Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
03/2007
03/06/2007US7186870 Cyclization by reacting 4-(2-CHLORO-4-TRIFLUOROMETHYL-PHENYL)-4-CYANO-BUT-3-ENOIC ACID METHYL ESTER in the presence of a palladium catalyst and a base; chemical intermediates for preparing 10-AZA-TRICYCLO[6.3.1.02,7] drugs; bind nicotinic acetylcholine receptor, modulate cholinergic function
03/06/2007US7186841 Antiinflammation agents
03/06/2007US7186832 anticancer agents; antidiabetic agents; autoimmune disease; restenosis; antiarthritic agents; skin disorders; cardiovascular disorders; antiinflammatory agents
03/06/2007US7186830 Tricyclic 2-pyrimidone compounds useful as HIV reverse transcriptase inhibitors
03/06/2007US7186753 nitroso derivatives of drugs such as antiinflammatory agents, antibiotics, expectorants, mucolytic agents, antidiabetics, antitumor, viricides, enzyme inhibitors bronchodilators and antiulcer agents
03/06/2007US7186743 drugs such as 1 -[4-(aminosulfonyl)phenyl]-8-{[(trifluoromethyl)sulfonyl]amino}-4,5-dihydro-1H-benzo[g]indazole-3-carboxamide, used as antiinflammatory agents, antiarthritic agents, antipyretics or analgesics
03/06/2007US7186732 For therapy and prophylaxis of upper airway allergic response, nasal congestion, or allergic rhinitis, dementia, mild cognitive impairment (pre-dementia), cognitive dysfunction, schizophrenia, depression, manic disorders
03/06/2007US7186731 2-cyanopyrrolidinecarboxamide compound
03/06/2007US7186730 Bicyclic nitrogen-containing heterocyclic derivatives for use as antibacterials
03/06/2007US7186724 central nervous system disorders; psychological disorders; Parkinson's disease; Huntington's disease ; sleep disorders
03/06/2007US7186721 Substituted hexahydropyrrolo[1,2-a]pyrazines, octahydropyrido[1,2-a]-pyrazines and decahydropyrazino[1,2-a]azepines
03/06/2007US7186716 3-Pyrrol-pyridopyrazoles and 3-pyrrolyl-indazoles as novel kinase inhibitors
03/06/2007US7186714 administering drugs such as 3-[2-(Cyclopentylamino)-4-pyrimidinyl]-2-(4-fluorophenyl)imidazo[1,2-a]pyridin-8-amine, for therapy of viral diseases caused by DNA viruses
03/06/2007US7186710 PDE4/7 inhibitors useful in treatment of airway disorders, autoimmune system disorders, skin disorders, arthritis, nerve system disorders
03/06/2007US7186709 Subjecting a vinyl ethers and an unsaturated ketoester to suitable conditions to generate a scaffold having the core dihydropyrancarboxamide or dihydropyrancarboxylic ester or acid; anticarcinogenic agents
03/06/2007US7186469 Bathophenanthroline compound and EL device
03/06/2007CA2294990C Pharmaceutical compositions and methods for effecting dopamine release
03/01/2007WO2007025090A2 Heterobicyclic and - tricyclic inhibitors of mapk/erk kinase
03/01/2007WO2007025069A2 Diazaspirodecane orexin receptor antagonists
03/01/2007WO2007024945A1 Condensed imidazolo derivatives for the inhibition of aldosterone synthase and aromatase
03/01/2007WO2007024814A1 HETEROARYL-SUBSTiTUTED DIAZATRICYCLOALKANES, METHODS FOR ITS PREPARATION AND USE THEREOF
03/01/2007WO2007024789A1 Pyrrolopyridine, pyrrolopyrimidine and pyrazolopyridine compounds, compositions comprising them, and methods of their use
03/01/2007WO2007023504A1 Process for the preparation of imidazopyridines
03/01/2007WO2007023382A2 Pyrimidine amino pyrazole compounds, potent kinase inhibitors
03/01/2007WO2007023110A2 P38 map kinase inhibitors and methods for using the same
