Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
09/2010
09/21/2010US7799782 P38 inhibitors and methods of use thereof
09/21/2010US7799775 Pyrimidine derivatives
09/21/2010US7799773 administering 7-Benzyloxy-3-cyclobutyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine, for the treatment of Alzheimer's disease, cognitive impairment, dementia, epilepsy, neuropathic pain, Parkinson's disease, schizophrenia, attention deficit disorder or depression in humans
09/21/2010CA2445068C Azo compounds for type i phototherapy
09/21/2010CA2405002C Antitumoral analogs of et-743
09/21/2010CA2359948C Triazole compounds with dopamine-d3-receptor affinity
09/16/2010WO2010103381A1 Spirocyclic piperidine derivatives as trpm 8 modulators
09/16/2010WO2010103240A1 10-amino-1,2,3,4-tetrahydropyrido[2,1-a]isoindol-6(10bh)-one derivatives, method for preparing same, and therapeutic uses thereof
09/16/2010WO2010054285A3 Fused bicyclic and tricyclic pyrimidine compounds as tyrosine kinase inhibitors
09/16/2010US20100234609 Fused ring spiroketal derivative and use thereof as anti-diabetic drug
09/16/2010US20100234528 Supports for oligomer synthesis
09/16/2010CA2755157A1 10-amino-1,2,3,4-tetrahydropyrido[2,1-a]isoindol-6(10bh)-one derivatives, method for preparing same, and therapeutic uses thereof
09/16/2010CA2754847A1 Halogenalkylmethylenoxy-phenyl-substituted ketoenols
09/15/2010EP2227474A1 Azo and diaza derivatives and uses thereof in phototherapy
09/15/2010EP2227467A1 Isoxazolo-pyridine derivatives
09/15/2010EP1899303B1 Novel 3-aza-spiro[5.5]undecane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
09/15/2010EP1861092B1 Potassium channel opener having benzofuroindole skeleton
09/15/2010CN101830905A Method for preparation and semi-synthesis of galanthamine hydrobromide
09/15/2010CN101245070B Novel technique for synthesizing toroid quinazoline protein tyrosine kinase restrainer
09/14/2010US7795440 N-substituted tricyclic 1-aminopyrazoles as inhibitors for the treatment of cell proliferative disorders
09/14/2010US7795434 Quaternary chelidonine and alkaloid derivatives, process for their preparation and their use in manufacture of medicaments
09/14/2010US7795431 Terrylene and quaterrylene derivatives
09/14/2010US7795299 11,15-dioxa-cyclopenta[a]phenanthren-12-one derivatives, used for the treatment of cancer; anticarcinogenic agents
09/14/2010US7795273 Pyrazolo[1,5-a]pyridine-3-carboxylic acids as EphB and VEGFR2 kinase inhibitors
09/14/2010US7795260 ecteinascidin analogues used for the treatment of of leukaemia, lung cancer, colon cancer, kidney cancer, melanoma, prostate cancer, ovarian cancer, breast cancer, pancreatic epitheloid carcinoma, and cervix epitheloid carcinoma; antitumor and anticarcinogenic agents
09/14/2010US7795259 pyrrolo[2,3-b]pyrazine derivatives used as enzyme inhibitors for the treatment of cardiovascular disorders, diabetes, Alzheimer's disease, immunodeficiency disorders, inflammatory diseases, hypertension, allergic diseases, autoimmune diseases, bone disorders, cancer and viral diseases
09/14/2010US7795255 4-[2-(4-nitro-phenyl)-6-oxo-4-thioxo-6H-1-oxa-3b,5-diaza-cyclopenta[a]pentalen-5-yl]-butyric acid, used for inhibiting heparin-binding proteins and in the treatment of pancreatic cancer; anticarcinogenic agents
09/14/2010US7795247 13-Cyclohexyl-5-(2-pyrrolidin-1-ylethoxy)-6,7-dihydro-5H-indolo[2.1-a][2]benzazepine-10-carboxylic acid, for example; use for the treatment or prevention of infection by hepatitis C virus
