Patents
Patents for C07D 487 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups (57,272)
08/2009
08/19/2009CN100528875C Crystal-free type Idi prone and its preparing method
08/19/2009CN100528874C Pyrrolo [2,3d] pyrimidine compositions and their use
08/19/2009CN100528873C 3 position substituted mesoazalene compounds and high efficiency synthesis method
08/19/2009CN100528350C Method for increasing the cutting hardness of a molded body
08/19/2009CN100528162C Pharmaceutical compositions
08/19/2009CN100528154C Malonyl-COA decarboxylase inhibitors useful as metabolic modulators
08/18/2009US7576245 Using a fluorinated phenyl compound containing electrophilic and nucleophilic groups; increasing the fluorous nature of an organic compound; 4-(1H,1H,2H,2H-Perfluorodecyl)benzenesulfonamide; N-[4-(1H,1H,2H,2H-perfluorodecyl)benzyloxycarbonyloxy]succinimide
08/18/2009US7576199 Near infrared dyes
08/18/2009US7576092 Benzofuro- and benzothienopyrimidine modulators of the histamine H4 receptor
08/18/2009US7576091 Thiazolo-, oxazalo and imidazolo-quinazoline compounds capable of inhibiting protein kinases
08/18/2009US7576090 Benzazole analogues and uses thereof
08/18/2009US7576087 3-(Phenylsulfonyl)-7-piperazin-1-yl-1H-pyrazolo[4,3-b]pyridine; 5-HT receptor subtype 5HT6; selective serotonin receptor antagonist; cognition actiators; alzheimer's disease; attention deficit disorder; antidepressant; antiepileptic agent; anxiolytic agents; obsessive compulsive disorder; Parkinson's
08/18/2009US7576085 Imidazo[1,2-a]pyrazine compounds; cancers
08/18/2009US7576084 1-(Phenylmethylaminocarbonyl-),4,7-di(oxo-),6-(4-(hydroxylphenyl),8-(piperidino(1,3-phenylene)methyl)-perhydro(pyrazino(2,1-c)-as-triazine); disorders modulated by Wnt-signaling pathway; anticarcinogenic agents; colorectal cancer; restenosis; polycystic kidney disease; angiogenesis inhibition
08/18/2009US7576082 rac-6-Chloro-3-(3-chloro-benzyl)-3-(1-methyl-1H-pyrazol-4-yl)-1,3-dihydro-indol-2-one; murine double minute (MDM2 ) oncogene inhibitor; feedback control loop of p53 mutant cells; inhibit the interaction between p53 and MDM2 proteins
08/18/2009US7576077 9-{[5-(3-Chlorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-3-pyridin-4-yl-6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a][1,3]diazepine; Group 1 receptor subtype; analgesics; psychological disorders; gastroesophageal reflux; neuroprotectans; antiischemic agents; hyperglycemic agents; neurodegenerative disease
08/18/2009US7576074 Receptor-type kinase modulators and methods of use
08/18/2009US7576072 Heterocyclic inhibitors of MEK and methods of use thereof
08/18/2009CA2585557C Pyrazolo[4,3-d] pyrimidine derivatives useful as pde-5 inhibitors
08/18/2009CA2429133C Novel imidazole derivatives, production method thereof and use thereof
08/18/2009CA2400268C Pyrrolopyrimidinone derivatives, process of preparation and use
08/18/2009CA2392030C Urea compounds having muscarinic receptor antagonist activity
08/18/2009CA2392028C Carbamate derivatives having muscarinic receptor antagonist activity
08/13/2009WO2009100431A1 Cysteine and cystine prodrugs to treat schizophrenia and reduce drug cravings
08/13/2009WO2009100375A1 Substituted imidazopyridazines useful as kinase inhibitors
08/13/2009WO2009100120A2 Pyridinyl-substituted piperazinyl oxoethyl tetrahydropyrazolopyridines
08/13/2009WO2009099982A1 2-aminopyridine kinase inhibitors
08/13/2009WO2009099929A1 Mesoionic pesticides
08/13/2009WO2009099596A2 Macrocyclic serine protease inhibitors
08/13/2009WO2009099163A1 Pyrrolopyrimidin derivative for use as pi3k inhibitor, and use thereof
08/13/2009WO2009098257A1 Composition for dyeing keratin fibres comprising at least one cationic diamino-n,n-dihydropyrazolone derivative
