Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
02/2005
02/10/2005US20050031899 Carbazole derivative, organic semiconductor element, light emitting element, and electronic device
02/10/2005CA2534893A1 A novel process for the manufacture of (+)-(s)-clopidogrel bisulfate form-i
02/10/2005CA2534649A1 Bicyclic imidazol derivatives against flaviviridae
02/10/2005CA2534460A1 Benzylamine derivative
02/10/2005CA2534263A1 Phenylazole compounds, production process and antioxidants
02/10/2005CA2534212A1 Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
02/10/2005CA2534038A1 Inhibitors of akt activity
02/10/2005CA2533774A1 Compounds and compositions as protein kinase inhibitors
02/10/2005CA2532965A1 3, 4-disubstituted 1h-pyrazole compounds and their use as cyclin dependent kinases (cdk) and glycogen synthase kinase-3 (gsk-3) modulators
02/10/2005CA2531291A1 Pyrazoloisoquinoline derivatives as kinase inhibitors
02/10/2005CA2520546A1 Benzo[1,2,5]thiadiazole compounds
02/09/2005EP1505061A1 Compound exhibiting pgd 2 receptor antagonism
02/09/2005EP1504040A1 Method for reduction of residual organic solvent in carbomer
02/09/2005EP1504008A1 7-aminoimidazotriazones
02/09/2005EP1504003A1 Nitrosated imidazopyridines
02/09/2005EP1503760A1 Camptothecin derivatives and polymeric conjugates thereof
02/09/2005EP1503757A2 Tyrosine kinase inhibitors
02/09/2005EP1385854B1 Thiazolopyrimidines and their use as modulators of chemokine receptor activity
02/09/2005EP1339717B1 Novel carbamate-substituted pyrazolopyridine derivatives
02/09/2005EP1292269B1 Agent for dyeing keratin containing fibers
02/09/2005EP1100789B1 Substituted benzoylcyclohexandiones
02/09/2005CN1578781A 1, 8 naphthyridine derivatives and their use to treat diabetes and related disorders
02/09/2005CN1578780A 1, 6-naphthyridine derivatives as antidiabetics and pharmaceutical compositions containing them
02/09/2005CN1578773A Methods and compositions of novel triazine compounds
02/09/2005CN1578661A Naphthyridine derivatives, their preparation and their use as phosphodiesterase isoenzyme 4 (pde4) inhibitors
02/09/2005CN1578660A Lactam-containing compounds and derivatives thereof as factor xa inhibitors
02/09/2005CN1575816A Compounds for the treatment of female sexual dysfunction
02/09/2005CN1188414C Method of stabilizing aqueous pyrazoloacridone derivative solution
02/09/2005CN1188413C Compound for treatment of pain
02/09/2005CN1188412C Process for preparing crystalline form 1 of cabergoline
02/08/2005US6852861 Preparation of 1H-imidazo [4,5-C] quinolin-4-amines via 1H-imidazo [4,5-C] quinolin-4-phthalimide intermediates
02/08/2005US6852855 Synthesis of piperazine ring
02/08/2005US6852745 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
02/08/2005US6852734 Indole wherein A is an oxygen atom or a nitrogen atom which nitrogen atom is optionally substituted with an alkyl group, and (i) R1 and R2 each stand for a hydrogen atom or an alkyl group, independently, or (ii) R1 and R2 as taken together form
02/08/2005US6852732 A tetrahydropyridino or piperidino heterocyclic derivative represented by the formula (I): has a high affinity for CRF receptors and is effective against diseases in which CRF is considered to be involved. (Corticotropin releasing factor
02/08/2005US6852730 Substituted fused pyrazolecarboxylic acid arylamides and related compounds
02/08/2005US6852727 Inhibitors of Janus protein tyrosine kinases (Jak), and as such are useful as immunosuppressants, and in the treatment of diseases including asthma, allergies, autoimmune diseases.
02/08/2005US6852725 Imidazolyl derivatives
02/08/2005US6852722 Administering a growth hormone secretagogue.
