Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
01/2006
01/25/2006EP1490363B1 Methods of preparation of the 2-(7-chloro-1,8-naphthyridine-2-yl)-3-(5-methyl-2-oxo-hexyl)-1-isoindolinone
01/25/2006EP1235825B1 Novel benzoimidazole derivatives useful as antiproliferative agents
01/25/2006EP1224189B1 Condensed dihydroquinolinone derivatives for inhibiting mrp1
01/25/2006EP0978392B1 Optical recording media
01/25/2006EP0697872B1 Tricyclopolyazamacrocyclophosphonic acids, complexes and derivatives thereof, for use as contrast agents
01/25/2006CN1726603A Charge transport compositions and electronic devices made with such compositions
01/25/2006CN1726215A [1,7]naphthyridines as PDE4 inhibitors
01/25/2006CN1726214A Enantiomer (-) of tenatoprazole and the therapeutic use thereof
01/25/2006CN1726213A Imidazoquinoline derivatives as adenosine A3 receptor ligands
01/25/2006CN1726212A Pre-organized tricyclic integrase inhibitor compounds
01/25/2006CN1726205A 2-substituted quinazolin-4-ylamine analogues as capsaicin receptor modulators
01/25/2006CN1726031A 8-trialkylsiloxy-2-methyl-9-phenyl-7-oxo-7,8,9,10-tetrahydroimidazo[1,2-h][1,7]naphthyridines
01/25/2006CN1724539A Purification method of catharanthine and vincristine
01/25/2006CN1724538A Method of chromatography preparing high purity catharanthine sulphate by continuous medium pressure column
01/24/2006US6989449 Containing nitroxide or hydroxylamine moieties; use stabilizing pulp or paper against yellowing and discoloration due to light
01/24/2006US6989398 Benzanilides as potassium channel openers
01/24/2006US6989393 Ccr5 modulators benzimidazoles or benzotriazoles
01/24/2006US6989391 Lactam-containing compounds and derivatives thereof as factor Xa inhibitors
01/24/2006US6989389 Immunomodulators; tetrahydroimidazo[4,5-c]quinoline-4-amine-1-(alkynyloxyalkyl) derivatives; induce cytokines biosynthesis; antitumor agents, viral diseases
01/24/2006US6989386 Pharmaceutically active ornithine derivatives, ammonium salts thereof and methods of making same
01/24/2006US6989385 Pyrazole compounds useful as protein kinase inhibitors
01/24/2006CA2261923C Pyridazino [4,5-b]-quinoline 5-oxide derivatives, their preparation and their use as glycine antagonists
01/19/2006WO2006005974A1 A process for the preparation of risperidone
01/19/2006WO2006005853A1 S-tenatoprazole sodium monohydrate salt and the use thereof in the form of a proton pump inhibitor
01/19/2006WO2006005726A2 Heterocyclic compounds
01/19/2006WO2006005725A2 N containing condensed heterocycles with antitumor effects
01/19/2006WO2005105805A9 Annelated carbamoylase-heterocycles, focused library, pharmaceutical compositions and methods for the production thereof
01/19/2006WO2005097129A3 6-azaindole compound
01/19/2006WO2005070930A3 Tetrahydrocarboline compounds as anticancer agents
01/19/2006US20060014951 4-amino-substituted pyrimidine derivatives
01/19/2006US20060014948 e.g 1-[3,5-bis(trifluoromethyl)benzoyl]-2-[3-[(2-methoxyethoxy)-methoxy]-4-methylbenzyl]-4-[2-[(3R)-3-methoxymethyl-morpholino]ethyl]piperazine; treating or preventing Tachykinin-mediated diseases in humans or animals
01/19/2006US20060014787 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
01/19/2006US20060014778 (+-)-cis 6-Methoxy-8-phenyl-2,3,3a,4,5,9b-hexahydro-1H-pyrrolo[3,4-c]quinoline; serotonin receptor modulators; obesity, diabetes, atherosclerosis, dyslipidemia; central nervous system diseases like anxiety, depression, OCD, panic disorder, psychosis, schizophrenia, sleep and sexual disorders,
01/19/2006US20060014777 Pyrrolo(oxo)isoquinolines as 5HT ligands
01/19/2006US20060014776 Antitumoral compounds
01/19/2006US20060014772 Phenanthroindolizidine alkaloids
01/19/2006US20060014765 For therapy of, for example, transplant rejection, inflammatory bowel syndrome, rheumatoid arthritis, psoriasis, restenosis, allergic asthma, Alzheimer's disease, Parkinson, stroke, osteoporosis, cancer, and benign hyperplasia
01/19/2006US20060014756 Benzimidazoles
01/19/2006US20060014750 Pharmaceutical compositions for the treatment of CNS and other disorders
01/19/2006US20060014749 (R)-2-{4-[(1H-Indol-2-ylmethyl)-amino]-piperidin-1-yl}-1-(6-methoxyquinolin-4-yl)-ethanol; effective against both gramnegative and grampositive bacteria
01/19/2006US20060014748 2-NH-heteroarylimidazoles with antibacterial activity
01/19/2006US20060014746 Heteroaryl substituted fused bicyclic heteroaryl compounds as GABAA receptor ligands
01/19/2006US20060014739 Androgen receptor modulators and method of treating disease using the same
01/19/2006US20060014682 Chemokine receptor antagonist peptide with a sequence homologous to SDF-1 wherein at least one amino acid at positions five to eight are substituted with proline; proliferative agents; self-regeneration of stem cells
01/19/2006CA2571491A1 Synthesis of heteroaryl acetamides from reaction mixtures having reduced water content
01/19/2006CA2568993A1 S-tenatoprazole sodium monohydrate salt and the use thereof in the form of a proton pump inhibitor
