Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
02/2010
02/18/2010CA2731108A1 Cmet inhibitors
02/17/2010EP2154223A1 Thermal insulating foam comprising HFO-1233zd as blowing agent
02/17/2010EP2154138A1 Novel compounds for treatment of psychotic disorders, preparation methods and uses thereof
02/17/2010EP2154137A1 Crystalline form of moxifloxacin base
02/17/2010EP2152710A2 4,4-disubstituted piperidine derivatives
02/17/2010EP2152709A1 Morphinan compounds
02/17/2010EP2152707A1 [6,5]-bicyclic gpr119 g protein-coupled receptor agonists
02/17/2010EP2152706A1 Pyrazolo-pyridinone and pyrazolo-pyrazinone compounds as p38 modulators, process for their preparation, and their pharmaceutical use
02/17/2010EP2152705A1 9- (pyrazol- 3 -yl) - 9h- purine-2 -amine and 3- (pyraz0l-3-yl) -3h-imidaz0 [4, 5-b]pyridin-5-amine derivatives and their use for the treatment of cancer
02/17/2010EP2152704A1 Pyrazolo-pyridinone compounds, process for their preparation, and their pharmaceutical use
02/17/2010EP2152695A2 Gamma secretase modulators
02/17/2010EP2152664A1 Dipeptide analogs as coagulation factor inhibitors
02/17/2010EP2152660A2 Photocrosslinkable materials comprising alicyclic group
02/17/2010EP1828200B1 Bi- and tricyclic substituted phenyl methanones as glycine transporter i (glyt-1) inhibitors for the treatment of alzheimer's disease.
02/17/2010EP1347950B1 Derivatives of 4-hydroxybutanoic acid and of its higher homologue as ligands of gamma-hydroxybutyrate (ghb) receptors, pharmaceutical compositions containing same and pharmaceutical uses
02/17/2010CN101652364A New indole derivative compounds and pharmaceutical compositions containing the same
02/17/2010CN100590124C Tricyclic androgen receptor modulator compounds and method
02/16/2010US7662833 metalloproteinases inhibitor, particular Peptide Deformylase (Pdf) inhibitor; antibiotic; e.g. 2-(6-fluoro-imidazo[1,2-a]pyridin-3-ylamino)-N-hydroxy-acetamide
02/16/2010US7662832 Pyrrolo[2,3-c]pyridine derivatives and processes for the preparation thereof
02/16/2010US7662831 N-5,6,9,10,11,12-hexahydro-4H,8H-cyclohepta[4,5]pyrrolo[3,2,1-ij]quinolin-2-yl-3,3-dimethylbutanamide; for treating cardiovascular disorders, nervous system disorders e.g epilepsy, episodic ataxia type 1, paroxysmal dyskinesia, neurodegenerative spincerebrallar ataxia, Parkinson's disease
02/16/2010US7662828 Substituted 5,6,7,8-tetrahydropyrido[4,3-d]pyrimidine-2-yl compounds and 5,6,7,8-tetrahydroquinazoline-2-yl compounds
02/16/2010US7662827 Pyrazole derivatives having tyrosine kinase inhibitory activity
02/16/2010US7662823 non-nucleoside reverse transcriptase inhibitors; for treatment of HIV and AIDS
02/16/2010US7662822 Substituted azaquinazolines having an antiviral action
02/16/2010US7662818 e.g. 4-[5-(piperidine-1-carbonyl)-furan-2-ylmethyl]-2H-phthalazin-1-one; enzyme poly(ADP-ribose)polymerase (synthase)-1 or poly ADP-ribosyltransferase (PARP-1) inhibitor; anticarcinogenic agent with BRCA2 deficient phenotype; septic shock; ischemic injury; hemorrhagic shock; and multiple sclerosis
02/16/2010US7662808 Diazabicyclic aryl derivatives as cholinergic receptor modulators
02/16/2010CA2571627C Substituted aryl-amine derivatives and methods of use
02/16/2010CA2478183C Substituted amides
02/16/2010CA2450922C Piperidines for use as orexin receptor antagonists
02/16/2010CA2406095C Synthetic process for the manufacture of an ecteinaschidin compound
