Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559) |
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04/18/1989 | US4822882 DC-52 derivatives and their antitumor use |
04/18/1989 | US4822801 4-oxo-1,4-dihydroquinoline-3-carboxylic acid derivative as antibacterial agents |
04/18/1989 | US4822799 Pyrazolopyridine analogs of mevalonolactone and derivatives thereof useful for inhibiting cholesterol biosynthesis in mammals |
04/18/1989 | US4822788 Microbiocides, beta-lactamase inhibitors |
04/18/1989 | CA1252790A1 4-aryl-4-piperidinecarbinols |
04/18/1989 | CA1252786A1 Substituted spiro-quinolines, spiro-naphthyridines and spiro-(aza-naphthyridines), pharmaceutical compositions containing them and processes for the preparation of such compounds and compositions |
04/12/1989 | EP0311313A2 Heterocyclic spiro compounds and their preparation |
04/12/1989 | EP0311303A2 4-aminopyridine derivatives |
04/12/1989 | EP0311135A2 Heterocyclic substituted azoles and azines, process for their preparation and their use as an agent with herbicide activity |
04/12/1989 | EP0311010A2 Alpha,Alpha-disubstituted aromatics and heteroaromatics as cognition enhancers |
04/12/1989 | EP0310950A1 Quinoline intermediates for the synthesis of 1H-imidazo[4,5-c]quinolines and 1H-imidazo[4,5-c]quinolin-4-amimes |
04/12/1989 | EP0310917A2 Quinolonecarboxylic acids bearing C(7) carbon-functionality and a method for their preparation |
04/11/1989 | US4820822 Antihistamine, antiserotonine agents |
04/11/1989 | US4820716 7-(1-Pyrrolidinyl)-quinolonecarboxylic acid derivatives |
04/11/1989 | US4820710 Benzimidazole derivatives and pharmaceutical compositions containing them |
04/11/1989 | CA1252467A1 Process for the preparation of eburnamonine derivatives |
04/11/1989 | CA1252466A1 Process for producing 1,2,5,6-tetrahydro-4h- pyrrolo¬3,2,1-ij|-quinolin-4-one, and 5- halo-1,2,3-(1,2-dihydropyrrolo)-4-quinolones as intermediates for carrying out the process |
04/06/1989 | WO1989002740A1 4-aminopyridine derivatives |
04/06/1989 | WO1989002739A1 4-aminopyridine derivatives |
04/05/1989 | EP0310386A2 4-Aryl-5-carbamoyl-1,4-dihydropyridines |
04/05/1989 | EP0309952A2 Anti-retroviral castanospermine esters |
04/04/1989 | US4818819 Process for the preparation of fused pyridine compounds |
04/04/1989 | US4818759 Rheumatoid arthritis |
04/04/1989 | US4818754 Certain anti-inflammatory pyrazolo [4,3-b] pyridine 7-amines |
04/04/1989 | CA1252100A1 (1h-tetrazol-5-yl)tetrazolo¬1,5-a|-quinolines and related compounds |
04/04/1989 | CA1252093A1 Quinazolines, process for their preparation and pharmaceutical compositions containing them |
03/30/1989 | DE3730222A1 3-Benzhydryl-3,7-diazabicyclo[3.3.1]nonane compounds, process for their preparation and medicaments containing these compounds |
03/30/1989 | DE3717071A1 Radical anion salts of derivatives of 1,4,5,8-naphthalene-tetracarboxylic acid, process for their preparation, and their use |
03/29/1989 | EP0309423A2 New benzimidazoline-2-oxo-1-carboxylic acid derivatives useful as 5-ht receptor antagonists |
03/29/1989 | EP0309422A2 New amidino tricycle derivatives |
03/29/1989 | EP0309402A1 N-substituted hindered amine stabilizers |
