Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
04/2002
04/25/2002US20020049223 Quinoline and naphthyridine carboxylic acid antibacterials
04/25/2002US20020049214 Aralkyl and aralkylidene heterocyclic lactams and imides as selective agonists and antagonists of serotonin 1 (5-HT1) recepor, used in treating hypertension and all forms of depression
04/25/2002US20020049212 Benzimidazole compounds and salts containing piperidine ring are useful in treatment or prevention or medical conditions selected from pain, and inflammatoy diseases; analgesics
04/25/2002US20020049211 Combination treatment for depression and anxiety
04/25/2002US20020049210 Heteroaryl amines as novel acetylcholinesterase inhibitors
04/25/2002US20020049209 Dopamine D4 ligands for the treatment of novelty-seeking disorders
04/25/2002US20020049207 Nitrogen containing heterobicyclic compounds for treating disorders manifesting hypersecretion of corticotropin releasign factor(CRF) in a warm-blooded animals, such as stroke
04/25/2002US20020049196 Hexahydro-pyrazolo-(4,3-c)pyridine derivatives useful for increasing the endogenous production or release of growth hormone in a human or other animal, thus treat or prevent osteoporosis
04/25/2002US20020049195 Urea compounds that are muscarinic receptor antagonists and agonists, administering to the mammal the urea compound to treat urinary incontinence, chronic pulmonary obstructive disease, asthma, hyper salivation, blurred vision etc.
04/25/2002US20020049194 A benzoazepin or benzodiazepin derivatives, shows excellent anti-vasopressin activity, vasopressin agonistic activity and oxytocin antagonistic activity, and are useful as antagonist
04/25/2002US20020049189 Vanadium (IV) complexes containing catecholate ligand and having spermicidal activity
04/25/2002CA2426487A1 Ep4 receptor inhibitors to treat rheumatoid arthritis
04/25/2002CA2423933A1 Pharmaceutically active sulfanilide derivatives
04/25/2002CA2423789A1 Bridged piperazine derivatives
04/24/2002EP1198233A1 Sulfonamide and sulfamide substituted imidazoquinolines
04/24/2002EP1198232A1 Urea substituted imidazoquinolines
04/24/2002CN1346354A Substituted benzoylpyrazoles as herbicides
04/24/2002CN1346351A 1,2-benzothiazepines for the treatment of hyperlipidemic diseases
04/24/2002CN1346282A Use of a cyclooxygenase-2 inhibitor and one or more antineoplastic agents as combination therapy method in treating neoplasia
04/24/2002CN1346271A Quinazoline derivatives as angiogenesis inhibitors
04/24/2002CN1083453C Fused imidazole derivatives as emultidrug resistance modulators
04/24/2002CN1083452C Pyrido (2,3-d) pyrimidines for inhibiting protein tyrosine kinase mediated cellular proliferation
04/24/2002CN1083450C Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
04/24/2002CN1083244C Zilpaterol hydrochloride in specific crystallized formits prepn. process and intermediate products used
04/23/2002US6376676 Intermediates in the synthesis of (±)-camptothecin and related compounds and synthesis thereof
04/23/2002US6376670 Bactericide for grampositive bacteria
04/23/2002US6376669 Dye labeled imidazoquinoline compounds