08/13/2009WO2009098236A1 Pyrrolo [2, 3-d] pyridines and use thereof as tyrosine kinase inhibitors
08/13/2009WO2009097971A1 Triazolium salts as par1 inhibitors, production thereof, and use as medicaments
08/13/2009WO2009097970A1 Triazolopyridazines as par1 inhibitors, production thereof, and use as medicaments
08/13/2009WO2009097709A1 Pyrazolopyrimidinone-containing phenyl guanidine derivatives, pharmaceutical compositions containing them, process for their preparation and their use
08/13/2009WO2009097695A1 Arylmethylidene heterocycles as novel analgesics
08/13/2009WO2009074575A3 Organic compounds
08/13/2009WO2009032754A3 Heterocyclodiazepine cannabinoid receptor modulators for treatment of disease
08/13/2009WO2005122682A3 Process for the preparation of esters of piperazic acid
08/13/2009US20090203901 Process for preparing pyrazole functionalized benzodiazepinones
08/13/2009US20090203757 Ethylene glycol esters as photoactive agents
08/13/2009US20090203719 Enhancing treatment of mdr cancer with adenosine a3 antagonists
08/13/2009US20090203717 Fused heterocyclic compound
08/13/2009US20090203702 INHIBITORS OF p38
08/13/2009US20090203672 Substituted Sulfonamide Compounds
08/13/2009US20090203665 Heterocyclic-substituted phenyl methanones
08/13/2009US20090203664 (1s,5s)-3-(5,6-dichloro-3-pyridinyl)-3,6- diazabicyclo[3.2.0]heptane
08/13/2009US20090203577 Azepinoindole Derivatives As Pharmaceutical Agents
08/13/2009US20090202480 Macrocyclic serine protease inhibitors
08/13/2009US20090202478 inhibit the function of the NS5A protein encoded by Hepatitis C virus (HCV); useful in establishing or determining the binding site of other antiviral compounds, for example, by competitive inhibition; used to treat or prevent viral contamination of materials
08/13/2009CA2714966A1 Arylmethylidene heterocycles as novel analgesics
08/13/2009CA2714226A1 Cysteine and cystine prodrugs to treat schizophrenia and reduce drug cravings
08/13/2009CA2714177A1 Pyrrolo [2,3-d] pyridines and use thereof as tyrosine kinase inhibitors
08/13/2009CA2713551A1 Triazolium salts as par1 inhibitors, production thereof, and use as medicaments
08/13/2009CA2713550A1 Triazolopyridazines as par1 inhibitors, production thereof, and use as medicaments
08/13/2009CA2713347A1 Mesoionic pesticides
08/13/2009CA2712971A1 Macrocyclic serine protease inhibitors
08/13/2009CA2711778A1 Pyrrolopyrimidine derivative as pi3k inhibitor and use thereof
08/13/2009CA2711777A1 Novel pyrazolo [3,4-d] pyrimidine derivatives as anti-cancer drugs
08/12/2009EP2088150A1 Fused pyrrolocarbazoles and methods for the preparation thereof
08/12/2009EP2086981A1 Compounds for inhibiting mitotic progression
08/12/2009EP2086980A1 Macrocyclic peptides as hepatitis c virus inhibitors
08/12/2009EP2086979A2 Imidazoý1,2-b¨pyridazine and pyrazoloý1,5-a¨pyrimidine derivatives and their use as protein kinase inhibitors
08/12/2009EP2086978A1 Amorphous form of n-{2-fluoro-5-[3-(thiophene-2-carbonyl)-pyrazolo [1,5-a]pyrimidin-7-yl]-phenyl-n-methyl-acetamide
08/12/2009EP2086967A2 Inhibitors of hepatitis c virus
08/12/2009EP1904461B1 Cyclic anilino-pyridinotriazines as gsk-3 inhibitors
08/12/2009EP1392328B1 Medicament for protection in radiotherapy
08/12/2009CN101506216A Fused imidazole derivatives for the treatment of disorders mediated by aldosterone synthase and/or 11-beta-hydroxylase and/or aromatase
08/12/2009CN101506215A Adenosine A2a receptor antagonists
08/12/2009CN101506214A Pyrazoloquinazolinones as PARP inhibitors
08/12/2009CN101506213A Amino- imidazolones and their use as a medicament for treating cognitive impairment. alzheimer disease, neurodegeneration and dementia.
