Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
02/2004
02/19/2004WO2004014910A1 Dihydropyrazolopyridine compounds
02/19/2004WO2004014909A1 Fused tetrahydropyridine derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014908A1 Heterobicylcic metalloproteinase inhibitors
02/19/2004WO2004014907A1 6-alkoxy-pyrido-pyrimidines as p-38 map kinase inhibitors
02/19/2004WO2004014906A2 Nitro and amino substituted dibenzonaphthyridines as topoisomerase agents
02/19/2004WO2004014900A1 Benzimidazoles and benzothiazoles as inhibitors of map kinase
02/19/2004WO2004014893A2 Antimicrobial aza-bicyclic derivates, their compositions and uses
02/19/2004WO2004014891A1 Pyridazine derivatives as ligands for gaba receptors
02/19/2004WO2004014869A2 5,6-fused 3,4-dihydropyrimidine-2-one derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014868A2 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014866A1 Azaisoquinoline derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014862A1 Nitro and amino substituted heterocycles as topoisomerase i targeting agents
02/19/2004WO2004014856A1 2,3-dihydro-isoindol-1-ones with mao-b inhibiting activity
02/19/2004WO2004014430A1 Compositions of a cyclooxygenase-2 selective inhibitor and a carbonic anhydrase inhibitor for the treatment of neoplasia
02/19/2004WO2004014389A1 3,4-dihydroquinolin-2-one, 5,6-fused oxazin-3-one, and 5,6-fused thiazin-3-one derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014380A1 Composition and antiviral activity of substituted azaindoleoxoacetic piperazine derivatives
02/19/2004WO2004014378A1 3-isoquinolinone derivatives as matrix metalloproteinase inhiitors
02/19/2004WO2004014374A1 Bicyclo-pyrazoles active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
02/19/2004WO2004014368A1 3-pyrrolyl-pyridopyrazoles and 3-pyrrolyl-indazoles as novel kinase inhibitors
02/19/2004WO2004014365A1 Phthalimide derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014361A1 Aminocyclohexene quinolines and their azaisosteric analogues with antibacterial activity
02/19/2004WO2004014352A2 Methods for treating carbonic anhydrase mediated disorders
02/19/2004WO2004014294A2 4,7-disubstituted indoles and methods of making
02/19/2004WO2004007481A3 Substituted amine derivatives and methods of use in the treatment of angiogenesis relates disorders
02/19/2004WO2002046314A3 Perylene pigment compositions
02/19/2004US20040034226 Imidazopyridine compounds as 5-HT4 receptor modulators
02/19/2004US20040034223 3-24 synthons independently selected from aryl, heteroaryl, alicyclic and heteroalicyclic, provided at least one of the synthon is different from other, and these synthons are bonded through linkers, thus forming a closed ring of synthon
02/19/2004US20040034221 Enzyme inhibitors for treating AIDS
02/19/2004US20040034081 Estrogen receptor modulators
02/19/2004US20040034063 Antiallergens for treating and prevention of asthma
02/19/2004US20040034061 An antagonist of corticotropin releasing factor receptor, treating depression, anxiety, Alzheimer's disease, Parkinson's disease, Huntington's chorea, eating disorder, hypertension, gastrointestinal disorders, drug dependence
02/19/2004US20040034055 For treating central nervous system disorders, immunomodulatory disorders, antimalaria, viral disease of Borna virus, Hepatitis; a 6-azatricyclo(6.3.1.01,6)dodecane derivatives
02/19/2004US20040034052 Antitumor agents
02/19/2004US20040034037 Heteroaryl compounds useful as inhibitors of GSK-3
02/19/2004US20040034032 Quinoline and quinazoline compounds useful in therapy
02/19/2004US20040034023 Dibenzophenanthrolines useful for treating cancer
02/19/2004US20040034015 Administering to a human patient suffering from addictive behavior associated with 5HT2C receptor modulation, a fused tetra or pentaheterocyclic compound containing nitrogen in the rings
02/19/2004US20040033935 Novel imidazole derivatives, production method thereof and use thereof
02/19/2004US20040033934 Antimalarial and antiproliferative pharmacophore models, novel tryptanthrin compounds having increased solubility, and methods of making and using thereof
02/19/2004CA2497656A1 Pyrimidine-2,4-dione derivatives as matrix metalloproteinase inhibitors
02/19/2004CA2495516A1 Compositions of a cyclooxygenase-2 selective inhibitor and a carbonic anhydrase inhibitor for the treatment of neoplasia
02/19/2004CA2495502A1 Methods for treating carbonic anhydrase mediated disorders
02/19/2004CA2495293A1 Azaisoquinoline derivatives as matrix metalloproteinase inhibitors
02/19/2004CA2495216A1 3-pyrrolyl-pyridopyrazoles and 3-pyrrolyl-indazoles as novel kinase inhibitors
02/19/2004CA2494785A1 Dihydropyrazolopyridine compounds
02/19/2004CA2493725A1 Antitumoral analogs of lamellarins