03/01/2007WO2007023105A1 FUSED PYRAZOLE AS p38 MAP KINASE INHIBITORS
03/01/2007WO2007022946A1 Heterocyclic compounds and their use as binding partners for 5-ht5 receptors
03/01/2007WO2007003961A3 Gpcr agonists
03/01/2007WO2006138347A3 Androgen receptor modulator compounds and methods
03/01/2007WO2006114520A3 Substituted pyrrolo-pyridines, composition containing them, method for their producing and use thereof
03/01/2007WO2006047528A3 Pyrazolobenzamides and derivatives as factor xa inhibitors
03/01/2007WO2006014325A3 C-met modulators and method of use
03/01/2007WO2005117876A8 Dual small molecule inhibitors of cancer and angiogenesis
03/01/2007US20070049620 Cyclic tertiary amine compound
03/01/2007US20070049616 Organic compounds
03/01/2007US20070049615 3-(6-Chloro-pyridin-3-ylmethyl)-4-phenyl-1H-pyrrolo[2,3-b]pyridine; molecular scaffolds
03/01/2007US20070049593 Tetracyclic fused heterocyclic compound and use thereof as HCV polymerase inhibitor
03/01/2007US20070049582 Substituted-3-indolyl-4-piperidino-alkyl heterocycles for the treatment of depression
03/01/2007US20070049580 Anxiolytic agents with reduced sedative and ataxic effects
03/01/2007US20070049574 4,5-Dicyclopropyl-1-methyl-2-phenyl-1,2-dihydro-pyrazol-3-one; 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1); 4-Cyclopropyl-5-(2,2-difluoro-cyclopropyl)-1-methyl-2-(2-trifluoromethyl-phenyl)-1,2-dihydro-pyrazol-3-one;
03/01/2007US20070048728 Hydroxylases and modulators thereof
03/01/2007US20070048215 Chemical compound and assay
03/01/2007CA2620254A1 P38 map kinase inhibitors and methods for using the same
03/01/2007CA2620104A1 Fused pyrazole as p38 map kinase inhibitors
03/01/2007CA2620052A1 Indenoisoquinolinone analogs and methods of use thereof
03/01/2007CA2619972A1 Pyrrolopyridine, pyrrolopyrimidine and pyrazolopyridine compounds, compositions comprising them, and methods of their use
03/01/2007CA2619660A1 Condensed imidazolo derivatives for the inhibition of aldosterone synthase and aromatase
03/01/2007CA2619111A1 Fused aminopiperidines as dipeptidyl peptidase-iv inhibitors for the treatment or prevention of diabetes
03/01/2007CA2618700A1 Heteroaryl-substituted diazatricycloalkanes, methods for its preparation and use thereof
02/2007
02/28/2007EP1757670A2 Organic electroluminescent element
02/28/2007EP1757608A1 New benzazepine derivatives, medicaments containing the same and their use in the preparation of medicaments
02/28/2007EP1757605A1 Cyclic amine compound
02/28/2007EP1757594A1 Quinazoline derivative
02/28/2007EP1756129A1 Novel dna threading intercalators
02/28/2007EP1756109A1 Novel indole derivatives as selective androgen receptor modulators (sarms)
02/28/2007EP1756108A2 Azaindoles useful as inhibitors of rock and other protein kinases
02/28/2007EP1756107A2 Aryl-substituted piperazine derivatives
02/28/2007EP1756106A1 Cyclohexylalanine derivatives as dipeptidyl peptidase-iv inhibitors for the treatment or prevention of diabetes
02/28/2007EP1756105A1 Substituted imidazo[1,2-a]pyridine compounds and drugs containing substituted imidazo[1,2-a]pyridine compounds
02/28/2007EP1756104A1 Tetrahydronaphthyridine derivatives useful as histamine h3 receptor ligands
02/28/2007EP1756103A2 Pyrrolopyridine derivatives and their use as hiv-integrase inhibitors
02/28/2007EP1756102A1 8-PHENOXY-GammaCARBOLINE DERIVATIVES
02/28/2007EP1756101A2 Androgen receptor modulators and method of treating disease using the same
