance, dyslipidemia, hypertriglyceridemia, and insulin resistance
04/20/2006US20060084643 6-Fluoro-10-[3-(2-methoxy-ethyl)-4-methyl-piperazin-1-yl]-2-methyl-4H-3-thia-4,9-diaza-benzo[f]azulene; dopamine D2 and serotonin receptor anatagonist; neuroleptic agent, antidepressnt; psychological, bipolar disorders, psychosis, schizophrenia, acute mania
04/20/2006CA2579288A1 Thiazolyldihydroindazoles
04/20/2006CA2579279A1 Tricyclic thiazole derivatives as pi3 kinases
04/19/2006EP1647553A1 2-acylaminothiazole derivative or salt thereof
04/19/2006EP1646615A1 Pyrimidine derivatives as modulators of atp-binding cassette transporters
04/19/2006EP1537112B1 Condensed pyridines and pyrimidines with tie2 (tek) activity
04/19/2006EP1212330B1 Androgen receptor modulator compounds and methods
04/19/2006EP1196167B1 Use of p38 MAPK inhibitors in the treatment of ophthalmic conditions
04/19/2006EP1189890B1 Dihydrobenzodiazepins and their use for treating dyslipidemia
04/19/2006CN1761673A Guanidine derivatives and use thereof as neuropeptide FF receptor antagonists
04/19/2006CN1761672A Thienopyrimidinediones and their use in the modulation of autoimmune disease
04/19/2006CN1761651A 2,4-dihalogen-6-(c2-c3-alkyl)-phenyl substituted tetramic acid derivatives
04/18/2006US7030135 A sulfonylamino-tetrahydro(1,3)thiazolo(5,4-c)pyridinyl or benzothiazole derivatives, for treating diabetes, syndrome X, obesity, glaucoma, hyperlipidemia, hyperglycemia, hyperinsulinemia, osteoporosis, tuberculosis, dementia
04/13/2006WO2005118549A3 Compounds having affinity for dopamine d3 receptor and uses thereof
04/13/2006WO2005049559A3 Novel piperidine-substituted indoles- or hetero-derivatives thereof and their use as modulators of chemokine receptor (ccr-3)
04/13/2006US20060079707 Cyclization by reacting 4-(2-CHLORO-4-TRIFLUOROMETHYL-PHENYL)-4-CYANO-BUT-3-ENOIC ACID METHYL ESTER in the presence of a palladium catalyst and a base; chemical intermediates for preparing 10-AZA-TRICYCLO[6.3.1.02,7] drugs; bind nicotinic acetylcholine receptor, modulate cholinergic function
04/13/2006US20060079677 Novel tricyclic azepine derivatives, method for production thereof and pharmaceutical compositions comprising the same
04/13/2006US20060079549 Administering a stimulantfor the endogenous production/ release of somatotropins; 3-((1-(2-aminoprop-2-yl)carbonylamino-),2-(phenylmethoxymethyl-)ethyl-),5-(morpholino-carbonyloxymethyl-)-5,6,7,8-tetrahydro-1,2,4-triazolo(4,3-)pyridine; osteoporosis; obesity;improving bone densisty, muscle mass/strength
04/13/2006DE102004048877A1 New tricyclic thiazole derivatives useful as PI3 kinase inhibitors, for treating e.g. inflammatory and allergic airway and skin diseases, autoimmune and kidney disease
04/12/2006EP1644337A1 Melanocortin-4 receptor binding compounds and methods of use thereof
04/12/2006EP1643998A1 Dual nk1/nk3 antagonists for treating schizophrenia
04/12/2006EP1643960A2 Arylsulfonamide derivatives
04/12/2006EP1087981B1 Prenyl transferase inhibitors
04/12/2006CN1757645A Material contg. thiophene spirane structure, its synthesis and application
04/11/2006US7026313 2-thia-1,6,8-triaza-naphthalene-2,2-dioxides are kinase inhibitors
04/06/2006CA2581375A1 Specific kinase inhibitors
04/05/2006EP1641805A1 Thiazolo-, oxazalo and imidazolo-quinazoline compounds capable of inhibiting protein kinases
04/05/2006EP1173427B1 Hydroxamic acid derivative
04/05/2006CN1249039C Inhibitors of 11-beta-hydroxy steroid dehydrogenase type I
04/04/2006US7022850 Bicyclicpyrimidones and their use to treat diseases
04/04/2006US7022701 for treatment of disorders (sleeping, feeding) relating to or affected by the 5-HT6 receptor; serotonin receptor antagonists
04/04/2006US7022667 Mycobacterium; grampositive bacteria bactericides, antibiotics
04/04/2006US7022317 Heterocyclic derivatives of 2-oxothiazolidine-4-carboxylic acid, and use as active photoprotective agents
04/04/2006CA2354123C New benzothiadiazine derivatives, their preparation process and the pharmaceutical compositions that contain them
04/04/2006CA2235133C Esters of 3-hydroxy-piperidinemethanol derivatives
03/2006
03/30/2006WO2006034113A2 Quinolone analogs as cell proliferation inhibitors
03/30/2006WO2005113536A3 Tri- and bi-cyclic heteroaryl histamine-3 receptor ligands
03/30/2006WO2005097107A3 Diphenyl - indol-2-on compounds and their use in the treatment of cancer
03/30/2006US20060069116 3-Amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
03/30/2006US20060069109 Therapeutic agents
03/30/2006CA2580749A1 Quinolone analogs
03/30/2006CA2580725A1 Novel heterocyclic nf-kb inhibitors
03/29/2006EP1638957A1 N-heterocyclyl phenyl-substituted cyclic ketoenols
