Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559) |
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07/03/2014 | US20140187576 Salt of naphthyridine carboxylic acid derivative |
07/03/2014 | US20140187559 Inhibitors of the fibroblast growth factor receptor |
07/03/2014 | US20140187553 Azole Compounds as PIM Inhibitors |
07/03/2014 | US20140187551 7-azaindole derivatives suitable for treatment of cancers |
07/03/2014 | US20140187550 Bicyclic organic compounds suitable for the treatment of inflammatory or allergic conditions |
07/03/2014 | US20140187549 Pyridonemorphinan Analogs and Biological Activity on Opioid Receptors |
07/03/2014 | US20140187547 Azaindenoisoquinoline topoisomerase i inhibitors |
07/03/2014 | US20140187535 Substituted benzimidazole-type piperidine compounds and uses thereof |
07/03/2014 | US20140187534 Nitrogen-containing spirocyclic compounds and pharmaceutical uses thereof |
07/03/2014 | US20140187530 AZA Spiro Alkane Derivatives as Inhibitors of Metalloproteases |
07/03/2014 | US20140186951 Novel opioid antagonists |
07/02/2014 | EP2749561A1 Radioactive quinolinone derivative and pharmaceutical drug comprising the same |
07/02/2014 | EP2748165A1 1,6- diazabicyclo [3,2,1]octan-7-one derivatives and their use in the treatment of bacterial infections |
07/02/2014 | EP2748164A1 Bicyclic heteroaromatic compounds |
07/02/2014 | EP2748163A1 New synthetic intermediates for manufacturing antibiotics |
07/02/2014 | CN103906733A Trpm8拮抗剂及其在治疗中的用途 Trpm8 antagonists and their use in the treatment of |
07/02/2014 | CN103896986A 一种含苯并噻唑的钌配合物的制备方法及其抗癌活性 A preparation and antitumor activity of benzene and thiazole ruthenium complexes |
07/02/2014 | CN103896943A 一种伐伦克林盐及其制备方法 An 伦克林 cutting salt and its preparation method |
07/02/2014 | CN103896942A 聚(adp-核糖)聚合酶(parp)的二氢吡啶并酞嗪酮抑制剂 Poly (adp- ribose) polymerase (parp) dihydropyridine and -phthalazinone inhibitor |
07/02/2014 | CN103896941A 6-氯咪唑并[1,2-a]吡啶-3-甲腈的合成方法 Synthesis of 6-chloro-imidazo [1,2-a] pyridine-3-carbonitrile |
07/02/2014 | CN103896940A 一种阿哌沙班的合成方法 A method of synthesis of apixaban |
07/02/2014 | CN103896939A 一种6-氯-8-羟基-咪唑并(1,2a)吡啶盐酸盐及其合成方法 One kind of 6-chloro-8-hydroxy - imidazo (1,2a) pyridine hydrochloride and synthetic method |
07/02/2014 | CN103896920A 红色磷光化合物和使用该化合物的有机发光二极管器件 Red phosphorescent compounds and using the compounds of organic light emitting diode device |
07/02/2014 | CN103896860A 含有锌结合基的不可逆egfr抑制剂 Zinc binding group containing irreversible inhibitors of egfr |
07/02/2014 | CN103896831A 4-(4-吡啶基)-苯甲酰胺及其作为rock活性调节剂的应用 4- (4-pyridinyl) - benzamide and its use as an active modifier rock Application |
07/02/2014 | CN103893173A 靶向人La蛋白的先导化合物及其在制备抗乙型肝炎病毒的药物中的用途 Lead compounds targeting human La protein and its anti-hepatitis B virus in the preparation of a medicament for |
07/02/2014 | CN102925529B 制备左旋吡喹酮的中间体及左旋吡喹酮的方法 Preparation of L and L praziquantel praziquantel intermediate approach |
07/02/2014 | CN102925528B 一种制备左旋吡喹酮的中间体及左旋吡喹酮的方法 A process for preparing L-L praziquantel praziquantel intermediates and methods |
07/02/2014 | CN102844305B 抗菌异喹啉-3-基脲衍生物 Antibacterial isoquinoline-3-yl urea derivatives |
07/02/2014 | CN102690264B 2-苯基-3-取代咪唑并[1,2-a]吡啶类衍生物及其制备方法 2-phenyl-3-substituted imidazo [1,2-a] pyridine derivatives and their preparation |
07/02/2014 | CN102617569B 一种具有抗肿瘤活性的β-咔啉类衍生物及其制备方法 Β- carboline derivatives and method for preparing anti-tumor activity |
