Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
07/2003
07/16/2003EP1326867A2 Bridged piperazine derivatives
07/16/2003EP1326866A1 Substituted 3.4-dihydro-pyrido[1,2-a]pyrimidines
07/16/2003EP1326865A2 Aza- and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors
07/16/2003EP1326864A2 Aryl or heteroaryl fused imidazole compounds as anti-inflammatory and analgesic agents
07/16/2003EP1326863A2 Octahydro-indolizines and quinolizines and hexahydro-pyrrolizines
07/16/2003EP1326856A1 Pyridine derivatives with ikb-kinase (ikk-beta) inhibiting activity
07/16/2003EP1326846A1 Process for preparation of integrin receptor antagonist intermediates
07/16/2003EP1326841A1 Pyridinone derivatives for treatment of atherosclerosis
07/16/2003EP1326836A1 Process for making 3-amino-2-chloro-4-methylpyridine
07/16/2003EP1326619A2 Pyrrolidine modulators of ccr5 chemokine receptor activity
07/16/2003EP1326615A1 Phosphoric acid salt of an integrin receptor antagonist
07/16/2003EP1326613A1 Use of substituted imidazo 1,2-a]pyridine-, imidazo 1,2-a]pyrimidine and imidazo 1,2-a]pyrazine-3-yl-amine derivatives for producing nos-inhibiting medicaments
07/16/2003EP1326611A1 Aza- and polyaza-naphthalenyl-carboxamides useful as hiv integrase inhibitors
07/16/2003EP1326610A2 Aza-and polyaza-naphthalenyl carboxamides useful as hiv integrase inhibitors
07/16/2003EP1326606A2 Ep4 receptor inhibitors to treat rheumatoid arthritis
07/16/2003EP1165555B1 Aryl fused 2,4-disubstituted pyridines: nk3 receptor ligands
07/16/2003EP0787720B1 Pyridonecarboxylate derivative or salt thereof and antibacterial containing the same as active ingredient
07/16/2003EP0550550B1 3,9-diazabicyclo (3.3.1) nonan-7-yl derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them
07/16/2003CN1114608C Novel camptothecine analogues, prepn. method therefor, use thereof, and pharmaceutical compositions contg. same
07/16/2003CN1114605C Novel camptothecine derivatives
07/15/2003US6593357 Treating disease states in mammals that are alleviated by a protein kinase inhibitor, particularly diseases such as cancer, inflammatory disorders, restenosis, and cardiovascular disease.
07/15/2003US6593346 Substituted 3-(piperidin-1-ylmethyl)cyclopentylamines, useful as modulators of the chemokine receptors CCR-5 and/or CC R-3.
07/15/2003US6593344 These substances have especially high cytostatic activities and pronounced immunosuppressive properties which make them suitable for therapeutic treatment in broad tumor spectrum and autoimmune diseases
07/15/2003US6593338 Inhibit the binding of integrins to their ligands and are of use in the prophylaxis and treatment of immuno or inflammatory disorders or disorders involving the inappropriate growth or migration of cells.
07/15/2003US6593337 Tricyclic compounds useful as HIV reverse transcriptase inhibitors
07/15/2003US6593325 Method for the treatment of anxiety which comprises administering to a patient in need of such treatment an effective amount of the compound of claim 1 or a pharmaceutically acceptable salt thereof.
07/15/2003US6593013 Electroluminescence device, cyclic azine compound and production process of cyclic azine dye
07/10/2003WO2003055881A1 Pyrido(2,1-a)isoquinoline derivatives as dpp-iv inhibitors
07/10/2003WO2003055876A1 Chemokine receptor binding heterocyclic compounds with enhanced efficacy
07/10/2003WO2003055856A2 BICYCLIC LACTAM DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-α CONVERTING ENZYME (TACE)
07/10/2003WO2003055447A2 Heterocyclic acridone inhibitors of impdh enzyme
07/10/2003WO2003050119A3 Urea substituted imidazopyridines
07/10/2003WO2003022274A3 2-aroylimidazole compounds for treating cancer
07/10/2003WO2003010140A3 Hepatitis c virus polymerase inhibitors with heterobicyclic structure
07/10/2003WO2003006440A8 Amide-containing compound having improved solubility and method of improving the solubility of an amide-containing compound
07/10/2003WO2002059267A3 Constitutively desensitized g protein-coupled receptors
07/10/2003WO2001098269A3 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
07/10/2003US20030130518 They induce the biosynthesis of various cytokines and are useful in the treatment of viral and neoplastic diseases.
07/10/2003US20030130516 E.g., reacting a 6H-imidazo(4,5-c) tetrazolo(1,5-a)quinoline with triphenylphosphine and hydrolyzing the product thereof.
