Patents
Patents for C07D 498 - Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms (21,960)
03/1981
03/25/1981EP0025546A2 Therapeutical use of tranquillizing benzodiazepine derivatives and mixtures containing them
03/25/1981EP0025496A1 Maytansinoids, their production and therapeutic compositions containing them
03/24/1981US4258049 Inhibiting phenylethanolamine N-methyltransferase with thiadiazolo and oxadiazolotetrahydroisoquinolines
03/24/1981EP0018991A4 1,5-diazabicyclo(3.3.0)octadienedione derivatives, preparation and use thereof as fluorescent labelling agents.
03/18/1981EP0025108A1 Maytansinoids, their production and therapeutic compositions containing them
03/17/1981US4256886 Hypotensive agents, vasodilation
03/17/1981US4256746 Antitumor agents; microbiocides; mitosis
03/17/1981CA1097627A1 Method for the production of maytansinoids
03/10/1981US4255568 2H-Pyrimido[4,5-d][1,3]oxazine-2,4(1H)-dione derivatives
03/10/1981US4255432 8-[2-3-Indolyl)ethyl]-1-oxa-3-,8-diazaspiro[4.5]decan-2-ones, pharmaceutical compositions thereof and methods of use thereof
03/10/1981CA1097340A1 No translation available
03/03/1981US4254135 3-Amino-4-hydroxypyrrolidines
03/03/1981US4254121 3-Oxo-5H-pyrimido[2,1-c][1,4 ]benzoxazines
03/03/1981US4254118 1-Oxo-5H-pyrimido[2,1-c][1,4]benzthiazine-2-carboxylic acid esters
03/03/1981CA1096862A1 Oxadiazolopyrimidine derivatives
02/1981
02/24/1981US4252964 Antitumor agent intermediate, propenyl 3-/dihydrocarbylamino/acrylate, substituted hydroxylamine
02/24/1981US4252953 Antibiotic crystalline epimer
02/24/1981US4252825 5-fluoro-2-(2-hydroxy-3-tert-butyl amino-propoxy) butyrophenone
02/17/1981US4251534 Antihypertensive polyfluorohydroxyisopropyl bicyclic and tricyclic carbostyrils
02/17/1981US4251533 Nitrogen-containing heterocyclic compounds
02/17/1981US4251529 Ergot peptide alkaloids
02/17/1981CA1095908A1 Morpholine derivatives as antibacterial agents
02/11/1981EP0023885A1 Method for the introduction of an oxygen-containing functional group into ansamycines, compounds thus obtained, and pharmaceutical compositions containing them
02/11/1981EP0023761A1 Tetrahydroisoquinoline derivatives, process for preparing them and compositions containing them
02/11/1981EP0023663A2 Method for the preparation of new heterocycles that contain oxygen
02/11/1981EP0023578A1 Aminoalkylbenzene derivatives, process for their preparation and pharmaceutical compositions
02/11/1981EP0023559A1 2-(Perhydro-1,4-diazino)-pyrimido(5,4-d)pyrimidines, their preparation and medicaments containing them
02/10/1981US4250268 Polysilylesters having a polyalkylpiperidine as part of the polymer useful as light stabilizers for plastics
02/10/1981US4250095 Imidazobenzodiazepines
02/03/1981US4248870 Microbiocides, antitumor agents, and antimitotics
02/03/1981CA1095041A1 0-2-isocephem antibacterial agents and processes and intermediates for their production
02/03/1981CA1095036A1 Process for producing 3-amino-rifamycins s and sv
02/03/1981CA1095035A1 Process for the production of rifamycins
01/1981
01/28/1981EP0022997A1 2,2,6,6-Tetramethyl-4-piperidyl carboxylic acid esters and amides of mono and poly alcohols, phenols and amines and synthetic polymer compositions stabilized thereby
01/27/1981US4247704 Hexahydro thieno imadazole intermediates for the synthesis of biotin
01/27/1981US4247449 Urea derivatives, process for their manufacture and their use as light protecting agents for polymers
01/21/1981EP0022628A1 Process for the preparation of oxazolinoazetidinones
01/20/1981CA1094063A1 Thieno ¬2,3-d| pyrimidine antiallergic agents
01/13/1981US4245104 Production of biotin
01/13/1981US4245089 Novel intermediates for β-lactams
01/13/1981US4244961 1-Oxa-3,8-diazaspiro[4.5]decan-2-ones antihypertensive agents
01/07/1981EP0022086A1 4-Oxa-6-aza-6(phenyl)-spiro(2.4)heptane-5,7-diones, preparation and use as microbicides
01/07/1981EP0021178A1 Maytansinoids, their production and use
01/07/1981EP0021177A1 Maytansinoids, their production and use
01/07/1981EP0021173A1 Maytansinoids, their production and use
01/06/1981US4243588 Cyclizing a 2-chloroazetidinone with lead fluoride in dimethyl sulfoxide to obtain the 4-oxa-2,6-diazabicyclo(3.2.0)heptane
01/06/1981US4243587 Process for 3β-aminoazetidin-2-ones
01/06/1981CA1093071A1 5.alpha.-BICYCLOMYCIN DERIVATIVES
01/06/1981CA1093070A1 8.beta.-ALKYL-SUBSTITUTED MORPHINAN-6-ONE COMPOUNDS