03/29/1989 | EP0309401A1 Stabilization of coatings with N-hydroxy hindered amines |
03/29/1989 | EP0309400A2 N-acyloxy hindered amine stabilizers |
03/29/1989 | EP0308917A2 Imidazopyridine compound, a process for preparation thereof and pharmaceutical compositions comprising them |
03/29/1989 | EP0308913A2 2,6-Methanopyrrolo-3-benzazocines, a process and intermediates for their preparation and their use as medicaments |
03/29/1989 | EP0308843A2 Bispidin derivatives as class III antiarrhythmics |
03/29/1989 | EP0308444A1 PYRROL 1.2-b]AZINES |
03/29/1989 | CN1032011A Pyrrolo 1,2-a) imidazole and pyrrolo 1,2-a) pyridine derivatives and their use as 5-lipoxygenase pathway inhibitors |
03/28/1989 | US4816463 Substituted diimidazo [1,5-a: 4',5'-d]pyridines having antihypertensive activity |
03/28/1989 | US4816459 Antiallergens |
03/28/1989 | US4816457 Hypotensive agents, bronchodilators, eyes |
03/28/1989 | US4816453 Antiemetics |
03/23/1989 | DE3730667A1 Novel ss-carbolines |
03/23/1989 | DE3730224A1 3-Cinnamyl-3,7-diazabicyclo[3.3.1]nonane compounds, process for their preparation and medicaments containing these compounds |
03/22/1989 | EP0308084A1 Pyridine derivative |
03/22/1989 | EP0307814A2 Tetracyclic quinazoline derivatives, preparation and use |
03/22/1989 | CN1031842A Diazole |
03/22/1989 | CN1031841A Improvements in or relating to specific 5-ht3 antagonists |
03/21/1989 | US4814457 2,2*-bipyridine or 1-10-phenantroline compounds |
03/21/1989 | US4814450 Central nervous system disorders |
03/21/1989 | CA1251449A1 TETRAHYDRO-.beta.-CARBOLINE DERIVATIVES AND PROCESS FOR THE PREPARATION THEREOF |
03/15/1989 | EP0307172A2 Improvements in or relating to specific 5-HT3 antagonists |
03/15/1989 | EP0307142A1 Thiadiazoles useful in the treatment of senile dementia |
03/15/1989 | EP0307078A1 Quinoline derivatives, process for their preparation and pharmaceutical compositions containing them |
03/15/1989 | EP0307014A1 Anti-allergic 2-(heterocyclyl alkyl) imidazo pyridines and 2-(heterocyclyl alkyl) purines |
03/15/1989 | EP0306871A2 3,7-Diazabicyclo [3,3,1] nonane compounds, process for their preparation and medicaments containing them |
03/15/1989 | EP0306826A1 N-(substituted alkylidene)fused bicycloalkylidene and hetero-alkylidene quinolinamines, a process for their preparation and their use as medicaments |
03/15/1989 | EP0306698A1 Condensed diazepinones, processes for their preparation, and medicaments containing these compounds |
03/14/1989 | US4812568 Cyclization of a 2,5-di(phenylamino)-3,6-dihydroterephthalate |
03/14/1989 | US4812462 4,5,6,7-tetrahydro-1H-imidazo[4,5-c]pyridine-6-carboxylic acid analogs having antihypertensive activity |
03/14/1989 | CA1251211A1 Process for the preparation of triazole derivatives |
03/14/1989 | CA1251208A1 Fused tricyclic derivatives of naphthyridinone, pyridone and quinolone and the corresponding thiones |
03/09/1989 | WO1989000571A3 Bicyclic compounds, their use as pharmaceuticals, their preparation, and intermediates useful in their preparation |
03/08/1989 | EP0306323A2 Lactam derivatives |
03/08/1989 | EP0306300A2 Pyrrolo(1,2-a)imidazole and imidazo(1,2-a)pyridine derivatives and their use as 5-lipoxygenase pathway inhibitors |
