Patents
Patents for C07D 487 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups (57,272)
03/2008
03/27/2008WO2007150011A3 Prolyl hydroxylase inhibitors
03/27/2008WO2007117381A9 2 -aminopyridine analogs as glucokinase activators
03/27/2008WO2007092879A3 Substituted thiatriazaacenaphthylene-6-carbonitrile kinase inhibitors
03/27/2008US20080076921 Inhibitors of bruton's tyrosine kinase
03/27/2008US20080076917 Intermediates of 2-Substituted Carbapenem Derivatives and Process for Production Thereof
03/27/2008US20080076781 Pseudobase benzo[c]phenanthridines with improved efficacy, stability, and safety
03/27/2008US20080076776 Therapeutic compounds
03/27/2008US20080076775 3-(2-alkoxycarbonyl-3-indolyl)-3-oxo-propionic acid ester or propionamide intermediates: methyl 3-[6-fluoro-2-(methoxycarbonyl)-1-methyl-1H-indol-3-yl]-3-oxopropanoate; peripheral neuropathy, Parkinson's disease, Alzheimer's disease
03/27/2008US20080076774 Kinase Modulators and Methods of Use
03/27/2008US20080076773 Such as (3R,4R)-1-Pyrimidin-4-yl-4-(2,4,5-trifluorophenyl)piperidin-3-amine bis-trifluoroacetic acid salt
03/27/2008US20080076755 4-(Adamantane-1-carbonylamino)-3-oxo-2-aza-bicyclo[2.2.2]octane; 5-(Adamantane-1-carbonylamino)-10-oxo-9-aza-bicyclo[3.3.2]decane for treating autoimmune diseases, vascular disorders, viral infection or replication, asthma, osteoporosis, tumor growth, rheumatoid arthritis, organ transplant rejection
03/27/2008US20080076754 Substituted spiroheterocycles
03/27/2008US20080076753 Substituted spiroheterocycles
03/27/2008US20080076748 Palladium 31-oxo-15- methoxycarbonylmethyl- Rhodobacteriochlorin-131-(2-N3- trimethylammoniumethyl)amide acetate (salt); bacteriochlorophylls free of carbamate group; as photosensitizer for thermodynamic therapy and diagnosis; cancer, age related macular degeneration; killing viruses and bacteria
03/27/2008US20080076738 antiviral: improved pharmacokinetics
03/27/2008DE102006043443A1 Neue aza-bicyclische Verbindungen und ihre Verwendung New aza-bicyclic compounds and their use
03/27/2008CA2665851A1 Spiro benzazepines as vasopressin antagonists
03/27/2008CA2665849A1 Spiro benzazepines used as vasopressin antagonists
03/27/2008CA2663791A1 Pyrazolo (1, 5-a) (1, 3, 5) triazine and pyrazolo (1, 5-a) pyrimidine derivatives useful as protein kinase inhibitors
03/27/2008CA2662835A1 Octahydropyrrolo [3, 4-c] pyrrole derivatives and their use as antiviral agents
03/26/2008EP1903045A1 Pyrazolopyrimidine derivative
03/26/2008EP1902716A1 Prophylactic and/or therapeutic agent for motor disorder
03/26/2008EP1902057A1 Macrocyclic heterocyclic aspartyl protease inhibitors
03/26/2008EP1902056A2 Raf inhibitor compounds and methods of use thereof
03/26/2008EP1902055A1 Pyridazine compounds as glycogen synthase kinase 3 inhibitors
03/26/2008EP1527075B1 Diazabicyclononane and -decane derivatives and their use as opioid receptor ligands
03/26/2008EP1509218A4 Peptide deformylase inhibitors
03/26/2008EP1467997B1 Pyrrolopyrimidine and pyrrolopyridine derivatives substituted with cyclic amino group
03/26/2008CN100377004C Image forming material and ammonium compound
03/26/2008CN100376581C [1,4]diazocino [7,8,1-hi]indole derivatives as antipsychotic and antiobesity agents
03/26/2008CN100376580C Pyrazolopyrimidines as cyclin-dependent kinase inhibitors
03/26/2008CN100376579C 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino[4,5-b]indole-1-carboxamide derivatives, their preparation and use in treating
03/26/2008CN100376576C Substituted 2-(diaza-bicyclo-alkyl)-pyrimidone derivatives
03/26/2008CN100376573C 1,3-dihydroimidazole fused-ring compound
03/26/2008CN100376571C 6-substituted pyrido-pyrimidines
03/26/2008CN100376569C Inhibitors of farnesyl protein transferase