12/1980
12/30/1980CA1092604A1 Rifamycin derivatives
12/23/1980US4241208 Stabilizers of synthetic polymers against heat and light
12/23/1980US4240962 Process for the preparation of imidazobenzodiazepines
12/23/1980CA1092110A1 Antibacterial agents
12/23/1980CA1092108A1 Oxadiazolopyrimidine derivatives
12/23/1980CA1092105A1 Pyrrolo(2,1-b) (3)benzazepines
12/16/1980US4239898 Novel 4-(substituted-aminophenoxy)-3-thiophenemethanols
12/16/1980US4239683 Antitumor
12/10/1980EP0019934A1 Antibiotic C-15003 PND and process for their preparation
12/10/1980EP0019788A2 Novel process for the manufacture of thiophene derivatives suited for the manufacture of biotin, process for the manufacture of biotin and novel intermediates in this process
12/09/1980US4238616 3-(Substituted)phenyl-5-(β-hydroxyphenethyl)-N-(alkyl)-isoxazole-4-carboxamides
12/09/1980US4238486 Treating hypertension and parkinson*s disease
12/09/1980CA1091230A1 7-acylamino-8-oxo-3-oxa-1-azabicyclo- ¬4.2.0|octane-2-carboxylic acid derivatives
12/02/1980US4237287 Diazotization with sodium nitrite and chlorination with thionyl chloride
12/02/1980CA1090806A1 Oxazolines
11/1980
11/26/1980EP0019457A2 Clavulanic acid derivatives, their preparation and pharmaceutical compositions
11/26/1980EP0018991A1 1,5-diazabicyclo(3.3.0)octadienedione derivatives, preparation and use thereof as fluorescent labelling agents
11/25/1980US4236004 Antisecretory, antiulcer, antiallergens
11/25/1980US4235920 Antibiotics
11/25/1980CA1090364A2 Azetidinones and their production and use
11/18/1980US4234596 3-(2-Aminoethylthio)-6-(1-hydroxyethyl)-7-oxo-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid
11/18/1980US4234581 Thieno[2,3-d]oxazines
11/18/1980US4234485 Process for preparing 4-desoxy-thiazolo[5,4-c]rifamycin derivatives
11/12/1980EP0018811A1 Antibiotic crystalline epimer, its preparation and pharmaceutical composition containing it
11/12/1980EP0018760A1 D-Sesquisodium salt of an oxa-beta-lactam diacid compound and its preparation
11/12/1980EP0018594A2 Process for the preparation of 3-(1-hydroxyethyl)-azetidinones
11/11/1980US4233446 5-Chloro-7,8-dihydro-7-oxo-pyrido[2,3-d]pyrimidine-6-carboxylic acid derivatives
11/11/1980CA1089491A1 Process for asymmetric synthesis of optically active 2-aklanoyl-1,2,3,4-tetrahydro-2-naphthol compounds
11/11/1980CA1089470A2 Oxazolidine compounds
11/11/1980CA1089469A2 Oxazolidine compounds
11/11/1980CA1089457A1 5-nor-bicyclomycin-5-one derivatives
11/11/1980CA1089453A1 Rifamycin compounds
11/04/1980US4232154 Carbocyclic analogs of cytosine nucleosides exhibiting antiviral and antineoplasticactivity
11/04/1980US4232036 6-, 1- and 2-Substituted-1-carbadethiapen-2-em-3-carboxylic acids
10/1980
10/29/1980EP0018139A2 Pyrido (2,3-d) pyrimidine derivatives, pharmaceutical compositions containing them and processes for preparing the pyrido (2,3-d) pyrimidine derivatives
10/29/1980EP0017992A1 2-Substituted-6-substituted-1-carbadethiapen-2-em-3-carboxylic acids, processes for preparing them, antibiotic pharmaceutical compositions containing same and process for preparing intermediates
10/28/1980US4230712 7-Methyl-8β-lower alkyl or 7-methyl-8-lower alkyl B/C cis or trans morphinan-6-one compounds and therapeutic method of treating pain employing them
10/21/1980US4229533 Method for producing antibiotic C-15003 P-4
10/15/1980EP0017617A2 Polyalkylpiperidine spirooxazolones, their application as light stabilisers and polymers stabilised therewith
10/14/1980US4228295 Novel cycloheptathiophene intermediates for the synthesis of biotin
10/14/1980US4228239 Method for producing antibiotic C-15003 P-3
10/07/1980US4226870 O-, N- and carboxyl derivatives of thienamycin
10/07/1980US4226771 Sedatives, anesthetics, imidazobenzodiazepine intermediates
10/07/1980US4226767 Intermediates for 3-aminoazetidin-2-ones
10/07/1980US4226765 Reaction with an aldehyde in the presence of iron or zinc and acetic acid; cyclization
10/07/1980CA1087194A1 Oxazolidine compounds
10/07/1980CA1087181A1 Aminoalkylpyrrolobenzoxazalkanes
09/1980
09/30/1980US4225494 Antibiotic c-15003, fungicide, antiprotozoa
09/23/1980US4224443 From crotonaldehyde and 5-chlorosalicylhydroxamic acid
09/23/1980US4224336 3-(2-Aminoethylthio)-6-amido-7-oxo-1-azabicyclo[3.2.0]-hept-2-ene-2-carboxylic acid
09/23/1980US4224323 Method for lowering serum uric acid