04/23/2002US6376521 A3 adenosine receptor antagonists
04/23/2002US6376509 Melanocortin receptor agonists
04/23/2002US6376507 NK-1 receptor antagonists for the treatment of neuronal injury and stroke
04/23/2002US6376500 Substituted 2-(4-piperidyl)-4(3H)-quinazolinones and 2-(4-piperidyl)-4(3H)-azaquinazolinones
04/23/2002US6376499 Piperazine-amide compound with anticoagulant activity
04/23/2002US6376487 Oxadiazine derivatives
04/23/2002US6376472 Compounds having antihypertensive, cardioprotective, anti-ischemic and antilipolytic properties
04/18/2002WO2002030933A1 Substituted 3.4-dihydro-pyrido[1,2-a]pyrimidines
04/18/2002WO2002030932A2 N8,n13-disubstituted quino[4,3,2-kl]acridinium salts as therapeutic agents
04/18/2002WO2002030931A2 Aza- and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors
04/18/2002WO2002030930A2 Aza- and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors
04/18/2002WO2002030911A1 Pyrimidinone derivatives and their use in the treatment of atherosclerosis
04/18/2002WO2002030906A1 Anti-tumour compounds
04/18/2002WO2002030904A1 Pyridinone derivatives for treatment of atherosclerosis
04/18/2002WO2002030901A1 Process for making 3-amino-2-chloro-4-methylpyridine
04/18/2002WO2002030890A1 Nitrogenous five-membered ring compounds
04/18/2002WO2002030886A2 Heterocyclic angiogenesis inhibitors
04/18/2002WO2002030428A1 Use of substituted imidazo[1,2-a]pyridine-, imidazo[1,2-a]pyrimidine and imidazo[1,2-a]pyrazine-3-yl-amine derivatives for producing nos-inhibiting medicaments
04/18/2002WO2002030426A1 Aza- and polyaza-naphthalenyl-carboxamides useful as hiv integrase inhibitors
04/18/2002WO2001064681A3 3-(pyrolyllactone)-2-indolinone compounds as kinase inhibitors
04/18/2002US20020045756 Preparation of camptothecin and of its derivatives
04/18/2002US20020045747 Treating Alzheimer's disease both prophylactically and therapeutically
04/18/2002US20020045637 Novel 20,21-dinor-eburnamenine
04/18/2002US20020045630 Antiproliferative, -carcinogenic, -tumor and -diabetic agents; binding to or modulating the human kinase insert-domain-containing receptor (KDR) or the murine fetal liver kinase 1 (FLK-1) receptor; vasculogenesis; angiogenesis
04/18/2002US20020045628 Antidepressants; anxiolytic agents; serotonin-affected nervous system disorders; acting at the 5-HT1a autoreceptors concommitantly with 5-HT transporters; antiserotonin agents; serotonin reuptake inhibitors; HT3 receptor antagonists
04/18/2002US20020045624 Treatment of central nervous system (CNS) dysfunctions, neurodegenerative diseases and neurotoxic injury following hypoxia, anoxia or ischemia of stroke, cardiac arrest or perinatal asphyxia; antipsychotic and -convulsant agents
04/18/2002US20020045623 Stable; potent; penetrates cell membranes; effectively hinders cellular apoptosis; Antiinflammatory agents, Ischemic agents, cancer, autoimmune diseases and nervous system disorders.
04/18/2002US20020045622 Growth hormone secretagogues
04/18/2002US20020045617 Act preferentially on M4 receptors; side effect reduction; used to treat nervous system disorders, psychological disorders and as an analgesic; Alzheimer's disease; Cognition activators.
