Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559) |
---|
12/23/2010 | WO2010146488A1 Bicyclic and tricyclic compounds as kat ii inhibitors |
12/23/2010 | WO2010146348A2 New crystalline form of pemirolast |
12/23/2010 | WO2010146104A1 Thiadiazole derivatives and their use for the treatment of disorders mediated by slpl receptors |
12/23/2010 | WO2010146025A1 Tricyclic azabicyclo [4.1.0] heptane derivatives as inhibitors of serotonin, dopamine and norepinephrine re-uptake |
12/23/2010 | WO2010145998A1 Substituted pyrimidinylpyrrolopyridinone derivatives, process for their preparation and their use as kinase inhibitors |
12/23/2010 | WO2010145883A1 Novel substituted indazole and aza-indazole derivatives as gamma secretase modulators |
12/23/2010 | WO2010145208A1 Diazahomoadamantane derivatives and methods of use thereof |
12/23/2010 | WO2010095042A3 Pyridocarbazole type compounds and applications thereof |
12/23/2010 | WO2010052161A3 Herbicidal compositions |
12/23/2010 | US20100324294 Process for the preparation of 2,3,4,9-tetrahydro-1h-beta-carbolin-3-carboxylic acid esters |
12/23/2010 | US20100324293 Monofunctionalized Perylenetetracarboxylic Acid Bismides |
12/23/2010 | US20100324082 ENANTIOMERIC COMPOSITIONS OF 2-AMINO-1-(2-ISOPROPYLPYRAZOLO[1,5-a]PYRIDIN-3-YL)PROPAN-1-ONE AND RELATED METHODS |
12/23/2010 | US20100324072 Pyrrolopyridine derivatives and their use as bace inhibitors |
12/23/2010 | US20100324065 Compounds and methods for development of Ret Modulators |
12/23/2010 | US20100324055 Solid states forms of varenicline salts and processes for preparation thereof |
12/23/2010 | US20100324054 Aminotetrahydropyrans as dipeptidyl peptidase-iv inhibitors for the treatment or prevention of diabetes |
12/23/2010 | US20100324052 Novel piperidine carboxylic acid amine derivatives |
12/23/2010 | US20100324049 Diaryl ketimine derivative having antagonism against melanin-concentrating hormone receptor |
12/23/2010 | US20100324043 Bicyclic And Tricyclic Compounds As KAT II Inhibitors |
12/23/2010 | US20100324042 Heterocyclic compounds and their use as glycogen synthase kinase 3 inhibitors |
12/23/2010 | US20100324040 9-(pyrazol-3-yl)-9h-purine-2-amine and 3-(pyrazol-3-yl) -3h-imidazo[4,5-b] pyridin-5- amine derivatives and their use for the treatment of cancer |
12/23/2010 | US20100324036 Substituted imidazopyridine derivatives as melanocortin-4 receptor antagonists |
12/23/2010 | US20100324035 Carboxamide Compounds and Their Use |
12/23/2010 | US20100324028 Novel compounds |
12/23/2010 | US20100324024 Quinolizidinone M1 Receptor Positive Allosteric Modulators |
12/23/2010 | US20100324021 (dihydro)imidazoiso[5,1-a]quinolines |
12/23/2010 | US20100324009 Substituted Sulfonamide Compounds |
12/23/2010 | US20100322901 5, 6-ring annulated indole derivatives and use thereof |
12/23/2010 | US20100319778 Perylene semiconductors and methods of preparation and use thereof |
12/23/2010 | CA2765466A1 Diazahomoadamantane derivatives and methods of use thereof |
12/23/2010 | CA2765415A1 Substituted -1,3,8-triazaspiro[4.5]decane-2,4-diones |
12/23/2010 | CA2765408A1 New crystalline form of pemirolast |
12/23/2010 | CA2763960A1 Bicyclic and tricyclic compounds as kat ii inhibitors |
12/23/2010 | CA2755467A1 Novel substituted indazole and aza-indazole derivatives as gamma secretase modulators |
12/22/2010 | EP2264033A1 3,5-DIPHENYL-SUBSTITUTED PYRROLO[2,3b]PYRIDINES USEFUL AS KINASE INHIBITORS |
12/22/2010 | EP2264032A2 Hiv protease inhibiting sulfonamides |
12/22/2010 | EP2264028A1 Pyrazole compounds useful as protein kinase inhibitors |
