Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
06/2001
06/26/2001US6251902 Dipeptide derivatives as growth hormone secretagogues
06/26/2001US6251894 1-(1,2-disubstituted piperidinyl)-4 (fused imidazole)-piperidine derivatives
06/26/2001US6251893 Bicyclic piperidine and piperazine compounds having 5-HT6 receptor affinity
06/26/2001CA1341261C Process for the synthesis of 3',4'-anhydrovinblastine, vinblastine and vincristine
06/21/2001WO2001044260A2 Novel purines
06/21/2001WO2001044259A1 Purine derivatives
06/21/2001WO2001044258A1 Novel heterocycles
06/21/2001WO2001044257A1 Proton pump inhibitors
06/21/2001WO2001044248A1 Imidazopyrimidinyl and imidazopyridinyl derivatives
06/21/2001WO2001044247A2 Agents and methods for the treatment of proliferative diseases
06/21/2001WO2001044246A1 Bicyclic inhibitors of glycogen synthase kinase 3
06/21/2001WO2001044245A1 Saccharin derivatives as orally active elastase inhibitors
06/21/2001WO2001044244A1 Pyrazolo-pyridine derivatives as ligands for gaba receptors
06/21/2001WO2001044243A2 Novel heteroaryl-diazabicycloalkanes
06/21/2001WO2001044239A2 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
06/21/2001WO2001044235A2 Agents and methods for the treatment of proliferative diseases
06/21/2001WO2001044193A1 1,3,4-substituted piperidine analogs and uses thereof in treating addictions
06/21/2001WO2001043741A1 Cytotoxic n-unsubstituted indoles and cyclopent(b)indoles and method of making and using same
06/21/2001US20010004669 For treatment of depression, anxiety, eating disorders, obesity, drug abuse, cluster headache, migraine, pain and chronic paroxysmal hemicrania and headache associated with vascular disorders
06/21/2001DE19961302A1 Treatment of erectile dysfunction using new or known imidazo(1,5-a)pyrido(3,2-e)pyrazinones as phosphodiesterase inhibitors, some of which are also useful for treating cardiovascular disorders
06/21/2001CA2395486A1 Saccharin derivatives as orally active elastase inhibitors
06/21/2001CA2395088A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
06/21/2001CA2395075A1 1,3,4-substituted piperidine analogs and uses thereof in treating addictions
06/21/2001CA2394654A1 Proton pump inhibitors
06/21/2001CA2394650A1 Novel heterocycles
06/21/2001CA2394646A1 Novel purines
06/21/2001CA2394573A1 Purine derivatives
06/21/2001CA2392992A1 Imidazopyrimidinyl and imidazopyridinyl derivatives
06/21/2001CA2392944A1 Pyrazolo-pyridine derivatives as ligands for gaba receptors
06/20/2001EP1108722A1 Trazodone hydrochloride and process for its preparation
06/20/2001EP1107966A2 Oxo-pyridoimidazole-carboxamides: gaba brain receptor ligands
06/20/2001EP1107959A2 Quinazoline derivatives as medicaments
06/20/2001EP1107758A2 Use of piperidines and/or piperazines as inhibitors of p38-alpha kinase
06/20/2001EP1107753A1 Multivalent agonists, partial agonists, inverse agonists and antagonists of the 5ht2 receptors
06/20/2001EP0808303B1 5-(4-subst.-piperidinyl-1)-3-aryl-pentanoic acid derivatives as tachykinin receptor antagonist
06/20/2001EP0714394B1 Antipsychotic method with thiadiazole and oxadiazole derivatives
06/20/2001CN1300285A Oxyiminoalkanoic acid derivatives
06/20/2001CN1300277A Novel substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
06/20/2001CN1067394C Process for preparation of enantiomerically pure cycloalkano-indol-and azaindol-and pyrimido [1,2a] indol-carbocylic acids and their activated derivatives
06/20/2001CN1067387C 1,2,3,4-tetrahydroquinoxalindione derivative
06/20/2001CN1067386C 5-heteroarylindole derivatives as benzodiazepine receptor site agnoists and analagonists
06/19/2001USRE37234 Nitrosated and nitrosylated phosphodiestrase inhibitor compounds, compositions and their uses
06/19/2001US6248884 Particularly well suited for use in automated fluorescence-based dna sequencing systems using an excitation light source having a wavelength greater than about 630 nm, e.g., a helium-neon gas laser or a solid state diode laser.