03/08/1989 | EP0306148A2 Azabicyclic ethers |
03/08/1989 | EP0305889A1 Process for the preparation of 4-alkoxyalkyl-beta-carbolines |
03/08/1989 | EP0305744A2 Quinoline, naphthyridine and benzoxazine-carboxylic acid derivatives and their use as antibacterial agents |
03/08/1989 | EP0305667A2 Improved process for producing 5,10-dideaza-(5,6,7,8)-tetrahydrofolic acid |
03/07/1989 | US4810828 Antiarthritic, psoriasis |
03/07/1989 | US4810711 1-(acylaminomethyl)imidazo(1,2-A)quinoline derivatives, their preparation and their application in therapy |
03/07/1989 | US4810708 Antiallergy, immunosuppressive |
03/07/1989 | CA1250846A1 6-fluoro-1,4-dihydro-4-oxo-7-(4-pyridyl)-1,8- naphthyridine-3 carboxylic acid compounds |
03/07/1989 | CA1250845A1 Imidazo¬1,5-a|pyridine derivatives |
03/07/1989 | CA1250844A1 Substituted imidazo¬1,5-a|pyridines, process for their manufacture, pharmaceutical preparations containing these compounds and their therapeutic application |
03/01/1989 | EP0305322A2 Isoxazole-beta-carboline derivatives |
03/01/1989 | EP0304889A2 Novel aristeromycin/adenosine derivatives |
03/01/1989 | EP0304624A2 Benzimidazol-2-yl-pyridinum compounds |
03/01/1989 | CN1031378A Antibiotic compounds |
03/01/1989 | CN1031376A Pyrazolopyridine compound andprocesses for preparation thereof |
02/28/1989 | US4808620 Pyrazolopyridine compounds, their preparation and use as platelet aggregation inhibitors |
02/28/1989 | US4808618 Antiallergens |
02/28/1989 | US4808605 Tetrahydronaphthalene derivatives as calcium antagonists |
02/28/1989 | US4808596 Imidazo[4,5-b]pyridine compounds and pharmaceutical compositions containing same |
02/28/1989 | US4808594 Anxidytic and hypnotic properties |
02/28/1989 | US4808587 5-substituted pyrido[2,3-d]pyrimidine-2,4-diones |
02/28/1989 | US4808585 Solutions of lactic acid salts of piperazinylquinolone- and piperazinyl-azaquinolone-carboxylic acids |
02/28/1989 | US4808583 Solutions of lactic acid salts of piperazinylquinolone- and piperazinyl-azaquinolone-carboxylic acids |
02/28/1989 | US4808506 Photoconductive imaging members with imidazole perinones |
02/28/1989 | CA1250582A1 Tetrahydrocorynantheine derivatives and process for their preparation |
02/28/1989 | CA1250579A1 Heterocycle-fused pyrazolo (3,4-d) pyridin-3-ones |
02/23/1989 | WO1989001474A1 Peroxide free radical initiators containing hindered amine light stabilizer groups |
02/22/1989 | EP0304330A1 Carbamoylpyrrolidone derivatives, their use and preparation |
02/22/1989 | EP0304223A2 Beta-carbolines as cholecy-stokinin and gastrin antagonist |
02/22/1989 | EP0304158A1 Cephalosporins, processes for their preparation and pharmaceutical compositions containing them |
02/22/1989 | EP0304087A2 Quinolone and naphthyridine antibacterial agents containing an alpha-amino acid in the side chain of the 7-substituent |
02/22/1989 | CN1031227A Acrylate fungicides |
02/21/1989 | US4806560 Imidazo[4,5-b]pyridin-2-one derivatives |
02/21/1989 | US4806545 (-)-1β-ethyl-1α-hydroxymethyl-1,2,3,4,6,7,12, 12Bα-octahydroindolo(2,3-A)quinolizine, process for its preparation and pharmaceutical compositions containing same |
02/21/1989 | US4806541 Antibacterial agents |