12/22/2010 | EP2263669A1 Pharmaceutically active isoindoline derivatives |
12/22/2010 | EP2262805A1 Polysubstituted derivatives of 2-heteroaryl-6-phenyl-imidazo[l,2-a] pyridines, and preparation and therapeutic use thereof |
12/22/2010 | EP2262804A1 Polysubstituted derivatives of 6-heteroaryl-imidazo[l,2- a] pyridines, and preparation and therapeutic use thereof |
12/22/2010 | EP2262803A1 Polysubstituted derivatives of 2-aryl-6-phenyl-imidazo[l,2-a] pyridines, and preparation and therapeutic use thereof |
12/22/2010 | EP2262784A1 Inhibitors of the chemokine receptor cxcr3 |
12/22/2010 | EP2262780A2 Amorphous varenicline tartrate |
12/22/2010 | EP2262769A1 Polysubstituted 2-aryl-6-phenyl-imidazo[1,2-a]pyridine derivatives, and preparation and therapeutic use thereof |
12/22/2010 | EP2262505A2 Substituted heterocycle fused gamma-carbolines solid |
12/22/2010 | EP2178873B1 6-phenyl-1h-imidazo[4,5-c]pyridine-4-carbonitrile derivatives as cathepsin inhibitors |
12/22/2010 | EP1891066B1 Compounds and compositions as protein kinase inhibitors |
12/22/2010 | CN1988907B Dual small molecule inhibitors of cancer and angiogenesis |
12/22/2010 | CN1809357B Small molecule Toll-like receptor (TLR) antagonists |
12/22/2010 | CN101925601A Enantiomerically pure (-) 2-[1-(7-methyl-2-(morpholin-4-yl)-4-oxo-4h-pyrido[1,2-a]pyrimidin-9-yl)ethylamino]benzoic acid, its use in medical therapy, and pharmaceutical composition comprising it - 026 |
12/22/2010 | CN101925383A Carboxamide compounds and their use as chemokine receptor agonists |
12/22/2010 | CN101921279A Spirocyclic heterocyclic derivatives and methods of their use |
12/22/2010 | CN101921272A Method for extracting and separating laburnine |
12/22/2010 | CN101921271A Pyridine [2,3-d] pyrimidone compounds and application thereof to pharmacy |
12/22/2010 | CN101921268A 5-thiazole amide compound and biology application thereof |
12/22/2010 | CN101921229A Synthesis method of stepholidine or derivative optical isomer thereof and intermediate thereof |
12/22/2010 | CN101445507B Method for preparing praziquantel |
12/22/2010 | CN101367823B Method for separating citrate, evodiamine and rutaecarpine from evodia rutaecarpa |
12/22/2010 | CN101302227B Method for synthesizing 3,3'-purrocoline compounds |
12/22/2010 | CN101302217B Triazole compounds, preparation and use thereof |
12/22/2010 | CN101208340B Pyrazolopyridine derivatives as inhibitors of beta-adrenergic receptor kinase 1 |
12/22/2010 | CN101137656B Crystal forms of an imidazole derivative |
12/22/2010 | CN101128461B Imidazo (1, 2-a) pyridine compounds as VEGF-R2 inhibitors |
12/22/2010 | CN101048406B Novel substituted imidazole derivatives |
12/22/2010 | CA2708723A1 Solid states forms of varenicline salts and processes for preparation thereof |
12/21/2010 | US7855295 Tetrahydrocarboline compounds as anticancer agents |
12/21/2010 | US7855294 (6R,8S)-6-(spiro[isobenzofuran-1-(3H), 4'-piperidin]-1'-ylmethyl)-5,6,7,8-tetrahydroquinolin-8-ol), exhibiting an antagonism to binding of nociceptin to opioid receptor-like-1 receptors, useful as medicines for diseases associated with pain and appetite control or memory and learning |
12/21/2010 | US7855216 e.g. 3-(4-Bromo-2-fluoro-phenylamino)-1-methyl-1H-pyrrolo[3,2-c]pyridine-2-carboxylic acid ethyl ester; MEK kinase (Mitogen-Activated protein kinase kinase) inhibitor; anticarcinogenic, antiinflammatory agent; rheumatoid arthritis |
12/21/2010 | US7855214 Autoimmune, inflammatory, proliferative, or hyperproliferative disease or an immunologically-mediated disease; inhibitors of the Tec family of non-receptor tyrosine kinases; compounds are quinazolino[3,2-a]quinazolin-12-ones |