07/02/2014 | CN102471338B 氮杂杂环化合物 Aza-heterocyclic compounds |
07/02/2014 | CN102239151B 硫代酰胺化合物,其制备方法和使用方法 Thioamide compounds, their preparation and use |
07/02/2014 | CN102137862B 作为nadph氧化酶抑制剂的吡唑并吡啶衍生物 As nadph oxidase inhibitors pyrazolo pyridine derivatives |
07/02/2014 | CN102099357B 用于治疗代谢障碍的甲酰胺化合物 For the treatment of metabolic disorders carboxamide compounds |
07/02/2014 | CN102015686B 杂环化合物及其用途 Heterocyclic compounds and their use |
07/02/2014 | CN101970435B 吡咯并嘧啶和吡咯并吡啶类化合物 Pyrrolopyrimidine and pyrrolopyridine compounds |
07/02/2014 | CN101784516B 作为凝血因子抑制剂的二肽类似物 As a coagulation factor inhibitor dipeptide analogs |
07/01/2014 | US8765954 1,8-naphthyridine compounds for the treatment of cancer |
07/01/2014 | US8765940 Heterocyclic compounds and their uses |
07/01/2014 | US8765791 Method of treating cancer using a neuropeptide Y 5R (NP Y5R) antagonist |
07/01/2014 | US8765784 Positive allosteric modulators of MGLUR2 |
07/01/2014 | US8765783 Pharmaceutical composition for treatment of disease due to vascular constriction or vasodilation |
07/01/2014 | US8765782 Indole derivatives as selective androgen receptor modulators (SARMS) |
07/01/2014 | US8765766 Pyrimidine derivatives which are antagonists of the vitronectin receptor |
07/01/2014 | US8765760 [1,2,4] triazol [1,5-a] pyrazines useful as inhibitors of phosphodiesterases |
07/01/2014 | US8765748 Indazolyl, benzimidazolyl, benzotriazolyl substituted indolinone derivatives as kinase inhibitors useful in the treatment of cancer |
07/01/2014 | US8765743 Compounds |
07/01/2014 | US8765734 Piperidin-4-yl azetidine derivatives as JAK1 inhibitors |
07/01/2014 | US8765728 [1,5]-diazocin derivatives |
06/26/2014 | WO2014100765A1 Substituted pyrimidine aminoalkyl-quinazolones as phosphatidylinositol 3-kinase inhibitors |
06/26/2014 | WO2014100735A2 Diazole amides |
06/26/2014 | WO2014100695A1 Prmt5 inhibitors and uses thereof |
06/26/2014 | WO2014100691A1 Tetracationic cyclophanes and their use in the sequestration of polyaromatic hydrocarbons by way of complexation |
06/26/2014 | WO2014100665A1 1,4-pyridone bicyclic heteroaryl compounds |
06/26/2014 | WO2014100646A1 1,4-pyridone compounds |
06/26/2014 | WO2014100323A1 Polycyclic-carbamoylpyridone compounds and their pharmaceutical use |
06/26/2014 | WO2014100065A1 Substituted imidazopyridines as hdm2 inhibitors |
06/26/2014 | WO2014098000A1 Process for preparation of a tricyclic heterocycle |
06/26/2014 | WO2014097711A1 Organic electroluminescent element and electronic device |
06/26/2014 | WO2014097272A2 Method for production of (s,s)-6-benzyloctahydro-1h-pyrrolo[3,4-b]pyridine, an intermediate of azabicyclo pyridine derivatives |
06/26/2014 | WO2014097150A1 Process for the preparation of tofacitinib and intermediates thereof |
06/26/2014 | WO2014097041A1 Aryl and heteroaryl fused lactams |
06/26/2014 | WO2014096212A1 NOVEL TRICYCLIC 3,4-DIHYDRO-2H-PYRIDO[1,2-α]PYRAZINE-1,6-DIONE DERIVATIVES AS GAMMA SECRETASE MODULATORS |
06/26/2014 | WO2014096098A1 (6r,10r)-6,10,14-trimetylpentadecan-2-one prepared from 6,10,14-trimetylpentadeca-5,9,13-trien-2-one or 6,10,14-trimetylpentadeca-5,9-dien-2-one |
06/26/2014 | WO2014096093A1 3,5-diarylazaindoles as dyrk1a protein inhibitors for the treatment of cognitive deficiences associated with down's syndrome and with alzheimer's disease |
06/26/2014 | WO2014096067A1 (6r,10r)-6,10,14-trimetylpentadecan-2-one prepared from (r)-6,10,14-trimetylpentadec-5-en-2-one |
