Patents
Patents for C07D 487 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups (57,272)
09/2004
09/23/2004US20040185002 condensation aerosol for delivery of a drug selected from chlordiazepoxide, betahistine, clonidine, testosterone, a conjugated estrogen, an estrogen ester, estradiol, an estradiol ester, ethinyl estradiol, an ethinyl estradiol ester and hyoscyamine
09/23/2004US20040185001 Delivery of physiologically active compounds through an inhalation route
09/23/2004US20040185000 Delivery of antihistamines through an inhalation route
09/23/2004US20040184999 Delivery of anti-migraine compounds through an inhalation route
09/23/2004US20040184998 Delivery of drug esters through an inhalation route
09/23/2004US20040184997 volatilizing a coating of drug on a solid support, having the surface texture of a metal foil, to a temperature sufficient to produce a heated vapor of drug and condensing the heated vapor to form condensation aerosol particles
09/23/2004US20040184996 Delivery of nonsteroidal antiinflammatory drugs through an inhalation route
09/23/2004DE10311300A1 New 2-alkoxy-4-halo-6-alkylphenyl-substituted (hetero)cyclic ketoenols, useful as total or selective herbicides and pesticides, e.g. insecticides, acaricides and nematocides for plant protection
09/23/2004CA2518759A1 Synergistically acting herbicidal mixtures
09/23/2004CA2518748A1 Antimicrobial agents and anticancer agents
09/23/2004CA2518743A1 Protein kinase inhibitors
09/23/2004CA2518395A1 Bicyclo-pyrazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
09/22/2004EP1460077A1 Novel pyrazolopyrimidones and their use as PDE inhibitors
09/22/2004EP1460076A1 Substituted 8-perfluoroalkyl-6,7,8,9-tetrahydropyrimido[1,2-a] pyrimidin-4-one derivatives
09/22/2004EP1460075A1 Substituted 8-Pyridinyl-6,7,8,9-Tetrahydropyrimido[1,2-a]Pyrimidin-4-one and 8-Phenyl-6-7,8,9-Tetrahydropyrimido[1,2-a]Pyrimidin-4-one derivatives
09/22/2004EP1458726A2 Mitotic kinesin inhibitors
09/22/2004EP1458723A1 Fused heterocyclic succinimidecompounds and analogs thereof, modulators of nuclear hormone receptor function
09/22/2004EP1458722A1 Pyrrolopyrimidines as phosphodiesterase vii inhibitors
09/22/2004EP1458721A1 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino 4,5-b]indole-1-carboxamide derivatives, their preparation and therapeutic use
09/22/2004EP1458714A1 3,4-dihydro-1h-isoquinoloin-2-yl-derivatives
09/22/2004EP1458395A1 New use
09/22/2004EP1458392A2 Acridone inhibitors of impdh enzyme
09/22/2004EP1458375A2 Compositions for decreasing activity of hormone-sensitive lipase
09/22/2004EP1458374A2 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
09/22/2004EP1383770B1 Method for the production of 4,6-diaminopyrimido 5,4-d]pyrimidines
09/22/2004EP1274709B1 Salts of bicyclic, n-acylated imidazo-3-amines and imidazo-5-amines
09/22/2004EP1200438B1 Method for making debromohymenialdisine and analogs thereof
09/22/2004EP1192165B1 Substituted heterocycle fused gamma-carbolines
09/22/2004EP1189904B1 Substituted heterocycle fused gamma-carbolines
09/22/2004EP1000062B1 Tricyclic vasopressin agonists
09/22/2004EP0966468B1 Crown ether-derivatised perylenes
09/22/2004CN1531540A Heterocyclic compounds and cerebral function improvers containing same as active
09/22/2004CN1531538A 4-amino-5-phenyl-7-cyclobutyl-pyrrolo (2,3-D) pyrimidie derivatives