02/19/2004CA2493625A1 Bicyclo-pyrazoles active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
02/19/2004CA2493146A1 Antimicrobial aza-bicyclic derivates, their compositions and uses
02/19/2004CA2493143A1 2,3-dihydro-isoindol-1-ones with mao-b inhibiting activity
02/19/2004CA2492112A1 6-alkoxy-pyrido-pyrimidines as p-38 map kinase inhibitors
02/18/2004EP1389618A1 Pyrazolo 1,5-a]pyridines and medicines containing the same
02/18/2004EP1389463A1 Medicine for inhibiting drug elimination pump
02/18/2004EP1389208A1 Substituted azabicyclic moieties for the treatment of disease (nicotinic acethylcholine receptor antagonists)
02/18/2004EP1389189A2 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
02/18/2004EP1389103A2 Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic agents
02/18/2004EP1389099A1 Delivery of beta-blockers through an inhalation route
02/18/2004EP1389098A1 Delivery of antipsychotics through an inhalation route
02/18/2004EP1389097A1 Delivery of compounds for the treatment of parkinsons through an inhalation route
02/18/2004EP1389096A1 Delivery of opioids through an inhalation route
02/18/2004EP1389095A1 Delivery of antidepressants through an inhalation route
02/18/2004EP1389094A1 Delivery of sedative-hypnotics trough an inhalation route
02/18/2004EP1213281B1 Novel amide derivatives
02/18/2004EP1196410B1 Respiratory syncytial virus replication inhibitors
02/18/2004EP1192156B1 Bispidine compounds useful in the treatment of cardiac arrhythmias
02/18/2004EP1183252B1 pharmaceutically active compounds
02/18/2004EP0983270B1 Process for preparing 6-o-monoesters of castanospermine
02/18/2004EP0944631B1 Novel substituted pyrazole derivatives for the treatment of cardiocirculatory diseases
02/18/2004EP0944627B1 8-azabicyclo 3.2.1]octane-, 8-azabicyclo 3.2.1]oct-6-ene-, 9-azabicyclo 3.3.1]nonane-, 9-aza-3-oxabicyclo 3.3.1]nonane- and 9-aza-3-thiabicyclo 3.3.1]nonane derivatives, their preparation and their use as insecticides
02/18/2004CN1476448A Aryl or heteroaryl fused imidazole compounds as anti-inflammatory and analgesic agents
02/18/2004CN1476446A Benzodiazepine derivative
02/18/2004CN1476442A Pyridine derivatives with IKB-kinase (IKK-beta) INhibiting activity
02/18/2004CN1476436A Novel compounds for use as HIV protease inhibitors
02/18/2004CN1138778C Bicyclic pyrimidines and bicyclic 3,4-dihydropyrimidines as inhibitors of cellular proliferation
02/18/2004CN1138776C Extraction method of pyrroquinolinequinone
02/18/2004CN1138775C Acetylcholine enhancers and its use
02/18/2004CN1138774C Substituted 6,6-hetero-bicyclic derivatives
02/18/2004CN1138765C Oxazolidinone antibacterial agents having thiocarbonyl functionality
02/18/2004CN1138760C Preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and TACE inhibitors
02/17/2004US6693199 Deprotecting carbamate group and amidating in presence of such as hydroxybenzotriazole hydrate promoter
02/17/2004US6693116 Adenosine receptor ligands
02/17/2004US6693114 N-(4-chlorobenzyl)-6-(3-hydroxy-1-propynyl)-1-7-dimethyl-4-oxo-1,4 -dihydro(1,8) naphthyridine-3-carboxamide for example; inhibiting viral dna polymerase; treating herpes virus infections
02/17/2004US6693113 As immunomodulators and for inducing cytokine biosynthesis in animals, for therapy of viral infections
02/17/2004US6693112 Compounds for enhancing chemotherapy
02/17/2004US6693111 Indole-2,3-dione-3-oxime derivatives
02/17/2004US6693109 Spiro compounds as inhibitors of fibrinogen-dependent platelet aggregation
02/17/2004US6693102 Pyridine-substituted pyrazolopyridine derivatives
02/17/2004US6693101 Alkanoic acid derivative; integrin receptor antagonist
02/17/2004CA2302965C Processes and intermediates for preparing anti-cancer compounds
02/17/2004CA2290918C Heteroaromatic bicyclic derivatives useful as anticancer agents
02/12/2004WO2004013143A2 Aza-bridged bicyclic amine derivatives for use as novel cholinergic receptor ligands
02/12/2004WO2004013142A1 A riboflavin derivative and its manufacture and uses
02/12/2004WO2004013140A1 Pyrazole compositions useful as inhibitors of gsk-3
02/12/2004WO2004013139A2 Process for preparing 7-azaindoles
02/12/2004WO2004013138A2 Imidazo`1,2-a!pyridines
02/12/2004WO2004013137A1 1h-pyrazole and 1h-pyrrole-azabicyclic compounds with alfa-7 nachr activity
02/12/2004WO2004013135A1 2-phenylpyridin-4-yl derivatives as alk5 inhibitors
02/12/2004WO2004013109A1 Resorcinol derivative
02/12/2004WO2004012776A1 Isotopically labelled indolinone derivatives and process for their preparation
02/12/2004WO2003103610A3 Mappicine analogs, methods of inhibiting retroviral reverse transcriptase and methods of treating retroviruses
02/12/2004WO2003070236A3 Tricyclic pyrazole derivatives, process for their preparation and their use as antitumor agents