Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
02/2003
02/25/2003US6525215 HIV protease inhibitors
02/25/2003US6525200 Multicyclic aromatic compounds and uses thereof
02/25/2003US6525196 5HT1 antagonists for antidepressant therapy
02/25/2003US6525072 Prevention and treatment of cellular disorders such as cancer
02/25/2003US6525070 Bipiperidine derivatives as modulators of CCR3 activity and as H1 antagonists
02/25/2003US6525069 Such as N-(t-butyl)-N'-(2-((3-(4-fluorophenyl)methyl)piperi -dinyl)methyl)cyclohexyl)urea; prevention of asthma and other allergic diseases
02/25/2003US6525064 Immune response modifiers; can induce the biosynthesis of various cytokines;
02/25/2003US6525063 3,7-dimethyl-1,5-diazaanthraquinone for example
02/25/2003US6525059 Substituted pyrazoles as p38 kinase inhibitors
02/25/2003US6525056 Heterocyclyl-substituted ring-fused pyridines and pyrimidines as corticotropin releasing hormone (CRH) antagonists, useful for treating cns and stress-related disorders
02/25/2003US6525049 Pyrroloquinolones as antiviral agents
02/25/2003US6525048 Aminomethylphenoxymethyl/benzisoxazole substituted azabicyclic compounds; depression, generalized anxiety disorder, obesity, migraine; 2-(5-Fluoro-benzo(d)isoxazol-3-y)-7-(3-morpholin-4-ylmethylphenoxymethyl) -octahydro-pyrido(1,2-a)pyrazine;
02/25/2003US6525047 Which are growth hormone secretogogues and increase the level of endogenous growth hormone; treating osteoporosis, congestive heart failure, frailty associated with aging, obesity; accelerating bone fracture repair
02/25/2003US6525044 Treatment of neurological disorders related to beta -amyloid production such as Alzheimer's disease and Down's Syndrome.
02/25/2003US6525036 Compounds and compositions as protease inhibitors
02/25/2003US6524761 Photosensitive with respect to light from the visible to near infrared range; charging; electrostatic stability; mass spectrophotometry
02/25/2003CA2073747C Process for the continuous preparation of perylenetetracarboxylic diimides
02/20/2003WO2003014128A2 Tumour inhibiting cerium compounds
02/20/2003WO2003014121A1 Compounds, derivatives, compositions, preparation and uses
02/20/2003WO2003014120A1 Amino-substituted imidazopyridines for the treatment of gastrointestinal diseases
02/20/2003WO2003014119A1 Tricyclic epoxides
02/20/2003WO2003014118A1 THERAPEUTIC 1H-PYRIDO[4,3-b]INDOLES
02/20/2003WO2003014117A1 3-substituted pyrrolo[2.1-a]isoquinoline derivatives
02/20/2003WO2003014116A1 Pyrrolo[2.1-a]isoquinoline derivatives
02/20/2003WO2003014115A1 3-substituted pyrrolo (2.1-a) isoquinoline derivatives
02/20/2003WO2003014083A1 Spiro compounds
02/20/2003WO2003014075A2 Novel gamma secretase inhibitors
02/20/2003WO2002096516A8 Use of compositions comprising cyclooxygenase-2 selective inhibitors in combination with radiation for inhibition or prevention of cardiovascular disease
02/20/2003WO2002078602A3 Transdermal delivery of pergolide
02/20/2003WO2002072585A3 Substituted pyrazolopyrimidines and thiazolopyrimidines used as analgesics
02/20/2003WO2002065979A3 (diazolo-pyridinyl)-pyrimidines for use in treatment of cns disorders and diabetes
02/20/2003WO2002049993A3 High affinity small molecule c5a receptor modulators
02/20/2003US20030036651 As phosphodiesterase inhibitor for prophylaxis and therapy of bronchial asthma; pneumonic diseases, pulmonary emphysema, chronic obstructive pulmonary disease acute respiratory distress syndrome (ARDS), and other respiratory diseases
02/20/2003US20030036543 Especially as inhibitors of Aurora-2 and GSK-3, for treating diseases such as cancer, diabetes and Alzheimer's disease.
