Patents
Patents for C07D 473 - Heterocyclic compounds containing purine ring systems (11,932)
02/2005
02/03/2005WO2005009348A2 Substituted purine derivatives
02/03/2005WO2005009343A2 A1 adenosine receptor antogonists
02/03/2005WO2005009334A2 Reversible inhibitors of s-adenosyl-l-homocysteine hydrolase and uses thereof
02/03/2005US20050026939 Metabolite of xanthine phosphodiesterase 5 inhibitor and derivatives thereof useful for treatment of erectile dysfunction
02/03/2005US20050026938 Purine inhibitors of protein kinases, G proteins and polymerases
02/03/2005US20050026174 Alternative heterocycles for DNA recognition
02/03/2005DE10130504B4 Xanthin- und Phenazon-Acesulfam-H-Komplexe mit verbessertem Geschmack, Verfahren zu ihrer Herstellung und ihre Verwendung Xanthine-phenazone and acesulfame-H-complexes with improved taste, process for their preparation and their use
02/03/2005CA2522338A1 Reversible inhibitors of s-adenosyl-l-homocysteine hydrolase and uses thereof
02/02/2005EP1502914A1 Process for the preparation of 1-amino-4-(hydroxymethyl)-2-cyclopentene derivatives
02/02/2005EP1501812A1 Pna monomer and precursor
02/02/2005EP0912575B1 Processes for the synthesis of chemical compounds having pde-iv inhibitory activity
02/02/2005CN1187354C Adenosine receptor antagonists and methods of making and using the same
02/02/2005CN1187051C Xanthine-based compound for preparation of medicine for enhancing insulin action
02/01/2005US6849737 Synthesis and purification of valacyclovir
02/01/2005US6849736 Crystalline forms of valacyclovir hydrochloride
02/01/2005US6849735 Making N-4-carboxyphenyl-3-(6-oxohydropurin-9-yl) propanamide starting from aminopropionic acid, ethyl p-aminobenzoate, and using aminocyanoacetamide
02/01/2005US6849660 Antimicrobial biaryl compounds
02/01/2005US6849623 For use as human and veterinary medicine
02/01/2005US6849270 Releasable linkage and compositions containing same
02/01/2005CA2320448C 6,9-disubstituted 2-[trans-(4-aminocyclohexyl)amino]purines
01/2005
01/27/2005WO2005007658A2 Fused-aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
01/27/2005WO2005007167A1 Solid pharmaceutical preparation
01/27/2005US20050020532 Partial and full agonists of A1 adenosine receptors
01/27/2005CA2532093A1 Solid formulation
01/26/2005EP1500657A1 Substituted pyrazoles as P38 kinase inhibitors
01/26/2005EP1499713A2 Genomic library of cyanophage s-2l and functional analysis
01/26/2005EP1499613A1 Thioxanthine derivatives as myeloperoxidase inhibitors
01/26/2005EP1499305A2 Use of ep4 receptor ligands in the treatment of il-6 involved diseases
01/25/2005US6846927 Multistep synthesis of penciclovir or famciclovir starting with 2-amino-6-chloropurine
01/20/2005US20050014943 Reacting 5-aminoimidazole-4-carboxamide with triethyl orthoformate; cyclization; hydrolysis
01/20/2005US20050014811 Such as 4-cyclopentylamino-benzenesulfonic acid 2-(3,4-dimethoxy-phenylamino)-1H-benzoimidazol-5-yl ester; cyclin-dependent kinase inhibitors that are aimed to be more active than flavopiridol
01/19/2005EP1496896A1 Inhibitors of akt activity
01/19/2005EP1124562B1 Combination therapy to treat hepatitis b virus
01/19/2005CN1566118A Antiviral activity possessed compound and preparation method thereof
01/13/2005WO2005003100A2 4-arylamino-quinazolines as activators of caspases and inducers of apoptosis
01/13/2005WO2004078943A3 Alternative heterocycles for dna recognition
01/13/2005WO2004050035A3 Benzimidazoles and analogs thereof as antivirals
01/13/2005US20050009846 2,6,9-Substituted purine derivatives and their use in the treatment of proliferative disorders
01/13/2005US20050009842 2-hydroxymethylcyclopropylidene methylpurines and -pyrimidines as antiviral agents
01/13/2005US20050009829 1-Substituted 2-carboxamide derivatives of fused ring imidazoles, e.g., -[5-(5-Chloro-thiophen-2-yl)-isoxazol-3-ylmethyl]-1H-benzoimidazole-2-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide
01/13/2005US20050009076 Conjugate of hormone (thyroxine) and inosine-5'-monophosphate dehydrogenase inhibitor (such as mycophenolic acid)
01/13/2005CA2531327A1 Compounds and therapeutical use thereof
01/12/2005CN1564688A Methods of treating pulmonary disease
01/12/2005CN1563007A 9-(2-fatty ester ethoxy methyl) guanine, liposome, and preparation emthod
01/12/2005CN1563006A Synthesizing nucleoside analog for antivirus
01/11/2005US6841549 Condensed imidazole compounds and a therapeutic agent for diabetes mellitus
01/06/2005WO2005000850A2 Novel crystalline forms of valacyclovir hydrochloride
01/06/2005WO2005000404A2 Heterocyclic compounds for preventing and treating disorders associated with excessive bone loss
01/06/2005WO2005000313A1 Antiepileptic agent
01/06/2005WO2004073595A3 Novel purine derivatives, preparation method thereof, application of same as medicaments, pharmaceutical compositions and novel use
01/06/2005US20050004207 Substituted isoindoles and the use thereof