09/14/2010US7795042 red-emitting fluorescent rhodamine dyes; photostable; useful as molecular probes; For use in assays involving staining of cells, protein binding, and/or analysis of nucleic acids (hybridization and sequencing)
09/14/2010CA2409715C .beta.-carboline derivatives useful as inhibitors of phosphodiesterase
09/10/2010WO2010102219A1 Methylenedioxybenzo [i] phenanthridine derivatives used to treat cancer
09/10/2010WO2010101128A1 Amide compound
09/10/2010WO2010101127A1 Indole compound
09/10/2010WO2010100178A1 Heterocyclic antiviral compounds
09/10/2010CA2753730A1 Inhibitors of beta-secretase
09/10/2010CA2752443A1 Heterocyclic antiviral compounds
09/09/2010US20100227878 Noscapine analogs and their use in treating cancers, including drug-resistant cancers
09/09/2010US20100227877 New camptothecin derivatives and uses thereof
09/09/2010US20100227873 Nitrogen-containing heterocyclic compounds and methods of use thereof
09/09/2010US20100227851 Method of preventing and/or treating a neurodegenerative disease by administering an extract of Lycoris chejuensis and/or a compound isolated therefrom
09/09/2010US20100226879 Heterocyclic antiviral compounds
09/08/2010EP0882717B1 Nitrogenous heterocyclic compounds
09/08/2010CN101824061A Baicalin ion pair medicine from traditional Chinese medicine of baikal skullcap root as well as preparation method and application thereof
09/08/2010CN101824060A Ion pair medicine from traditional Chinese medicine extracts as well as preparation method and application thereof
09/08/2010CN101824043A Compositions useful as inhibitors of protein kinases
09/08/2010CN101824038A Camptothecin and method for preparing analogues thereof
09/08/2010CN101044123B Pyrimidine derivative fused with nonaromatic ring
09/07/2010US7790883 5-[[(2,3-difluorophenyl)methyl]thio]-7-[[(1R)-2-hydroxy-1-methylethyl]amino]-3-[2-(phenylsulfonyl)ethyl]thiazolo[4,5-d]pyrimidin-2-(3H)-one; protection of the thiazole nitrogen atom while reacting a 7- leaving group with an amine for an amination reaction to result in improved yields; efficiency
09/07/2010US7790748 N-alkyl-4-methyleneamino-3-hydroxy-2-pyridones
09/07/2010US7790729 vascular endothelial growth factor (VEGF) and hepatocyte growth factor (HGF), receptor antagonists, such as N-(3-Fluoro-4-(2- (thiophen-2-yl)thieno[3,2- b]pyridin-7- yloxy)phenylcarbamothio- yl)-2-phenylacetamide, used for treating angiogenesis-mediated cell proliferative diseases or as antitumor agents
09/07/2010US7790713 Inhibitors of interleukin-1β converting enzyme
09/07/2010US7790709 Heterocyclic compounds, methods of making them and their use in therapy
09/07/2010CA2493680C Condensed heterocyclic pyrazole derivatives as kinase inhibitors
09/07/2010CA2370344C Thieno- and furopyrimidine derivatives as a2a-receptor antagonists
09/02/2010WO2010099159A1 Cyclopropyl fused indolobenzazepine hcv ns5b inhibitors
09/02/2010WO2010097469A1 Novel dioxo-imidazolidine derivatives, which inhibit the enzyme soat-1, and pharmaceutical and cosmetic compositions containing them
09/02/2010WO2010097468A1 Novel dioxo-imidazolidine derivatives, which inhibit the enzyme soat-1, pharmaceutical and cosmetic compositions containing them
09/02/2010WO2010097087A1 Catecholamine derivatives and prodrugs thereof
09/02/2010WO2010067078A8 3,6-disubstituted xanthylium salts
09/02/2010US20100222585 Preparation of dihydrothieno [3, 2-d] pyrimidines and intermediates used therein
09/02/2010US20100222374 Spirocyclic heterocyclic derivatives and methods of their use
09/02/2010US20100222352 Compounds and Methods for the Treatment of Viruses and Cancer