08/12/2009CN101506212A Amino- imidazolones and their use as a medicament for treating cognitive impairment. alzheimer disease, neurodegeneration and dementia.
08/12/2009CN101506211A 激酶拮抗剂 Kinase antagonists
08/12/2009CN101505752A Prolyl hydroxylase inhibitors
08/12/2009CN100526316C Triazole miazines derivative
08/11/2009US7572914 2-hydroxy-1H-indol derivatives enzyme inhibitors for preventing or treating inflammation, inflammatory bowel disease, psoriasis, dementia related diseases Alzheimer's Disease, Cognitive Impairment, arthritis, neurodegenerative diseases, amyotrophic lateral sclerosis, Down syndrome, Huntington's Disease
08/11/2009US7572817 Carboxypeptidase U inhibitors; thrombosis, atherosclerosis, adhesions, dermal scarring, cancer, fibrotic conditions, inflammatory diseases; e.g. 2-[(6-Aminopyridin-3-yl)methyl]-3-mercapto-5-[3-(pyrrolidin-1-ylcarbonyl)phenyl]pentanoic acid
08/11/2009US7572816 Therapeutic agents for the treatment of cancer, metabolic diseases and skin disorders
08/11/2009US7572806 PPAR active compounds
08/11/2009US7572802 For central nervous system diseases, in particular Parkinson's disease, Extra Pyramidal Syndrome, restless legs syndrome and attention deficit hyperactivity disorder
08/11/2009US7572799 Pyrazolo[4,3-d]pyrimidines as Phosphodiesterase Inhibitors
08/11/2009US7572795 Pyrrolotriazine aniline prodrug compounds useful as kinase inhibitors
08/11/2009US7572787 Substituted naphthalene sulfonamides
08/11/2009US7572784 Inhibit Aurora kinase; cancer; 4-[9-Chloro-7-(2-fluoro-phenyl)-5H-benzo[c]pyrimido[4,5-e]azepin-2-ylamino]-N-(2-methylamino-ethyl)-benzamide; 9-Chloro-N-(4-{[3-(dimethylamino)azetidin-1-yl]carbonyl}phenyl)-7-(2-fluoro-6-methoxyphenyl)-5H-pyrimido[5,4-d][2]benzazepin-2-amine
08/11/2009CA2482551C 1-(4-piperidinyl) benzimidazolones as histamine h3 antagonists
08/11/2009CA2433874C Improved process for carbapenem synthesis
08/11/2009CA2417590C Prophylactic or ameliorative agent for insulin resistance and/or obesity
08/11/2009CA2359772C Cyclic substituted fused pyrrolocarbazoles and isoindolones
08/11/2009CA2222552C N-oxides as antibacterial agents
08/06/2009WO2009097578A1 Oxim derivatives as hsp90 inhibitors
08/06/2009WO2009097515A2 [a]-fused indole compounds, their use as mtor kinase and pi3 kinase inhibitors, and their syntheses
08/06/2009WO2009097490A1 1H-PYRAZOLO[3,4-D]PYRIMIDINE, PURINE, 7H-PURIN-8(9H)-ONE, 3H-[1,2,3]TRIAZOLO[4,5-D]PYRIMIDINE, AND THIENO[3,2-D]PYRIMIDINE COMPOUNDS, THEIR USE AS mTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES
08/06/2009WO2009097446A1 Pyrazolopyrimidine pi3k inhibitor compounds and methods of use
08/06/2009WO2009097405A2 Compounds and methods for preparing diazaspiro derivatives
08/06/2009WO2009097233A1 Imidazopyrazines as protein kinase inhibitors
08/06/2009WO2009096445A1 Nerve trunk cell propagation accelerator
08/06/2009WO2009096435A1 Condensed heterocyclic derivatives and uses thereof
08/06/2009WO2009095923A2 Corroles for neuroprotection and neurorescue
08/06/2009WO2009095789A1 Substituted arylamide diazepinopyrimidone derivatives for the treatment of neurodegenerative diseases caused by abnormal activity of gsk3-beta
08/06/2009WO2009095282A2 Photolatent amidine bases for redox curing of radically curable formulations