Patents
Patents for C07D 501 - Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula: , e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring (7,574)
03/1981
03/10/1981US4255423 Cephalosporin compounds
03/10/1981CA1097341A1 Method of preparing a rapidly dissolving powder of sterile crystalline cefozolin sodium for parenteral administration
03/10/1981CA1097340A1 No translation available
03/04/1981EP0024347A1 Organic sulfoxides having a latent allyl group, process for preparing the same and pharmaceutical enzyme inhibiting composition comprising the same
03/03/1981US4254260 3-Substituted-7-substituted alkanamido-3-cephem-4-carboxylic acid compounds
03/03/1981US4254119 3-Unsubstituted-3-cephem compounds
03/03/1981US4254117 Bactericides
03/03/1981US4254029 Process for preparing β-lactam antibiotics
02/1981
02/24/1981US4252973 Process for chemically removing the acyl sidechain from cephalosporins and penicillins
02/24/1981US4252952 7-(α-Substituted glycinamido)-3-substituted methyl-3-cephem-4-carboxylic acids and their derivatives
02/24/1981US4252951 Isolation of syn-7-(2-amino-4-thiazolyl)-(methoxyimino)acetamido-3-acetoxymethyl-3-cephem-4-carboxylic acid
02/24/1981US4252950 3-Halo cephalosporins
02/24/1981US4252802 Hydroxamic acid derivatives of 7-[(2-amino-4-thiazolyl)-oximino] cephalosporins
02/24/1981CA1096373A1 Ureido substituted cephalosporin antibiotics
02/17/1981US4251657 Deacylation of a halogenoacetylamino compound using an n-substituted dithiocarbamic acid
02/17/1981US4251524 β-Lactam antibiotics
02/10/1981US4250307 N-substituted derivatives of cephalosporin extracted and cleaved
02/04/1981EP0023453A1 Process for the preparation of derivatives of 7-(2-aryl)-2-hydroxyimino-acetamido cephalosporanic acid
02/03/1981US4248868 For treating systemic infections by grampositive and gram negative bacteria
02/03/1981CA1095026A2 Cyclization to form cephem ring and intermediates therefor
02/03/1981CA1095025A1 Process for preparing 2-acyloxymethylpenams and 3- acyloxy-cephams
01/1981
01/28/1981EP0023045A1 Imidazolecarboxylic acid derivatives of penicillins and cephalosporins
01/27/1981US4247548 7α-Methoxycephalosporin derivatives and their pharmaceutical compositions having antibacterial activity
01/27/1981US4247461 Reaction with a penicillin or cephalosporin in an anhydrous solvent containing a base
01/27/1981CA1094547A1 Preparation process of 3-carbamoyloxymethyl 7-(amino thyazolyl acetamido) cephalosporanic acid derivatives
01/27/1981CA1094546A1 Process for the preparation of derivatives of 7-amino thiazolyl acetamido cephalosporanic acid
01/27/1981CA1094545A1 Cephalosporin antibiotics
01/21/1981EP0022494A1 Beta-lactam-compounds, process for their preparation and therapeutic agents containing them
01/20/1981US4246405 7-substituted-3-organic sulfonyloxy-3-cephem-4-carboxylate subjected to hydrogenolysis to from the 7-substituted-3-cephem-4-carboxylic acid
01/20/1981CA1094085A1 Azetidinone mercury sulfides and process therefor
01/20/1981CA1093997A1 Process of producing 7-methoxy cephalosporins
01/14/1981EP0022326A1 Process for chemically removing the acyl sidechain from cephalosporins and penicillins
01/14/1981EP0022245A2 Aminothiadiazolyl derivatives, process for their preparation, pharmaceutical compositions containing them;starting compounds and process for their preparation
01/13/1981US4245107 Antibiotics
01/13/1981US4245088 Novel 3-acyloxymethyl-cephem compounds useful as intermediates for preparing cephalosporin antibiotics
01/13/1981CA1093550A1 Cephalosporin derivatives
01/13/1981CA1093549A1 Cephalosporin antibiotics
01/13/1981CA1093548A1 Process for preparation of 3-halomethylcephems
01/07/1981EP0021688A1 7-(Thiazolylpropionamido) cephalosporins, their preparation, and pharmaceutical compositions containing them
01/07/1981EP0021176A2 Cephalosporin derivatives, process for their preparation and pharmaceutical compositions containing them
01/06/1981US4243810 3,5-dichloro-4-pyridone-1-acetic acid; a cephalosporin-derivative intermediate
01/06/1981US4243803 Hydrogenation of the 2-azido derivative using an amine-borane complex and raney nickel
01/06/1981CA1093068A1 Cephalosporin antibiotics
12/1980
12/30/1980US4242510 Cephalosporin compounds and processes for the preparation thereof
12/30/1980US4242509 The 7-imminohalide reacted with a primary lower alkanol or deuterated methanol
12/23/1980US4241057 Cephalosporins
12/23/1980US4240988 Method of stabilization of kinetically controlled triaryl phosphite-halogen compounds
12/23/1980CA1092096A1 Oxygen analogs of cephalosporins
12/23/1980CA1092095A1 3-acyloxymethyl-cephem compounds