06/19/2001US6248755 Antiinflammatory agents; antiallergens; autoimmune diseases
06/19/2001US6248753 Bicyclic compounds
06/19/2001US6248717 Tartrate salt of a substituted dipeptide as growth hormone secretagogue
06/19/2001CA2095444C Fused pyrazine derivatives
06/14/2001WO2001042247A1 Fused heterotricyclic compounds, process for preparing the compounds and drugs containing the same
06/14/2001WO2001042245A1 Neurotrophic bicyclic diamides
06/14/2001WO2001042244A1 Novel 1,8-naphthyridin-2(1h)-one derivatives
06/14/2001WO2001042243A2 Protein kinase inhibitors
06/14/2001WO2001042242A1 Antibacterial heterobicyclic substituted phenyl oxazolidinones
06/14/2001WO2001042216A2 Caspase inhibitors and uses thereof
06/14/2001WO2001042213A1 Urea compounds having muscarinic receptor antagonist activity
06/14/2001WO2001042212A1 Carbamate derivatives having muscarinic receptor antagonist activity
06/14/2001WO2001027111A3 Bicyclic imidazo-3-yl-amine derivatives
06/14/2001WO2001016133A3 8-substituted-6-trifluoromethyl-9-pyrido[3,2-g]quinoline compounds as androgen receptor modulators
06/14/2001WO1999067250A8 Syntheses of a variety of lamellarin compounds and analogues
06/14/2001US20010003779 Camptothecin analogs and methods of preparation thereof
06/14/2001CA2733434A1 Caspase inhibitors and uses thereof
06/13/2001EP1106178A1 Remedies for multiple sclerosis
06/13/2001EP1105393A1 Bicyclic piperidine and piperazine compounds having 5-ht 6? receptor affinity
06/13/2001EP1105391A2 New compounds
06/13/2001EP1105390A2 New compounds
06/13/2001EP1105389A1 Integrin receptor antagonists
06/13/2001EP1105387A1 Prodrugs of proton pump inhibitors
06/13/2001EP1105368A1 Photoactivatable bases containing nitrogen
06/13/2001EP1105120A2 NON-PEPTIDE GnRH AGENTS, METHODS AND INTERMEDIATES FOR THEIR PREPARATION
06/13/2001EP0805812B1 Bicyclic substituted hexahydrobenz(e)isoindole alpha-1- adrenergic antagonists
06/13/2001EP0666858B1 5-arylindole derivatives and their use as serotonin (5-ht 1) agonists
06/13/2001DE19955634A1 Kupplungs-Kondensations-Synthese von Heterocyclen Clutch condensation synthesis of heterocycles
06/13/2001CN1299361A Hypnotic beta-carboline derivatives, process for their prepn. and their use as medicinal products
06/13/2001CN1299282A Vitronectin receptor antagonists
06/13/2001CN1067072C Tricycle compounds, their prodn. and use
06/13/2001CN1067071C Carboline derivatives
06/12/2001US6245808 Oxy-vanadium (IV) complexes having spermicidal activity
06/12/2001US6245779 Naphthyridine derivatives
06/12/2001US6245778 1,6-naphthyridine anti-convulsants
06/12/2001US6245776 Drug mixture of immune response modifier, fatty acid, preservative and carbomer
06/12/2001US6245775 Anticholesterol agents; cardiovascular disorders
06/12/2001US6245774 Tri-substituted phenyl or pyridine derivatives
06/12/2001US6245770 Fungicidal pyrimidinones
06/12/2001US6245769 Heterocyclyl-substituted ring-fused pyridines and pyrimidines as corticotropin releasing hormone(CRH) antagonists, useful for treating CNS and stress-related disorders
06/12/2001US6245403 Using lasers
06/12/2001CA2207784C Certain pyrrolopyridine derivatives; novel crf1 specific ligands
06/11/2001WO2001044230A1 1-(aminophenyl)-2-pyrrolidones as integrin inhibitors
06/11/2001CA2393310A1 1-(aminophenyl)-2-pyrrolidones as integrin inhibitors
06/07/2001WO2001040227A1 Triazaspiro[5.5]undecane derivatives and drugs containing the same as the active ingredient
06/07/2001WO2001040226A1 Agents for improving learning or memory
06/07/2001WO2001040225A1 Remedies or preventives for frequent urination or urinary incontinence
06/07/2001WO2001040224A1 Diketopiperazine derivatives to inhibit thrombin
06/07/2001WO2001040217A1 Novel benzoimidazole derivatives useful as antiproliferative agents
06/07/2001WO2001040189A1 Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
06/07/2001WO2001040185A1 Compounds, compositions, and methods for stimulating neuronal growth and elongation
06/07/2001WO2001039759A2 Sulfonic acid or sulfonylamino n-(heteroaralkyl)-azaheterocyclylamide compounds
06/07/2001WO2001039723A2 Triazospiro compounds having nociceptin receptor affinity
06/07/2001WO2001025213A3 Pyrrolo imidazole derivatives and their use as medicaments
06/07/2001WO1999063940A3 INHIBITORS OF H+K+-ATPase
06/07/2001DE19952146A1 Arylalkane, Arylalkene und Aryl-azaalkane, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung Arylalkanes, aryl alkenes and aryl azaalkane, pharmaceutical compositions containing them and methods for their preparation
06/07/2001DE19948438A1 New azino-fused bicyclic imidazolyl-amine compounds, obtained by reacting amide, amine and aldehyde, useful as analgesics