02/16/2010CA2385938C Cyclic amine compounds as ccr5 antagonists
02/16/2010CA2308551C Phenanthroline derivatives
02/11/2010WO2010017105A1 Urotensin ii receptor antagonists
02/11/2010WO2010016846A1 Heterocyclic modulators of tgr5 for treatment of disease
02/11/2010WO2010016549A1 Tricyclic compound
02/11/2010WO2010016490A1 Imidazopyridin-2-on derivative
02/11/2010WO2010016005A1 6 substituted 2-heterocyclylamino pyrazine compounds as chk-1 inhibitors
02/11/2010WO2010015985A1 Tricyclic alkylaminomethyloxazolidinone derivatives
02/11/2010WO2010015803A1 Diazaindole derivatives and their use in the inhibition of c-jun n-terminal kinase
02/11/2010WO2010015636A1 Beta-carbolin-derivates as substrates for an enzyme
02/11/2010WO2010015589A1 Benzyl-substituted tetracyclic heterocyclic compounds as pde5 inhibitors
02/11/2010WO2010015588A1 Benzyl-substituted tetracyclic heterocyclic compounds
02/11/2010WO2010015587A1 5-benzyl-1,2,3,6-tetrahydro-4,6-diaza-cyclopenta[c]fluorene compounds and 5-benzyl-1,2,3,6-tetrahydro-4,6-diaza-cyclohepta[c]fluorene compounds
02/11/2010WO2010015586A2 2,3,4,7-tetrahydro-indolo[2,3-c]quinoline compounds
02/11/2010WO2010015585A1 6-benzyl-2,3,4,7-tetrahydro-indolo[2,3-c]quinoline compounds
02/11/2010WO2010015524A1 Method for stereoselective synthesis of bicyclic heterocyclene
02/11/2010WO2010015520A1 Substituted naphthyridines and use thereof as medicines
02/11/2010WO2010015518A2 4-dimethylamino-phenyl-substituted naphthyridines, and use thereof as medicaments
02/11/2010WO2010015090A1 Functionalized pyrrolidines and use thereof as iap inhibitors
02/11/2010WO2009138386A3 Alicyclic carboxylic acid derivatives of benzomorphans and related scaffolds, medicaments containing such compounds and their use
02/11/2010US20100036129 Process for the preparation of imidazopyridines
02/11/2010US20100036118 Fused Ring Heterocycle Kinase Modulators
02/11/2010US20100036102 Novel chelating agents and highly luminescent and stable chelates and their use
02/11/2010US20100035920 SUBSTITUTED PYRAZOLO[1,5-a] PYRIDINE COMPOUNDS AND THEIR METHODS OF USE
02/11/2010US20100035919 Compounds useful as inhibitors of protein kinases
02/11/2010US20100035918 Imidazolone Compounds and Methods of Making and Using the Same
02/11/2010US20100035917 Pyrrolo[2,3-b]pyridin-4-yl-benzenesulfonamide compounds as 1kk2 inhibitors
02/11/2010US20100035916 Azabicycloalkane derivatives, preparation thereof and use thereof in therapy
02/11/2010US20100035915 Indolizine derivatives and the use thereof as antidiabetics
02/11/2010US20100035912 Small Molecule Inhibitors of Retroviral Assembly and Maturation
02/11/2010US20100035902 5-aryl-substituted dihydropyridopyrimidines and dihydropyridazines and use thereof as mineral corticoid antagonists
02/11/2010US20100035898 Organic compounds
02/11/2010US20100035893 Triazolopyridine carboxamide derivatives, preparation thereof and therapeutic use thereof
02/11/2010US20100035892 Method for assembling high-purity chemical libraries, compounds suppressing acetyl coenzyme a carboxylase activities discovered by same
02/11/2010US20100035884 Kinase inhibitor
02/11/2010US20100035883 Dihydropyridophthalazinone inhibitors of poly(adp-ribose)polymerase (parp)
02/11/2010US20100035878 Inhibitors of c-jun n-terminal kinases for the treatment of neurodegenerative disorders relating to apoptosis and/or inflammation