06/26/2014 | WO2014095798A1 Novel dihydropyrimidinoisoquinolinones and pharmaceutical compositions thereof for the treatment of inflammatory disorders (gpr84 antagonists) |
06/26/2014 | WO2014095775A1 Bet-protein-inhibiting dihydroquinoxalinones |
06/26/2014 | WO2014095774A1 Bet-protein-inhibiting dihydropyridopyrazinones |
06/26/2014 | WO2014094816A1 P38 mapk inhibitors for the treatment of inflammatory diseases |
06/26/2014 | WO2014094664A1 Crystal form of compound used as mineralocorticoid receptor antagonist and preparation method therefor |
06/26/2014 | US20140179924 Process for the preparation of cathepsin S inhibitors |
06/26/2014 | US20140179733 Diazole amides |
06/26/2014 | US20140179732 Tricyclic lactam derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors |
06/26/2014 | US20140179730 Novel methysergide derivatives |
06/26/2014 | US20140179724 Spirocyclic Morphinans and Their Use |
06/26/2014 | US20140179696 Indazole inhibitors of the wnt signal pathway and therapeutic uses thereof |
06/26/2014 | US20140179685 Substituted noribogaine |
06/26/2014 | US20140179684 Substituted noribogaine |
06/26/2014 | US20140179682 Metabotrophic glutamate receptor 5 modulators and methods of use thereof |
06/26/2014 | US20140179680 Substituted Imidazopyridines as HDM2 Inhibitors |
06/26/2014 | US20140179675 Quinolone compound |
06/26/2014 | US20140179672 Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use |
06/26/2014 | US20140179671 Fused ring azadecalin glucocorticoid receptor modulators |
06/26/2014 | US20140179669 Alicyclic carboxylic acid derivatives of benzomorphans and related scaffolds, medicaments containing such compounds and their use |
06/26/2014 | US20140179667 Aryl and heteroaryl fused lactams |
06/26/2014 | US20140179666 Bicyclic heterocycle compounds and their uses in therapy |
06/26/2014 | US20140179662 Pharmaceutically active disubstituted triazine derivatives |
06/26/2014 | US20140179017 Tetracationic cyclophanes and their use in the sequestration of polyaromatic hydrocarbons by way of complexation |
06/25/2014 | EP2746282A1 Triazolopyridine compound, and action thereof as prolyl hydroxylase inhibitor and erythropoietin production inducer |
06/25/2014 | EP2746281A2 7-azaindole derivatives |
06/25/2014 | EP2746272A1 Nitrogen-containing compounds and pharmaceutical compositions thereof for the treatment of atrial fibrillation |
06/25/2014 | EP2744809A1 4-(8-methoxy-1-((1-methoxypropan-2-yl)-2-(tetrahydro-2h-pyran-4-yl)-1 h-imidazo[4,5-c]quinolin-7-yl)-3,5-dimethylisoxazole and its use as bromodomain inhibitor |
06/25/2014 | CN103889986A 新杂环衍生物及其应用 New heterocyclic derivatives and its application |
06/25/2014 | CN103889985A 作为有机半导体的萘-二酰亚胺-杂环-萘二酰亚胺低聚物以及自其产生的晶体管 As the organic semiconductor naphthalene - imide - heterocycle - naphthalene imide oligomer, and from which the produced transistors |
06/25/2014 | CN103889984A 4-(8-甲氧基-1-((1-甲氧基丙烷-2-基)-2-(四氢-2H-吡喃-4-基)-1H-咪唑并[4,5-c]喹啉-7-基)-3,5-二甲基异噁唑及其作为溴结构域抑制剂的用途 4- (8-methoxy-1 - ((1-methoxy-propan-2-yl) -2- (tetrahydro -2H- pyran-4-yl) -1H- imidazo [4,5- c] quinolin-7-yl) -3,5-dimethyl-isoxazole and their use as inhibitors of the use of bromine domain |
06/25/2014 | CN103889983A 新型酶抑制剂化合物 Novel inhibitor compound |
06/25/2014 | CN103889976A 吲唑化合物、组合物及使用方法 Indazole compounds, compositions and methods of use |
06/25/2014 | CN103889972A 作为磷酸二酯酶抑制剂的1-苯基-2-吡啶基烷基醇的衍生物 A phosphodiesterase inhibitor 1-phenyl-2-pyridinyl alkyl alcohols derivatives |