12/21/2010 | US7855206 antidiabetic agents such as (1S,2R,5S)-5-(2-Methyl-6,8-dihydro-7H-pyrazolo[1,5-a]pyrrolo[3,4-e]pyrimidin-7-yl)-2-(2,4,5-trifluorophenyl)cyclohexanamine bis-hydrochloride salt, used for treating non-insulin dependent diabetes |
12/21/2010 | US7855202 useful in the treatment respiratory system disorders, allergic diseases, inflammation, reperfusion injury, ischemia, atherosclerosis, hypertension, retinopathy, diabetes, gastrointestinal disorders and/or autoimmune diseases |
12/21/2010 | US7855198 Benzamide derivative or salt thereof |
12/21/2010 | US7855194 Pyrimidine, quinazoline, pteridine and triazine derivatives |
12/21/2010 | CA2543201C ((ir, 3s)-3-isopropyl-3-{ [3-(trifluoromethyl)-7, 8-dihydro-1, 6-naphthyridin-6 (5h)-yl] carbonyl} cyclopentyl) [(3s, 4s)-3-methoxytetrahydro-2h-pyran-4-yl] amine succinate salt, composition thereof, and its use in the treatment of inflammatory diseases |
12/21/2010 | CA2480046C Improved method of making nevirapine |
12/21/2010 | CA2426654C 2,4,8-trisubstituted-8h-pyrido[2,3-d}pyrimidin-7-one compounds |
12/21/2010 | CA2404594C Agent for prophylaxis and treatment of renal disease |
12/16/2010 | WO2010144647A1 Nicotinamide compounds useful as kinase modulators |
12/16/2010 | WO2010144486A1 Dihydropyrrolonaphtyridinone compounds as inhibitors of jak |
12/16/2010 | WO2010144416A1 SUBSTITUTED PYRAZOLO [1,5-a] PYRIDINE COMPOUNDS HAVING MULTI-TARGET ACTIVITY |
12/16/2010 | WO2010143733A1 Novel fused cyclic compound and use thereof |
12/16/2010 | WO2010143664A1 Tetracyclic compound |
12/16/2010 | WO2010142974A1 mCPP IMMUNOASSAY |
12/16/2010 | WO2010142628A1 Pyrazole oxadiazole derivatives as s1p1 agonists |
12/16/2010 | WO2010142576A1 Novel sterically hindered amine light stabilizers |
12/16/2010 | WO2010142426A1 Hedgehog pathway antagonists and therapeutic applications thereof |
12/16/2010 | WO2010142402A1 Substituted benzimidazoles, benzothiazoles and benzoxazoles |
12/16/2010 | WO2010116122A3 Herbicidal quinoline and 1,8 -naphthyridine compounds |
12/16/2010 | US20100317689 Prodrugs of proton pump inhibitors including the 1h-imidazo[4,5-b] pyridine moiety |
12/16/2010 | US20100317688 2-HETEROAROYLIMIDAZOL[1,2-a]PYRIDINE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF |
12/16/2010 | US20100317687 2-BENZOYLIMIDAZO[1,2-a]PYRIDINE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF |
12/16/2010 | US20100317686 N-HETEROCYCLIC-6-HETEROCYCLIC-IMIDAZO[1,2-a]PYRIDINE-2-CARBOXAMIDE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF |
12/16/2010 | US20100317685 N-PHENYL-IMIDAZO[1,2-a]PYRIDINE-2-CARBOXAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
12/16/2010 | US20100317684 Amide and Carbamate Derivatives of N-{2-[4-Amino-2- (Ethoxymethyl)-1H-Imidazo[4,5-c] Quinolin-1-Yl]-1,1-Dimethylethyl} Methanesulfonamide and Methods |
12/16/2010 | US20100317676 Fused heterocyclic compounds, and compositions and uses thereof |
12/16/2010 | US20100317675 6-HETEROCYCLIC-IMIDAZO[1,2-a]PYRIDINE-2-CARBOXAMIDE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF |
12/16/2010 | US20100317673 N-HETEROCYCLIC-IMIDAZO[1,2-a]PYRIDINE-2-CARBOXAMIDE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
12/16/2010 | US20100317672 Monomaleate Monohydrate Salt of a 5HT1A Receptor Antagonist |
12/16/2010 | US20100317667 1-aryl-or 1-heteroaryl-pyrido[B]indoles and uses thereof |
12/16/2010 | US20100317660 Mediators of hedgehog signaling pathways, compositions and uses related thereto |