03/29/2006CN1753899A Spirotetrathiocarbamates and spirooxothiocarbamates
03/29/2006CN1753897A Fused bicyclic nitrogen-containing heterocycles
03/28/2006US7018960 Formed by inter-molecular interaction of one or more keto-enol tautomeric compounds; for mechanical friction sliding members
03/23/2006US20060063798 Heterocyclic aromatic compounds useful as growth hormone secretagogues
03/23/2006US20060063782 3-Hetero arylmethoxy ! pyridines and their analogues as p38 map kinase inhibitors
03/23/2006US20060063769 Preventives/remedies for urinary disturbance
03/22/2006EP1637533A1 Substituted thiazolopyrimidines as analgetics
03/22/2006EP1636242A1 Acylated imidazo (2,1-b) -1,3,4,-thiadia zole-2-sulfonamides, and uses thereof
03/22/2006EP1636241A1 Imidazo (2,1-b) -1,3,4-thiadiazole sulfoxides and sulfones
03/22/2006EP1635829A1 8-(3-biaryl)phenylquinoline phosphodiesterase-4-inhibitors
03/22/2006EP0915700B1 Use of beta-sheet mimetics as protease and kinase inhibitors and as inhibitors of transcription factors
03/22/2006CN1751052A Therapeutic agents
03/22/2006CN1751047A Triazole compounds useful in therapy
03/21/2006US7015328 Substituted coumarins and quinolines and analogs as activators of caspases and inducers of apoptosis and the use thereof
03/21/2006US7015321 Synthesis of non-symmetrical sulfamides using burgess-type reagents
03/21/2006US7015212 Thiazepine inhibitors of HIV-1 integrase
03/16/2006WO2006028284A1 Morpholine compound
03/16/2006WO2005016235A3 Combined use of impdh inhibitors with toll-like receptor agonists
03/16/2006US20060058298 Inhibitors of histone deacetylase
03/16/2006US20060058287 Gramnegative and Grampositive bacterial infections; substituted Piperidine derivatives specially optionally substituted pyrido [3,2, -b][1,4] thiazin-yl; 6-({(3R,4S)-3-Fluoro-1-[(R)-2-hydroxy-2-(2-methoxy-quinolin-8-yl)-ethyl]-piperidin-4-ylamino }-methyl)-4H-pyrido[3,2-b][1,4]thiazin-3-one; nontoxic
03/16/2006US20060058259 Human t-cell,lymphocyte virus; hepatitis virus
03/15/2006EP1633758A2 Imidazothiazoles and imidazoxazole derivatives as inhibitors of p38
03/15/2006EP1633725A1 Hepatitis c virus inhibitors
03/15/2006EP1448566B1 Chemokine receptor antagonists and methods of use thereof
03/15/2006CN1747957A Intermediate for 2-substituted carbapenem derivative and production process
03/15/2006CN1747951A Novel 2-pyridinecarboxamide derivatives
03/15/2006CN1747949A Acyclic pyrazole compounds
03/15/2006CN1746172A Preparation of plurichari
03/15/2006CN1245660C Color coupler for forming dye, silver halide photosensitive material and azomethine dyes compounds
03/14/2006US7012087 Anticancer agents
03/14/2006US7012085 As antipsychotics in therapy of schizophrenia, depression, bipolar disorders, cognition deficits, Parkinson disease, drug abuse, attention deficit hyperactivity disorders, glaucoma, diabetes and erectile dysfunction
03/14/2006CA2165800C Antiallergic imidazoazepines
03/09/2006WO2006024535A1 Substituted indole compounds and their use as 5-ht6 receptor modulators
03/09/2006US20060052612 Bis-4,7-(5'-(2-fluorophenyl)-2'-thienyl)-2,1,3-benzothiadiazole; emission color of the compounds of can be adjusted over the entire visible region, i.e. from deep blue to deep red, by choice of an appropriate substitution pattern; high current densities
03/09/2006US20060052406 Methods and compositions for treatment of central and peripheral nervous system disorders and novel compounds useful therefor
03/09/2006US20060052400 Immunosuppressants; respiratory system disorders; asthma; chronic obstructive pulmonary disease
03/09/2006US20060052372 N-(Heterocycloalkyl)alkylsulfonamides, e.g., N-[3-[4-(3-Chlorophenyl)piperazin-1-yl]propyl]-N-(4-methoxyphenyl)-propanesulfonamide; improve blood flow to the optic nerve head and the retina ; used to treat retinal diseases, sleep disorders, depression, schizophrenia, anxiety, OCD, etc.
03/09/2006CA2577925A1 Substituted indole compounds and their use as 5-ht6 receptor modulators
03/08/2006EP1632494A1 Vasopressin v1a antagonists
03/08/2006EP1632491A1 Substituted indole compounds and their use as 5-HT6 receptor modulators
03/08/2006EP1445252B1 Sulphonamide derivatives, the preparation thereof and the application of same as medicaments
03/08/2006EP1339723B1 Process and ester derivatives useful for preparation of cephalosporins
03/08/2006EP1325009B1 Amino-substituted tetracyclic compounds useful as anti-inflammatory agents and pharmaceutical compositions comprising same
03/08/2006CN1745087A Novel tricyclic azepine derivatives, method for production therof and pharmaceutical compositions comprising the same
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