02/28/2007EP1756084A2 Substituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto
02/28/2007EP1756069A2 Hiv integrase inhibitors
02/28/2007EP1756063A1 Amido compounds and their use as pharmaceuticals
02/28/2007EP1756044A1 Therapeutic compounds
02/28/2007EP1756037A2 Amino alcohol derivatives and their activity as renin inhibitors
02/28/2007EP1755603A2 3,3-disubstituted tetrahydropyranyl cyclopentyl amide modulators of chemokine receptor activity
02/28/2007EP1509522B1 1-(aminoalkyl)-3-sulfonylazaindoles as 5-hydroxytryptamine-6 ligands
02/28/2007EP1507776B1 2-oxo-1,3,4-trihydroquinazolinyl derivatives for the treatment of cell proliferation-related disorders
02/28/2007EP1465893B1 Derivatives of 5-(pyridin-3-yl)-1-azabicyclo (3.2.1) octane, the preparation thereof and the application of same in therapeutics
02/28/2007EP1441734B1 Dihydroxypyrimidine carboxamide inhibitors of hiv integrase
02/28/2007EP1415987B1 Nitrogenous aromatic ring compounds as anti cancer agents
02/28/2007EP1370531B1 Phenylalanine enamide derivatives possessing a cyclobutene group, for use as integrin inhibitors
02/28/2007EP1309592B9 Substituted pyrazoles
02/28/2007EP1178988B1 Compounds and therapeutic methods
02/28/2007EP1102753B1 Pyrazoles as estrogen receptor modulators
02/28/2007CN1922189A Spirocyclic cyclohexane derivatives with affinity for the ORL1-receptor
02/28/2007CN1922186A Diazabicyclic aryl derivatives as nicotinic acetylcholine receptor ligands
02/28/2007CN1922178A Piperazine, [1,4]diazepane, [1,4]diazocane, and [1,5]diazocane fused imidazo ring compounds
02/28/2007CN1922177A Aryl- and heteroaryl-piperidinecarboxylate derivatives, the preparation and the use thereof in the form of FAAH enzyme inhibitors
02/28/2007CN1922174A 病毒聚合酶抑制剂 Viral polymerase inhibitor
02/28/2007CN1922171A Pyrimidine derivative
02/28/2007CN1922169A Spirocyclic heterocyclic derivatives and methods of their use
02/28/2007CN1922155A Novel sulfone amide derivative
02/28/2007CN1922141A Novel heterocyclic compound
02/28/2007CN1921854A Heterocyclic GABAA subtype selective receptor modulators
02/27/2007US7183415 Melanin-concentrating hormone antagonistic action for treating obesity, for example 4'-fluoro-N-[8-methyl-3-(1-pyrrolidinylmethyl)-7-quinolinyl][1,1'-biphenyl]-4-carboxamide
02/27/2007US7183413 Aminoquinoline compounds
02/27/2007US7183412 Ester or amide derivatives
02/27/2007US7183318 Substituted cyclic compounds, preparation method and pharmaceutical compositions containing them
02/27/2007US7183313 Keto cannabinoids with therapeutic indications
02/27/2007US7183284 Aminium salts of 1,2,3-triazoles as prodrugs of drugs including antiviral agents
02/27/2007US7183282 N'-methyl-2-[(p-fluorophenyl)-4-oxo-butyl]piperazino[1,2-fg]gamma-carboline; N'-methyl-2-[p-fluorophenoxypropyl]piperazino[1,2-fg]gamma-carboline; serotonin modulators; sleep disorders; central nervous system disorders
02/27/2007US7183273 Administering compounds such as N-(2-pyridinylmethyl)-N'-(6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-9-yl)-1,4-benzenedimethanamine for therapy of disease mediated by a chemokine receptor
02/27/2007US7183270 Cyclic derivatives as modulators of chemokine receptor activity
02/27/2007CA2163400C Process for the preparation of organic pigments
02/22/2007WO2007022529A2 Method of treating inflammatory diseases
02/22/2007WO2007022305A2 2-aminoimidazopyridines for treating neurodegenerative diseases