12/16/1980US4239758 Bactericides
12/10/1980EP0019739A1 2-Aminoalkyl-5-pyridinoles, process for their preparation and pharmaceutical preparations containing them
12/09/1980US4238608 Antibiotics
12/02/1980US4237298 Aromatic acetic acid derivatives having sulfur atom at alpha-position and process for their preparation
12/02/1980US4237280 Intermediate for cephalosporin type compound
12/02/1980US4237279 Antibiotics
12/02/1980US4237128 7-[2-(2-Amino-4-thiazolyl)-2-[(1-carboxy-1,1-dialkyl)alkoxyimino]acetamido]cephem sulfoxides
12/02/1980US4237051 Stereospecific production of 6- or 7-carbon-substituted-β-lactams
11/1980
11/26/1980EP0019401A1 Process for preparing enamine derivatives, compounds so produced and process for preparing a 3-hydroxy-cephalosporin
11/26/1980EP0019387A1 Thiazolinoazetidinone compounds useful as intermediates for preparing cephalosporins and a process for their preparation
11/26/1980EP0019345A1 Process for the preparation of a (D-alpha-amino-(p-hydroxyphenyl)-acetamido) group containing cephalosporanic acid derivatives
11/26/1980EP0019308A1 Tetrazole derivatives and a process for their preparation
11/26/1980EP0019067A1 5,10-Dioxo-5,10-dihydrodiimidazo(1,5-a,1',5'-d)pyrazine-1,6-dicarboxylic acid and a process for producing imidazoledicarboxylic acid amido-derivatives
11/25/1980US4236002 Antibiotics
11/25/1980US4236001 7β-Acyloxy-3-heterocyclicthiomethyl cephalosporins
11/25/1980CA1090331A1 Process for the manufacture of heterocyclic compounds containing an alkylsulphonylamino group
11/18/1980US4234721 Process for the preparation of the crystalline monohydrate of 7-[D-amino-(p-hydroxyphenyl]acetamido)-3-methyl-3-cephen-4-carboxylic acid
11/18/1980US4234578 Aminoethyl-methoxy-cephalosporin compounds
11/18/1980CA1089848A1 Arylmalonamido methoxycephalosporins
11/12/1980EP0018669A1 1-(2-Sulfamoylaminoethyl)-1,4-dihydro-5H-tetrazole-5-thione and its salts
11/12/1980EP0018595A2 7-N-Heterocyclyl cephalosporins, a process for preparing and a pharmaceutical composition comprising the same
11/11/1980CA1089447A2 Sodium cefamandole crystalline forms
11/11/1980CA1089446A2 Sodium cefamandole crystalline forms
11/11/1980CA1089445A1 3-cephem derivatives
11/11/1980CA1089444A1 Unsaturated aliphatic halogenated heterocyclic compounds
10/1980
10/29/1980EP0018001A2 Chromophoric cephalosporin derivatives, process for their preparation and their utilisation, compositions containing them and their preparation
10/28/1980US4230849 Conversion to amides and esters
10/28/1980US4230644 Derived from triaryl phosphites and chlorine or bromine
10/28/1980CA1088519A1 Diazole and tetrazole derivatives of cyanomethylthioacetylcephalosporins
10/28/1980CA1088518A1 Cyanomethylthioacetylcephalosporins
10/28/1980CA1088517A1 3-heterothiomethyl ureido cephalosporins
10/21/1980US4229575 Antibiotics
10/21/1980US4229574 Indole cephalosporin derivatives
10/21/1980US4229573 7α-Methoxycephalosporin derivatives
10/21/1980US4229363 Intermediates for cephalosporin and penicillin derivatives
10/21/1980US4229349 Production of semi-synthetic β-lactam antibiotics
10/21/1980CA1088049A1 3-substituted-7-substituted alkanamido-3-cephem-4- carboxylic acid compounds and processes for preparation thereof
10/15/1980EP0017238A1 Cephalosporin derivatives and process for their preparation and pharmaceutical compositions containing them
10/15/1980EP0017170A1 Improved process for the preparation of cephamycin antibiotics
10/15/1980EP0016900A1 Intermediates in the preparation of cephalosporin derivatives, process for their preparation and use
10/07/1980US4226986 7-acylamino-3-hydroxy-3-cephem compound, triaryl phosphite dihalide
10/07/1980US4226864 7-Substituted aminoacetamido oxadethiacephalosporins
10/07/1980US4226863 7-Methoxy cephalosporins
10/07/1980US4226806 Chemical intermediates
10/07/1980CA1087170A1 N-substituted aminomethyl-methoxy-heterocyclic compounds
10/07/1980CA1087169A1 Process for converting 3-methylene cephalosporins to 3-heterothiomethyl cephalosporins
10/01/1980EP0016725A1 Process for the preparation of 3-hydroxycepham compounds
10/01/1980EP0016296A1 Cephalosporin derivatives, process for their preparation, compositions containing them, and intermediates and their preparation
09/1980
09/30/1980US4225707 2-Lower alkyl-7-substituted-2 or 3-cephem-4-carboxylic acid compounds
09/30/1980US4225706 Polychalcogen ester of cephem compound, process for preparing the same and method for removing the protective group of the same
09/30/1980CA1086739A1 Mercury intermediates useful in the preparation of 2- alkoxy cephalosporins
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