07/10/2003US20030130504 Antidepressants
07/10/2003US20030130302 Bactericides
07/10/2003US20030130299 Administering dosage of immunology response moderator
07/10/2003US20030130287 Psychological disorders; central nervous system disorders; antidepressants; Parkinson's disease; Alzheimer's disease;cardiovascular disorders
07/10/2003US20030130285 Controlling cell differentiation, cell proliferation
07/10/2003US20030130284 Animal growth regulators; osteoporosis; congestive heart failure; muscular disorders
07/10/2003US20030130283 CRF receptor antagonists and methods relating thereto
07/10/2003US20030130281 DPP IV inhibitors
07/10/2003US20030130278 Alkynylated fused ring pyrimidine compounds
07/10/2003US20030130277 Pyrazoloquinolinone derivatives as protein kinase C inhibitors
07/10/2003US20030130273 Hydantoins and related heterocycles as inhibitors of matrix metalloproteinases and/or TNF-alpha converting enzyme (TACE)
07/10/2003US20030130261 Central nervous system disorders; psychological disorders; inflammatory bowel disorders
07/10/2003US20030130260 Aryl fused azapolycyclic compounds
07/10/2003US20030130259 Quinoline and quinazoline compounds useful in therapy
07/10/2003US20030130257 Bicyclic hydroxamates as inhibitors of matrix metalloproteinases and/or TNF-alpha converting enzyme (TACE)
07/10/2003US20030130255 Pyridoquinoxaline antivirals
07/10/2003US20030130122 Aryl ether derivatives and processes for their preparation and herbicidal and desiccant compositions containing them
07/09/2003EP1325910A1 Aliphatic nitrogenous five-membered ring compounds
07/09/2003EP1325009A2 Amino-substituted tetracyclic compounds useful as anti-inflammatory agents and pharmaceutical compositions comprising same
07/09/2003EP1325007A2 Hexahydropyrazino[1'2':1,6]-pyrido[3,4-b]indole-1,4-dione derivatives for the treatment of cardiovascular disorders and erectile disfunction
07/09/2003EP1325006A2 Heterocyclic compounds as ligands of the gaba a? receptor
07/09/2003EP1325005A1 1,2,5,10-tetrahydropyridazino 4,5-b]quinoline-1,10-diones and their use for the treatment of pain
07/09/2003EP1325004A1 1,2,5,10-tetrahydropyridazino[4,5-b]quinoline-1,10-diones and their use for the treatment of pain
07/09/2003EP1325003A1 7-chloro-4-hydroxy-2-(2-pyridylethyl)-1,2,5,10-tetrahydropyridazino 4,5-b]quinoline-1,10-dione and the use thereof for the treatment of pain
07/09/2003EP1325002A1 1,2,5,10-tetrahydropyridazino[4,5-b]quinoline-1,10-diones and their use for the treatment of pain
07/09/2003EP1324991A1 Compounds useful in the treatment of inflammatory diseases
07/09/2003EP1324985A1 Inhibitors of prenyl-protein transferase
07/09/2003CN1113895C Growth hormone secretagogues
07/09/2003CN1113894C Process for preparing intermediates of inhibitors of enkephalinase and angiotensin coverting enzyme and intermediates thereof
07/09/2003CN1113885C Process for producing beta-lactam derivs.
07/09/2003CN1113881C 8-substituted-1,3,8-triaza-spiro [4.5] decan-4-on derivatives
07/09/2003CN1113880C Process for production of endotropine
07/09/2003CN1113875C Substituted aromatic thiocarboxylic acid amides and their use as herbicides
07/09/2003CN1113648C Use of tetrahydro-beta-carboline derivative as antimetastatic carcinoma preparation
07/08/2003US6589954 Indoles, benzimidazoles and benztriazoles which are substituted at the 5 or 6 position with a substituent comprising an aromatic moiety linked through a piperazine ring to said indole, benzimidazole or benztriazole are useful
07/08/2003US6589934 Methods of treatment of non insulin dependent diabetes mellitus, antagonists of the delayed rectifier potassium channel Kv2.1, methods of using and preparing the antagonists and assays for identifying such antagonist
07/08/2003CA2278845C Process for preparing quinolone and naphthyridone carboxylic acids
07/08/2003CA2226784C Use of cgmp-phosphodiesterase inhibitors to treat impotence
07/03/2003WO2003053972A1 Pyridoquinoxaline antivirals
07/03/2003WO2003053971A1 Pyridoquinoxaline antivirals
07/03/2003WO2003053970A1 Azaindolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands
07/03/2003WO2003053969A1 Imidazoquinoline derivatives
07/03/2003WO2003053968A1 Triazolo-quinolin derivatives useful as adenosine receptor ligands
07/03/2003WO2003053967A1 Aroyl pyridinones
07/03/2003WO2003053941A2 Barbituric acid derivatives as inhibitors of tnf-alpha converting enzyme (tace) and/or matrix metalloproteinases
07/03/2003WO2003053939A1 Benzimidazole derivatives and their use as gnrh antagonists
07/03/2003WO2003053926A1 Novel phenylalanine derivative
07/03/2003WO2003053444A1 New use
07/03/2003WO2003053433A1 Indolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands
07/03/2003WO2003053368A2 Chalcone derivatives and their use to treat diseases
07/03/2003WO2003053366A2 Pyrimidine a2b selective antagonist compounds, their synthesis and use
07/03/2003WO2003053354A2 Fused cyclic modulators of nuclear hormone receptor function
07/03/2003WO2003053344A2 Substituted 2-methyl-benzimidazole respiratory syncytial virus antiviral agents
07/03/2003WO2003018548A3 Halogenated calixpyrroles, calixpyridinopyrroles and calixpyridines, and uses thereof
07/03/2003WO2002079189A3 Spiroisoquinoline compounds, methods for their preparation and intermediates
07/03/2003WO2002016340A8 Aminoalkoxybenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
07/03/2003US20030125561 Triazole or imidazole oxide compound with a positively charged electron withdrawing group (a quaternary nitrogen containing amidine or imine group); useful in effecting the acylation step in amide formation (peptide synthesis)
07/03/2003US20030125354 Aromatic compounds containing urea or thiourea groups are useful for terating cytokine mediated diseases
07/03/2003US20030125351 Administering a heterocyclic amide compound to a glaucoma patient for inhibiting contraction of ciliary muscle; Rho kinase inhibitor
07/03/2003US20030125339 Substituted alkylamine derivatives and methods of use
07/03/2003US20030125327 Prodrugs of imidazopyridine derivatives