02/11/2010US20100035875 Triazolopyridine jak inhibitor compounds and methods
02/11/2010US20100035869 Targeted nitroxide agents
02/11/2010US20100035756 Triazolophyridine derivatives as herbicides
02/11/2010US20100035279 Fluorescent Substrates for Monoamine Transporters as Optical False Neurotransmitters
02/11/2010DE102008036495A1 New naphthalene, perylene, benzoperylene, terrylene, quaterrylene bisimide and trisimide anions, as salts, e.g. tetrabutylammonium- or potassium-salts, useful e.g. to prepare dyes, preferably vats dye, to color cotton, paper and nylon
02/11/2010CA2732950A1 Imidazopyridin-2-one derivatives
02/11/2010CA2732762A1 Urotensin ii receptor antagonists
02/11/2010CA2732520A1 Therapeutic compounds
02/11/2010CA2732087A1 Substituted naphthyridines and their use as medicaments
02/11/2010CA2731926A1 4-dimethylamino-phenyl-substituted naphthyridines, and use thereof as medicaments
02/11/2010CA2731895A1 Process for the stereoselective preparation of bicyclic heterocycles
02/11/2010CA2731368A1 6 substituted 2-heterocyclylamino pyrazine compounds as chk-1 inhibitors
02/11/2010CA2731365A1 Tricyclic alkylaminomethyloxazolidinone derivatives
02/10/2010EP2151441A1 Beta-carbolin-derivates as substrates for an enzyme
02/10/2010EP2151435A1 Pharmaceutical composition for treatment of alzheimer's disease
02/10/2010EP2150552A1 1,3,8-trisubstituted-1,3,8-triaza-spiro[4.5]decan-4-one derivatives as ligands of the orl-i receptor for the treatment of anxiety and depression
02/10/2010EP2150543A2 Heterocyclic compounds with affinity to muscarinic receptors
02/10/2010EP2150255A1 Quinoxaline derivatives as p13 kinase inhibitors
02/10/2010EP2086965B1 Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
02/10/2010EP1747196B1 Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
02/10/2010EP1490365B1 Azaindoles as inhibitors of c-jun n-terminal kinases
02/10/2010CN101646668A Heterocycles as orexin antagonists
02/10/2010CN101643475A Amide substituted imidazole[1,2-a] pyridine compounds, preparation method thereof and application thereof
02/09/2010US7659398 Heating 4-chloro-1-isobutyl-1H-imidazo[4,5-c]quinoline with ammonia in a polar aprotic solvent to produce imiquimod; purification; industrial scale; dechlorination; precipitation, crystallization, slurrying, washing in a suitable solvent, filtration through a packed-bed column, dissolution in solvent
02/09/2010US7659298 2-(3-Phenyl-5-chloro-1-methyl-1H-pyrazol-4-ylmethylsulphanyl)-N-quinolin-3-ylbenzamide; 2-(3-Phenyl-5-chloro-1-methyl-1H-pyrazol-4-ylmethoxy)-N-naphthalin-2-ylbenzamide; obesity, including obesity of the non-insuline-dependent diabetes patients, sleeping disorders, stroke, nausea and vomiting
02/09/2010US7659283 Pyrrolo [3,2-C] pyridines useful as inhibitors of protein kinases
02/09/2010CA2557576C Novel benzothiazepine and benzothiepine compounds
02/09/2010CA2451962C Ecl labels having improved non-specific binding properties, methods of using and kits containing the same
02/09/2010CA2440760C Substituted pyrazolopyrimidines and thiazolopyrimidines used as analgesics
02/09/2010CA2430690C Perylene pigment compositions
02/09/2010CA2291065C Raf kinase inhibitors
02/09/2010CA2274201C Di-or triaza-spiro[4,5]decane derivatives
02/09/2010CA2201863C Substituted 4-biarylbutyric or 5-biarylpentanoic acids and derivatives as matrix metalloprotease inhibitors