09/22/2004CN1531537A Novel tricyclic pyridyl benzazepine carboxyamides and derivatives their tocolytic oxytocin leceptor antagonists
09/22/2004CN1531536A Process for preparation of pyrazolo[4,3-D] pyrimidine derivative
09/22/2004CN1531531A Novel arylsusfonamide compounds for treatment of obesity, type II diabetes and CNS-disorders
09/22/2004CN1167711C Octahydro-6,10-dioxo-6h-pyridazino/1,2-a//1,2/diazepin-1-carboxylic derivatives, prepn. method and use for preparing therapeutically active compounds
09/22/2004CN1167701C Method for preparing oxazolidone amine
09/22/2004CN1167405C Karatin fibre dyeing composition containing pyrazolo-(1,5-alpha)- pyrimidine derivatives, dyeing method, and pyrazolo-(1,5-alpha) pyrimidine derivatives and preparation thereof
09/21/2004US6794545 Conformationally restricted polyamine analogs as disease therapies
09/21/2004US6794544 Method for the preparation of tetrahydrobenzothiepines
09/21/2004US6794505 Chlorins possessing fused ring systems useful as photoselective compounds for photodynamic therapy
09/21/2004US6794387 Pharmaceutically active compounds
09/21/2004US6794382 Benzimidazole derivatives, preparation and therapeutic use thereof
09/21/2004US6793839 Forming methylene bridges between glycoluril units; attaining oligimers with up to twelve units at high yield
09/21/2004CA2280587C Growth hormone secretagogues
09/21/2004CA2167673C Condensed benzazepine derivative and pharmaceutical composition thereof
09/16/2004WO2004078761A1 Enantiomerically pure cilazapril,process for preparation
09/16/2004WO2004078760A1 SUBSTITUTED 8'-PYRIDINYL-DIHYDROSPIRO-[CYCLOALKYL]-PYRIMIDO [1,2-a] PYRIMIDIN-6-ONE AND 8'-PYRIMIDINYL-DIHYDROSPIRO-[CYCLOALKYL]-PYRIMIDO [1,2-a] PYRIMIDIN-6-ONE DERIVATIVES AND THEIR USE AGAINST NEUROGENERATIVE DISEASES
09/16/2004WO2004078759A1 Substituted 2-(diaza-bicyclo-alkyl)-pyrimidone derivatives
09/16/2004WO2004078758A1 Novel fused heterocycles and uses thereof
09/16/2004WO2004078733A1 Quinazolines useful as modulators of ion channels
09/16/2004WO2004078714A2 Processes for preparing imidazoquinoxalinones, heterocyclic-substituted imidazopyrazinones, imidazouinoxalines and heterocyclic-substituted imidazopyrazines
09/16/2004WO2004078116A2 P38 inhibitors and methods of use thereof
09/16/2004WO2004078110A2 Fused imizadoles as transforming growth factor (tgf) inhibitors
09/16/2004WO2004058176A3 Acyclic pyrazole compounds
09/16/2004US20040181069 modulators of the monoamine receptors, in particular the serotonin, dopamine and norepinephrine receptors, and the biogenic amine transporters for serotonin, dopamine and norepinephrine;
09/16/2004US20040181063 such as 1-C-(5-N-benzyloxymethyl-4-methoxy pyrrolo[3,2-d]pyrimidin-7-yl)-1,4-dideoxy-1,4-imino-2,3-O-isopropylidene-D-ribitol; potent inhibitors of purine nucleoside phosphorylase and useful for suppressing T-cell function and/or treating and/or preventing infections caused by protozoan parasites
09/16/2004US20040181052 Process for the production of pentostatin aglycone and pentostatin
09/16/2004US20040180947 Sulfonamide compounds and pharmaceutical use thereof
09/16/2004US20040180944 Pyrazolopyrimidinones which inhibit type 5 cyclic guanosine 3',5'-monophosphate phosphodiesterase (cGMP-PDE5) for the treatment of sexual dysfunction
09/16/2004US20040180934 Dihydropyrrolo[1,2-a]indole and tetrahydropyrido[1,2-a]-indole derivatives as prostaglandin d2 receptor antagonists