02/08/2005US6852721 Compounds capable of activating nicotinic cholinergic receptors; N-aryl diazabicyclic compounds such as (1S,4S)-2-(5-(3-methoxyphenoxy)-3-pyridyl)-2,5-diazabicyclo(2. 2.1)-heptane; treating central nervous system disorders
02/08/2005US6852716 Central nervous system disorders; psychological disorders
02/08/2005US6852712 Controlling cell differentiation; antiinflammatory agents
02/08/2005CA2287316C Process for preparing 6-o-monoesters of castanospermine
02/03/2005WO2005010003A1 Sulfonyldihydroimid- azopyridinone compounds as 5-hydroxytryptamine-6 ligands
02/03/2005WO2005010002A1 Process for the synthesis of zolpidem
02/03/2005WO2005010001A1 Nicotinamide derivatives useful as pdea4 inhibitors
02/03/2005WO2005010000A2 Aryl-condensed 3-arylpyridine compounds and use thereof for controlling pathogenic fungi
02/03/2005WO2005009995A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005WO2005009994A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005WO2005009978A1 2-aminopyrimidine and 2-aminopyridine-4-carbamates for use in the treatment of autoimmune diseases
02/03/2005WO2005009967A2 Quinolinone derivatives as inhibitors of c-fms kinase
02/03/2005WO2005009962A1 Hydroxypyridine cgrp receptor antagonists
02/03/2005WO2005009958A1 Ppar active compounds
02/03/2005WO2005009947A2 Aryl heteroaromatic products, compositions comprising the same and use thereof
02/03/2005WO2005009398A2 Tetracyclic benzamide derivatives and methods of use thereof
02/03/2005WO2005009389A2 Anaplastic lymphoma kinase modulators and methods of use
02/03/2005WO2005009370A2 Beta-carboline compounds and analogues thereof and their use as mitogen-activated protein kinase-activated protein kinase-2 inhibitors
02/03/2005WO2004101565A3 Jnk inhibitors
02/03/2005WO2004054581A3 Cyclohexyl compounds as ccr5 antagonists
02/03/2005WO2003106450A8 Phenylaminopyrimidines and their use as rho-kinase inhibitors
02/03/2005US20050027130 Rhodamine dye compounds for patterns with DNA sequences for kits
02/03/2005US20050027122 Compounds for modulators of chemokine activity
02/03/2005US20050026947 1H-imidazo dimers
02/03/2005US20050026946 GSK-3 inhibitors
02/03/2005US20050026942 Chemokine receptor binding heterocyclic compounds
02/03/2005US20050026941 preferential inhibitors of cyclic guanosine 3',5'-monophosphate specific phosphodiesterase used for prophylaxis of erectile dysfunction and cardiovascular disorders
02/03/2005US20050026929 2-Phenyl-4-(piperidin-1-ylcarbonyl)-oxazole derivatives; capsase activators; cancer, autoimmune diseases, rheumatoid arthritis, inflammatory bowel disease, or psoriasis
02/03/2005US20050026925 1,2,3,4,9,9a-Hexahydro-2,4a,5-triaza-fluorene derivatives for obesity treatment
02/03/2005US20050026922 For treating CNS or other disorders, including concurrent treatment of disorders such as schizophrenia and depression; side effect reduction; for example, (7R,9aS)-trans-7-[6-(2,6-Dimethyl-piperidin-1-ylmethyl)-pyridin-2-yloxymethyl]-2-(5-fluoro-benzo[d]isoxazol-3-yl)-octahydro-pyrido[1,2-a]pyrazine
02/03/2005US20050026921 New imidazopyridazinone and imidazopyridone derivatives, the preparation thereof and their use as pharmaceutical compositions
02/03/2005US20050026917 Tricyclic indanyls as integrin inhibitors
02/03/2005US20050026915 As melanin concentrating hormone (MCH)receptor antagonists, for prevention or treatment of obesity or eating disorders; (2E)-3-(4-chlorophenyl)-N-[2-(dimethylamino)quinolin-6-yl]prop-2-enamide
02/03/2005US20050026914 Pyrimidine or pyridine carbamate compounds as for example 1,1-dimethylethyl 4-(4-((4-((((2,6-dimethylphenyl)oxy)carbonyl)(4-(methyloxy)phenyl)amino)-2-pyrimidinyl)amino)phenyl)-1-piperazinecarboxylate; for the treatment of protein tyrosine kinase-associated disorders
02/03/2005US20050026901 Antihistaminic spiro compounds
02/03/2005US20050026174 Alternative heterocycles for DNA recognition
02/03/2005DE10330358A1 New arylalkanol derivatives used for treating e.g. respiratory diseases, joint diseases, vascular inflammations, skin disorders, kidney and liver diseases and neurological diseases
02/03/2005CA2536383A1 Nicotinamide compounds useful as pde4 inhibitors
02/03/2005CA2533681A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005CA2533626A1 Quinolinone derivatives as inhibitors of c-fms kinase
02/03/2005CA2533624A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005CA2533494A1 Aryl heteroaromatic products, compositions comprising the same and use thereof
02/03/2005CA2532980A1 2-aminopyrimidine and 2-aminopyridine-4-carbamates for use in the treatment of autoimmune diseases
02/03/2005CA2532917A1 Aryl-condensed 3-arylpyridine compounds and use thereof for controlling pathogenic fungi
02/03/2005CA2532800A1 Anaplastic lymphoma kinase modulators and methods of use
02/03/2005CA2532403A1 Ppar active compounds
02/03/2005CA2532249A1 Nicotinamide derivatives useful as pde4 inhibitors
02/03/2005CA2532076A1 Sulfonyldihydroimid- azopyridinone compounds as 5-hydroxytryptamine-6 ligands
02/03/2005CA2532064A1 Hydroxypyridine cgrp receptor antagonists
02/03/2005CA2517260A1 Tetracyclic benzamide derivatives and methods of use thereof
02/02/2005EP1502917A1 Use of mono- and dicationic naphthalene-based imide dyes in optical layers for optical data recording
02/02/2005EP1501841A2 Non nucleoside reverse transcriptase inhibitors
02/02/2005EP1501830A1 7-aryl-3,9-diazabicyclo[3.3.1]non-6-ene derivatives and their use as renin inhibitors in the treatment of hypertension, cardiovascular or renal diseases
02/02/2005EP1501827A2 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acid and their use as protease inhibitors
02/02/2005EP1501507A2 Tetrahydropyranyl cyclopentyl tetrahydropyridopyridine modulators of chemokine receptor activity
02/02/2005EP1390365B1 Novel sulfonate substituted pyrazol pyridine dervivatives
02/02/2005EP1373267B1 Non-nucleoside reverse transcriptase inhibitors
02/02/2005EP1137413B1 Non-peptide antagonists of glp-1 receptor and methods of use
02/02/2005EP0828754B1 Dipeptides which promote release of growth hormone
02/02/2005CN1575289A 6-hydroxy isoflavon compounds, their derivatives and medicaments involving the same
02/02/2005CN1575177A Cxcr3 antagonists