04/18/2002US20020045613 1-aroyl-piperidinyl benzamidines
04/18/2002US20020045550 Uracil substituted phenyl sulfamoyl carboxamides
04/18/2002US20020044899 Controlled, super-fine grinding so particles react completely during leaching; extraction of copper from copper sulfide ores and concentrates
04/18/2002US20020043656 1-Phenyl-5-(p-methoxyphenyl)-3-(1,8-naphthoylene-1',2' -benzimidazol-4-yl)-2-pyrazol
04/18/2002DE10050663A1 Use of amino-substituted imidazo(1,2-a)pyridine, imidazo(1,2-a)pyrimidine and imidazo(1,2-a)pyrazine derivatives as NO synthase inhibitors, e.g. in treatment of migraine and neurodegenerative diseases
04/18/2002DE10050662A1 New substituted dihydropyrido-pyrimidine derivatives, useful for treating e.g. pain, urinary incontinence and tinnitus
04/18/2002CA2459746A1 Pyrimidinone derivatives and their use in the treatment of atherosclerosis
04/18/2002CA2425672A1 Use of substituted imidazo[1,2-a]-pyridin-,pyrimidin-and -pyrazin-3-yl-amine derivatives in the preparation of medicaments for inhibiting nos
04/18/2002CA2425666A1 Substituted 3.4-dihydro-pyrido[1,2-a]pyrimidines
04/17/2002EP1197485A1 Cyclobuten-dione derivatives for use in the treatment of artherosclerosis
04/17/2002EP1196418A1 METHOD FOR PREPARING SUBSTITUTED 1,4]DIAZEPINO 6,7,1- i hi /i ]INDOL-4-ONES
04/17/2002EP1196410A1 Respiratory syncytial virus replication inhibitors
04/17/2002EP1196409A2 Respiratory syncytial virus replication inhibitors
04/17/2002EP1196408A1 Respiratory syncytial virus replication inhibitors
04/17/2002EP1196397A1 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases
04/17/2002EP1196391A1 Benzimidazolone derivatives and their use as phosphodiesterase inhibitors
04/17/2002EP1196390A2 Pyrazole compositions useful as inhibitors of erk
04/17/2002EP1196384A1 1-(aromatic- or heteroaromatic-substituted)-3-(heteroaromatic substituted)-1,3-propanediones and uses thereof
04/17/2002EP1196380A2 Indoles and indazoles for the treatment of migraine
04/17/2002EP1196167A1 Method of reducing neuronal injury or apoptosis
04/17/2002EP1042322B1 Kv2.1 ANTAGONISTS
04/17/2002EP1015434B1 Novel pyrimidin-4-one and pyrimidin-4-thione as fungicide
04/17/2002CN1345320A Diazabicyclic derivatives as nicotinic acetylcholine receptor ligands
04/17/2002CN1344717A Quaternary ammonium salt compound of piperazine with pain relieving effect
04/17/2002CN1082963C Isoxazolidine derivatives
04/17/2002CN1082962C 1,7-diaroxy-or 1,7-diarylthio-substituted perylene-3,4,9,10-tetracarboxylic acid and their dianhydrides and diimides, prep. and use thereof
04/16/2002US6372919 (+)-1-(3,4-dichlorophenyl)-3-azabicyclo[3.1.0]hexane, compositions thereof, and uses as an anti-depressant agent
04/16/2002US6372775 Reversal of multidrug resistance in human colon carcinoma cells
04/16/2002US6372767 Benzanilides as potassium channel openers
04/16/2002US6372758 Sulfamato hydroxamic acid metalloprotease inhibitor
04/16/2002US6372757 Phenylurea and phenylthio urea derivatives
04/16/2002US6372750 Heterocyclic compounds, process for their preparation and pharmaceutical compounds containing them and their use in the treatment of diabetes and related diseases
04/16/2002CA2103556C Bicyclopolyazamacrocyclophosphonic acids, their complexes and conjugates, for use as contrast agents, and processes for their preparation
04/16/2002CA2076948C Isatineoxime derivatives, their preparation and use
04/11/2002WO2002028865A2 Condensed pyridoindole derivatives
04/11/2002WO2002028860A2 Amino-substituted tetracyclic compounds useful as anti-inflammatory agents and pharmaceutical compositions comprising same
04/11/2002WO2002028859A2 Condensed pyridoindole derivatives
04/11/2002WO2002028858A2 Hexahydropyrazino `1'2' : 1, 6!- pyrido `3, 4-b! indole-1, 4-dione derivatives for the treatment of cardiovascular disorders and erectile disfunction
04/11/2002WO2002028840A1 Process for preparation of integrin receptor antagonist intermediates
04/11/2002WO2002028837A1 Metabotropic glutamate receptor antagonists
04/11/2002WO2002028831A1 Inhibitors of prenyl-protein transferase
04/11/2002WO2002028830A1 Novel phenylalanine derivatives
04/11/2002WO2002028395A1 Phosphoric acid salt of an integrin receptor antagonist
04/11/2002WO2002000683A3 Novel chain-breaking antioxidants