09/16/2004US20040180911 for the treatment of a proliferative disease, such as a tumor
09/16/2004US20040180902 3-Substituted quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists
09/16/2004US20040180898 chemical reduction reaction
09/16/2004US20040180897 anticarcinogenic agents
09/16/2004US20040180896 P38 inhibitors and methods of use thereof
09/16/2004US20040180877 Nicotinic acetylcholine receptor cholinergic ligands, monoamine receptor and transporter modulators; such as 1-(2-Benzo[b]thiophenyl-1,1-dioxide)-imidazolidine
09/16/2004US20040180875 Obesity, anorexia, bulemia, depression, anxiety, psychosis, schizophrenia, migraine, addictive behavior, obsessive-compulsive disorder, sexual disorders
09/16/2004US20040180872 Method for the preparation of selectively-substituted corroles and new substituted corroles
09/16/2004US20040180871 Anti-inflammatory compositions and methods
09/16/2004US20040180837 Porphyrin compound, albumin inclusion compound thereof and artificial oxygen carrier
09/16/2004US20040180235 Fluorescent diketopyrrolopyrroles
09/16/2004DE10350280A1 New complex comprising cucurbituril and fullerene coupled with each other by molecular interaction, useful as a medicine delivery means in the field of pharmaceutics
09/16/2004DE10309927A1 New trisubstituted dihydro-imidazo-pyridazinone or imidazo-pyridinone derivatives, useful as dipeptidylpeptidase-IV inhibitors for e.g. treating diabetes mellitus type I or II, arthritis or obesity
09/16/2004CA2517962A1 Enantiomerically pure cilazapril, process for preparation
09/16/2004CA2517844A1 Quinazolines useful as modulators of ion channels
09/15/2004EP1457490A1 5-membered N-heterocyclic compounds with hypoglycemic and hypolipidemic activity
09/15/2004EP1457488A1 Intermediates for use in the preparation of urea compounds having muscarinic receptor antagonist activity
09/15/2004EP1456211A1 N-carbacycle monosubstituted indolocarbazoles as protein kinase inhibitors
09/15/2004EP1456210A1 Pyrazolyl-substituted triazoloquinoxalines
09/15/2004EP1456207A2 Heterocyclic acridone inhibitors of impdh enzyme
09/15/2004EP1456205A1 Imidazoquinoline derivatives
09/15/2004EP1456201A1 Benzhydryl derivatives
09/15/2004EP1455792A1 Ureas of 2-aminobenzothiazoles as adenosine modulators
09/15/2004EP1305317B1 Dihydroporphyrin derivatives and their uses
09/15/2004EP1295878B1 Pyrazinone derivatives
09/15/2004EP1173440B1 Tetracyclic azepinoindole compounds as 5-ht receptor ligands
09/15/2004EP1129095B1 Process for preparing cross-bridged tetraaza macrocycles
09/15/2004EP0986384A4 Inhibitors of protein isoprenyl transferases
09/15/2004EP0968254B1 Fluorescent materials and their use
09/15/2004EP0710109B1 Method for identifying a PDE IV inhibitor
09/15/2004EP0693072B9 Method for the synthesis of 4- and/or 5-(di)substituted 2-aminoimidazoles from 2-aminoimidazoles and aldehydes
09/15/2004CN1529706A 哌嗪衍生物 Piperazine derivatives
09/15/2004CN1529705A Tri-and tetraaza-acenaphthylen derivatives as CRF receptor antagonists
09/15/2004CN1529594A Injectable galenic formulation for use in diagnosis or photodynamic therapy and method for preparing same
09/15/2004CN1528762A 6-2-(2-halogen-4-alkoxypenyl)-triazo-pyrimidine of killing fungus
09/15/2004CN1166668C Method for preparing substituted [1,4] diazepino (6,7,1-hi) indol-4-ones
09/15/2004CN1166667C Imidazoimidazoles and trizoles as anti-inflammatory agents
09/14/2004US6790884 Nondeforming; for crystalline plastics