01/06/2005US20050004117 Such as 2-[2-(3-Amino-piperidin-1-yl)4-oxo-4H-quinazolin-3-ylmethyl]-benzonitrile; type 2 diabetes mellitus, diabetic dislipidemia, impaired glucose tolerance
01/06/2005US20050004110 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease
01/06/2005CA2530649A1 Antiepileptic agent
01/06/2005CA2527708A1 Crystalline forms of valacyclovir hydrochloride
01/06/2005CA2527079A1 Heterocyclic compounds for preventing and treating disorders associated with excessive bone loss
01/05/2005EP1493743A1 Substituted bipiperidine intermediates and derivatives thereof
01/05/2005EP1492803A1 New analogs of nitrobenzylthioinosine
01/05/2005EP1492791A1 Crystal and solvate of 2-amino-6-benzyloxypurine and production methods thereof
01/05/2005CN1183133C 2-amino-6-anilino-purines and their use as medicaments
01/04/2005US6838559 Such as 2-((6-(((4-(3,4-dimethoxyphenyl)methyl)amino)-7-ethyl-7H-purin-2-yl)amino) -4,5-methyl-N-phenyl-5-thiazole-carboxamide for treatment of lymphocyte mediated diseases such as transplant rejection and graft versus host disease
01/04/2005CA2350854C 1,4-dihydropyridine derivatives and methods of producing the same
12/2004
12/30/2004US20040267034 Hydrogenation process
12/30/2004US20040266795 reacting a compound of formula I (acetic acid 2-acetoxymethyl-4-(5-amino-7-chloro-imidazo[4,5-b]pyridin-3-yl)-butyl ester) in the presence of a catalyst in a C1-C6 alkyl acetate and ammonium formate
12/30/2004US20040266780 Inhibitors of human phosphatidyl-inositol 3-kinase delta
12/29/2004WO2004113357A2 Nucleoside analog inhibitors of reverse transcriptase
12/29/2004WO2004009091A8 Purine derivatives as liver x receptor agonists
12/29/2004EP1490369A1 Production method of 2,6-dihalopurine
12/29/2004EP1490368A2 2,2-bis(hydroxymethyl)cyclopropylidenemethyl - purines and -pyrimidines as antiviral agents
12/29/2004EP1490367A1 Imidazopyridine derivatives as kinase inhibitors
12/29/2004EP1490366A1 Novel alkoxypyridine-derivatives
12/29/2004EP1490015A2 Novel 2-amino-9-((2-hydroxymethyl) cyclopropylidenemethyl) purines as antiviral agents
12/29/2004CN1558761A Substituted benzimidazole compounds and their use for the treatment of cancer
12/29/2004CN1557841A Process for synthetic extraction of polysaccharides, tea-polyphenol, theanine, caffeine from tea
12/29/2004CN1182137C Preparation method and use of sodium Penciclovir sodium hydrate
12/23/2004WO2004111049A1 Ganciclovir sodium salt in crystalline form
12/23/2004WO2004111007A1 1-aryl-4-(aryloxycarbonyl)-piperazine derivatives for use as inhibitors of hormone sensitive lipase
12/23/2004WO2004110379A2 A1 adenosine receptor antagonists
12/23/2004WO2004110343A2 2-amino-9-(2-substituted ethyl)purines and preparing methods for 9-[4-acetoxy-3-(acetoxymethyl)but-1-yl]- 2- aminopurine using the same
12/23/2004WO2004074270A3 Inhibitors of hepatitis c virus rna-dependent rna polymerase, and compositions and treatments using the same
12/23/2004WO2004040003A3 Nucleotide-binding protein-directed probes and methods of their synthesis and use
12/23/2004US20040259889 Vasconstriction ; administering adenosine receptor antagonist
12/23/2004US20040259870 Antidiabetic agents; obesity; controlling appetite
12/23/2004US20040259833 DNA methyl transferase inhibitors
12/23/2004US20040259832 Synergistic mixture of thymidine kinase inhibitor and viricides
12/23/2004CA2798163A1 Inosine derivatives and production methods therefor
12/23/2004CA2727748A1 Inosine derivatives and production methods therefor
12/23/2004CA2528367A1 A1 adenosine receptor antagonists
12/23/2004CA2526518A1 1-aryl-4-(aryloxycarbonyl)-piperazine derivatives for use as inhibitors of hormone sensitive lipase
12/22/2004CN1556808A Heterocyclic compound based on N6-substituted adenine, methods of their preparation, their use for preparation of drugs, cosmetic preparations and growth regulators, pharmaceutical preparations, cosme
12/21/2004US6833378 Pyridines, pyrimidines, purinones, pyrrolopyrimidinones and pyrrolopyridinones; useful in the treatment disorders including CNS and stress-related disorders.
12/21/2004US6833375 As inhibitors of the retinoic acid-metabolism, as drugs
12/16/2004WO2004035740A3 Aromatic bicyclic heterocyles to modulate 1l - 12 production
12/16/2004US20040254201 Substituted-1,3-oxathiolanes and substituted-1,3-dioxolanes with antiviral properties
12/16/2004US20040254141 Therapy for hepatitis B virus infection ; antiproliferative agents; antitumor agents; anticancer agents
12/16/2004US20040253647 Evaluating modulators effectiveness as treatment for alzheimer's via quantifying amyloid precursor protein peptide cleavage products present after exposure agonist/antagonist
12/15/2004EP1485388A2 Topiramate salts and compositions comprising and methods of making and using the same
12/15/2004EP0788507B1 L-pyranosyl nucleosides
12/15/2004CN1554350A Nucleotide analog composition and synthesis method
12/14/2004US6831174 Processes for preparing substituted 1, 3-oxathiolanes with antiviral properties
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