02/20/2003US20030036542 Derivatives of pyrimido[6.1-a]isoquinolin-4-one
02/20/2003US20030036473 Catalysts and methods for catalytic oxidation
02/20/2003CA2456599A1 Spiro compounds
02/20/2003CA2456550A1 Tumour inhibiting cerium compounds
02/20/2003CA2453537A1 Therapeutic 1h-pyrido¬4,3-b|indoles
02/20/2003CA2452802A1 Tricyclic epoxides
02/19/2003EP1284266A1 Novel indole derivatives exhibiting chymase-inhibitory activities and process for preparation thereof
02/19/2003EP1283836A2 Neuroprotective and anti-proliferative compounds
02/19/2003EP1283825A1 N-substituted peptidyl nitriles as cysteine cathepsin inhibitors
02/19/2003EP1283711A1 Peptide deformylase inhibitors
02/19/2003EP1165559B1 1,4-diazabicyclo[3.2.2]nonane-4-carboxylate and carboxamide derivatives, production and use thereof in therapeutics
02/19/2003EP0988302B1 Benzonaphthyridines
02/19/2003EP0920429B1 Substituted pyrido- or pyrimido-containing 6,6- or 6,7-bicyclic derivatives
02/19/2003CN1398189A Combination therapy of radiation and COX-2 inhibitor for treatment of neoplasia
02/19/2003CN1397557A NOvel octahydro-2H-pyridino-[1,2-a] pyrazine compound, its prepn. process and medicinal compound contg. them
02/19/2003CN1397551A N-([1,2,4]triazoleo azine group) benzene sulfonamide and pyridine sulfamide compound and their use as herbicide
02/19/2003CN1397549A Novel derivative of 2-azadicyclo-(2,2,1) heptane, its prepn. and use
02/19/2003CN1101649C Herbicidal synergistic compsn. and method of controlling weeds
02/18/2003WO2002016329A1 Novel phenylalanine derivatives
02/18/2003US6521656 Contacting sperm with a pyrazolo(1,5-a)pyridine acrosomal reaction induction promoter then joining with ovum
02/18/2003US6521638 2,3-dihydro-1H-isoindole derivatives useful as modulators of dopamine D3 receptors (antipsychotic agents)
02/18/2003US6521636 Imidazo-pyridines as corticotropin releasing factor antagonists
02/18/2003US6521629 2-amine substituted quinoline or quinozoline derivatives useful for treating benign prostatic hyperplasia
02/18/2003US6521623 N,N'-disubstituted benzimidazolone derivatives with affinity at the serotonin and dopamine receptors
02/18/2003US6521621 1-(1,2-disubstituted piperidinyl)-4-substituted piperazine derivatives
02/18/2003US6521620 Suppressing tumors, especially breast cancers; antiproli-ferative agents; arthritis, vascular restenosis, psoriasis and angiogenesis; extremely low cytotoxicity
02/18/2003US6521592 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
02/13/2003WO2003011864A1 DERIVATIVES OF TRIAZOLYL-IMIDAZOPYRIDINE AND OF THE TRIAZOLYLPURINES USEFUL AS LIGANDS OF THE ADENOSINE A2a RECEPTOR AND THEIR USE AS MEDICAMENTS
02/13/2003WO2003011862A1 Non-nucleoside reverse transcriptase inhibitors
02/13/2003WO2003011834A1 Novel vinyl n-(2-benzoylphenyl)-l-tyrosine derivatives and their use as antidiabetics etc
02/13/2003WO2003011824A1 Bicyclic modulators of androgen receptor function
02/13/2003WO2003011450A1 Processes for the production of amino-protected derivatives of 4-aminomethylene-pyrrolidin-3-one and/or 4-aminomethylene-pyrrolidin-3-alkoxyimino derivatives and/or gemifloxacin or a salt thereof
02/13/2003WO2003011297A1 N3-substituted 6-anilinopyrimidines and methods to treat gram-positive bacterial and mycoplasmal infections
02/13/2003WO2003011285A1 BENZIMIDAZO[4,5-f]ISOQUINOLINONE DERIVATIVES
02/13/2003WO2003011264A2 Betacarboline derivatives as gaba a-receptor-modulators having nmda-antagonistic activity for treating diseases of the central nervous system
02/13/2003WO2002087574A3 Use of pyridoindolone derivatives for preparing anticancer medicines
02/13/2003WO2002076988A3 Tert. alkylphenoxy substituted polycyclic compounds
02/13/2003WO2002059082A8 Aryl and aminoaryl substituted serotonin receptor agonist and antagonist ligands
02/13/2003WO2002046192A3 Thioether substituted imidazoquinolines
02/13/2003WO2002037927A3 Compounds and methods for promoting smoking cessation
02/13/2003WO2001072754A8 Alkylated imidazopyridine derivatives
02/13/2003US20030032805 Process for the preparation of high purity pemirolast
02/13/2003US20030032652 Hydroxamic and carboxylic acid derivatives
02/13/2003US20030032647 Aromatic nitrogen-containing 6-membered cyclic compounds
02/13/2003US20030028975 For dyeing hair
02/12/2003EP1282732A1 Fluorescent monomers and tagged treatment polymers containing same for use in industrial water systems
02/12/2003EP1282622A1 Crf receptor antagonists and methods relating thereto
02/12/2003EP1282621A1 Novel vitronectin receptor antagonists
02/12/2003EP1282600A1 Inhibitors of dipeptidyl peptidase iv
02/12/2003EP1282404A2 Method for preparing microparticles having a selected polymer molecular weight
02/12/2003EP0947514B1 Novel phenanethridinium derivatives
02/12/2003EP0816338B1 3-(bis-substituted-phenylmethylene)oxindole derivatives
02/12/2003EP0770079B1 Heterobicyclic derivatives
02/12/2003CN1396923A 4-Pyridyl-and 2,4-pyrimidinyl-substituted pyrrole derivatives and their use in pharmacy
02/12/2003CN1396921A Pyrrolo-isoquinoline and tetrahydropyrrolo-isoquinoline derivatives and their use as mediators of 5-HT7 reactor
02/12/2003CN1396915A Heterocylic derivative, its preparation method and medicine composition containing them
02/12/2003CN1396833A Integrin expression inhibitors
02/12/2003CN1396165A Zilpaterol hydrochcoride monohydrate
02/11/2003US6518426 Pyrimidine derivatives and methods of making and using these derivatives
02/11/2003US6518297 Selective 5-HT6 receptor ligands
02/11/2003US6518286 Compounds
02/11/2003US6518283 Squaric acid derivatives
02/11/2003US6518280 Antiviral and antitumor properties; immunomodulators and for inducing cytokine biosynthesis in animals
02/11/2003US6518276 Treating a p38 mediated disorders
02/11/2003US6518271 1H-imidazo[4,5-d]pyridazin-7-one, and corresponding thiones as corticotropin releasing factor (CRF) receptor ligands
02/11/2003US6518270 Heterocyclic compounds for inhibition of gastric acid secretion, processes for their preparation and pharmaceutical compositions thereof