01/18/2006EP1615944A2 Antiandrogens with marginal agonist activity and methods of use
01/18/2006EP1615925A1 Imidazopyridine derivatives as melanocortin receptor agonists
01/18/2006EP1615924A1 Water soluble salts of risperidone
01/18/2006EP1615923A1 Risperidone monohydrochloride
01/18/2006EP1615922A1 Azaindole derivatives, preparations thereof, uses thereof and compositions containing them
01/18/2006EP1615921A2 Pyrido 2,3-d pyrimidin-7-carboxylic acid derivatives, their manufacture and use as pharmaceutical agents
01/18/2006EP1615919A1 7-([1,4]dioxan-2-yl)-benzothiazole derivatives as adenosine receptor ligands
01/18/2006EP1615904A2 Substituted benzosulphonamide as potentiators of glutamate receptors
01/18/2006EP1615889A2 Biphenyl derivatives having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity
01/18/2006EP1615886A1 [c]-fused bicyclic proline derivatives and their use for treating arthritic conditions
01/18/2006EP1615647A2 Pharmaceutical use of fused 1,2,4-triazoles
01/18/2006EP1615645A1 A crystalline form iii of anhydrous moxifloxacin hydrochloride and a process for preparation thereof
01/18/2006EP1615643A1 4-phenyl-piperidine compounds and their use as modulators of opioid receptors
01/18/2006EP1615636A1 Bicyclic compounds as nr2b receptor antagonists
01/18/2006EP1435951B1 Phenyl substituted 5-membered nitrogen containing heterocycles for the tretment of obesity
01/18/2006EP1207161B1 Novel isoindole derivatives
01/18/2006EP0973727B8 Activated iododerivatives for the treatment of cancer and aids
01/18/2006CN1721412A 7-oxo pyridopyrimidines
01/18/2006CN1237061C Chemokine receptor binding heterocyclic compounds
01/18/2006CN1237060C Quinzolone derivatives as alpha IA/B adrenergic receptor antagonists
01/18/2006CN1236767C Vitronectin receptor antagonists
01/17/2006US6987188 3a,4,5,9b-tetrahydro-1H-benz[e]indol-2-yl amine-derived neuropeptideYreceptors ligands useful in the treatment of obesity and other disorders
01/17/2006US6987187 Process for preparation of amidine derivatives
01/17/2006US6987186 Synthesis of small particle size quinacridone of beta crystal phase
01/17/2006US6987120 Pharmaceutical compounds
01/17/2006US6987115 Treating bacterial infections with a 1,2,3,4-tetrahydrobeta-carbolin-2-yl-alkyl-1-one; chemical intermediates, amidation
01/17/2006US6987109 Solubilized topoisomerase poison agents
01/17/2006US6987106 Nootropic agents; Alzheimer's Disease, Schizophrenia; ligands for the a7 subunits of the nicotinic receptor; 4-Bromophenyl-1,4-diazabicyclo[3.2.2]nonane-4-carboxylate
01/17/2006CA2300069C Naphthalimidobenzamide derivatives
01/17/2006CA2118812C 5-ht4 receptor antagonists
01/12/2006WO2006004925A1 Tetrahydroquinazolin-4(3h)-one-related and tetrahydropyrido[2,3-d]pyrimidin-4(3h)-one-related compounds, compositions and methods for their use
01/12/2006WO2006004884A2 Processes and intermediates useful for preparing fused heterocyclic kinase inhibitors
01/12/2006WO2006004833A2 Pyrrolotriazine kinase inhibitors
01/12/2006WO2006004702A1 Condensed triazoles and indazoles useful in treating citokines mediated diseases and other diseases
01/12/2006WO2006004636A2 Fused heterocyclic kinase inhibitors
01/12/2006WO2006003440A1 3,4-disubstituted pyrazoles as cyclin dependent kinases (cdk) or aurora kinase or glycogen synthase 3 (gsk-3) inhibitors
01/12/2006WO2006003090A1 Fluorescent quinacridones
01/12/2006WO2005103037A3 Selected cgrp antagonists, methods for the production thereof, and use thereof as medicaments
01/12/2006WO2005092066A3 Imidazole compounds
01/12/2006WO2005060959A8 Pyrazole derivatives and use thereof as orexin receptor antagonists
01/12/2006WO2004089951A8 Imidazopyridine derivatives having an affinity for melanocortin receptors
01/12/2006US20060009517 Tricyclic inhibitors of poly(ADP-ribose) polymerases
01/12/2006US20060009511 N-(2-arylethyl) benzylamines as antagonists of the 5-ht6 receptor
01/12/2006US20060009482 Screening method for identifying compounds that selectively induce interferon alpha
01/12/2006US20060009471 Amido compounds and their use as pharmaceuticals
01/12/2006US20060009465 Treatment of sleep disorders using sleep target modulators
01/12/2006US20060009453 Protein kinase modulators and method of use
01/12/2006CA2572084A1 Tetrahydroquinazolin-4(3h)-one-related and tetrahydropyrido[2,3-d]pyrimidin-4(3h)-one-related compounds, compositions and methods for their use
01/12/2006CA2572083A1 Fused pyrimidine derivatives and compositions thereof as cxcr3 receptor modulators, useful in prevention and treatment of inflammatory and immunoregulatory disorders and diseases
01/12/2006CA2572058A1 Azaindoles useful as inhibitors of protein kinases
01/12/2006CA2571680A1 Fused heterocyclic kinase inhibitors
01/12/2006CA2571588A1 Pyrazolopyridine derivatives
01/12/2006CA2570319A1 Condensed triazoles and indazoles useful in treating citokines mediated diseases and other diseases
01/11/2006EP1614683A1 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use