09/02/2010US20100222342 Pyrrolopyrazole, potent kinase inhibitors
09/02/2010US20100222338 Beta-secretase modulators and methods of use
09/02/2010US20100222324 Substituted Indole Compounds
09/02/2010US20100222316 Inhibitors of the 11-beta-hydroxysteroid dehydrogenase type 1 enzyme
09/02/2010CA2751299A1 Novel dioxo-imidazolidine derivatives, which inhibit the enzyme soat-1, and pharmaceutical and cosmetic compositions containing them
09/02/2010CA2751279A1 Novel dioxo-imidazolidine derivatives, which inhibit the enzyme soat-1, pharmaceutical and cosmetic compositions containing them
09/01/2010EP2223914A1 Tricyclic condensed pyrazole derivatives as CB1 inhibitors
09/01/2010EP2223913A1 Tricyclic pyrazole derivatives and microemulsions thereof as CB1- and/or CB2-inhibitors
09/01/2010EP2222680A1 Process improvement
09/01/2010EP1709047B1 Azabenzofuran substituted thioureas as inhibitors of viral replication
09/01/2010EP1469809B1 Multiple acting anti-angiogenic and cytotoxic compounds and methods for using the same
09/01/2010CN101821265A Substituted bicyclic piperidinyl-and piperazinyl- sulfonamides useful to inhibit 11ss-hydroxysteroid dehydrogenase type-1
09/01/2010CN101821253A Piperidine derivative
09/01/2010CN101817833A DPP-IV inhibitor
09/01/2010CN101817815A Compounds with antibacterial activity
09/01/2010CN101337928B Quinoline compounds, synthesizing method, applications in synthesis of alkaloid of camptothecins
08/2010
08/31/2010USRE41614 Synthetic analogs of ecteinascidin-743
08/31/2010US7786162 Agents useful for reducing amyloid precursor protein and treating dementia and methods of use thereof
08/31/2010US7786134 camptothecin derivatives such as 10-(benzyl succinate)-7-ethylcamptothecin in the form of an emulsion or micelle, used for treating lung, mammary gland, colon or ovarian cancer
08/31/2010US7786131 Anticancer agents; restenosis; atherosclerosis; skin disorders
08/31/2010US7786108 Compounds and method for treating dyslipidemia
08/31/2010US7786048 Condensed heterocyclic pyrazole derivatives as kinase inhibitors
08/31/2010CA2227235C Novel galanthamine derivatives, preparation method therefor, use thereof as drugs, and pharmaceutical compositions containing such derivatives
08/26/2010WO2010096115A1 Compounds, compositions and methods for control of hepatitis c viral infections
08/26/2010WO2010094405A1 Bi- and tricyclic indazole-substituted 1,4-dihydropyridine derivatives and uses thereof
08/26/2010WO2010094210A1 Preparation method of (4s,5r)-half-ester
08/26/2010WO2010094120A1 Novel spiro compounds useful as inhibitors of stearoyl-coenzyme a delta-9 desaturase
08/26/2010US20100217012 COMPOUNDS AND PROCESSES FOR PREPARING SUBSTITUTED AMINOMETHYL-2,3,8,9-TETRAHYDRO-7H-1,4-DIOXINO[2,3-e]INDOL-8-ONES
08/26/2010US20100216988 Regioselective metal catalyzed synthesis of annelated benzimidazoles and azabenzimidazoles
08/26/2010US20100216789 Rho-kinase inhibitors
08/26/2010US20100216785 Pharmaceutical compositions
08/26/2010US20100216726 Substituted-Quinoxaline-Type Piperidine Compounds and the Uses Thereof
08/26/2010US20100215741 Pharmaceutical compounds
08/26/2010US20100215590 Micronization Method
08/26/2010CA2752603A1 Bi- and tricyclic indazole-substituted 1,4-dihydropyridine derivatives and uses thereof
08/26/2010CA2750564A1 Novel spiro compounds useful as inhibitors of stearoyl-coenzyme a delta-9 desaturase
08/25/2010EP2221347A1 Sulfonated diarylrhodamine dyes
08/25/2010EP2221309A1 Novel naphthyridine derivative monohydrate and method for producing the same
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