03/25/2008US7348429 Process for purifying N-[3-(3-cyanopyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-N-ethylacetamide(zaleplon) and crystalline forms of zaleplon accessible with the process
03/25/2008US7348343 N-(N-heteroaryl)1-pyridyl- or -pyrimidyl-hydropyridine-4-carboxamides; e.g., 3'-Chloro-3,6-dihydro-2H-[1,2']bipyridinyl-4-carboxylic acid (6-trifluoromethyl-pyridin-3-yl)-amide and 1-pyrimidin-2-yl-1,2,3,6-tetrahydro-pyridine-4-carboxylic acid (6-trifluoromethyl-pyridin-3-yl)-amide
03/25/2008US7348338 PPAR active compounds
03/25/2008US7348336 Inhibitors of IkB kinase (I Kappa B Kinase); 1-acetyl-7-bromo- beta -carboline; antiinflammatory and anticarcinogenic agent; asthma, osteoarthritis, rheumatoid arthritis, Alzheimer's disease, infections, and cardiac infarct
03/25/2008US7348325 Pyrrolotriazine kinase inhibitors
03/25/2008US7348324 Cyclic amine compounds as CCR5 antagonists
03/25/2008US7348323 [5-(4-cyclopentyl-piperazin-1-yl)-1H-pyrrolo[2,3-c]pyridin-2-yl]-pyrrolidin-1-yl-methanone; antagonists or inverse agonists at histamine 3 receptor; obesity, antidepressant, dementia and cognitive disorders, neurological disorders
03/25/2008US7348321 Flumazenil for the treatment of alcohol dependency
03/25/2008CA2173319C Radiation sensitization using texaphyrins
03/20/2008WO2008033960A2 Systems and methods for transferring funds from a sending account
03/20/2008WO2008033798A2 A pyrrolopyrazin as syk-kinase inhibitor
03/20/2008WO2008033468A2 Azetidine and azetidone derivatives useful in treating pain and disorders of lipid metabolism
03/20/2008WO2008033447A1 Azetidine and azetidone derivatives useful in treating pain and disorders of lipid metabolism
03/20/2008WO2008032764A1 Fused heterocyclic derivative
03/20/2008WO2008032060A1 4-benzimidaz0lyl-6-m0rph0lin0-2-piperazinylpyrimidine derivatives as p13k and mtor inhibitors for the treatment of proliferative disorders
03/20/2008WO2008032033A1 4-benzimidazolyl-2-morpholino-6-piperazinylpyrimidine derivatives as pi3k and mtor inhibitors for the treatment of proliferative disorders
03/20/2008WO2008031513A1 Pyrazolopyridine, indazole, imidazopyridine, imidazopyrimidine, pyrazolopyrazine and pyrazolopyridine derivates as stimulators of guanylate cyclase for cardiovascular disorders
03/20/2008WO2008014108A3 Antimicrobial oxazolidinone prodrugs
03/20/2008WO2008004698A3 Pyrazolo [1, 5-a] pyrimidine compounds as cb1 receptor antagonist
03/20/2008WO2007146615A3 Long lived anion-selective sensors based on a covalently attached metalloporphyrin as anion receptor
03/20/2008WO2006094187A3 Phthalazine, aza- and diaza-phthalazine compounds and methods of use
03/20/2008WO2001003644A3 Pyrazolopyrimidinone derivatives conjugated to thiophene moieties or benzo [fused] 5-membered heterocycles for erectile dysfunction
03/20/2008US20080071093 Forming, purification of dipyrromethane and porphrin ; condensation, oxidation, cyclization
03/20/2008US20080071092 Oxidation color dye; reavcting a hydrazine compound
03/20/2008US20080070941 Derivatives of n-heterocyclylmethylbenzamides, preparation method thereof and application of same in therapeutics
03/20/2008US20080070936 Compounds specific to adenosine A1 receptors and uses thereof
03/20/2008US20080070932 unexpectedly potent antagonists of A2a adenosine receptor; Parkinson's; neurodegenerative diseases; 2-furan-2-yl-N5-[1-(5-methyl-isoxazol-3-ylmethyl)-pyrrolidin-2-ylmethyl]-[1,2,4]triazolo[1,5-a]pyrimidine-5,7-diamine
03/20/2008US20080070906 Quinolinone derivatives
03/20/2008US20080070902 Cinnamide Compound
03/20/2008US20080070896 Insulin secretagogue and hypoglycemic agent; pyrimidine derivatives condensed with a non-aromatic ring selected from dihydrothiophene, dihydrofuran, cycloalkane moiety; 1-[2-(4-chloro-2,5-difluorophenyl)-6,6-dioxido-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]-4-(3-hydroxypropyl)piperidin-4-ol for example
03/20/2008US20080070893 Cancer, neurological disorders, autoimmune disorders; inhibitors of CK2, a serine/threonine kinase; based upon macrocyclic pyrazolo[1,5-a][1,3,5]triazine and pyrazolo[1,5-a]pyrimidine compounds
03/20/2008US20080070891 (1s,5s)-3-(5,6-dichloro-3-pyridinyl)-3,6-diazabicyclo[3.2.0]heptane
03/20/2008US20080070889 Spirocyclic azetidin(one); e.g. 2,7-diazaspiro[3.5]nonan-1-one; T-type calcium channel blockers; Niemann-Pick C1-like (NPC1L1) antagonists
03/20/2008US20080069817 Heteroaryl-fused pyrimidinyl compounds as anticancer agents
03/20/2008DE102006040915A1 New oxindole derivatives useful for treating vasopressin- or oxytocin-dependent diseases
03/20/2008CA2663947A1 Azetidine and azetidone derivatives useful in treating pain and disorders of lipid metabolism
03/20/2008CA2663504A1 Azetidine and azetidone derivatives useful in treating pain and disorders of lipid metabolism
03/20/2008CA2663297A1 Pyrazolopyridine, indazole, imidazopyridine, imidazopyrimidine, pyrazolopyrazine and pyrazolopyridine derivatives as stimulators of guanylate cyclase for cardiovascular disorders
03/19/2008EP1900739A1 Diazolodiazine derivatives as kinase inhibitors
03/19/2008EP1899350A1 Pyrazolo ý3 , 4-d¨azepine derivatives as histamine h3 antagonists
03/19/2008EP1899349A1 Intermediates useful in preparing certain pyrrolotriazine compounds and process for making such intermediates
03/19/2008EP1899348A1 Pyrrolotriazine compounds useful as kinase inhibitors and methods of treating kinase-associated conditions therewith
03/19/2008EP1899347A2 Intermediates useful in preparing certain pyrrolotriazine compounds and process for making such intermediates
03/19/2008EP1899346A1 Pyrrolotriazine compounds useful as kinase inhibitors
03/19/2008EP1899345A1 Pyrrolotriazine compounds useful as kinase inhibitors
03/19/2008EP1899344A1 Compounds that maintain pluripotency of embryonic stem cells
03/19/2008EP1899343A1 Halogenated pyrazolo [1,5-a]pyrimidines, processes, uses as gaba-a receptors ligand, compositions and intermediates
03/19/2008EP1899342A1 [1, 2, 4]triazolo [1, 5-a]pyrimidine derivatives as chromatographic adsorbent for the selctive adsorption of igg
03/19/2008EP1899330A1 Substituted glycinamides having an antithrombotic and factor xa-inhibiting effect
03/19/2008EP1899318A1 New azetidine derivatives as neurokinin receptor antagonists for the treatment of gastrointestinal diseases
03/19/2008EP1711174B1 Adjuvant compositions
03/19/2008EP1638966B1 4-SUBSTITUTED DERIVATIVES OF PYRAZOLO ¬3,4-d PYRIMIDINE AND USES THEREOF
03/19/2008EP1628979B1 Diaminopyrroloquinazolines compounds as protein tyrosine phosphatase inhibitors
03/19/2008EP1581535B9 Pyrrolopyridazine derivatives
03/19/2008EP1530573B1 Condensed heterocyclic pyrazole derivatives as kinase inhibitors
03/19/2008EP1511751B1 Pyrazolo[1,5-a]pyrimidine compounds as antiviral agents
03/19/2008EP1490344B1 Anxiolytic agents with reduced sedative and ataxic side effects
03/19/2008EP1432715B1 Pyrimidine derivatives
03/19/2008CN101147286A Electrode for use in oxygen reduction
03/19/2008CN101146889A Luminous compound containing lanthanide ion
03/19/2008CN101146812A Optically active ammonium salt compound, production intermediate thereof and method for producing same
03/19/2008CN101146811A Hiv整合酶抑制剂 Hiv integrase inhibitors
03/19/2008CN101146540A Hiv整合酶抑制剂 Hiv integrase inhibitors
03/19/2008CN101143866A Chlorophyll derivatives, preparation method and application thereof in medical agricultural chemicals